GB1355033A

GB1355033A – Antimalarial medicines comprising thiazolyl thioureas
– Google Patents

GB1355033A – Antimalarial medicines comprising thiazolyl thioureas
– Google Patents
Antimalarial medicines comprising thiazolyl thioureas

Info

Publication number
GB1355033A

GB1355033A
GB2108473A
GB2108471A
GB1355033A
GB 1355033 A
GB1355033 A
GB 1355033A
GB 2108473 A
GB2108473 A
GB 2108473A
GB 2108471 A
GB2108471 A
GB 2108471A
GB 1355033 A
GB1355033 A
GB 1355033A
Authority
GB
United Kingdom
Prior art keywords
thioureas
thiazolyl
alkyl
antimalarial medicines
july
Prior art date
1970-07-24
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
GB2108473A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

F Hoffmann La Roche AG

Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1970-07-24
Filing date
1971-07-23
Publication date
1974-06-05

1971-07-23
Application filed by F Hoffmann La Roche AG
filed
Critical
F Hoffmann La Roche AG

1974-06-05
Publication of GB1355033A
publication
Critical
patent/GB1355033A/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings

C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings

C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members

C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D277/38—Nitrogen atoms

C07D277/44—Acylated amino or imino radicals

C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines

Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS

Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE

Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE

Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather

Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

1355033 Antimalarial medicines F HOFFMANN-LA ROCHE & CO AG 23 July 1971 [24 July 1970] 21084/73 Divided out of 1330930 Heading A5B Compositions in unit dosage form for treating or preventing malaria comprise a carrier and a compound (or a salt thereof) of the formula: wherein R1 is H or C 1-4 alkyl, R2=C 1-4 alkyl or aryl and R3 is H or C 1-4 alkyl, provided that when R3 is H, R1 and R2 are not both ethyl and when R3 is CH 3 , R1 and R2 are not both ethyl or methyl. They may be in conventional forms for oral, rectal and parenteral administration.

GB2108473A
1970-07-24
1971-07-23
Antimalarial medicines comprising thiazolyl thioureas

Expired

GB1355033A
(en)

Applications Claiming Priority (1)

Application Number
Priority Date
Filing Date
Title

CH1123970A

CH543535A
(en)

1970-07-24
1970-07-24

Process for the preparation of thiazole derivatives

Publications (1)

Publication Number
Publication Date

GB1355033A
true

GB1355033A
(en)

1974-06-05

Family
ID=4371497
Family Applications (2)

Application Number
Title
Priority Date
Filing Date

GB2108473A
Expired

GB1355033A
(en)

1970-07-24
1971-07-23
Antimalarial medicines comprising thiazolyl thioureas

GB3475571A
Expired

GB1330930A
(en)

1970-07-24
1971-07-23
Thiazole derivatives and a process for the manufacture thereof

Family Applications After (1)

Application Number
Title
Priority Date
Filing Date

GB3475571A
Expired

GB1330930A
(en)

1970-07-24
1971-07-23
Thiazole derivatives and a process for the manufacture thereof

Country Status (15)

Country
Link

AR
(1)

AR192413A1
(en)

AT
(2)

AT315168B
(en)

AU
(1)

AU3041871A
(en)

BE
(1)

BE770402A
(en)

BR
(1)

BR7104636D0
(en)

CA
(1)

CA954514A
(en)

CH
(1)

CH543535A
(en)

DE
(1)

DE2137046A1
(en)

ES
(1)

ES393554A1
(en)

FR
(2)

FR2100949B1
(en)

GB
(2)

GB1355033A
(en)

HU
(1)

HU163282B
(en)

IL
(1)

IL37234A0
(en)

NL
(1)

NL7109995A
(en)

ZA
(1)

ZA714030B
(en)

Cited By (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

CN108938628A
(en)

*

2018-08-29
2018-12-07
锁浩
A kind of composition and its application with anti-malarial activity

Families Citing this family (2)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US5593993A
(en)

*

1991-08-02
1997-01-14
Medivir Ab
Method for inhibition of HIV related viruses

IL102548A
(en)

*

1991-08-02
1998-08-16
Medivir Ab
Thiourea derivatives for use in the preparation of medicaments for the inhibition of hiv and the treatment of aids and some such novel compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

FR1265810A
(en)

*

1956-04-13
1961-07-07
Merck & Co Inc

Process for the preparation of urea and thiourea derivatives

FR1533184A
(en)

*

1965-04-06
1968-07-19
Pechiney Saint Gobain

Thiazole derivatives

1970

1970-07-24
CH
CH1123970A
patent/CH543535A/en
not_active
IP Right Cessation

1971

1971-06-21
ZA
ZA714030A
patent/ZA714030B/en
unknown

1971-06-24
AU
AU30418/71A
patent/AU3041871A/en
not_active
Expired

1971-07-05
IL
IL37234A
patent/IL37234A0/en
unknown

1971-07-07
CA
CA117,594A
patent/CA954514A/en
not_active
Expired

1971-07-20
NL
NL7109995A
patent/NL7109995A/xx
unknown

1971-07-22
BR
BR4636/71A
patent/BR7104636D0/en
unknown

1971-07-22
FR
FR7126841A
patent/FR2100949B1/fr
not_active
Expired

1971-07-22
HU
HUHO1397A
patent/HU163282B/hu
unknown

1971-07-23
ES
ES393554A
patent/ES393554A1/en
not_active
Expired

1971-07-23
GB
GB2108473A
patent/GB1355033A/en
not_active
Expired

1971-07-23
AR
AR236970A
patent/AR192413A1/en
active

1971-07-23
BE
BE770402A
patent/BE770402A/en
unknown

1971-07-23
DE
DE19712137046
patent/DE2137046A1/en
active
Pending

1971-07-23
AT
AT847272A
patent/AT315168B/en
not_active
IP Right Cessation

1971-07-23
AT
AT642271A
patent/AT309420B/en
not_active
IP Right Cessation

1971-07-23
GB
GB3475571A
patent/GB1330930A/en
not_active
Expired

1972

1972-11-16
FR
FR7240728A
patent/FR2158578B1/fr
not_active
Expired

Cited By (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

CN108938628A
(en)

*

2018-08-29
2018-12-07
锁浩
A kind of composition and its application with anti-malarial activity

Also Published As

Publication number
Publication date

AR192413A1
(en)

1973-02-21

BR7104636D0
(en)

1973-03-08

CA954514A
(en)

1974-09-10

BE770402A
(en)

1972-01-24

AT309420B
(en)

1973-08-27

FR2158578B1
(en)

1976-03-05

FR2158578A1
(en)

1973-06-15

AT315168B
(en)

1974-05-10

DE2137046A1
(en)

1972-01-27

ES393554A1
(en)

1974-11-16

IL37234A0
(en)

1971-10-20

CH543535A
(en)

1973-10-31

FR2100949A1
(en)

1972-03-24

GB1330930A
(en)

1973-09-19

AU3041871A
(en)

1973-01-04

FR2100949B1
(en)

1975-02-07

HU163282B
(en)

1973-07-28

ZA714030B
(en)

1972-03-29

NL7109995A
(en)

1972-01-26

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(en)

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(en)

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Pharmaceutical compositions comprising aminoguanidine derivatives

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(en)

1978-04-19

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(en)

1972-06-14

Antiinflammatory compositions

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(en)

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Ethanolamine derivatives

GB1277993A
(en)

1972-06-14

Amebicidal compositions and processes

Legal Events

Date
Code
Title
Description

1974-10-09
PS
Patent sealed [section 19, patents act 1949]

1976-02-18
PLNP
Patent lapsed through nonpayment of renewal fees

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