AU2123797A

AU2123797A – 2-thioxotetrahydropyrimidin-4-one derivatives
– Google Patents

AU2123797A – 2-thioxotetrahydropyrimidin-4-one derivatives
– Google Patents
2-thioxotetrahydropyrimidin-4-one derivatives

Info

Publication number
AU2123797A

AU2123797A
AU21237/97A
AU2123797A
AU2123797A
AU 2123797 A
AU2123797 A
AU 2123797A
AU 21237/97 A
AU21237/97 A
AU 21237/97A
AU 2123797 A
AU2123797 A
AU 2123797A
AU 2123797 A
AU2123797 A
AU 2123797A
Authority
AU
Australia
Prior art keywords
thioxotetrahydropyrimidin
derivatives
Prior art date
1996-03-07
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU21237/97A
Other versions

AU707732B2
(en

Inventor
Sie-Yearl Chai
Hassan Mahmoud Elokdah
Theodore Sylvester Sulkowski
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Wyeth LLC

Original Assignee
American Home Products Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1996-03-07
Filing date
1997-02-12
Publication date
1997-09-22

1997-02-12
Application filed by American Home Products Corp
filed
Critical
American Home Products Corp

1997-09-22
Publication of AU2123797A
publication
Critical
patent/AU2123797A/en

1999-07-15
Application granted
granted
Critical

1999-07-15
Publication of AU707732B2
publication
Critical
patent/AU707732B2/en

2017-02-12
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings

C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings

C07D239/20—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members

C07D239/22—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES

A61K31/00—Medicinal preparations containing organic active ingredients

A61K31/33—Heterocyclic compounds

A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins

A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines

A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P9/00—Drugs for disorders of the cardiovascular system

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P9/00—Drugs for disorders of the cardiovascular system

A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

AU21237/97A
1996-03-07
1997-02-12
2-thioxotetrahydropyrimidin-4-one derivatives

Ceased

AU707732B2
(en)

Applications Claiming Priority (3)

Application Number
Priority Date
Filing Date
Title

US1299396P

1996-03-07
1996-03-07

US60/012993

1996-03-07

PCT/US1997/002281

WO1997032855A1
(en)

1996-03-07
1997-02-12
2-thioxotetrahydropyrimidin-4-one derivatives

Publications (2)

Publication Number
Publication Date

AU2123797A
true

AU2123797A
(en)

1997-09-22

AU707732B2

AU707732B2
(en)

1999-07-15

Family
ID=21757747
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU21237/97A
Ceased

AU707732B2
(en)

1996-03-07
1997-02-12
2-thioxotetrahydropyrimidin-4-one derivatives

Country Status (15)

Country
Link

US
(1)

US5807864A
(en)

EP
(1)

EP0885197A1
(en)

JP
(1)

JP2000507926A
(en)

KR
(1)

KR19990087582A
(en)

CN
(1)

CN1217715A
(en)

AR
(1)

AR005986A1
(en)

AU
(1)

AU707732B2
(en)

BR
(1)

BR9708310A
(en)

CA
(1)

CA2247933A1
(en)

HU
(1)

HU9901968A3
(en)

IL
(1)

IL125974A0
(en)

NZ
(1)

NZ332199A
(en)

TW
(1)

TW422840B
(en)

WO
(1)

WO1997032855A1
(en)

ZA
(1)

ZA971911B
(en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

WO1998021190A1
(en)

*

1996-11-14
1998-05-22
American Home Products Corporation
Substituted tetrahydro-1,3,5-triazin-2[1h]-thiones as anti-atherosclerotic agents

WO2002028845A1
(en)

*

2000-10-02
2002-04-11
Wyeth
3-thioxo-[1,2,4]-oxadiazinan-5-one and their use as anti-antherosclerotic agents

US20050096319A1
(en)

*

2003-02-21
2005-05-05
Balzarini Jan M.R.
Identification of compounds that inhibit replication of human immunodeficiency virus

CN102423314A
(en)

*

2011-11-26
2012-04-25
济南环肽医药科技有限公司
Medicine for treating immunological liver injury or immunological liver fibrosis

Family Cites Families (7)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

JPS55108858A
(en)

*

1979-02-14
1980-08-21
Kyowa Hakko Kogyo Co Ltd
Novel dihydrouracil derivative and herbicide

JPS5939875A
(en)

*

1982-08-31
1984-03-05
Sagami Chem Res Center
Preparation of 5-trifluoromethyldihydrouracils

JPS60243017A
(en)

*

1984-05-16
1985-12-03
Kyowa Hakko Kogyo Co Ltd
Antispasmodic composition

JPH0651682B2
(en)

*

1986-09-05
1994-07-06
株式会社上野製薬応用研究所

Method for producing uracil derivative

US4927451A
(en)

*

1988-12-30
1990-05-22
Uniroyal Chemical Company, Inc.
3-aryldihydrouracils

DE4318550A1
(en)

*

1993-06-04
1994-12-08
Boehringer Mannheim Gmbh

Arylidene-4-oxo-2-thioxo-3-thiazolidinecarboxylic acids, process for their preparation and pharmaceutical compositions containing them

US5554607A
(en)

*

1995-11-28
1996-09-10
American Home Products Corporation
Use of 2-thioxo-imidazolin-4-one derivatives in the treatment of atherosclerosis

1997

1997-02-12
WO
PCT/US1997/002281
patent/WO1997032855A1/en
not_active
Application Discontinuation

1997-02-12
NZ
NZ332199A
patent/NZ332199A/en
unknown

1997-02-12
IL
IL12597497A
patent/IL125974A0/en
unknown

1997-02-12
EP
EP97906583A
patent/EP0885197A1/en
not_active
Withdrawn

1997-02-12
JP
JP9531771A
patent/JP2000507926A/en
active
Pending

1997-02-12
HU
HU9901968A
patent/HU9901968A3/en
unknown

1997-02-12
CA
CA002247933A
patent/CA2247933A1/en
not_active
Abandoned

1997-02-12
BR
BR9708310A
patent/BR9708310A/en
not_active
Application Discontinuation

1997-02-12
CN
CN97194335A
patent/CN1217715A/en
active
Pending

1997-02-12
KR
KR1019980707023A
patent/KR19990087582A/en
not_active
Application Discontinuation

1997-02-12
AU
AU21237/97A
patent/AU707732B2/en
not_active
Ceased

1997-02-20
TW
TW086102010A
patent/TW422840B/en
active

1997-02-24
AR
ARP970100745A
patent/AR005986A1/en
unknown

1997-02-27
US
US08/807,164
patent/US5807864A/en
not_active
Expired – Lifetime

1997-03-05
ZA
ZA971911A
patent/ZA971911B/en
unknown

Also Published As

Publication number
Publication date

KR19990087582A
(en)

1999-12-27

US5807864A
(en)

1998-09-15

NZ332199A
(en)

1999-03-29

JP2000507926A
(en)

2000-06-27

EP0885197A1
(en)

1998-12-23

TW422840B
(en)

2001-02-21

WO1997032855A1
(en)

1997-09-12

ZA971911B
(en)

1998-09-07

CA2247933A1
(en)

1997-09-12

IL125974A0
(en)

1999-04-11

BR9708310A
(en)

1999-08-03

HU9901968A2
(en)

1999-10-28

AU707732B2
(en)

1999-07-15

HU9901968A3
(en)

2000-01-28

CN1217715A
(en)

1999-05-26

AR005986A1
(en)

1999-07-21

Similar Documents

Publication
Publication Date
Title

AU1151099A
(en)

1999-05-17

Azaoxindole derivatives

AU1825899A
(en)

1999-07-05

Dota-biotin derivatives

AU2070795A
(en)

1995-10-17

3-aryl-4-hydroxy-delta3-dihydrothiophenone derivatives

AU7935398A
(en)

1999-01-25

Diaminorhodamine derivatives

AU6117998A
(en)

1998-10-20

3-oxadiazolylquinoxaline derivatives

AU1594697A
(en)

1997-08-20

New substituted 19-nor-pregnane derivatives

AU3867997A
(en)

1998-03-19

Chromene-3-carboxylate derivatives

AU1735497A
(en)

1997-09-10

Sulfonylureidopyrazole derivatives

AU7738098A
(en)

1998-07-15

Novel tetrahydrobenzindolone derivatives

AU2956097A
(en)

1997-12-05

Alkylaminobenzothiazole and -benzoxazole derivatives

EP1008579A3
(en)

2003-01-29

Cyclopentenebutanol derivatives

AU2485595A
(en)

1996-01-25

1-Pyridyltetrazolinone derivatives

AU2090897A
(en)

1997-09-16

Hydroxyhexahydropyridazines

AU2961097A
(en)

1998-01-05

Substituted pyrazolylpyrazole derivatives

AU7813598A
(en)

1998-12-21

Betulinol derivatives

AU4962097A
(en)

1998-05-22

2-methoxyphenylpiperazine derivatives

AU1793197A
(en)

1997-09-10

Pyrazole-4-yl-hetaroyl derivatives

AU1174199A
(en)

1999-06-15

Biphenylamidine derivatives

AU6729498A
(en)

1998-10-20

Thiazolimine derivatives

AU4117396A
(en)

1996-06-19

Morpholinoethylamide derivatives

AU3685097A
(en)

1998-03-12

N-benzylazolium derivatives

AU689566B2
(en)

1998-04-02

DC-89 derivatives

AU1900097A
(en)

1997-11-06

Cremators

AU6115798A
(en)

1998-09-18

Saponarin derivatives

AU1562199A
(en)

1999-06-16

Amino-benzothiazole derivatives

Legal Events

Date
Code
Title
Description

2002-09-12
MK14
Patent ceased section 143(a) (annual fees not paid) or expired

Download PDF in English

None