GB1214010A – New acylating agents, their production, and their use in peptide synthesis
– Google Patents
GB1214010A – New acylating agents, their production, and their use in peptide synthesis
– Google Patents
New acylating agents, their production, and their use in peptide synthesis
Info
Publication number
GB1214010A
GB1214010A
GB58359/67A
GB5835967A
GB1214010A
GB 1214010 A
GB1214010 A
GB 1214010A
GB 58359/67 A
GB58359/67 A
GB 58359/67A
GB 5835967 A
GB5835967 A
GB 5835967A
GB 1214010 A
GB1214010 A
GB 1214010A
Authority
GB
United Kingdom
Prior art keywords
acylating agents
production
peptide synthesis
dec
tert
Prior art date
1966-12-23
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB58359/67A
Inventor
Ivar Ugi
Erich Klauke
Eugen Schnabel
Peter Hoffmann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1966-12-23
Filing date
1967-12-22
Publication date
1970-11-25
1967-12-22
Application filed by Bayer AG
filed
Critical
Bayer AG
1970-11-25
Publication of GB1214010A
publication
Critical
patent/GB1214010A/en
Status
Expired
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
C07D307/40—Radicals substituted by oxygen atoms
C07D307/42—Singly bound oxygen atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07K—PEPTIDES
C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
C07K1/063—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for alpha-amino functions
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07K—PEPTIDES
C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
C07K1/064—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for omega-amino or -guanidino functions
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07K—PEPTIDES
C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
C07K1/068—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for heterocyclic side chains
Abstract
1,214,010. Acylating agents. FARBENFABRIKEN BAYER A.G. 22 Dec., 1967 [23 Dec., 1966; 26 June, 1967; 26 Aug., 1967(2)], No. 58359/67. Heading C2C. Compounds of the general formula where R is tert.-butyl, furfuryl or benzyl radical substituted on the benzene ring by 1 or 3 methoxy groups are made by reacting carbonyl fluoride chloride with the appropriate alcohol at 0 to -70 C. in an inert solvent containing an acid binding agent. An amino or imino acid may be acylated by these compounds at +20 to- 20 C. in the presence of an acid binding agent and preferably at constant pH. In the case of tert.- butyloxy carbonyl fluoride the temperature range may be – 70 to +30 C.
GB58359/67A
1966-12-23
1967-12-22
New acylating agents, their production, and their use in peptide synthesis
Expired
GB1214010A
(en)
Applications Claiming Priority (3)
Application Number
Priority Date
Filing Date
Title
DEF0051062
1966-12-23
DEF0053339
1967-08-26
DEF0053338
1967-08-26
Publications (1)
Publication Number
Publication Date
GB1214010A
true
GB1214010A
(en)
1970-11-25
Family
ID=27210520
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
GB58359/67A
Expired
GB1214010A
(en)
1966-12-23
1967-12-22
New acylating agents, their production, and their use in peptide synthesis
Country Status (6)
Country
Link
US
(1)
US3592836A
(en)
BE
(1)
BE708453A
(en)
DE
(2)
DE1543630A1
(en)
FR
(1)
FR1549816A
(en)
GB
(1)
GB1214010A
(en)
NL
(1)
NL6717406A
(en)
Families Citing this family (8)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
US3711458A
(en)
*
1969-08-21
1973-01-16
Research Corp
Substituted and unsubstituted vinyloxycarbonyl groups as amino protecting groups in the syntheses of peptides
US4293706A
(en)
*
1980-06-19
1981-10-06
Ppg Industries, Inc.
Preparation of N-benzyloxycarbonyl aspartic acid
US4484001A
(en)
*
1983-11-18
1984-11-20
Ppg Industries, Inc.
Method for preparing N-benzyloxycarbonyl amino acids containing additional functionality
FR2559764B1
(en)
*
1984-02-16
1988-01-29
Poudres & Explosifs Ste Nale
NOVEL A-CHLORINE CARBONATES, THEIR MANUFACTURING PROCESS AND THEIR APPLICATION TO PROTECT THE AMINE FUNCTIONS OF AMINO ACIDS
US4500726A
(en)
*
1984-05-23
1985-02-19
Ppg Industries, Inc.
Method for preparing N-benzyloxycarbonyl amino acids containing additional functionality
GB9625895D0
(en)
1996-12-13
1997-01-29
Riley Patrick A
Novel compound useful as therapeutic agents and assay reagents
EP1916256A3
(en)
*
2001-09-25
2008-07-16
JAPAN as represented by PRESIDENT OF NATIONAL CANCER CENTER
Search for cancer markers by a novel screening method
JP6326825B2
(en)
*
2013-02-18
2018-05-23
住友化学株式会社
Salt, resist composition and method for producing resist pattern
1966
1966-12-23
DE
DE19661543630
patent/DE1543630A1/en
active
Pending
1967
1967-08-26
DE
DE19671643350
patent/DE1643350A1/en
active
Pending
1967-12-20
NL
NL6717406A
patent/NL6717406A/xx
unknown
1967-12-21
US
US692272A
patent/US3592836A/en
not_active
Expired – Lifetime
1967-12-22
FR
FR1549816D
patent/FR1549816A/fr
not_active
Expired
1967-12-22
BE
BE708453D
patent/BE708453A/xx
unknown
1967-12-22
GB
GB58359/67A
patent/GB1214010A/en
not_active
Expired
Also Published As
Publication number
Publication date
DE1543630A1
(en)
1969-07-31
NL6717406A
(en)
1968-06-24
BE708453A
(en)
1968-06-24
US3592836A
(en)
1971-07-13
FR1549816A
(en)
1968-12-13
DE1643350A1
(en)
1971-04-15
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Legal Events
Date
Code
Title
Description
1971-05-19
PS
Patent sealed [section 19, patents act 1949]
1973-06-06
PLNP
Patent lapsed through nonpayment of renewal fees
