AU534802B2

AU534802B2 – Pyrimidone derivatives and their use as histamine h2- antagonists
– Google Patents

AU534802B2 – Pyrimidone derivatives and their use as histamine h2- antagonists
– Google Patents
Pyrimidone derivatives and their use as histamine h2- antagonists

Info

Publication number
AU534802B2

AU534802B2
AU52722/79A
AU5272279A
AU534802B2
AU 534802 B2
AU534802 B2
AU 534802B2
AU 52722/79 A
AU52722/79 A
AU 52722/79A
AU 5272279 A
AU5272279 A
AU 5272279A
AU 534802 B2
AU534802 B2
AU 534802B2
Authority
AU
Australia
Prior art keywords
histamine
antagonists
pyrimidone derivatives
pyrimidone
derivatives
Prior art date
1978-11-13
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Ceased

Application number
AU52722/79A
Other versions

AU5272279A
(en

Inventor
Thomas Henry Brown
Robert John Ife
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Smith Kline and French Laboratories Ltd

Original Assignee
Smith Kline and French Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1978-11-13
Filing date
1979-11-12
Publication date
1984-02-16

1979-11-12
Application filed by Smith Kline and French Laboratories Ltd
filed
Critical
Smith Kline and French Laboratories Ltd

1980-05-22
Publication of AU5272279A
publication
Critical
patent/AU5272279A/en

1984-02-16
Application granted
granted
Critical

1984-02-16
Publication of AU534802B2
publication
Critical
patent/AU534802B2/en

1999-11-12
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings

C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings

C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members

C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms

C07D239/46—Two or more oxygen, sulphur or nitrogen atoms

C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS

Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE

Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS

Y02P20/00—Technologies relating to chemical industry

Y02P20/50—Improvements relating to the production of bulk chemicals

Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

AU52722/79A
1978-11-13
1979-11-12
Pyrimidone derivatives and their use as histamine h2- antagonists

Ceased

AU534802B2
(en)

Applications Claiming Priority (4)

Application Number
Priority Date
Filing Date
Title

GB7844260

1978-11-13

GB7844260

1978-11-13

GB7929013

1979-08-21

GB7929013

1979-08-21

Publications (2)

Publication Number
Publication Date

AU5272279A

AU5272279A
(en)

1980-05-22

AU534802B2
true

AU534802B2
(en)

1984-02-16

Family
ID=26269556
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU52722/79A
Ceased

AU534802B2
(en)

1978-11-13
1979-11-12
Pyrimidone derivatives and their use as histamine h2- antagonists

Country Status (22)

Country
Link

US
(1)

US4496567A
(en)

EP
(1)

EP0013071B1
(en)

JP
(1)

JPS55500898A
(en)

AU
(1)

AU534802B2
(en)

CA
(1)

CA1137984A
(en)

CS
(1)

CS214813B2
(en)

DD
(1)

DD146953A5
(en)

DE
(1)

DE2966413D1
(en)

DK
(1)

DK298180A
(en)

ES
(1)

ES485912A1
(en)

FI
(1)

FI793533A
(en)

GR
(1)

GR78338B
(en)

HU
(1)

HU182740B
(en)

IE
(1)

IE49205B1
(en)

IL
(1)

IL58676A
(en)

NO
(1)

NO793642L
(en)

NZ
(1)

NZ192096A
(en)

PH
(1)

PH15579A
(en)

PL
(1)

PL126169B1
(en)

PT
(1)

PT70441A
(en)

RO
(1)

RO78491A
(en)

WO
(1)

WO1980000966A1
(en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

CA1140129A
(en)

*

1979-08-21
1983-01-25
Ronald J. King
4-pyrimidone derivatives

DE3275291D1
(en)

*

1981-07-24
1987-03-05
Glaxo Group Ltd
Heterocyclic derivatives

US4745110A
(en)

*

1983-04-29
1988-05-17
Rorer Pharmaceutical Corporation
Bicyclic benzenoid aminoalkylene ethers and thioethers, pharmaceutical compositions and use

GB8318638D0
(en)

*

1983-07-09
1983-08-10
Smith Kline French Lab
Chemical compounds

GB8320505D0
(en)

*

1983-07-29
1983-09-01
Smith Kline French Lab
Chemical compounds

US4772704A
(en)

*

1983-09-21
1988-09-20
Bristol-Myers Company
2,5-disubstituted-4(3H)-pyrimidones having histamine H2 -receptor antagonist activity

GB8332091D0
(en)

*

1983-12-01
1984-01-11
Smith Kline French Lab
Chemical compounds

GB8421427D0
(en)

*

1984-08-23
1984-09-26
Smith Kline French Lab
Chemical compounds

JO1410B1
(en)

*

1984-11-03
1986-11-30
سميث كلاين اند فرينش لابوراتوريز ليمتد
Compounds

JPS61155373A
(en)

*

1984-12-28
1986-07-15
Yamanouchi Pharmaceut Co Ltd
Novel 2-substituted amino-4(1h)-pyrimidone derivative and production thereof

JP2807577B2
(en)

*

1990-06-15
1998-10-08
エーザイ株式会社

Cyclic amide derivative

EP3909449A1
(en)

2020-05-11
2021-11-17
Bisaf Spolka Z Ograniczona Odpowiedzialnoscia
Protective filtering half mask

Family Cites Families (10)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US3980781A
(en)

*

1966-03-31
1976-09-14
Imperial Chemical Industries Limited
Fungicidal composition and method containing 2-amino-pyrimidines

GB1223686A
(en)

*

1967-02-24
1971-03-03
Ici Ltd
Salts of pyrimidine derivatives and the use thereof as fungicides

GB1419994A
(en)

*

1973-05-03
1976-01-07
Smith Kline French Lab
Heterocyclicalkylaminotheterocyclic compounds methods for their preparation and compositions comprising them

IN146736B
(en)

*

1975-10-02
1979-08-25
Smith Kline French Lab

US4145546A
(en)

*

1975-10-02
1979-03-20
Smith Kline & French Laboratories Limited
4-Pyrimidone compounds

MW5076A1
(en)

*

1975-12-29
1978-02-08
Smith Kline French Lab
Pharmacologicalle active compounds

US4154834A
(en)

*

1975-12-29
1979-05-15
Smith Kline & French Laboratories Limited
Substituted isocytosines having histamine H2 -antagonist activity

US4117131A
(en)

*

1976-12-07
1978-09-26
Warner-Lambert Company
Method of inhibiting gastric acid secretions with 2-(4-pyrimidinyl)thioacetamides

GB1604674A
(en)

*

1977-05-17
1981-12-16
Allen & Hanburys Ltd
Aminoalkyl-benzene derivatives

ZA793443B
(en)

*

1978-07-26
1980-12-31
Glaxo Group Ltd
Heterocyclic derivatives

1979

1979-11-06
US
US06/091,850
patent/US4496567A/en
not_active
Expired – Lifetime

1979-11-08
JP
JP50182279A
patent/JPS55500898A/ja
active
Pending

1979-11-08
EP
EP79302509A
patent/EP0013071B1/en
not_active
Expired

1979-11-08
WO
PCT/GB1979/000184
patent/WO1980000966A1/en
unknown

1979-11-08
CA
CA000339434A
patent/CA1137984A/en
not_active
Expired

1979-11-08
DE
DE7979302509T
patent/DE2966413D1/en
not_active
Expired

1979-11-09
IL
IL58676A
patent/IL58676A/en
unknown

1979-11-09
PH
PH23272A
patent/PH15579A/en
unknown

1979-11-12
PT
PT70441A
patent/PT70441A/en
unknown

1979-11-12
DD
DD79216837A
patent/DD146953A5/en
unknown

1979-11-12
NO
NO793642A
patent/NO793642L/en
unknown

1979-11-12
NZ
NZ192096A
patent/NZ192096A/en
unknown

1979-11-12
AU
AU52722/79A
patent/AU534802B2/en
not_active
Ceased

1979-11-12
PL
PL1979219563A
patent/PL126169B1/en
unknown

1979-11-12
HU
HU79SI1728A
patent/HU182740B/en
unknown

1979-11-12
GR
GR60483A
patent/GR78338B/el
unknown

1979-11-12
IE
IE2169/79A
patent/IE49205B1/en
unknown

1979-11-12
FI
FI793533A
patent/FI793533A/en
not_active
Application Discontinuation

1979-11-13
ES
ES485912A
patent/ES485912A1/en
not_active
Expired

1979-11-13
RO
RO7999212A
patent/RO78491A/en
unknown

1979-11-13
CS
CS797734A
patent/CS214813B2/en
unknown

1980

1980-07-10
DK
DK298180A
patent/DK298180A/en
not_active
Application Discontinuation

Also Published As

Publication number
Publication date

IL58676A0
(en)

1980-02-29

HU182740B
(en)

1984-03-28

ES485912A1
(en)

1980-07-01

DK298180A
(en)

1980-07-10

US4496567A
(en)

1985-01-29

PH15579A
(en)

1983-02-17

IE792169L
(en)

1980-05-13

NO793642L
(en)

1980-05-14

AU5272279A
(en)

1980-05-22

PL126169B1
(en)

1983-07-30

RO78491A
(en)

1982-02-26

PT70441A
(en)

1979-12-01

FI793533A
(en)

1980-05-14

EP0013071B1
(en)

1983-11-16

CA1137984A
(en)

1982-12-21

EP0013071A1
(en)

1980-07-09

DD146953A5
(en)

1981-03-11

NZ192096A
(en)

1981-11-19

IL58676A
(en)

1983-07-31

JPS55500898A
(en)

1980-11-06

IE49205B1
(en)

1985-08-21

CS214813B2
(en)

1982-06-25

WO1980000966A1
(en)

1980-05-15

GR78338B
(en)

1984-09-26

PL219563A1
(en)

1980-12-01

DE2966413D1
(en)

1983-12-22

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(en)

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