AU551338B2

AU551338B2 – 6-(aminomethyl) penicillanic acid 1,1-dioxide esters
– Google Patents

AU551338B2 – 6-(aminomethyl) penicillanic acid 1,1-dioxide esters
– Google Patents
6-(aminomethyl) penicillanic acid 1,1-dioxide esters

Info

Publication number
AU551338B2

AU551338B2
AU29078/84A
AU2907884A
AU551338B2
AU 551338 B2
AU551338 B2
AU 551338B2
AU 29078/84 A
AU29078/84 A
AU 29078/84A
AU 2907884 A
AU2907884 A
AU 2907884A
AU 551338 B2
AU551338 B2
AU 551338B2
Authority
AU
Australia
Prior art keywords
aminomethyl
penicillanic acid
dioxide esters
esters
dioxide
Prior art date
1983-06-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Ceased

Application number
AU29078/84A
Other versions

AU2907884A
(en

Inventor
Wayne Ernest Barth
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pfizer Inc

Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1983-06-06
Filing date
1984-06-05
Publication date
1986-04-24

1984-06-05
Application filed by Pfizer Inc
filed
Critical
Pfizer Inc

1984-12-13
Publication of AU2907884A
publication
Critical
patent/AU2907884A/en

1986-04-24
Application granted
granted
Critical

1986-04-24
Publication of AU551338B2
publication
Critical
patent/AU551338B2/en

2004-06-05
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom

C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems

C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans

C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Abstract

6-alpha- and 6-beta-(Aminomethyl)penicillanic acid, 1,1-dioxide esters which are hydrolyzable under physiological conditions, particularly those wherein the ester radical is 1H-isobenzofuran-3-on-1-yl or (5-methyl-1,3-dioxol-2-on-4-yl)methyl, and an improved process and intermediates used in their synthesis.

AU29078/84A
1983-06-06
1984-06-05
6-(aminomethyl) penicillanic acid 1,1-dioxide esters

Ceased

AU551338B2
(en)

Applications Claiming Priority (4)

Application Number
Priority Date
Filing Date
Title

US50145183A

1983-06-06
1983-06-06

US501451

1983-06-06

US06/577,478

US4536393A
(en)

1983-06-06
1984-02-06
6-(Aminomethyl)penicillanic acid 1,1-dioxide esters and intermediates therefor

US577478

1984-02-06

Publications (2)

Publication Number
Publication Date

AU2907884A

AU2907884A
(en)

1984-12-13

AU551338B2
true

AU551338B2
(en)

1986-04-24

Family
ID=27053819
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU29078/84A
Ceased

AU551338B2
(en)

1983-06-06
1984-06-05
6-(aminomethyl) penicillanic acid 1,1-dioxide esters

Country Status (19)

Country
Link

US
(1)

US4536393A
(en)

EP
(1)

EP0128719B1
(en)

KR
(1)

KR870000323B1
(en)

AT
(1)

ATE23862T1
(en)

AU
(1)

AU551338B2
(en)

CA
(1)

CA1206957A
(en)

DE
(1)

DE3461467D1
(en)

DK
(1)

DK275784A
(en)

ES
(1)

ES533146A0
(en)

FI
(1)

FI842254A
(en)

GR
(1)

GR82215B
(en)

HU
(1)

HU193930B
(en)

IL
(1)

IL72005A
(en)

NO
(1)

NO842249L
(en)

NZ
(1)

NZ208382A
(en)

PH
(1)

PH19077A
(en)

PL
(1)

PL143943B1
(en)

PT
(1)

PT78688A
(en)

YU
(1)

YU97384A
(en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4590073A
(en)

*

1984-10-22
1986-05-20
Pfizer Inc.
6-substituted penicillanic acid 1,1-dioxide compounds

US4613462A
(en)

*

1985-07-02
1986-09-23
Pfizer, Inc.
6-substituted penicillanic acid 1,1-dioxide compounds

US5006661A
(en)

*

1987-06-16
1991-04-09
University Of Cincinnati
Selective stereospecific biologically active beta-lactams

US4855419A
(en)

*

1987-06-16
1989-08-08
University Of Cincinnati
Application of 4-[1-oxoalkyl]-2,5-oxazolidinediones in selective stereospecific formation of biologically active α-lactams

GB2206579B
(en)

*

1987-07-10
1991-05-29
Erba Farmitalia
6a and 6b-(substituted methyl)-penicillanic acid derivatives

Family Cites Families (15)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US3487079A
(en)

*

1966-01-14
1969-12-30
Bristol Myers Co
Certain alpha-amino bicyclic beta-lactam carboxylic acids

US4207323A
(en)

*

1975-11-21
1980-06-10
Merck & Co., Inc.
6-Substituted methyl penicillins, derivatives and analogues thereof

US4234579A
(en)

*

1977-06-07
1980-11-18
Pfizer Inc.
Penicillanic acid 1,1-dioxides as β-lactamase inhibitors

IE49880B1
(en)

*

1979-02-13
1986-01-08
Leo Pharm Prod Ltd
Penicillin derivatives

US4237051A
(en)

*

1979-04-19
1980-12-02
Schering Corporation
Stereospecific production of 6- or 7-carbon-substituted-β-lactams

US4309347A
(en)

*

1979-05-16
1982-01-05
Pfizer Inc.
Penicillanoyloxymethyl penicillanate 1,1,1′,1′-tetraoxide

US4244951A
(en)

*

1979-05-16
1981-01-13
Pfizer Inc.
Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide

DE2927004A1
(en)

*

1979-07-04
1981-05-27
Bayer Ag, 5090 Leverkusen

PENICILLANIC ACID 1,1-DIOXIDES, THEIR PRODUCTION AND THEIR USE AS MEDICINAL PRODUCTS AS MEDICINAL PRODUCTS

US4287181A
(en)

*

1979-10-22
1981-09-01
Pfizer Inc.
Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors

US4342768A
(en)

*

1979-10-22
1982-08-03
Pfizer Inc.
Bis-esters of 1,1-alkanediols with 6-beta-hydroxymethylpenicillanic acid 1,1-dioxide and beta-lactam antibiotics

US4260598A
(en)

*

1979-10-22
1981-04-07
Pfizer Inc.
Method for increasing antibacterial effectiveness of a β-lactam antibiotic

JPS6019908B2
(en)

*

1980-04-30
1985-05-18
カネボウ株式会社

1,3-dioxolen-2-one derivative

CA1212105A
(en)

*

1980-04-30
1986-09-30
Shoji Ikeda
Ampicillin esters and production thereof

EP0069962B1
(en)

*

1981-07-15
1985-01-02
Kanebo, Ltd.
Novel ester of 1,1-dioxopenicillanic acid, process for production thereof, and use thereof as beta-lactamase inhibitor

JPS5832882A
(en)

*

1981-07-18
1983-02-25
Kanebo Ltd
Novel ester of 6-((hexahydro-1h-azepin-1-yl)- methyleneamino)penicillanic acid and its preparation

1984

1984-02-06
US
US06/577,478
patent/US4536393A/en
not_active
Expired – Lifetime

1984-06-01
PH
PH30754A
patent/PH19077A/en
unknown

1984-06-04
AT
AT84303736T
patent/ATE23862T1/en
not_active
IP Right Cessation

1984-06-04
EP
EP84303736A
patent/EP0128719B1/en
not_active
Expired

1984-06-04
CA
CA000455813A
patent/CA1206957A/en
not_active
Expired

1984-06-04
PT
PT78688A
patent/PT78688A/en
unknown

1984-06-04
IL
IL72005A
patent/IL72005A/en
unknown

1984-06-04
DE
DE8484303736T
patent/DE3461467D1/en
not_active
Expired

1984-06-04
DK
DK275784A
patent/DK275784A/en
not_active
Application Discontinuation

1984-06-04
GR
GR74910A
patent/GR82215B/el
unknown

1984-06-04
PL
PL1984248044A
patent/PL143943B1/en
unknown

1984-06-05
NO
NO842249A
patent/NO842249L/en
unknown

1984-06-05
NZ
NZ208382A
patent/NZ208382A/en
unknown

1984-06-05
FI
FI842254A
patent/FI842254A/en
not_active
Application Discontinuation

1984-06-05
AU
AU29078/84A
patent/AU551338B2/en
not_active
Ceased

1984-06-05
YU
YU00973/84A
patent/YU97384A/en
unknown

1984-06-05
KR
KR1019840003121A
patent/KR870000323B1/en
not_active
IP Right Cessation

1984-06-05
ES
ES533146A
patent/ES533146A0/en
active
Granted

1984-06-05
HU
HU842177A
patent/HU193930B/en
unknown

Also Published As

Publication number
Publication date

ATE23862T1
(en)

1986-12-15

PL143943B1
(en)

1988-03-31

EP0128719A1
(en)

1984-12-19

PT78688A
(en)

1984-07-01

FI842254A0
(en)

1984-06-05

PH19077A
(en)

1985-12-19

FI842254A
(en)

1984-12-07

NO842249L
(en)

1984-12-07

IL72005A0
(en)

1984-10-31

NZ208382A
(en)

1987-05-29

US4536393A
(en)

1985-08-20

DK275784A
(en)

1984-12-07

HU193930B
(en)

1987-12-28

AU2907884A
(en)

1984-12-13

DE3461467D1
(en)

1987-01-15

CA1206957A
(en)

1986-07-02

PL248044A1
(en)

1985-03-26

ES8506023A1
(en)

1985-06-01

KR850000445A
(en)

1985-02-27

EP0128719B1
(en)

1986-11-26

KR870000323B1
(en)

1987-02-27

ES533146A0
(en)

1985-06-01

YU97384A
(en)

1986-06-30

IL72005A
(en)

1988-02-29

DK275784D0
(en)

1984-06-04

GR82215B
(en)

1984-12-13

HUT34202A
(en)

1985-02-28

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