GB1368225A

GB1368225A – 1-aminouracil compounds a processf for their production and their use ans herbicides
– Google Patents

GB1368225A – 1-aminouracil compounds a processf for their production and their use ans herbicides
– Google Patents
1-aminouracil compounds a processf for their production and their use ans herbicides

Info

Publication number
GB1368225A

GB1368225A
GB776173A
GB776173A
GB1368225A
GB 1368225 A
GB1368225 A
GB 1368225A
GB 776173 A
GB776173 A
GB 776173A
GB 776173 A
GB776173 A
GB 776173A
GB 1368225 A
GB1368225 A
GB 1368225A
Authority
GB
United Kingdom
Prior art keywords
optionally substituted
alkyl
formula
aryl
optionally
Prior art date
1972-02-18
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
GB776173A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bayer AG

Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1972-02-18
Filing date
1973-02-16
Publication date
1974-09-25

1973-02-16
Application filed by Bayer AG
filed
Critical
Bayer AG

1974-09-25
Publication of GB1368225A
publication
Critical
patent/GB1368225A/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings

C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings

C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members

C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms

C07D239/46—Two or more oxygen, sulphur or nitrogen atoms

C07D239/52—Two oxygen atoms

C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings

C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings

C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members

C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms

C07D239/46—Two or more oxygen, sulphur or nitrogen atoms

C07D239/52—Two oxygen atoms

C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals

C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms

C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms

C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines

C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems

Abstract

1368225 Herbicidal 1-aminouracils BAYER AG 16 Feb 1973 [18 Feb 1972 14 Sept 1972] 7761/73 Heading C2C New herbicidal compounds are 1-aminouracils or salts thereof, the 1-aminouracils being of the general formula in which R1 represents alkyl, alkenyl, alkynyl, cycloalkyl, alkylcycloalkyl, halocycloalkyl, terpenyl, haloalkyl, cyanoalkyl, alkoxyalkyl, alkoxycarbonylalkyl, alkoxycarbonyl, alkylthiocarbonyl, alkylcarbonyl, alkoxyalkylcarbonyl, aroxyalkylcarbonyl, alkylthioalkyl, optionally substituted arylsulphonyl, aralkyl optionally substituted in the aryl part, optionally substituted arylcarbonyl, optionally substituted phenoxycarbonyl, optionally substituted phenylthiocarbonyl, optionally substituted aryl or an optionally substituted heterocyclic structure, norbornylmethyl or cyclohexylmethyl) R2 represents hydrogen, halogen, the thiocyanate radical, alkyl or optionally substituted aryl, and R3 represents alkyl or aralkyl optionally substituted in the aryl part, or R2 and R3 together represent a multi-membered methylene bridge which forms, with the two carbon atoms in the 5- and 6-position of the heterocyclic structure, a fused ring which is optionally substituted by alkyl. The above compounds may be made by (a) reacting a dihydro-oxazine-dione of formula with hydrazine, optionally in the presence of a diluent at – 30 to +100 C. or (b) reacting a 1- aminouracil of formula in which R4 is alkyl or aralkyl (which may be substituted in the aryl part) with halogen or thiocyanogen, optionally in the presence of an acid binding agent or diluent at 0 to 50 C. The dihydro-oxazine-diones of Formula II may be made by reacting a dioxinone of formula in which R5 is hydrogen or alkyl and R6 is alkyl or aryl with isocyanates of formula optionally in the presence of an inert solvent at +80 to +200C.

GB776173A
1972-02-18
1973-02-16
1-aminouracil compounds a processf for their production and their use ans herbicides

Expired

GB1368225A
(en)

Applications Claiming Priority (1)

Application Number
Priority Date
Filing Date
Title

DE2207549A

DE2207549B2
(en)

1972-02-18
1972-02-18

1-aminouracils and their salts, processes for their preparation and their use as herbicides

Publications (1)

Publication Number
Publication Date

GB1368225A
true

GB1368225A
(en)

1974-09-25

Family
ID=5836269
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

GB776173A
Expired

GB1368225A
(en)

1972-02-18
1973-02-16
1-aminouracil compounds a processf for their production and their use ans herbicides

Country Status (29)

Country
Link

US
(1)

US3920653A
(en)

JP
(2)

JPS4892533A
(en)

AT
(2)

AT325887B
(en)

AU
(1)

AU466590B2
(en)

BE
(1)

BE795549A
(en)

BR
(1)

BR7301190D0
(en)

CA
(1)

CA1027122A
(en)

CH
(1)

CH585512A5
(en)

CS
(1)

CS179408B2
(en)

CY
(1)

CY943A
(en)

DD
(1)

DD103791A5
(en)

DE
(1)

DE2207549B2
(en)

DK
(1)

DK132497C
(en)

ES
(1)

ES411733A1
(en)

FR
(1)

FR2172345B1
(en)

GB
(1)

GB1368225A
(en)

HU
(1)

HU166671B
(en)

IE
(1)

IE37572B1
(en)

IL
(1)

IL41546A
(en)

IT
(1)

IT979209B
(en)

NL
(1)

NL7302152A
(en)

NO
(1)

NO137320C
(en)

PH
(1)

PH12198A
(en)

PL
(1)

PL89226B1
(en)

RO
(1)

RO62816A
(en)

SE
(1)

SE398879B
(en)

SU
(1)

SU580800A3
(en)

TR
(1)

TR17446A
(en)

ZA
(1)

ZA731117B
(en)

Families Citing this family (20)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4448961A
(en)

*

1980-09-14
1984-05-15
Zoecon Corporation
Substituted anilino pyrimidines

FR2549060B1
(en)

*

1983-07-11
1986-06-27
Roussel Uclaf

NOVEL SUBSTITUTED URACILS COMPRISING IN POSITION 1 A SUBSTITUTED PHENYLOXY GROUP, THEIR PREPARATION METHOD AND THE HERBICIDAL COMPOSITIONS CONTAINING THEM

US4526965A
(en)

*

1983-09-16
1985-07-02
Polaroid Corporation
Uracil derivatives of thio- and selenourea compounds

EP0260621A3
(en)

*

1986-09-18
1989-03-15
F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft
3-aryl uracil-enol ethers and their use as herbicides

US5314864A
(en)

*

1989-09-26
1994-05-24
Sumitomo Chemical Company, Limited
N-aminouracil derivatives, and their production and use

JP3064374B2
(en)

*

1989-10-02
2000-07-12
住友化学工業株式会社

Uracil derivative, method for producing the same, and herbicide containing the same as an active ingredient

CA2051942A1
(en)

*

1990-09-21
1992-03-22
Masayuki Enomoto
Uracil derivatives, and their production and use

EP0517181B1
(en)

*

1991-06-07
1995-09-20
Sumitomo Chemical Company Limited
Amino uracil derivatives, and their production and use

WO1994004511A1
(en)

*

1992-08-21
1994-03-03
Nissan Chemical Industries, Ltd.
Pyrimidine derivative and weedkiller

DE4326649A1
(en)

*

1993-08-09
1995-02-16
Bayer Ag

Aminoaryl-1,3-oxazine-2,4-diones

DE19528186A1
(en)

*

1995-08-01
1997-02-06
Bayer Ag

Substituted phenyluracile

DE19532344A1
(en)

*

1995-09-04
1997-03-06
Bayer Ag

Substituted aminouracile

WO1997012886A1
(en)

*

1995-10-04
1997-04-10
Fmc Corporation
Herbicidal heterocyclic benzisoxazoles and benzisoxazolidinones

WO1997042188A1
(en)

*

1996-05-08
1997-11-13
Kumiai Chemical Industry Co., Ltd.
Indolyl-substituted uracil derivatives and herbicides comprising them as active ingredients

DE19651036A1
(en)

*

1996-12-09
1998-06-10
Bayer Ag

3-amino-1-cyanophenyl-uracile

DE19652432A1
(en)

*

1996-12-17
1998-06-18
Bayer Ag

Process for the preparation of 3-amino-1-phenyl-uracil derivatives

DE19652431A1
(en)

*

1996-12-17
1998-06-18
Bayer Ag

Heterocyclyluracile

DE19755926A1
(en)

*

1997-12-17
1999-06-24
Basf Ag

Herbicidal 3- (benzazol-4-yl) pyrimidinedione derivatives

AU3702699A
(en)

*

1998-04-08
1999-11-01
Bayer Aktiengesellschaft
Substituted oxazolyle and thiazolyl uracil herbicides

US6140270A
(en)

*

1998-09-14
2000-10-31
American Cyanamid Company
Process for the preparation of 6-(perfluoroalkyl) uracil compounds from 2-(N,N-disubstituted) amino-4-(perfluoroalkyl)-1,3-oxazin-6-one compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB923608A
(en)

*

1960-03-11
1963-04-18

GB1035097A
(en)

*

1962-12-07
1966-07-06
Du Pont
Improvements relating to herbicides

0

BE
BE795549D
patent/BE795549A/en
unknown

1972

1972-02-18
DE
DE2207549A
patent/DE2207549B2/en
not_active
Withdrawn

1973

1973-02-06
RO
RO7300073745A
patent/RO62816A/en
unknown

1973-02-07
US
US330524A
patent/US3920653A/en
not_active
Expired – Lifetime

1973-02-08
SU
SU7301883551A
patent/SU580800A3/en
active

1973-02-12
PH
PH14340A
patent/PH12198A/en
unknown

1973-02-14
DD
DD168852A
patent/DD103791A5/xx
unknown

1973-02-15
IL
IL7341546A
patent/IL41546A/en
unknown

1973-02-15
TR
TR17446A
patent/TR17446A/en
unknown

1973-02-15
NL
NL7302152A
patent/NL7302152A/xx
not_active
Application Discontinuation

1973-02-16
CH
CH228073A
patent/CH585512A5/xx
not_active
IP Right Cessation

1973-02-16
GB
GB776173A
patent/GB1368225A/en
not_active
Expired

1973-02-16
IT
IT7320511A
patent/IT979209B/en
active

1973-02-16
AT
AT138973A
patent/AT325887B/en
not_active
IP Right Cessation

1973-02-16
ZA
ZA731117A
patent/ZA731117B/en
unknown

1973-02-16
IE
IE244/73A
patent/IE37572B1/en
unknown

1973-02-16
BR
BR731190A
patent/BR7301190D0/en
unknown

1973-02-16
AT
AT599074*7A
patent/AT329076B/en
active

1973-02-16
PL
PL1973160786A
patent/PL89226B1/pl
unknown

1973-02-16
FR
FR7305548A
patent/FR2172345B1/fr
not_active
Expired

1973-02-16
HU
HUBA2872A
patent/HU166671B/hu
unknown

1973-02-16
DK
DK84573*#A
patent/DK132497C/en
active

1973-02-16
CA
CA163,869A
patent/CA1027122A/en
not_active
Expired

1973-02-16
NO
NO73640A
patent/NO137320C/en
unknown

1973-02-16
CY
CY943A
patent/CY943A/en
unknown

1973-02-17
ES
ES411733A
patent/ES411733A1/en
not_active
Expired

1973-02-17
JP
JP48018918A
patent/JPS4892533A/ja
active
Pending

1973-02-17
JP
JP48018917A
patent/JPS4892383A/ja
active
Pending

1973-02-19
CS
CS7300001183A
patent/CS179408B2/en
unknown

1973-02-19
AU
AU52338/73A
patent/AU466590B2/en
not_active
Expired

1973-02-19
SE
SE7302286A
patent/SE398879B/en
unknown

Also Published As

Publication number
Publication date

AU466590B2
(en)

1975-10-30

FR2172345B1
(en)

1977-12-30

DE2207549A1
(en)

1973-08-23

FR2172345A1
(en)

1973-09-28

CY943A
(en)

1978-06-23

AU5233873A
(en)

1974-08-22

JPS4892383A
(en)

1973-11-30

NL7302152A
(en)

1973-08-21

ZA731117B
(en)

1973-11-28

ATA599074A
(en)

1975-07-15

DK132497C
(en)

1976-05-17

NO137320B
(en)

1977-10-31

SE398879B
(en)

1978-01-23

US3920653A
(en)

1975-11-18

CA1027122A
(en)

1978-02-28

CH585512A5
(en)

1977-03-15

ES411733A1
(en)

1976-06-16

PH12198A
(en)

1978-11-28

JPS4892533A
(en)

1973-11-30

ATA138973A
(en)

1975-01-15

IE37572B1
(en)

1977-08-31

AT325887B
(en)

1975-11-10

PL89226B1
(en)

1976-11-30

HU166671B
(en)

1975-05-28

BR7301190D0
(en)

1973-09-25

NO137320C
(en)

1978-02-08

IE37572L
(en)

1973-08-18

DD103791A5
(en)

1974-02-12

BE795549A
(en)

1973-08-16

IL41546A
(en)

1977-05-31

RO62816A
(en)

1978-05-15

CS179408B2
(en)

1977-10-31

DK132497B
(en)

1975-12-15

AT329076B
(en)

1976-04-26

SU580800A3
(en)

1977-11-15

IL41546A0
(en)

1973-04-30

TR17446A
(en)

1975-07-23

IT979209B
(en)

1974-09-30

DE2207549B2
(en)

1979-07-26

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Legal Events

Date
Code
Title
Description

1975-02-05
PS
Patent sealed [section 19, patents act 1949]

1980-10-01
PCNP
Patent ceased through non-payment of renewal fee

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