AU2547584A - Creación de Inventos y Patentes con Inteligencia Artificial

AU2547584A – 1- phenyl-2-azole-ethylamino-carbonyl derivatives
– Google Patents

AU2547584A – 1- phenyl-2-azole-ethylamino-carbonyl derivatives
– Google Patents
1- phenyl-2-azole-ethylamino-carbonyl derivatives

Info

Publication number
AU2547584A

AU2547584A
AU25475/84A
AU2547584A
AU2547584A
AU 2547584 A
AU2547584 A
AU 2547584A
AU 25475/84 A
AU25475/84 A
AU 25475/84A
AU 2547584 A
AU2547584 A
AU 2547584A
AU 2547584 A
AU2547584 A
AU 2547584A
Authority
AU
Australia
Prior art keywords
azole
ethylamino
phenyl
carbonyl derivatives
carbonyl
Prior art date
1983-03-11
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU25475/84A
Other versions

AU571494B2
(en

Inventor
Helmut Egger
Anton Stutz
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sandoz AG

Original Assignee
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1983-03-11
Filing date
1984-03-09
Publication date
1984-09-13

1984-03-09
Application filed by Sandoz AG
filed
Critical
Sandoz AG

1984-09-13
Publication of AU2547584A
publication
Critical
patent/AU2547584A/en

1988-04-21
Application granted
granted
Critical

1988-04-21
Publication of AU571494B2
publication
Critical
patent/AU571494B2/en

2004-03-09
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members

C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D213/62—Oxygen or sulfur atoms

C07D213/70—Sulfur atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS

C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds

C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups

C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings

C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings

C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members

C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings

C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members

C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms

C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings

C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms

C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms

C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms

C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof

C07D295/182—Radicals derived from carboxylic acids

C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof

C07D295/215—Radicals derived from nitrogen analogues of carbonic acid

AU25475/84A
1983-03-11
1984-03-09
1- phenyl-2-azole-ethylamino-carbonyl derivatives

Ceased

AU571494B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

CH1332/83

1983-03-11

CH1332/83A

CH655103A5
(en)

1983-03-11
1983-03-11

AZOLE DERIVATIVES, METHOD FOR THEIR PRODUCTION AND THEIR USE.

Publications (2)

Publication Number
Publication Date

AU2547584A
true

AU2547584A
(en)

1984-09-13

AU571494B2

AU571494B2
(en)

1988-04-21

Family
ID=4207992
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU25475/84A
Ceased

AU571494B2
(en)

1983-03-11
1984-03-09
1- phenyl-2-azole-ethylamino-carbonyl derivatives

Country Status (24)

Country
Link

JP
(1)

JPS59175472A
(en)

KR
(1)

KR890000377B1
(en)

AU
(1)

AU571494B2
(en)

BE
(1)

BE899073A
(en)

CA
(1)

CA1242723A
(en)

CH
(1)

CH655103A5
(en)

DE
(1)

DE3408127A1
(en)

DK
(1)

DK149784A
(en)

ES
(1)

ES530461A0
(en)

FI
(1)

FI840968A
(en)

FR
(1)

FR2542315B1
(en)

GB
(1)

GB2136801B
(en)

GR
(1)

GR81869B
(en)

HU
(1)

HUT36098A
(en)

IL
(1)

IL71203A
(en)

IT
(1)

IT1199085B
(en)

LU
(1)

LU85245A1
(en)

NL
(1)

NL8400730A
(en)

NZ
(1)

NZ207453A
(en)

PH
(1)

PH24667A
(en)

PL
(1)

PL146072B1
(en)

PT
(1)

PT78226B
(en)

SE
(1)

SE8401321L
(en)

ZA
(1)

ZA841782B
(en)

Families Citing this family (24)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB8618188D0
(en)

1986-07-25
1986-09-03
Ici Plc
Diamine compounds

DE3644615A1
(en)

1986-12-29
1988-07-07
Lentia Gmbh

IMIDAZOLE AND TRIAZOLE DERIVATIVES FOR USE AS AN ANTIMYCOTIC AGENTS

DE3644616A1
(en)

1986-12-29
1988-07-07
Lentia Gmbh

IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION AND USE THEREOF

US5252594A
(en)

1992-06-17
1993-10-12
Rohm And Haas Company
Fungicidal (2-aryl-2-substituted)ethyl-1,2,4-triazoles

US5358939A
(en)

1992-06-25
1994-10-25
Rohm And Haas Company
Fungicidal 2-aryl-2,2-disubstituted ethyl-1,2,4-triazoles

DE4412358A1
(en)

1994-04-11
1995-10-12
Bayer Ag

Cyclopropyl ethyl azoles

GB9409882D0
(en)

1994-05-18
1994-07-06
Sandoz Ltd
Organic compounds

JP3214987B2
(en)

1994-09-05
2001-10-02
日本碍子株式会社

Semiconductor device and method of manufacturing the same

AU2003299750A1
(en)

2002-12-20
2004-07-22
Irm Llc
Differential tumor cytotoxocity compounds and compositions

WO2004056744A1
(en)

2002-12-23
2004-07-08
Janssen Pharmaceutica N.V.
Adamantyl acetamides as hydroxysteroid dehydrogenase inhibitors

KR101192861B1
(en)

2004-05-07
2012-10-19
얀센 파마슈티카 엔.브이.
Pyrrolidin-2-one and piperidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors

DE602005017159D1
(en)

2004-08-30
2009-11-26
Janssen Pharmaceutica Nv

OXYSTEROID DEHYDROGENASE INHIBITORS

NZ553159A
(en)

2004-08-30
2010-05-28
Janssen Pharmaceutica Nv
N-Adamantan-2-yl-2-phenoxy-acetamide derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors

AU2005279209B2
(en)

2004-08-30
2011-03-24
Janssen Pharmaceutica N.V.
Tricyclic lactam derivatives as 11-BETA hydroxysteroid dehydrogenase inhibitors

CN101084207A
(en)

2004-09-20
2007-12-05
泽农医药公司
Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors

AR051092A1
(en)

2004-09-20
2006-12-20
Xenon Pharmaceuticals Inc

HETEROCICLIC DERIVATIVES AND THEIR USE AS INHIBITORS OF ESTEAROIL-COA

CA2580844A1
(en)

2004-09-20
2006-03-30
Xenon Pharmaceuticals Inc.
Heterocyclic derivatives and their use as mediators of stearoyl-coa desaturase

CN101083982A
(en)

2004-09-20
2007-12-05
泽农医药公司
Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes

AU2005329423A1
(en)

2004-09-20
2006-09-28
Xenon Pharmaceuticals Inc.
Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors

WO2006034279A1
(en)

2004-09-20
2006-03-30
Xenon Pharmaceuticals Inc.
Heterocyclic derivatives and their use as therapeutic agents

CN101083992A
(en)

2004-09-20
2007-12-05
泽农医药公司
Pyridazine derivatives for inhibiting human stearoyl-coa-desaturase

BRPI0611187A2
(en)

2005-06-03
2010-08-24
Xenon Pharmaceuticals Inc

amino thiazide derivatives as inhibitors of human stearoyl coa desaturase

CN104530038A
(en)

2014-12-10
2015-04-22
沈阳药科大学
Amide imidazole derivative and application thereof

CN112142673B
(en)

2020-09-18
2023-06-30
聊城大学
Aryl alkene azole derivative and preparation method and application thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

SU557755A3
(en)

1968-08-19
1977-05-05
Янссен Фармасьютика Н.В. (Фирма)

Method for preparing imidazole derivatives

CA1189857A
(en)

1981-03-27
1985-07-02
Janssen Pharmaceutica Naamloze Vennootschap
Antimicrobial triazole derivatives

AU8314482A
(en)

1981-05-19
1982-11-25
Imperial Chemical Industries Plc
3-triazolyl(imidazolyl)-2,2 bis phenyl-propionamides

EP0117462A3
(en)

1983-02-28
1986-08-20
American Cyanamid Company
N-(2-4-(1h-imidazol-1-yl)alkyl)arylamides

1983

1983-03-11
CH
CH1332/83A
patent/CH655103A5/en
not_active
IP Right Cessation

1984

1984-02-27
HU
HU84780A
patent/HUT36098A/en
unknown

1984-02-29
DK
DK149784A
patent/DK149784A/en
not_active
Application Discontinuation

1984-03-05
BE
BE1/10974A
patent/BE899073A/en
not_active
IP Right Cessation

1984-03-05
FR
FR8403733A
patent/FR2542315B1/en
not_active
Expired

1984-03-06
DE
DE19843408127
patent/DE3408127A1/en
not_active
Withdrawn

1984-03-07
NL
NL8400730A
patent/NL8400730A/en
not_active
Application Discontinuation

1984-03-07
GB
GB08405900A
patent/GB2136801B/en
not_active
Expired

1984-03-08
IT
IT47817/84A
patent/IT1199085B/en
active

1984-03-09
PT
PT78226A
patent/PT78226B/en
not_active
IP Right Cessation

1984-03-09
CA
CA000449330A
patent/CA1242723A/en
not_active
Expired

1984-03-09
FI
FI840968A
patent/FI840968A/en
not_active
Application Discontinuation

1984-03-09
IL
IL71203A
patent/IL71203A/en
unknown

1984-03-09
PL
PL1984246600A
patent/PL146072B1/en
unknown

1984-03-09
SE
SE8401321A
patent/SE8401321L/en
not_active
Application Discontinuation

1984-03-09
PH
PH30375A
patent/PH24667A/en
unknown

1984-03-09
LU
LU85245A
patent/LU85245A1/en
unknown

1984-03-09
NZ
NZ207453A
patent/NZ207453A/en
unknown

1984-03-09
AU
AU25475/84A
patent/AU571494B2/en
not_active
Ceased

1984-03-09
ES
ES530461A
patent/ES530461A0/en
active
Granted

1984-03-09
ZA
ZA841782A
patent/ZA841782B/en
unknown

1984-03-10
KR
KR1019840001218A
patent/KR890000377B1/en
not_active
IP Right Cessation

1984-03-10
JP
JP59046384A
patent/JPS59175472A/en
active
Pending

1984-03-12
GR
GR74070A
patent/GR81869B/el
unknown

Also Published As

Publication number
Publication date

FR2542315A1
(en)

1984-09-14

BE899073A
(en)

1984-09-05

GB8405900D0
(en)

1984-04-11

CH655103A5
(en)

1986-03-27

ZA841782B
(en)

1985-10-30

SE8401321D0
(en)

1984-03-09

KR890000377B1
(en)

1989-03-15

KR850006386A
(en)

1985-10-05

LU85245A1
(en)

1984-11-14

DE3408127A1
(en)

1984-09-13

FR2542315B1
(en)

1986-02-07

ES8506639A1
(en)

1985-07-16

PL146072B1
(en)

1988-12-31

FI840968A
(en)

1984-09-12

GB2136801B
(en)

1987-03-04

IT1199085B
(en)

1988-12-30

GR81869B
(en)

1984-12-12

NZ207453A
(en)

1987-09-30

PT78226A
(en)

1984-04-01

ES530461A0
(en)

1985-07-16

IL71203A0
(en)

1984-06-29

FI840968A0
(en)

1984-03-09

PH24667A
(en)

1990-09-07

CA1242723A
(en)

1988-10-04

NL8400730A
(en)

1984-10-01

HUT36098A
(en)

1985-08-28

PL246600A1
(en)

1985-03-12

GB2136801A
(en)

1984-09-26

DK149784D0
(en)

1984-02-29

PT78226B
(en)

1986-07-15

IL71203A
(en)

1988-10-31

AU571494B2
(en)

1988-04-21

DK149784A
(en)

1984-09-12

JPS59175472A
(en)

1984-10-04

IT8447817D0
(en)

1984-03-08

SE8401321L
(en)

1984-09-12

Información de contacto