AU616351B2 - Creación de Inventos y Patentes con Inteligencia Artificial

AU616351B2 – Processes for preparing 1,5-benzothiazepine derivatives
– Google Patents

AU616351B2 – Processes for preparing 1,5-benzothiazepine derivatives
– Google Patents
Processes for preparing 1,5-benzothiazepine derivatives

Info

Publication number
AU616351B2

AU616351B2
AU53856/90A
AU5385690A
AU616351B2
AU 616351 B2
AU616351 B2
AU 616351B2
AU 53856/90 A
AU53856/90 A
AU 53856/90A
AU 5385690 A
AU5385690 A
AU 5385690A
AU 616351 B2
AU616351 B2
AU 616351B2
Authority
AU
Australia
Prior art keywords
preparing
formula
processes
benzothiazepine derivatives
chem
Prior art date
1989-04-28
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
AU53856/90A
Other versions

AU5385690A
(en

Inventor
Hironori Hayashi
Masashi Kitano
Sadao Maeda
Shigeru Nishimoto
Tamotsu Okuno
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Tanabe Seiyaku Co Ltd

Original Assignee
Tanabe Seiyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1989-04-28
Filing date
1990-04-26
Publication date
1991-10-24

1990-04-26
Application filed by Tanabe Seiyaku Co Ltd
filed
Critical
Tanabe Seiyaku Co Ltd

1990-11-01
Publication of AU5385690A
publication
Critical
patent/AU5385690A/en

1991-10-24
Application granted
granted
Critical

1991-10-24
Publication of AU616351B2
publication
Critical
patent/AU616351B2/en

2010-04-26
Anticipated expiration
legal-status
Critical

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms

C07D281/02—Seven-membered rings

C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4

C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems

C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Abstract

There is disclosed a process for preparing 1,5-benzothiazepine derivatives represented by the formula: wherein R is a lower alkyl group, which comprises subjecting a propionic acid compound represented by the formula: wherein R has the same meaning as defined above, to intramolecular ring closing reaction in the presence of a sulfonic acid compound represented by the formula: R<1>SO3H (III) wherein R<1> represents a lower alkyl group or a substituted or unsubstituted phenyl group.

AU53856/90A
1989-04-28
1990-04-26
Processes for preparing 1,5-benzothiazepine derivatives

Expired

AU616351B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

JP1109795A

JPH0798813B2
(en)

1989-04-28
1989-04-28

Process for producing 1,5-benzothiazepine derivative

JP1-109795

1989-04-28

Publications (2)

Publication Number
Publication Date

AU5385690A

AU5385690A
(en)

1990-11-01

AU616351B2
true

AU616351B2
(en)

1991-10-24

Family
ID=14519414
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU53856/90A
Expired

AU616351B2
(en)

1989-04-28
1990-04-26
Processes for preparing 1,5-benzothiazepine derivatives

Country Status (16)

Country
Link

EP
(1)

EP0395323B1
(en)

JP
(1)

JPH0798813B2
(en)

KR
(1)

KR970002466B1
(en)

CN
(3)

CN1031708C
(en)

AT
(1)

ATE154348T1
(en)

AU
(1)

AU616351B2
(en)

DE
(1)

DE69030897T2
(en)

DK
(1)

DK0395323T3
(en)

ES
(1)

ES2106018T3
(en)

FI
(1)

FI109533B
(en)

FR
(1)

FR2646424B1
(en)

GR
(1)

GR3023767T3
(en)

HK
(1)

HK1003789A1
(en)

HU
(1)

HU203882B
(en)

IL
(1)

IL94208A0
(en)

SG
(1)

SG47004A1
(en)

Cited By (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

AU628217B2
(en)

1989-08-31
1992-09-10
Marion Merrell Dow Inc.
Heterogeneous synthesis of azepinones from esters

Families Citing this family (8)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

ES2069003T3
(en)

1989-04-28
1995-05-01
Tanabe Seiyaku Co

PROCEDURE FOR PREPARING 1,5-BENZOTIAZEPINE DERIVATIVES.

IT1234387B
(en)

1989-07-12
1992-05-18
Zambon Spa

PURIFICATION PROCESS OF USEFUL INTERMEDIATES IN THE PREPARATION OF DILTIAZEM

JPH085869B2
(en)

1990-03-08
1996-01-24
田辺製薬株式会社

Process for producing 1,5-benzothiazepine derivative

IT1249318B
(en)

1991-05-23
1995-02-22
Zambon Spa

BENZOTIAZEPINE PREPARATION PROCESS FOR CYCLING WITH PHOSPHONIC ACIDS

DE4206714A1
(en)

1992-03-04
1993-09-09
Sandoz Ag

WAX DISPERSIONS, THEIR PRODUCTION AND USE

NL1002687C2
(en)

1996-03-22
1997-09-23
Dsm Nv

Process for the preparation of a benzothiazepine.

IL123352A0
(en)

1997-02-27
1998-09-24
Tanabe Seiyaku Co
Process for preparing an optically active trans-3-substituted glycidic acid ester

IT1295376B1
(en)

1997-10-22
1999-05-12
Zambon Spa

PROCESS FOR THE RECYCLING OF A BY-PRODUCT OF THE SYNTHESIS OF DILTIAZEM

Citations (3)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

AU3509989A
(en)

1988-05-24
1989-11-30

F. Hoffmann-La Roche Ag

Process for the manufacture of optically active naphthothiazepinones

AU5385890A
(en)

1989-04-28
1990-11-01

Tanabe Seiyaku Co., Ltd.

Processes for preparing 1,5-benzothiazepine derivatives

AU7199391A
(en)

1990-03-08
1991-09-12

Tanabe Seiyaku Co., Ltd.

Processes for preparing 1,5-benzothiazepine derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

DE3374865D1
(en)

1982-07-07
1988-01-21
Siegfried Ag
Process for preparing 4-hydroxy-2-methyl-n-2-pyridyl-2h-1,2-benzothiazine-3-carboxamide 1,1-dioxide

US4552695A
(en)

1983-04-21
1985-11-12
Shionogi & Co., Ltd.
Process for production of diltiazem hydrochloride

FR2641535B1
(en)

1989-01-11
1991-03-15
Synthelabo

PROCESS FOR THE PREPARATION OF (+) – (2S, 3S) -HYDROXY-3 (METHOXY-4 PHENYL) -2 DIHYDRO-2,3 5H-BENZOTHIAZEPINE-1,5 ONE-4

1989

1989-04-28
JP
JP1109795A
patent/JPH0798813B2/en
not_active
Expired – Lifetime

1990

1990-04-20
AT
AT90304299T
patent/ATE154348T1/en
not_active
IP Right Cessation

1990-04-20
DK
DK90304299.2T
patent/DK0395323T3/en
active

1990-04-20
ES
ES90304299T
patent/ES2106018T3/en
not_active
Expired – Lifetime

1990-04-20
EP
EP90304299A
patent/EP0395323B1/en
not_active
Expired – Lifetime

1990-04-20
DE
DE69030897T
patent/DE69030897T2/en
not_active
Expired – Lifetime

1990-04-20
SG
SG1996001748A
patent/SG47004A1/en
unknown

1990-04-23
FI
FI902030A
patent/FI109533B/en
active
IP Right Grant

1990-04-25
IL
IL94208A
patent/IL94208A0/en
unknown

1990-04-26
FR
FR9005323A
patent/FR2646424B1/en
not_active
Expired – Lifetime

1990-04-26
AU
AU53856/90A
patent/AU616351B2/en
not_active
Expired

1990-04-27
HU
HU902607A
patent/HU203882B/en
unknown

1990-04-28
CN
CN90102552A
patent/CN1031708C/en
not_active
Expired – Lifetime

1990-04-28
KR
KR1019900006059A
patent/KR970002466B1/en
not_active
IP Right Cessation

1994

1994-12-28
CN
CN94120033A
patent/CN1052479C/en
not_active
Expired – Lifetime

1997

1997-06-12
GR
GR970401275T
patent/GR3023767T3/en
unknown

1998

1998-04-08
HK
HK98102939A
patent/HK1003789A1/en
not_active
IP Right Cessation

1999

1999-01-28
CN
CNB991017072A
patent/CN1136205C/en
not_active
Expired – Lifetime

Patent Citations (3)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

AU3509989A
(en)

1988-05-24
1989-11-30
F. Hoffmann-La Roche Ag
Process for the manufacture of optically active naphthothiazepinones

AU5385890A
(en)

1989-04-28
1990-11-01
Tanabe Seiyaku Co., Ltd.
Processes for preparing 1,5-benzothiazepine derivatives

AU7199391A
(en)

1990-03-08
1991-09-12
Tanabe Seiyaku Co., Ltd.
Processes for preparing 1,5-benzothiazepine derivatives

Cited By (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

AU628217B2
(en)

1989-08-31
1992-09-10
Marion Merrell Dow Inc.
Heterogeneous synthesis of azepinones from esters

Also Published As

Publication number
Publication date

CN1031708C
(en)

1996-05-01

CN1245802A
(en)

2000-03-01

SG47004A1
(en)

1998-03-20

DE69030897D1
(en)

1997-07-17

CN1110684A
(en)

1995-10-25

HU203882B
(en)

1991-10-28

EP0395323A1
(en)

1990-10-31

JPH0798813B2
(en)

1995-10-25

DK0395323T3
(en)

1997-09-08

GR3023767T3
(en)

1997-09-30

ES2106018T3
(en)

1997-11-01

FR2646424A1
(en)

1990-11-02

ATE154348T1
(en)

1997-06-15

HU902607D0
(en)

1990-09-28

CN1136205C
(en)

2004-01-28

CN1052479C
(en)

2000-05-17

AU5385690A
(en)

1990-11-01

HUT55373A
(en)

1991-05-28

JPH02286672A
(en)

1990-11-26

FI902030A0
(en)

1990-04-23

FI109533B
(en)

2002-08-30

IL94208A0
(en)

1991-01-31

KR900016171A
(en)

1990-11-12

EP0395323B1
(en)

1997-06-11

CN1046901A
(en)

1990-11-14

KR970002466B1
(en)

1997-03-05

FR2646424B1
(en)

1994-05-20

DE69030897T2
(en)

1997-09-25

HK1003789A1
(en)

1998-11-06

Información de contacto