AU545491B2

AU545491B2 – Benzodiazepine derivatives
– Google Patents

AU545491B2 – Benzodiazepine derivatives
– Google Patents
Benzodiazepine derivatives

Info

Publication number
AU545491B2

AU545491B2
AU66819/81A
AU6681981A
AU545491B2
AU 545491 B2
AU545491 B2
AU 545491B2
AU 66819/81 A
AU66819/81 A
AU 66819/81A
AU 6681981 A
AU6681981 A
AU 6681981A
AU 545491 B2
AU545491 B2
AU 545491B2
Authority
AU
Australia
Prior art keywords
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
1980-02-08
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Ceased

Application number
AU66819/81A
Other versions

AU6681981A
(en

Inventor
Quirico Branca
Albert Eduard Fischli
Andre Szente
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

F Hoffmann La Roche AG

Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1980-02-08
Filing date
1981-02-02
Publication date
1985-07-18

1981-02-02
Application filed by F Hoffmann La Roche AG
filed
Critical
F Hoffmann La Roche AG

1981-08-13
Publication of AU6681981A
publication
Critical
patent/AU6681981A/en

1985-07-18
Application granted
granted
Critical

1985-07-18
Publication of AU545491B2
publication
Critical
patent/AU545491B2/en

2001-02-02
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms

C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4

C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems

C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines

C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals

C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms

C07D243/24—Oxygen atoms

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P3/00—Drugs for disorders of the metabolism

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P5/00—Drugs for disorders of the endocrine system

A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P9/00—Drugs for disorders of the cardiovascular system

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P9/00—Drugs for disorders of the cardiovascular system

A61P9/12—Antihypertensives

AU66819/81A
1980-02-08
1981-02-02
Benzodiazepine derivatives

Ceased

AU545491B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

CH1039/80

1980-02-08

CH103980

1980-02-08

Publications (2)

Publication Number
Publication Date

AU6681981A

AU6681981A
(en)

1981-08-13

AU545491B2
true

AU545491B2
(en)

1985-07-18

Family
ID=4201027
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU66819/81A
Ceased

AU545491B2
(en)

1980-02-08
1981-02-02
Benzodiazepine derivatives

Country Status (8)

Country
Link

US
(1)

US4361511A
(en)

EP
(1)

EP0033973B1
(en)

JP
(1)

JPS56125375A
(en)

AU
(1)

AU545491B2
(en)

CA
(1)

CA1145333A
(en)

DE
(1)

DE3160986D1
(en)

DK
(1)

DK39581A
(en)

ZA
(1)

ZA81694B
(en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

CA1163266A
(en)

*

1980-07-31
1984-03-06
Albert E. Fischli
Benzodiazepine derivatives

PT100631B
(en)

*

1991-06-28
1999-06-30
Smithkline Beecham Corp

BICYCLE FIBRINOGENIC ANTAGONISTS, ITS USE AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM

US5939412A
(en)

*

1992-06-26
1999-08-17
Smithkline Beecham Corporation
Bicyclic fibrinogen antagonists

US6403578B1
(en)

1993-12-21
2002-06-11
Smithkline Beecham Corporation
Bicyclic fibrinogen antagonists

MA23420A1
(en)

*

1994-01-07
1995-10-01
Smithkline Beecham Corp

BICYCLIC FIBRINOGEN ANTAGONISTS.

US6458784B1
(en)

1994-06-29
2002-10-01
Smithkline Beecham Corporation
Vitronectin receptor antagonists

US5977101A
(en)

*

1995-06-29
1999-11-02
Smithkline Beecham Corporation
Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity

WO2006132295A1
(en)

*

2005-06-09
2006-12-14
Dainippon Sumitomo Pharma Co., Ltd.
Regulator of aldosterone receptor

Family Cites Families (5)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US3371085A
(en)

*

1959-12-10
1968-02-27
Hoffmann La Roche
5-aryl-3h-1,4-benzodiazepin-2(1h)-ones

US3464978A
(en)

*

1967-04-21
1969-09-02
Hoffmann La Roche
1-substituted urea alkyl 1,2-dihydro-1,4-benzodiazepines and benzodiazepin – 2-ones

BE787117A
(en)

*

1971-08-04
1973-02-05
Hoffmann La Roche

BENZODIAZEPINE DERIVATIVES

JPS5084590A
(en)

*

1973-11-28
1975-07-08

US4251444A
(en)

*

1980-04-07
1981-02-17
American Home Products Corporation
Thiazepino-[4,3-b]-isoquinoline-1,5-dione derivatives and precursors

1980

1980-12-01
CA
CA000365868A
patent/CA1145333A/en
not_active
Expired

1981

1981-01-16
US
US06/225,746
patent/US4361511A/en
not_active
Expired – Fee Related

1981-01-29
DK
DK39581A
patent/DK39581A/en
not_active
Application Discontinuation

1981-02-02
AU
AU66819/81A
patent/AU545491B2/en
not_active
Ceased

1981-02-02
ZA
ZA00810694A
patent/ZA81694B/en
unknown

1981-02-05
JP
JP1511681A
patent/JPS56125375A/en
active
Pending

1981-02-09
DE
DE8181100906T
patent/DE3160986D1/en
not_active
Expired

1981-02-09
EP
EP81100906A
patent/EP0033973B1/en
not_active
Expired

Also Published As

Publication number
Publication date

AU6681981A
(en)

1981-08-13

EP0033973B1
(en)

1983-09-28

JPS56125375A
(en)

1981-10-01

DK39581A
(en)

1981-08-09

DE3160986D1
(en)

1983-11-03

US4361511A
(en)

1982-11-30

CA1145333A
(en)

1983-04-26

EP0033973A1
(en)

1981-08-19

ZA81694B
(en)

1982-03-31

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(en)

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