GB2013683B

GB2013683B – Metronidazole derivatives
– Google Patents

GB2013683B – Metronidazole derivatives
– Google Patents
Metronidazole derivatives

Info

Publication number
GB2013683B

GB2013683B
GB7903940A
GB7903940A
GB2013683B
GB 2013683 B
GB2013683 B
GB 2013683B
GB 7903940 A
GB7903940 A
GB 7903940A
GB 7903940 A
GB7903940 A
GB 7903940A
GB 2013683 B
GB2013683 B
GB 2013683B
Authority
GB
United Kingdom
Prior art keywords
metronidazole
derivatives
metronidazole derivatives
Prior art date
1978-02-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
GB7903940A
Other versions

GB2013683A
(en

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pharmacia and Upjohn Co

Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1978-02-06
Filing date
1979-02-05
Publication date
1982-06-30

1979-02-05
Application filed by Upjohn Co
filed
Critical
Upjohn Co

1979-08-15
Publication of GB2013683A
publication
Critical
patent/GB2013683A/en

1982-06-30
Application granted
granted
Critical

1982-06-30
Publication of GB2013683B
publication
Critical
patent/GB2013683B/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM

C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System

C07F9/02—Phosphorus compounds

C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom

C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms

C07F9/6503—Five-membered rings

C07F9/6506—Five-membered rings having the nitrogen atoms in positions 1 and 3

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics

GB7903940A
1978-02-06
1979-02-05
Metronidazole derivatives

Expired

GB2013683B
(en)

Applications Claiming Priority (1)

Application Number
Priority Date
Filing Date
Title

US05/875,393

US4160827A
(en)

1978-02-06
1978-02-06
Metronidazole phosphate and salts

Publications (2)

Publication Number
Publication Date

GB2013683A

GB2013683A
(en)

1979-08-15

GB2013683B
true

GB2013683B
(en)

1982-06-30

Family
ID=25365724
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

GB7903940A
Expired

GB2013683B
(en)

1978-02-06
1979-02-05
Metronidazole derivatives

Country Status (16)

Country
Link

US
(1)

US4160827A
(en)

JP
(1)

JPS54115375A
(en)

AU
(1)

AU523423B2
(en)

BE
(1)

BE873973A
(en)

CA
(1)

CA1108622A
(en)

CH
(1)

CH638535A5
(en)

DE
(1)

DE2903269A1
(en)

ES
(1)

ES477265A1
(en)

FR
(1)

FR2416234A1
(en)

GB
(1)

GB2013683B
(en)

GR
(1)

GR67623B
(en)

IT
(1)

IT1116516B
(en)

NL
(1)

NL7900858A
(en)

PH
(1)

PH14464A
(en)

SE
(1)

SE445221B
(en)

ZA
(1)

ZA79282B
(en)

Families Citing this family (45)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4386079A
(en)

*

1981-11-23
1983-05-31
The Upjohn Company
Method of treating depression

US4531004A
(en)

*

1981-11-23
1985-07-23
The Upjohn Company
Dimetronidazole phosphates

US5059591B1
(en)

*

1983-05-26
2000-04-25
Liposome Co Inc
Drug preparations of reduced toxicity

CA1237670A
(en)

*

1983-05-26
1988-06-07
Andrew S. Janoff
Drug preparations of reduced toxicity

PT78628B
(en)

*

1984-05-02
1986-06-18
Liposome Co Inc
Pharmaceutical composition with reduced toxicity

US4943579A
(en)

*

1987-10-06
1990-07-24
The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services
Water soluble prodrugs of camptothecin

US7223421B2
(en)

*

2000-06-30
2007-05-29
Mcneil-Ppc, Inc.
Teste masked pharmaceutical particles

US8512718B2
(en)

2000-07-03
2013-08-20
Foamix Ltd.
Pharmaceutical composition for topical application

US6423707B1
(en)

2000-08-28
2002-07-23
California Pacific Medical Center
Nitroimidazole ester analogues and therapeutic applications

WO2002076398A2
(en)

*

2001-03-27
2002-10-03
R.P. Scherer Technologies, Inc.
Improved forms of pharmaceutically active agents and method for manufacture thereof

IL152486A0
(en)

2002-10-25
2003-05-29
Meir Eini
Alcohol-free cosmetic and pharmaceutical foam carrier

MXPA05004278A
(en)

2002-10-25
2005-10-05
Foamix Ltd
Cosmetic and pharmaceutical foam.

US7704518B2
(en)

2003-08-04
2010-04-27
Foamix, Ltd.
Foamable vehicle and pharmaceutical compositions thereof

US8119109B2
(en)

2002-10-25
2012-02-21
Foamix Ltd.
Foamable compositions, kits and methods for hyperhidrosis

US7820145B2
(en)

2003-08-04
2010-10-26
Foamix Ltd.
Oleaginous pharmaceutical and cosmetic foam

US8486376B2
(en)

2002-10-25
2013-07-16
Foamix Ltd.
Moisturizing foam containing lanolin

US9668972B2
(en)

2002-10-25
2017-06-06
Foamix Pharmaceuticals Ltd.
Nonsteroidal immunomodulating kit and composition and uses thereof

US7700076B2
(en)

2002-10-25
2010-04-20
Foamix, Ltd.
Penetrating pharmaceutical foam

US8119150B2
(en)

2002-10-25
2012-02-21
Foamix Ltd.
Non-flammable insecticide composition and uses thereof

US9265725B2
(en)

2002-10-25
2016-02-23
Foamix Pharmaceuticals Ltd.
Dicarboxylic acid foamable vehicle and pharmaceutical compositions thereof

US10117812B2
(en)

2002-10-25
2018-11-06
Foamix Pharmaceuticals Ltd.
Foamable composition combining a polar solvent and a hydrophobic carrier

US8900554B2
(en)

2002-10-25
2014-12-02
Foamix Pharmaceuticals Ltd.
Foamable composition and uses thereof

US9211259B2
(en)

2002-11-29
2015-12-15
Foamix Pharmaceuticals Ltd.
Antibiotic kit and composition and uses thereof

US20080138296A1
(en)

2002-10-25
2008-06-12
Foamix Ltd.
Foam prepared from nanoemulsions and uses

US7575739B2
(en)

2003-04-28
2009-08-18
Foamix Ltd.
Foamable iodine composition

GB0315671D0
(en)

*

2003-07-04
2003-08-13
Chelsea And Westminster Nhs Tr
Improvements in or relating to organic compounds

US8486374B2
(en)

2003-08-04
2013-07-16
Foamix Ltd.
Hydrophilic, non-aqueous pharmaceutical carriers and compositions and uses

US8795693B2
(en)

2003-08-04
2014-08-05
Foamix Ltd.
Compositions with modulating agents

WO2005041853A2
(en)

*

2003-10-28
2005-05-12
Ems S.A.
Antibacterial and/or antiprotozoal nitroimidazole derivative compounds with urease inhibitor activity, process for preparing these compounds and use in pharmaceutical compositions and medicines.

JP2008540508A
(en)

2005-05-09
2008-11-20
フォーミックス エルティーディー.

Foaming vehicle and pharmaceutical composition thereof

US20080260655A1
(en)

2006-11-14
2008-10-23
Dov Tamarkin
Substantially non-aqueous foamable petrolatum based pharmaceutical and cosmetic compositions and their uses

US8636982B2
(en)

2007-08-07
2014-01-28
Foamix Ltd.
Wax foamable vehicle and pharmaceutical compositions thereof

WO2009069006A2
(en)

2007-11-30
2009-06-04
Foamix Ltd.
Foam containing benzoyl peroxide

WO2010041141A2
(en)

2008-10-07
2010-04-15
Foamix Ltd.
Oil-based foamable carriers and formulations

WO2009090495A2
(en)

2007-12-07
2009-07-23
Foamix Ltd.
Oil and liquid silicone foamable carriers and formulations

WO2009090558A2
(en)

2008-01-14
2009-07-23
Foamix Ltd.
Poloxamer foamable pharmaceutical compositions with active agents and/or therapeutic cells and uses

WO2010125470A2
(en)

2009-04-28
2010-11-04
Foamix Ltd.
Foamable vehicle and pharmaceutical compositions comprising aprotic polar solvents and uses thereof

WO2011013009A2
(en)

2009-07-29
2011-02-03
Foamix Ltd.
Non surfactant hydro-alcoholic foamable compositions, breakable foams and their uses

CA2769677A1
(en)

2009-07-29
2011-02-03
Foamix Ltd.
Non surface active agent non polymeric agent hydro-alcoholic foamable compositions, breakable foams and their uses

CN102686205A
(en)

2009-10-02
2012-09-19
弗艾米克斯有限公司
Topical tetracycline compositions

US9849142B2
(en)

2009-10-02
2017-12-26
Foamix Pharmaceuticals Ltd.
Methods for accelerated return of skin integrity and for the treatment of impetigo

CN102516299A
(en)

*

2011-12-09
2012-06-27
陕西合成药业有限公司
S-Ornidazole phosphate amino acid salt, its preparation method and application

CN102516298A
(en)

*

2011-12-09
2012-06-27
陕西合成药业有限公司
Stable pharmaceutical salt of L-aonitrate phosphate ester, its preparation method and application

CA2978573A1
(en)

2016-09-08
2018-03-08
Foamix Pharmaceuticals Ltd.
Compositions and methods for treating rosacea and acne

CN108295039A
(en)

*

2018-02-28
2018-07-20
重庆希尔安药业有限公司
Metronidazole vagina effervescent tablet and preparation method thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

BE571291A
(en)

*

1957-09-20
1962-01-12
Rhone Poulenc Sa

NEW DERIVATIVES OF IMIDAZOLE AND THEIR PREPARATION.

US2944061A
(en)

*

1957-09-20
1960-07-05

Acyl derivatives and process

GB1280355A
(en)

*

1969-06-20
1972-07-05
Rech S Et D Applic Scient Et M
Substituted 5-nitro-imidazoles and their preparation

FR2054504B1
(en)

*

1969-07-18
1973-06-08
Rhone Poulenc Sa

US3910945A
(en)

*

1972-10-04
1975-10-07
Searle & Co
2-(2-Methyl-5-nitro-1-imidazolyl)ethyl-N-arylalkyldithiocarbamates

US3882136A
(en)

*

1973-11-16
1975-05-06
Searle & Co
S-{8 omega-(1-imidazolyl) alkyl{9 hydrogen monothiosulfates and salts thereof

1978

1978-02-06
US
US05/875,393
patent/US4160827A/en
not_active
Expired – Lifetime

1979

1979-01-17
CA
CA319,763A
patent/CA1108622A/en
not_active
Expired

1979-01-23
ZA
ZA79282A
patent/ZA79282B/en
unknown

1979-01-26
AU
AU43705/79A
patent/AU523423B2/en
not_active
Ceased

1979-01-29
DE
DE2903269A
patent/DE2903269A1/en
not_active
Ceased

1979-01-29
GR
GR58208A
patent/GR67623B/el
unknown

1979-01-30
ES
ES477265A
patent/ES477265A1/en
not_active
Expired

1979-02-02
IT
IT47874/79A
patent/IT1116516B/en
active

1979-02-02
NL
NL7900858A
patent/NL7900858A/en
not_active
Application Discontinuation

1979-02-02
SE
SE7900952A
patent/SE445221B/en
not_active
IP Right Cessation

1979-02-05
GB
GB7903940A
patent/GB2013683B/en
not_active
Expired

1979-02-05
FR
FR7902950A
patent/FR2416234A1/en
active
Granted

1979-02-05
PH
PH22156A
patent/PH14464A/en
unknown

1979-02-06
CH
CH116479A
patent/CH638535A5/en
not_active
IP Right Cessation

1979-02-06
BE
BE0/193304A
patent/BE873973A/en
not_active
IP Right Cessation

1979-02-06
JP
JP1275979A
patent/JPS54115375A/en
active
Pending

Also Published As

Publication number
Publication date

AU4370579A
(en)

1979-08-16

IT1116516B
(en)

1986-02-10

GR67623B
(en)

1981-09-01

US4160827A
(en)

1979-07-10

NL7900858A
(en)

1979-08-08

ES477265A1
(en)

1980-10-01

FR2416234A1
(en)

1979-08-31

IT7947874D0
(en)

1979-02-02

BE873973A
(en)

1979-08-06

FR2416234B1
(en)

1983-02-04

JPS54115375A
(en)

1979-09-07

CA1108622A
(en)

1981-09-08

SE7900952L
(en)

1979-08-07

GB2013683A
(en)

1979-08-15

PH14464A
(en)

1981-07-29

ZA79282B
(en)

1980-01-30

SE445221B
(en)

1986-06-09

DE2903269A1
(en)

1979-08-09

CH638535A5
(en)

1983-09-30

AU523423B2
(en)

1982-07-29

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Legal Events

Date
Code
Title
Description

1988-09-28
PCNP
Patent ceased through non-payment of renewal fee

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