AU534992B2

AU534992B2 – Novel bis-and mono-quaternary ammonium derivatives of 2beta, 16beta-dipiperidino-5alpha-androstanes, processes for their preparation and pharmaceutical preparations
– Google Patents

AU534992B2 – Novel bis-and mono-quaternary ammonium derivatives of 2beta, 16beta-dipiperidino-5alpha-androstanes, processes for their preparation and pharmaceutical preparations
– Google Patents
Novel bis-and mono-quaternary ammonium derivatives of 2beta, 16beta-dipiperidino-5alpha-androstanes, processes for their preparation and pharmaceutical preparations

Info

Publication number
AU534992B2

AU534992B2
AU66405/81A
AU6640581A
AU534992B2
AU 534992 B2
AU534992 B2
AU 534992B2
AU 66405/81 A
AU66405/81 A
AU 66405/81A
AU 6640581 A
AU6640581 A
AU 6640581A
AU 534992 B2
AU534992 B2
AU 534992B2
Authority
AU
Australia
Prior art keywords
16beta
dipiperidino
2beta
androstanes
5alpha
Prior art date
1979-12-12
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Ceased

Application number
AU66405/81A
Other versions

AU6640581A
(en

Inventor
J. Kelder
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Akzo NV

Original Assignee
Akzo NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1979-12-12
Filing date
1980-12-09
Publication date
1984-02-23

1980-12-09
Application filed by Akzo NV
filed
Critical
Akzo NV

1981-07-06
Publication of AU6640581A
publication
Critical
patent/AU6640581A/en

1984-02-23
Application granted
granted
Critical

1984-02-23
Publication of AU534992B2
publication
Critical
patent/AU534992B2/en

2000-12-09
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07J—STEROIDS

C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton

C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P25/00—Drugs for disorders of the nervous system

A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies

AU66405/81A
1979-12-12
1980-12-09
Novel bis-and mono-quaternary ammonium derivatives of 2beta, 16beta-dipiperidino-5alpha-androstanes, processes for their preparation and pharmaceutical preparations

Ceased

AU534992B2
(en)

Applications Claiming Priority (3)

Application Number
Priority Date
Filing Date
Title

GB7942883

1979-12-12

GB7942883

1979-12-12

PCT/EP1980/000143

WO1981001710A1
(en)

1979-12-12
1980-12-09
Mono and bis piperidinium androstanes derivatives

Publications (2)

Publication Number
Publication Date

AU6640581A

AU6640581A
(en)

1981-07-06

AU534992B2
true

AU534992B2
(en)

1984-02-23

Family
ID=10509800
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU66405/81A
Ceased

AU534992B2
(en)

1979-12-12
1980-12-09
Novel bis-and mono-quaternary ammonium derivatives of 2beta, 16beta-dipiperidino-5alpha-androstanes, processes for their preparation and pharmaceutical preparations

Country Status (12)

Country
Link

US
(1)

US4348390A
(en)

EP
(1)

EP0032261B1
(en)

JP
(1)

JPH026360B2
(en)

AU
(1)

AU534992B2
(en)

CA
(1)

CA1153366A
(en)

DE
(1)

DE3065088D1
(en)

DK
(1)

DK158741C
(en)

ES
(1)

ES8204443A1
(en)

FI
(1)

FI66394C
(en)

HU
(1)

HU185865B
(en)

IE
(1)

IE50675B1
(en)

WO
(1)

WO1981001710A1
(en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

IE53463B1
(en)

*

1981-06-15
1988-11-23
Akzo Nv
Mono-and bisquaternary ammonium derivatives of 2 beta,16 beta-d-amino-5 alpha-androstane derivatives and pharmaceutical preparations containing same

US4726275A
(en)

*

1983-05-10
1988-02-23
Synthaxe Limited
Electronic musical instrument

US5418226A
(en)

*

1992-04-22
1995-05-23
Akzo N.V.
Monoquaternary 2,16-bispiperidinylandrostane derivatives

US5926516A
(en)

*

1995-05-24
1999-07-20
Siemens Aktiengesellschaft
Absorption structure for absorbing neutrons and method for producing an absorption structure

IT1277700B1
(en)

*

1995-12-22
1997-11-11
Poli Ind Chimica Spa

PROCESS OF PREPARATION OF 2-BETA, 16-BETA-DIAMINO 3-ALPHA, 17-BETA-DIACYLOSS 5-ALPHAANDROSTANS, STRUCTURED NEUROMUSCULAR BLOCKERS

US5990124A
(en)

1997-10-24
1999-11-23
Gyermek; Laszlo
Neuromuscular relaxants

Family Cites Families (4)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB1138605A
(en)

*

1965-02-19
1969-01-01
Organon Labor Ltd
Improvements in or relating to new 2-ß,16-ß-diamino-androstanes

GB1454749A
(en)

*

1972-11-29
1976-11-03
Akzo Nv
2beta, 16beta-diamino-androstanes and their preparation

HU172522B
(en)

*

1975-08-01
1978-09-28
Richter Gedeon Vegyeszet
Process for preparing new derivatives of 2beta-16beta-diamino-androstane and derivatives / quaternary salts / thereof

DE2962627D1
(en)

*

1978-09-05
1982-06-09
Akzo Nv
Acid addition salts of 16-beta-monoquaternary ammonium derivatives of 2-beta, 16-beta-bis-piperidino-androstanes and pharmaceutical preparations containing same

1980

1980-12-08
IE
IE2566/80A
patent/IE50675B1/en
not_active
IP Right Cessation

1980-12-09
DE
DE8080201186T
patent/DE3065088D1/en
not_active
Expired

1980-12-09
AU
AU66405/81A
patent/AU534992B2/en
not_active
Ceased

1980-12-09
HU
HU811180A
patent/HU185865B/en
unknown

1980-12-09
EP
EP80201186A
patent/EP0032261B1/en
not_active
Expired

1980-12-09
WO
PCT/EP1980/000143
patent/WO1981001710A1/en
active
IP Right Grant

1980-12-09
JP
JP56500158A
patent/JPH026360B2/ja
not_active
Expired – Lifetime

1980-12-10
US
US06/214,650
patent/US4348390A/en
not_active
Expired – Lifetime

1980-12-11
CA
CA000366536A
patent/CA1153366A/en
not_active
Expired

1980-12-12
ES
ES497724A
patent/ES8204443A1/en
not_active
Expired

1981

1981-06-15
DK
DK260881A
patent/DK158741C/en
not_active
IP Right Cessation

1981-06-15
FI
FI811857A
patent/FI66394C/en
not_active
IP Right Cessation

Also Published As

Publication number
Publication date

WO1981001710A1
(en)

1981-06-25

JPH026360B2
(en)

1990-02-08

EP0032261A1
(en)

1981-07-22

IE50675B1
(en)

1986-06-11

IE802566L
(en)

1981-06-12

CA1153366A
(en)

1983-09-06

US4348390A
(en)

1982-09-07

JPS56501761A
(en)

1981-12-03

FI66394C
(en)

1984-10-10

DK158741C
(en)

1990-11-26

DK260881A
(en)

1981-06-25

AU6640581A
(en)

1981-07-06

DK158741B
(en)

1990-07-09

FI811857L
(en)

1981-06-15

EP0032261B1
(en)

1983-09-28

ES497724A0
(en)

1982-05-01

HU185865B
(en)

1985-04-28

ES8204443A1
(en)

1982-05-01

DE3065088D1
(en)

1983-11-03

FI66394B
(en)

1984-06-29

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