AU6504586A

AU6504586A – N-«««1-«(6-fluoro-2-naphthalenyl)methyl«-4-piperidinyl` amino«carbonyl«-pyridinecarboxamide derivatives
– Google Patents

AU6504586A – N-«««1-«(6-fluoro-2-naphthalenyl)methyl«-4-piperidinyl` amino«carbonyl«-pyridinecarboxamide derivatives
– Google Patents
N-«««1-«(6-fluoro-2-naphthalenyl)methyl«-4-piperidinyl` amino«carbonyl«-pyridinecarboxamide derivatives

Info

Publication number
AU6504586A

AU6504586A
AU65045/86A
AU6504586A
AU6504586A
AU 6504586 A
AU6504586 A
AU 6504586A
AU 65045/86 A
AU65045/86 A
AU 65045/86A
AU 6504586 A
AU6504586 A
AU 6504586A
AU 6504586 A
AU6504586 A
AU 6504586A
Authority
AU
Australia
Prior art keywords
naphthalenyl
piperidinyl
fluoro
carbonyl
amino
Prior art date
1985-11-15
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU65045/86A
Other versions

AU585087B2
(en

Inventor
John Leheup Archibald
Terence James Ward
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

John Wyeth and Brother Ltd

Original Assignee
John Wyeth and Brother Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1985-11-15
Filing date
1986-11-12
Publication date
1987-05-21

1986-11-12
Application filed by John Wyeth and Brother Ltd
filed
Critical
John Wyeth and Brother Ltd

1987-05-21
Publication of AU6504586A
publication
Critical
patent/AU6504586A/en

1989-06-08
Application granted
granted
Critical

1989-06-08
Publication of AU585087B2
publication
Critical
patent/AU585087B2/en

2006-11-12
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings

C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom

C07D211/98—Nitrogen atom

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom

C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings

C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P25/00—Drugs for disorders of the nervous system

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P25/00—Drugs for disorders of the nervous system

A61P25/20—Hypnotics; Sedatives

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P25/00—Drugs for disorders of the nervous system

A61P25/24—Antidepressants

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P25/00—Drugs for disorders of the nervous system

A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Abstract

The invention relates to compounds of formula wherein R represents hydrogen or fluorine and R<1> represents 3-pyridyl or 4-pyridyl or a salt thereof which compounds exhibit psychotropic activity and are useful as antidepressants.

AU65045/86A
1985-11-15
1986-11-12
N-«««1-«(6-fluoro-2-naphthalenyl)methyl«-4-piperidinyl` amino«carbonyl«-pyridinecarboxamide derivatives

Ceased

AU585087B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

GB858528235A

GB8528235D0
(en)

1985-11-15
1985-11-15
Heterocyclic compounds

GB8528235

1985-11-15

Publications (2)

Publication Number
Publication Date

AU6504586A
true

AU6504586A
(en)

1987-05-21

AU585087B2

AU585087B2
(en)

1989-06-08

Family
ID=10588307
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU65045/86A
Ceased

AU585087B2
(en)

1985-11-15
1986-11-12
N-«««1-«(6-fluoro-2-naphthalenyl)methyl«-4-piperidinyl` amino«carbonyl«-pyridinecarboxamide derivatives

Country Status (18)

Country
Link

EP
(1)

EP0228795B1
(en)

JP
(1)

JPH0723371B2
(en)

KR
(1)

KR940008303B1
(en)

AT
(1)

ATE60770T1
(en)

AU
(1)

AU585087B2
(en)

CA
(1)

CA1276150C
(en)

DE
(1)

DE3677486D1
(en)

DK
(1)

DK170776B1
(en)

ES
(1)

ES2031823T3
(en)

FI
(1)

FI85699C
(en)

GB
(2)

GB8528235D0
(en)

GR
(1)

GR3001483T3
(en)

HU
(1)

HU197739B
(en)

IE
(1)

IE59007B1
(en)

IL
(1)

IL80639A
(en)

PH
(1)

PH22436A
(en)

PT
(1)

PT83715B
(en)

ZA
(1)

ZA868557B
(en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB9508438D0
(en)

*

1995-04-26
1995-06-14
Wyeth John & Brother Ltd
Medical treatment

Family Cites Families (7)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB1573066A
(en)

*

1977-09-08
1980-08-13
Wyeth John & Brother Ltd
Piperidylureas and thioreas

EP0007525A1
(en)

*

1978-07-18
1980-02-06
Hoechst Aktiengesellschaft
2-(4-Aminopiperidino)-3.4-dihydroquinoline derivatives, processes for their preparation, pharmaceutical compositions containing them and their use

GB2034305B
(en)

*

1978-10-24
1982-12-22
Wyeth John & Brother Ltd
Preparation of piperidine derivatives

GB2073176B
(en)

*

1980-03-01
1984-01-18
Wyeth John & Brother Ltd
Piperidine derivatives

PL128409B1
(en)

*

1980-03-01
1984-01-31
Wyeth John & Brother Ltd
Process for preparing novel derivatives of piperidine

GB2108489B
(en)

*

1980-03-01
1984-06-06
Wyeth John & Brother Ltd
Pharmaceutical composition comprising piperidine derivatives

GB2106108B
(en)

*

1981-09-10
1985-05-01
Wyeth John & Brother Ltd
Piperidine derivatives

1985

1985-11-15
GB
GB858528235A
patent/GB8528235D0/en
active
Pending

1986

1986-11-11
ZA
ZA868557A
patent/ZA868557B/en
unknown

1986-11-11
PT
PT83715A
patent/PT83715B/en
not_active
IP Right Cessation

1986-11-12
CA
CA000522789A
patent/CA1276150C/en
not_active
Expired – Fee Related

1986-11-12
AU
AU65045/86A
patent/AU585087B2/en
not_active
Ceased

1986-11-13
PH
PH34478A
patent/PH22436A/en
unknown

1986-11-13
JP
JP61270812A
patent/JPH0723371B2/en
not_active
Expired – Lifetime

1986-11-14
IL
IL80639A
patent/IL80639A/en
not_active
IP Right Cessation

1986-11-14
FI
FI864641A
patent/FI85699C/en
not_active
IP Right Cessation

1986-11-14
KR
KR1019860009618A
patent/KR940008303B1/en
not_active
IP Right Cessation

1986-11-14
IE
IE301586A
patent/IE59007B1/en
not_active
IP Right Cessation

1986-11-14
HU
HU864708A
patent/HU197739B/en
not_active
IP Right Cessation

1986-11-14
AT
AT86308899T
patent/ATE60770T1/en
not_active
IP Right Cessation

1986-11-14
DE
DE8686308899T
patent/DE3677486D1/en
not_active
Expired – Fee Related

1986-11-14
DK
DK546386A
patent/DK170776B1/en
active

1986-11-14
ES
ES198686308899T
patent/ES2031823T3/en
not_active
Expired – Lifetime

1986-11-14
EP
EP86308899A
patent/EP0228795B1/en
not_active
Expired – Lifetime

1986-11-14
GB
GB8627301A
patent/GB2182934B/en
not_active
Expired

1991

1991-02-19
GR
GR91400200T
patent/GR3001483T3/en
unknown

Also Published As

Publication number
Publication date

FI864641A0
(en)

1986-11-14

DK546386A
(en)

1987-05-16

AU585087B2
(en)

1989-06-08

IL80639A
(en)

1990-07-12

DK170776B1
(en)

1996-01-15

ES2031823T3
(en)

1993-01-01

CA1276150C
(en)

1990-11-13

PT83715A
(en)

1986-12-01

FI864641A
(en)

1987-05-16

PT83715B
(en)

1989-06-30

GB8627301D0
(en)

1986-12-17

GB2182934A
(en)

1987-05-28

GR3001483T3
(en)

1992-10-08

HUT43842A
(en)

1987-12-28

PH22436A
(en)

1988-09-12

IE863015L
(en)

1987-05-15

DE3677486D1
(en)

1991-03-14

IL80639A0
(en)

1987-02-27

ZA868557B
(en)

1988-06-29

GB2182934B
(en)

1989-09-27

ATE60770T1
(en)

1991-02-15

KR870004958A
(en)

1987-06-02

DK546386D0
(en)

1986-11-14

GB8528235D0
(en)

1985-12-18

FI85699B
(en)

1992-02-14

FI85699C
(en)

1992-05-25

JPS62135471A
(en)

1987-06-18

KR940008303B1
(en)

1994-09-12

HU197739B
(en)

1989-05-29

EP0228795A1
(en)

1987-07-15

JPH0723371B2
(en)

1995-03-15

EP0228795B1
(en)

1991-02-06

IE59007B1
(en)

1993-12-15

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Legal Events

Date
Code
Title
Description

2002-06-13
MK14
Patent ceased section 143(a) (annual fees not paid) or expired

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