AU3177271A

AU3177271A – Piperazine derivatives, processes for their preparation and pharmaceutical compositions containing thesame
– Google Patents

AU3177271A – Piperazine derivatives, processes for their preparation and pharmaceutical compositions containing thesame
– Google Patents
Piperazine derivatives, processes for their preparation and pharmaceutical compositions containing thesame

Info

Publication number
AU3177271A

AU3177271A
AU31772/71A
AU3177271A
AU3177271A
AU 3177271 A
AU3177271 A
AU 3177271A
AU 31772/71 A
AU31772/71 A
AU 31772/71A
AU 3177271 A
AU3177271 A
AU 3177271A
AU 3177271 A
AU3177271 A
AU 3177271A
Authority
AU
Australia
Prior art keywords
processes
preparation
pharmaceutical compositions
compositions containing
piperazine derivatives
Prior art date
1970-07-30
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
AU31772/71A
Other versions

AU463957B2
(en

Inventor
KURT SCHRAMM ANTON MENTRUP and ROLF GIESEMANN ERNST-OTTO RENTH
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Boehringer Ingelheim GmbH

Original Assignee
CH Boehringer Sohn AG and Co KG
Boehringer Ingelheim GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1970-07-30
Filing date
1971-07-29
Publication date
1973-02-01

1971-07-29
Application filed by CH Boehringer Sohn AG and Co KG, Boehringer Ingelheim GmbH
filed
Critical
CH Boehringer Sohn AG and Co KG

1973-02-01
Publication of AU3177271A
publication
Critical
patent/AU3177271A/en

1975-08-14
Application granted
granted
Critical

1975-08-14
Publication of AU463957B2
publication
Critical
patent/AU463957B2/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms

C07D295/02—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements

C07D295/027—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring

C07D295/03—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring with the ring nitrogen atoms directly attached to acyclic carbon atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings

C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems

C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring

C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms

C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3

C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems

C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring

C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring

C07D317/56—Radicals substituted by sulfur atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms

C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3

C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems

C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring

C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring

C07D317/58—Radicals substituted by nitrogen atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms

C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes

C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems

C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring

C07D319/18—Ethylenedioxybenzenes, not substituted on the hetero ring

AU31772/71A
1970-07-30
1971-07-29
Piperazine derivatives, processes for their preparation and pharmaceutical compositions containing thesame

Expired

AU463957B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

DEDE820378

1970-07-30

DE2037852A

DE2037852C3
(en)

1970-07-30
1970-07-30

New piperazine derivatives and processes for their preparation

Publications (2)

Publication Number
Publication Date

AU3177271A
true

AU3177271A
(en)

1973-02-01

AU463957B2

AU463957B2
(en)

1975-08-14

Family
ID=5778382
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU31772/71A
Expired

AU463957B2
(en)

1970-07-30
1971-07-29
Piperazine derivatives, processes for their preparation and pharmaceutical compositions containing thesame

Country Status (19)

Country
Link

US
(1)

US3808212A
(en)

JP
(1)

JPS5716989B1
(en)

AT
(6)

AT311987B
(en)

AU
(1)

AU463957B2
(en)

BE
(1)

BE770800A
(en)

BG
(5)

BG20594A3
(en)

CH
(6)

CH565166A5
(en)

CS
(1)

CS172929B2
(en)

DE
(1)

DE2037852C3
(en)

DK
(1)

DK137990C
(en)

ES
(6)

ES393738A1
(en)

FR
(1)

FR2100972B1
(en)

GB
(1)

GB1344720A
(en)

NL
(1)

NL173643C
(en)

PL
(6)

PL84347B1
(en)

RO
(6)

RO60597A
(en)

SE
(2)

SE375308B
(en)

SU
(5)

SU437290A3
(en)

YU
(7)

YU34530B
(en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US3991036A
(en)

*

1973-02-28
1976-11-09
Uniroyal Inc.
Preparation of polyurethane using 1,2,3,4,4a,5,7,7a-Octahydrothieno[3,4-b]py

US3940396A
(en)

*

1973-02-28
1976-02-24
Uniroyal Inc.
1,2,3,4,4A,5,7,7A-Octahydrothieno[3,4-b]pyrazines 6,6-dioxides

GB1407552A
(en)

*

1973-04-02
1975-09-24
Science Union & Cie
Disubstituted piperazines processes for their preparation and pharmaceutical compositions containing them

GB1432660A
(en)

*

1973-10-30
1976-04-22
Science Union & Cie
Piperazine derivatives processes for their preparation and and pharamacueitcal compositions containing them

US3960863A
(en)

*

1974-06-25
1976-06-01
Sankyo Company Limited
Pyrido[1,2-a]pyrimidinone derivatives

DE2604838A1
(en)

*

1976-02-07
1977-08-11
Knoll Ag

ALKYLENE DIOXYPIPERAZINE DERIVATIVES

AU561190B2
(en)

*

1983-01-21
1987-04-30
Fisons Plc
Aromatic amines

EP0190472B1
(en)

*

1984-12-21
1989-07-12
Duphar International Research B.V
New pharmaceutical compositions having anti-psychotic properties

FR2692264B1
(en)

*

1992-06-12
1994-08-05
Adir

NOVEL 1,4-DISUBSTITUTED PIPERAZINES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.

FR2734819B1
(en)

*

1995-05-31
1997-07-04
Adir

NOVEL COMPOUNDS OF PIPERAZINE, PIPERIDINE AND 1,2,5,6-TETRAHYDROPYRIDINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

US6002005A
(en)

*

1995-06-02
1999-12-14
Neurogen Corporation
Certain 1-substituted aminomethyl imidazole and pyrrole derivatives: novel dopamine receptor subtype specific ligands

FR2737724B1
(en)

*

1995-08-09
1997-09-05
Synthelabo

DERIVATIVES OF 1- [2- (2,3-DIHYDRO-1H-INDEN-1-YL) ETHYL] -4- (NAPHTALEN-1-YL) PIPERAZINE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

JPH09124643A
(en)

*

1995-08-14
1997-05-13
Bristol Myers Squibb Co
Antidepressant 1-arylalkyl-4-(alkoxypyrimidinyl)- or 4-(alkoxypyrimidinyl)piperazine derivative

US6040448A
(en)

*

1997-10-24
2000-03-21
Neurogen Corporation
Certain 1-(2-naphthyl) and 1-(2-azanaphthyl)-4-(1-phenylmethyl) piperazines, dopamine receptor subtype specific ligands

MA41169A
(en)

*

2014-12-17
2017-10-24
Acraf

WIDE-SPECTRUM ANTIBACTERIAL COMPOUNDS

Family Cites Families (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

NL132357C
(en)

*

1966-09-03

1970

1970-07-30
DE
DE2037852A
patent/DE2037852C3/en
not_active
Expired

1971

1971-06-23
RO
RO69219A
patent/RO60597A/ro
unknown

1971-06-23
RO
RO69220A
patent/RO60598A/ro
unknown

1971-06-23
RO
RO69218A
patent/RO61040A/ro
unknown

1971-06-23
RO
RO67429A
patent/RO59997A/ro
unknown

1971-06-23
RO
RO69217A
patent/RO60596A/ro
unknown

1971-06-23
RO
RO69222A
patent/RO60599A/ro
unknown

1971-07-08
US
US00160891A
patent/US3808212A/en
not_active
Expired – Lifetime

1971-07-27
CH
CH524075A
patent/CH565166A5/xx
not_active
IP Right Cessation

1971-07-27
CH
CH524175A
patent/CH565167A5/xx
not_active
IP Right Cessation

1971-07-27
CH
CH1106871A
patent/CH565780A5/xx
not_active
IP Right Cessation

1971-07-27
CH
CH523875A
patent/CH565165A5/xx
not_active
IP Right Cessation

1971-07-27
CH
CH523975A
patent/CH565781A5/xx
not_active
IP Right Cessation

1971-07-27
CH
CH524275A
patent/CH575412A5/xx
not_active
IP Right Cessation

1971-07-28
SU
SU1815878A
patent/SU437290A3/en
active

1971-07-28
SU
SU1815881A
patent/SU437292A3/en
active

1971-07-28
BG
BG21486A
patent/BG20594A3/xx
unknown

1971-07-28
CS
CS5538A
patent/CS172929B2/cs
unknown

1971-07-28
BG
BG18177A
patent/BG21029A3/xx
unknown

1971-07-28
BG
BG21487A
patent/BG19598A3/xx
unknown

1971-07-28
SU
SU1688445A
patent/SU416945A3/en
active

1971-07-28
JP
JP5608071A
patent/JPS5716989B1/ja
active
Pending

1971-07-28
SU
SU1815879A
patent/SU440840A3/ru
active

1971-07-28
BG
BG21484A
patent/BG20369A3/xx
unknown

1971-07-28
BG
BG21488A
patent/BG20370A3/xx
unknown

1971-07-28
SU
SU1815875A
patent/SU437289A3/en
active

1971-07-29
PL
PL1971178480A
patent/PL84347B1/pl
unknown

1971-07-29
AT
AT1100372A
patent/AT311987B/en
active

1971-07-29
ES
ES393738A
patent/ES393738A1/en
not_active
Expired

1971-07-29
PL
PL1971178478A
patent/PL84349B1/pl
unknown

1971-07-29
PL
PL1971149717A
patent/PL84664B1/pl
unknown

1971-07-29
AT
AT1100172A
patent/AT311985B/en
not_active
IP Right Cessation

1971-07-29
AU
AU31772/71A
patent/AU463957B2/en
not_active
Expired

1971-07-29
AT
AT664271A
patent/AT311976B/en
active

1971-07-29
AT
AT1100472A
patent/AT311988B/en
active

1971-07-29
DK
DK373271A
patent/DK137990C/en
active

1971-07-29
YU
YU1986/71A
patent/YU34530B/en
unknown

1971-07-29
PL
PL1971178479A
patent/PL84348B1/pl
unknown

1971-07-29
SE
SE7109767A
patent/SE375308B/xx
unknown

1971-07-29
GB
GB3577271A
patent/GB1344720A/en
not_active
Expired

1971-07-29
AT
AT1100072A
patent/AT311984B/en
not_active
IP Right Cessation

1971-07-29
AT
AT1100272A
patent/AT311986B/en
not_active
IP Right Cessation

1971-07-29
PL
PL1971182554A
patent/PL91965B1/pl
unknown

1971-07-29
PL
PL1971178481A
patent/PL84610B1/pl
unknown

1971-07-30
NL
NLAANVRAGE7110538,A
patent/NL173643C/en
not_active
IP Right Cessation

1971-07-30
BE
BE770800A
patent/BE770800A/en
not_active
IP Right Cessation

1971-07-30
FR
FR7128074A
patent/FR2100972B1/fr
not_active
Expired

1971-10-21
ES
ES396214A
patent/ES396214A1/en
not_active
Expired

1971-10-21
ES
ES396215A
patent/ES396215A1/en
not_active
Expired

1971-10-21
ES
ES396216A
patent/ES396216A1/en
not_active
Expired

1971-10-21
ES
ES396213A
patent/ES396213A1/en
not_active
Expired

1971-10-21
ES
ES396212A
patent/ES396212A1/en
not_active
Expired

1974

1974-06-27
SE
SE7408533A
patent/SE403288B/en
unknown

1978

1978-03-13
YU
YU596/78A
patent/YU34888B/en
unknown

1978-03-13
YU
YU60078A
patent/YU34891B/en
unknown

1978-03-13
YU
YU598/78A
patent/YU34889B/en
unknown

1978-03-13
YU
YU597/78A
patent/YU35248B/en
unknown

1978-03-13
YU
YU599/78A
patent/YU34890B/en
unknown

1978-06-12
YU
YU01388/78A
patent/YU138878A/en
unknown

Also Published As

Publication number
Publication date

CH565780A5
(en)

1975-08-29

PL84348B1
(en)

1976-03-31

PL84664B1
(en)

1976-04-30

FR2100972A1
(en)

1972-03-24

DE2037852C3
(en)

1980-06-26

CH565166A5
(en)

1975-08-15

NL173643C
(en)

1984-02-16

NL7110538A
(en)

1972-02-01

JPS5716989B1
(en)

1982-04-08

SU437293A3
(en)

1974-07-25

BG20594A3
(en)

1975-12-05

DK137990C
(en)

1978-11-13

SE375308B
(en)

1975-04-14

SE7408533L
(en)

1974-06-27

YU34530B
(en)

1979-09-10

ES396213A1
(en)

1974-04-16

AT311988B
(en)

1973-12-10

YU59878A
(en)

1979-10-31

YU34888B
(en)

1980-04-30

YU35248B
(en)

1980-10-31

CH565167A5
(en)

1975-08-15

RO60599A
(en)

1976-08-15

YU60078A
(en)

1979-10-31

CH565781A5
(en)

1975-08-29

AT311987B
(en)

1973-12-10

SU437291A3
(en)

1974-07-25

DK137990B
(en)

1978-06-19

ES393738A1
(en)

1974-07-01

PL84347B1
(en)

1976-03-31

BG21029A3
(en)

1976-01-20

YU59778A
(en)

1980-04-30

CS172929B2
(en)

1977-01-28

SU437289A3
(en)

1974-07-25

YU138878A
(en)

1982-10-31

PL84349B1
(en)

1976-03-31

RO60598A
(en)

1976-07-15

YU34891B
(en)

1980-04-30

CH575412A5
(en)

1976-05-14

YU59678A
(en)

1979-10-31

SU440840A3
(en)

1974-08-25

AU463957B2
(en)

1975-08-14

SU416945A3
(en)

1974-02-25

BG19598A3
(en)

1975-06-25

BE770800A
(en)

1972-01-31

AT311986B
(en)

1973-12-10

ES396215A1
(en)

1974-04-16

SE403288B
(en)

1978-08-07

AT311985B
(en)

1973-12-10

ES396214A1
(en)

1974-04-16

CH565165A5
(en)

1975-08-15

AT311976B
(en)

1973-12-10

FR2100972B1
(en)

1974-11-15

ES396212A1
(en)

1974-04-16

GB1344720A
(en)

1974-01-23

YU34890B
(en)

1980-04-30

BG20370A3
(en)

1975-11-05

DE2037852A1
(en)

1972-02-03

RO59997A
(en)

1976-06-15

NL173643B
(en)

1983-09-16

RO61040A
(en)

1976-08-15

RO60596A
(en)

1976-08-15

PL91965B1
(en)

1977-03-31

US3808212A
(en)

1974-04-30

YU34889B
(en)

1980-04-30

SU437292A3
(en)

1974-07-25

DE2037852B2
(en)

1979-10-11

ES396216A1
(en)

1974-04-16

YU198671A
(en)

1979-02-28

AT311984B
(en)

1973-12-10

RO60597A
(en)

1976-08-15

YU59978A
(en)

1979-10-31

PL84610B1
(en)

1976-04-30

BG20369A3
(en)

1975-11-05

SU437290A3
(en)

1974-07-25

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IL36261A0
(en)

1971-04-28

Substituted piperazine derivatives,their preparation and pharmaceutical compositions containing them

IL37846A0
(en)

1971-12-29

Phenylalanine derivatives,their manufacture and pharmaceutical compositions containing them

IL36352A0
(en)

1971-05-26

Pregnatetraene derivatives,their preparation and pharmaceutical compositions containing them

IL38310A0
(en)

1972-02-29

Benzopyranobenzopyran derivatives,their preparation and pharmaceutical compositions containing them

IL36370A0
(en)

1971-05-26

Benzocycloheptathiophene derivatives,their preparation and pharmaceutical compositions containing them

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