AU5806286A – 11-B substituted steroids and process for their preparation
– Google Patents
AU5806286A – 11-B substituted steroids and process for their preparation
– Google Patents
11-B substituted steroids and process for their preparation
Info
Publication number
AU5806286A
AU5806286A
AU58062/86A
AU5806286A
AU5806286A
AU 5806286 A
AU5806286 A
AU 5806286A
AU 58062/86 A
AU58062/86 A
AU 58062/86A
AU 5806286 A
AU5806286 A
AU 5806286A
AU 5806286 A
AU5806286 A
AU 5806286A
Authority
AU
Australia
Prior art keywords
preparation
substituted steroids
steroids
substituted
Prior art date
1985-05-31
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU58062/86A
Other versions
AU587031B2
(en
Inventor
Roberto D’alessio
Enrico Di Salle
Franco Faustini
Vittoria Villa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1985-05-31
Filing date
1986-05-29
Publication date
1986-12-04
1986-05-29
Application filed by Farmitalia Carlo Erba SRL
filed
Critical
Farmitalia Carlo Erba SRL
1986-12-04
Publication of AU5806286A
publication
Critical
patent/AU5806286A/en
1989-08-03
Application granted
granted
Critical
1989-08-03
Publication of AU587031B2
publication
Critical
patent/AU587031B2/en
2006-05-29
Anticipated expiration
legal-status
Critical
Status
Ceased
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P5/00—Drugs for disorders of the endocrine system
A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
C07J1/0051—Estrane derivatives
C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
C07J1/0074—Esters
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
C07J1/0051—Estrane derivatives
C07J1/0081—Substituted in position 17 alfa and 17 beta
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
C07J21/005—Ketals
C07J21/006—Ketals at position 3
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
C07J71/0005—Oxygen-containing hetero ring
C07J71/001—Oxiranes
AU58062/86A
1985-05-31
1986-05-29
11-B substituted steroids and process for their preparation
Ceased
AU587031B2
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
GB858513723A
GB8513723D0
(en)
1985-05-31
1985-05-31
11-beta substituted steroids
GB8513723
1985-05-31
Publications (2)
Publication Number
Publication Date
AU5806286A
true
AU5806286A
(en)
1986-12-04
AU587031B2
AU587031B2
(en)
1989-08-03
Family
ID=10579949
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU58062/86A
Ceased
AU587031B2
(en)
1985-05-31
1986-05-29
11-B substituted steroids and process for their preparation
Country Status (21)
Country
Link
JP
(1)
JPS6212796A
(en)
KR
(1)
KR860009035A
(en)
AU
(1)
AU587031B2
(en)
BE
(1)
BE904846A
(en)
CH
(1)
CH669385A5
(en)
DE
(1)
DE3617883A1
(en)
DK
(1)
DK251386A
(en)
ES
(1)
ES8707972A1
(en)
FI
(1)
FI862278A
(en)
FR
(1)
FR2582654B1
(en)
GB
(2)
GB8513723D0
(en)
GR
(1)
GR861405B
(en)
HU
(1)
HU197925B
(en)
IL
(1)
IL78957A
(en)
IT
(1)
IT1190014B
(en)
NL
(1)
NL8601387A
(en)
NZ
(1)
NZ216325A
(en)
PT
(1)
PT82665B
(en)
SE
(1)
SE8602449L
(en)
SU
(1)
SU1508963A3
(en)
ZA
(1)
ZA864065B
(en)
Cited By (1)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
AU613433B2
(en)
*
1987-12-12
1991-08-01
Akzo N.V.
New 11-arylsteroik compounds
Families Citing this family (6)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
ES2045082T3
(en)
*
1987-04-24
1994-01-16
Akzo Nv
A METHOD FOR THE PREPARATION OF NEW DERIVATIVES 11-ARILESTRANO AND 11-ARILPREGNANO.
FR2665901B2
(en)
*
1989-02-24
1994-07-29
Roussel Uclaf
NEW 19-NOR STEROUIDES HAVING IN THE 11BETA POSITION A CARBON CHAIN COMPRISING AN AMIDE FUNCTION, THEIR PREPARATION, THEIR APPLICATION AS MEDICAMENTS.
FR2643638B1
(en)
*
1989-02-24
1991-06-14
Roussel Uclaf
NOVEL 19-NOR STEROIDS HAVING IN THE 11BETA POSITION A CARBON CHAIN COMPRISING AN AMIDE OR CARBAMATE FUNCTION, THEIR PREPARATION METHOD AND INTERMEDIATES THEREOF, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
TWI265167B
(en)
*
1999-11-29
2006-11-01
Akzo Nobel Nv
3-methylene steroid derivatives
DE19961219A1
(en)
*
1999-12-15
2001-07-19
Jenapharm Gmbh
11beta-phenyltratriene derivatives with fluoroalkyl groups in the aromatic side chain, their preparation and pharmaceutical compositions containing these compounds
TW200531977A
(en)
2004-03-25
2005-10-01
Akzo Nobel Nv
Progesterone receptor modulators
Family Cites Families (10)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
CH488682A
(en)
*
1965-07-30
1970-04-15
Ciba Geigy
Process for the preparation of 4,9,11-trienes of the 19-nor-androstane series
FR205F
(en)
*
1965-10-22
FR5913M
(en)
*
1965-12-02
1968-04-01
NL128375C
(en)
*
1966-02-18
FR2054525B1
(en)
*
1969-07-28
1973-01-12
Roussel Uclaf
FR2054527B1
(en)
*
1969-07-28
1973-06-08
Roussel Uclaf
FR2377418A1
(en)
*
1977-01-13
1978-08-11
Roussel Uclaf
NEW 4,9-DIENIC 11B-SUBSTITUTE STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS
ZA8231B
(en)
*
1981-01-09
1982-11-24
Roussel Uclaf
New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained
FR2522328B1
(en)
*
1982-03-01
1986-02-14
Roussel Uclaf
NEW PRODUCTS DERIVED FROM THE STRUCTURE 3-CETO 4,9 19-NOR STEROIDS, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
NZ214998A
(en)
*
1985-02-07
1989-06-28
Schering Ag
13-(methyl or ethyl)-11-beta-phenyl-gonane derivatives; preparatory processes and pharmaceutical compositions
1985
1985-05-31
GB
GB858513723A
patent/GB8513723D0/en
active
Pending
1986
1986-05-23
ES
ES555298A
patent/ES8707972A1/en
not_active
Expired
1986-05-27
GB
GB08612866A
patent/GB2175905B/en
not_active
Expired
1986-05-27
HU
HU862228A
patent/HU197925B/en
not_active
IP Right Cessation
1986-05-28
PT
PT82665A
patent/PT82665B/en
not_active
IP Right Cessation
1986-05-28
DE
DE19863617883
patent/DE3617883A1/en
not_active
Withdrawn
1986-05-28
CH
CH2152/86A
patent/CH669385A5/de
not_active
IP Right Cessation
1986-05-28
NZ
NZ216325A
patent/NZ216325A/en
unknown
1986-05-28
IT
IT20598/86A
patent/IT1190014B/en
active
1986-05-28
IL
IL78957A
patent/IL78957A/en
unknown
1986-05-28
FR
FR8607660A
patent/FR2582654B1/en
not_active
Expired
1986-05-29
SE
SE8602449A
patent/SE8602449L/en
not_active
Application Discontinuation
1986-05-29
SU
SU864027509A
patent/SU1508963A3/en
active
1986-05-29
DK
DK251386A
patent/DK251386A/en
not_active
Application Discontinuation
1986-05-29
AU
AU58062/86A
patent/AU587031B2/en
not_active
Ceased
1986-05-29
GR
GR861405A
patent/GR861405B/en
unknown
1986-05-29
FI
FI862278A
patent/FI862278A/en
not_active
Application Discontinuation
1986-05-29
NL
NL8601387A
patent/NL8601387A/en
not_active
Application Discontinuation
1986-05-30
JP
JP61123893A
patent/JPS6212796A/en
active
Pending
1986-05-30
KR
KR1019860004283A
patent/KR860009035A/en
not_active
Application Discontinuation
1986-05-30
ZA
ZA864065A
patent/ZA864065B/en
unknown
1986-05-30
BE
BE0/216722A
patent/BE904846A/en
not_active
IP Right Cessation
Cited By (1)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
AU613433B2
(en)
*
1987-12-12
1991-08-01
Akzo N.V.
New 11-arylsteroik compounds
Also Published As
Publication number
Publication date
SE8602449D0
(en)
1986-05-29
NZ216325A
(en)
1989-01-27
FR2582654B1
(en)
1988-06-03
FI862278A
(en)
1986-12-01
GB2175905B
(en)
1989-01-18
ES8707972A1
(en)
1987-09-01
SE8602449L
(en)
1986-12-01
KR860009035A
(en)
1986-12-19
IL78957A0
(en)
1986-09-30
HUT44575A
(en)
1988-03-28
DK251386A
(en)
1986-12-01
AU587031B2
(en)
1989-08-03
FI862278A0
(en)
1986-05-29
GB8513723D0
(en)
1985-07-03
SU1508963A3
(en)
1989-09-15
GR861405B
(en)
1986-09-26
ES555298A0
(en)
1987-09-01
IT1190014B
(en)
1988-02-10
IT8620598A1
(en)
1987-11-28
NL8601387A
(en)
1986-12-16
PT82665B
(en)
1988-08-17
BE904846A
(en)
1986-12-01
IT8620598D0
(en)
1986-05-28
JPS6212796A
(en)
1987-01-21
FR2582654A1
(en)
1986-12-05
DE3617883A1
(en)
1986-12-04
PT82665A
(en)
1986-06-01
ZA864065B
(en)
1987-01-28
DK251386D0
(en)
1986-05-29
GB8612866D0
(en)
1986-07-02
GB2175905A
(en)
1986-12-10
IL78957A
(en)
1990-11-29
HU197925B
(en)
1989-06-28
CH669385A5
(en)
1989-03-15
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