AU7022391A – Triazole antifungal agents
– Google Patents
AU7022391A – Triazole antifungal agents
– Google Patents
Triazole antifungal agents
Info
Publication number
AU7022391A
AU7022391A
AU70223/91A
AU7022391A
AU7022391A
AU 7022391 A
AU7022391 A
AU 7022391A
AU 70223/91 A
AU70223/91 A
AU 70223/91A
AU 7022391 A
AU7022391 A
AU 7022391A
AU 7022391 A
AU7022391 A
AU 7022391A
Authority
AU
Australia
Prior art keywords
antifungal agents
triazole antifungal
triazole
agents
antifungal
Prior art date
1990-02-02
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU70223/91A
Other versions
AU625188B2
(en
Inventor
Stephen James Ray
Kenneth Richardson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1990-02-02
Filing date
1991-02-01
Publication date
1991-09-05
Family has litigation
First worldwide family litigation filed
litigation
Critical
https://patents.darts-ip.com/?family=10670334&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU7022391(A)
«Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
1991-02-01
Application filed by Pfizer Inc
filed
Critical
Pfizer Inc
1991-09-05
Publication of AU7022391A
publication
Critical
patent/AU7022391A/en
1992-07-02
Application granted
granted
Critical
1992-07-02
Publication of AU625188B2
publication
Critical
patent/AU625188B2/en
2016-02-01
Adjusted expiration
legal-status
Critical
Status
Expired
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
C07D239/30—Halogen atoms or nitro radicals
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
A61P31/04—Antibacterial agents
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
A61P31/10—Antimycotics
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D213/61—Halogen atoms or nitro radicals
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
AU70223/91A
1990-02-02
1991-02-01
Triazole antifungal agents
Expired
AU625188B2
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
GB909002375A
GB9002375D0
(en)
1990-02-02
1990-02-02
Triazole antifungal agents
GB9002375
1990-02-02
Publications (2)
Publication Number
Publication Date
AU7022391A
true
AU7022391A
(en)
1991-09-05
AU625188B2
AU625188B2
(en)
1992-07-02
Family
ID=10670334
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU70223/91A
Expired
AU625188B2
(en)
1990-02-02
1991-02-01
Triazole antifungal agents
Country Status (42)
Country
Link
US
(2)
US5567817A
(en)
EP
(1)
EP0440372B1
(en)
JP
(2)
JP2625584B2
(en)
KR
(1)
KR930011039B1
(en)
CN
(2)
CN1026788C
(en)
AP
(2)
AP223A
(en)
AT
(1)
ATE90090T1
(en)
AU
(1)
AU625188B2
(en)
BA
(1)
BA97298A
(en)
BG
(1)
BG60032A3
(en)
BR
(1)
BR9100435A
(en)
CA
(2)
CA2285891C
(en)
CZ
(1)
CZ279339B6
(en)
DE
(2)
DE10299035I2
(en)
DK
(1)
DK0440372T3
(en)
EG
(1)
EG19750A
(en)
ES
(1)
ES2055523T4
(en)
FI
(3)
FI107608B
(en)
GB
(1)
GB9002375D0
(en)
HK
(1)
HK219396A
(en)
HU
(2)
HU205351B
(en)
IE
(1)
IE64774B1
(en)
IL
(2)
IL110322A
(en)
IN
(1)
IN176148B
(en)
IS
(1)
IS1629B
(en)
LU
(1)
LU90960I2
(en)
LV
(1)
LV10615B
(en)
MA
(1)
MA22054A1
(en)
MX
(1)
MX24363A
(en)
MY
(1)
MY105494A
(en)
NL
(1)
NL300100I2
(en)
NO
(2)
NO176796C
(en)
NZ
(1)
NZ247205A
(en)
OA
(1)
OA09480A
(en)
PE
(1)
PE31691A1
(en)
PL
(3)
PL169332B1
(en)
PT
(1)
PT96617B
(en)
RO
(1)
RO109648B1
(en)
RU
(2)
RU2114838C1
(en)
SK
(1)
SK278215B6
(en)
YU
(1)
YU48105B
(en)
ZA
(1)
ZA91761B
(en)
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HETEROCYCLICALLY SUBSTITUTED HYDROXYALKYL-AZOLYL DERIVATIVES
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Aromatase inhibitors
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Antifungal azole compounds
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PROCEDURE TO PREPARE 4,6-DICLORO-PYRIMIDINE.
1990
1990-02-02
GB
GB909002375A
patent/GB9002375D0/en
active
Pending
1991
1991-01-24
DK
DK91300553.4T
patent/DK0440372T3/en
active
1991-01-24
DE
DE2002199035
patent/DE10299035I2/en
active
Active
1991-01-24
AT
AT91300553T
patent/ATE90090T1/en
active
1991-01-24
DE
DE9191300553T
patent/DE69100095T2/en
not_active
Expired – Lifetime
1991-01-24
ES
ES91300553T
patent/ES2055523T4/en
not_active
Expired – Lifetime
1991-01-24
EP
EP91300553A
patent/EP0440372B1/en
not_active
Expired – Lifetime
1991-01-25
IL
IL11032291A
patent/IL110322A/en
not_active
IP Right Cessation
1991-01-25
IN
IN74DE1991
patent/IN176148B/en
unknown
1991-01-25
IL
IL9704591A
patent/IL97045A/en
not_active
IP Right Cessation
1991-01-28
AP
APAP/P/1991/000237A
patent/AP223A/en
active
1991-01-28
RO
RO146821A
patent/RO109648B1/en
unknown
1991-01-28
AP
AP90/00237A
patent/AP9000237A0/en
unknown
1991-01-29
NZ
NZ247205A
patent/NZ247205A/en
unknown
1991-01-29
BG
BG93726A
patent/BG60032A3/en
unknown
1991-01-29
PE
PE1991180888A
patent/PE31691A1/en
not_active
IP Right Cessation
1991-01-30
CA
CA002285891A
patent/CA2285891C/en
not_active
Expired – Lifetime
1991-01-30
IS
IS3671A
patent/IS1629B/en
unknown
1991-01-30
CA
CA002035314A
patent/CA2035314C/en
not_active
Expired – Lifetime
1991-01-31
JP
JP3031977A
patent/JP2625584B2/en
not_active
Expired – Lifetime
1991-01-31
PL
PL91306940A
patent/PL169332B1/en
unknown
1991-01-31
NO
NO910368A
patent/NO176796C/en
not_active
IP Right Cessation
1991-01-31
PL
PL91288901A
patent/PL167294B1/en
unknown
1991-01-31
KR
KR1019910001613A
patent/KR930011039B1/en
not_active
IP Right Cessation
1991-01-31
PL
PL91306941A
patent/PL169307B1/en
unknown
1991-01-31
MY
MYPI91000155A
patent/MY105494A/en
unknown
1991-01-31
PT
PT96617A
patent/PT96617B/en
not_active
IP Right Cessation
1991-01-31
MX
MX2436391A
patent/MX24363A/en
unknown
1991-02-01
OA
OA59945A
patent/OA09480A/en
unknown
1991-02-01
CZ
CS91249A
patent/CZ279339B6/en
not_active
IP Right Cessation
1991-02-01
RU
SU5010394A
patent/RU2114838C1/en
active
1991-02-01
HU
HU91366A
patent/HU205351B/en
unknown
1991-02-01
FI
FI910508A
patent/FI107608B/en
active
Protection Beyond IP Right Term
1991-02-01
RU
SU914894374A
patent/RU2036194C1/en
active
1991-02-01
BR
BR919100435A
patent/BR9100435A/en
not_active
Application Discontinuation
1991-02-01
YU
YU17591A
patent/YU48105B/en
unknown
1991-02-01
ZA
ZA91761A
patent/ZA91761B/en
unknown
1991-02-01
MA
MA22327A
patent/MA22054A1/en
unknown
1991-02-01
IE
IE34291A
patent/IE64774B1/en
active
Protection Beyond IP Right Term
1991-02-01
SK
SK249-91A
patent/SK278215B6/en
active
Protection Beyond IP Right Term
1991-02-01
AU
AU70223/91A
patent/AU625188B2/en
not_active
Expired
1991-02-02
EG
EG6591A
patent/EG19750A/en
active
1991-02-02
CN
CN91100706A
patent/CN1026788C/en
not_active
Expired – Lifetime
1993
1993-11-15
LV
LVP-93-1224A
patent/LV10615B/en
unknown
1994
1994-02-26
CN
CN94102354A
patent/CN1040504C/en
not_active
Expired – Lifetime
1995
1995-05-01
US
US08/432,414
patent/US5567817A/en
not_active
Expired – Lifetime
1995-06-09
HU
HU95P/P00179P
patent/HU211582A9/en
active
Protection Beyond IP Right Term
1996
1996-07-18
US
US08/683,694
patent/US5773443A/en
not_active
Expired – Lifetime
1996-07-19
JP
JP8190918A
patent/JP2848811B2/en
not_active
Expired – Lifetime
1996-12-24
HK
HK219396A
patent/HK219396A/en
not_active
IP Right Cessation
1997
1997-03-25
FI
FI971238A
patent/FI971238A/en
unknown
1998
1998-03-30
BA
BA970298A
patent/BA97298A/en
unknown
2000
2000-01-17
FI
FI20000084A
patent/FI20000084A/en
unknown
2002
2002-09-05
NO
NO2002006C
patent/NO2002006I2/en
unknown
2002-09-06
NL
NL300100C
patent/NL300100I2/en
unknown
2002-09-11
LU
LU90960C
patent/LU90960I2/en
unknown
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FI971238A0
(en)
1997-03-25
DE69100095D1
(en)
1993-07-08
IL97045A0
(en)
1992-03-29
IS3671A7
(en)
1991-08-03
LV10615A
(en)
1995-04-20
IL110322A0
(en)
1994-10-21
GB9002375D0
(en)
1990-04-04
JP2848811B2
(en)
1999-01-20
DE10299035I2
(en)
2003-06-26
AP9000237A0
(en)
1991-01-31
DK0440372T3
(en)
1993-06-28
BR9100435A
(en)
1991-10-22
RU2114838C1
(en)
1998-07-10
NL300100I1
(en)
2002-11-01
BA97298A
(en)
2001-09-14
DE10299035I1
(en)
2003-05-22
KR930011039B1
(en)
1993-11-20
FI971238A
(en)
1997-03-25
EP0440372A1
(en)
1991-08-07
RU2036194C1
(en)
1995-05-27
CN1026788C
(en)
1994-11-30
CN1100421A
(en)
1995-03-22
PT96617B
(en)
1998-07-31
EP0440372B1
(en)
1993-06-02
FI20000084A
(en)
2000-01-17
CN1053787A
(en)
1991-08-14
RO109648B1
(en)
1995-04-28
PE31691A1
(en)
1991-11-29
PL169307B1
(en)
1996-06-28
HU205351B
(en)
1992-04-28
PL169332B1
(en)
1996-07-31
NO176796B
(en)
1995-02-20
HK219396A
(en)
1997-01-03
CZ279339B6
(en)
1995-04-12
SK278215B6
(en)
1996-04-03
ES2055523T3
(en)
1994-08-16
IL110322A
(en)
1996-10-31
JPH09208583A
(en)
1997-08-12
EG19750A
(en)
1996-01-31
FI910508A0
(en)
1991-02-01
US5567817A
(en)
1996-10-22
NO910368D0
(en)
1991-01-31
IS1629B
(en)
1996-07-19
CN1040504C
(en)
1998-11-04
NL300100I2
(en)
2003-01-06
PL288901A1
(en)
1992-01-27
CA2285891C
(en)
2004-01-06
JP2625584B2
(en)
1997-07-02
PT96617A
(en)
1991-10-15
LV10615B
(en)
1995-12-20
YU48105B
(en)
1997-03-07
LU90960I2
(en)
2003-04-02
NO2002006I2
(en)
2004-10-11
MA22054A1
(en)
1991-10-01
NO910368L
(en)
1991-08-05
KR910021398A
(en)
1991-12-20
FI107608B
(en)
2001-09-14
IE64774B1
(en)
1995-09-06
JPH04211078A
(en)
1992-08-03
FI910508A
(en)
1991-08-03
IN176148B
(en)
1996-02-10
IE910342A1
(en)
1991-08-14
MX24363A
(en)
1993-09-01
BG60032A3
(en)
1993-07-15
CS9100249A2
(en)
1991-09-15
ES2055523T4
(en)
2011-04-11
OA09480A
(en)
1992-11-15
MY105494A
(en)
1994-10-31
ATE90090T1
(en)
1993-06-15
CA2035314A1
(en)
1991-08-03
CA2035314C
(en)
2000-01-18
US5773443A
(en)
1998-06-30
AP223A
(en)
1992-08-27
PL167294B1
(en)
1995-08-31
IL97045A
(en)
1995-11-27
NO176796C
(en)
1995-05-31
HU211582A9
(en)
1995-12-28
ZA91761B
(en)
1992-09-30
YU17591A
(en)
1994-01-20
AU625188B2
(en)
1992-07-02
DE69100095T2
(en)
1993-09-09
HUT56361A
(en)
1991-08-28
NZ247205A
(en)
1993-09-27
CA2285891A1
(en)
1991-08-03
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