AU1869983A – 5-piperazinyl-2,4-pyrimidinediamine derivatives
– Google Patents
AU1869983A – 5-piperazinyl-2,4-pyrimidinediamine derivatives
– Google Patents
5-piperazinyl-2,4-pyrimidinediamine derivatives
Info
Publication number
AU1869983A
AU1869983A
AU18699/83A
AU1869983A
AU1869983A
AU 1869983 A
AU1869983 A
AU 1869983A
AU 18699/83 A
AU18699/83 A
AU 18699/83A
AU 1869983 A
AU1869983 A
AU 1869983A
AU 1869983 A
AU1869983 A
AU 1869983A
Authority
AU
Australia
Prior art keywords
piperazinyl
pyrimidinediamine
derivatives
pyrimidinediamine derivatives
Prior art date
1982-09-09
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU18699/83A
Other versions
AU560971B2
(en
Inventor
Jocelyn H. Hung
Leslie M. Werbel
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Warner Lambert Co LLC
Original Assignee
Warner Lambert Co LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1982-09-09
Filing date
1983-09-05
Publication date
1984-03-15
1983-09-05
Application filed by Warner Lambert Co LLC
filed
Critical
Warner Lambert Co LLC
1984-03-15
Publication of AU1869983A
publication
Critical
patent/AU1869983A/en
1987-04-30
Application granted
granted
Critical
1987-04-30
Publication of AU560971B2
publication
Critical
patent/AU560971B2/en
2003-09-05
Anticipated expiration
legal-status
Critical
Status
Ceased
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
C07D239/32—One oxygen, sulfur or nitrogen atom
C07D239/42—One nitrogen atom
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
C07D239/50—Three nitrogen atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
C07D239/52—Two oxygen atoms
C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
C07D239/52—Two oxygen atoms
C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil
AU18699/83A
1982-09-09
1983-09-05
5-piperazinyl-2,4-pyrimidinediamine derivatives
Ceased
AU560971B2
(en)
Applications Claiming Priority (4)
Application Number
Priority Date
Filing Date
Title
US41640482A
1982-09-09
1982-09-09
US416404
1982-09-09
US520653
1983-08-09
US06/520,653
US4532240A
(en)
1982-09-09
1983-08-09
Diaminopyrimidines
Related Child Applications (1)
Application Number
Title
Priority Date
Filing Date
AU68787/87A
Division
AU568997B2
(en)
1982-09-09
1987-02-13
Substituted 5-(1,4-piperazinyl)-2,4-diaminopyridine
Publications (2)
Publication Number
Publication Date
AU1869983A
true
AU1869983A
(en)
1984-03-15
AU560971B2
AU560971B2
(en)
1987-04-30
Family
ID=27023342
Family Applications (2)
Application Number
Title
Priority Date
Filing Date
AU18699/83A
Ceased
AU560971B2
(en)
1982-09-09
1983-09-05
5-piperazinyl-2,4-pyrimidinediamine derivatives
AU68787/87A
Ceased
AU568997B2
(en)
1982-09-09
1987-02-13
Substituted 5-(1,4-piperazinyl)-2,4-diaminopyridine
Family Applications After (1)
Application Number
Title
Priority Date
Filing Date
AU68787/87A
Ceased
AU568997B2
(en)
1982-09-09
1987-02-13
Substituted 5-(1,4-piperazinyl)-2,4-diaminopyridine
Country Status (9)
Country
Link
US
(1)
US4532240A
(en)
EP
(1)
EP0103464B1
(en)
AU
(2)
AU560971B2
(en)
CA
(1)
CA1251447A
(en)
DE
(1)
DE3378469D1
(en)
DK
(1)
DK158310C
(en)
ES
(2)
ES8502989A1
(en)
GR
(1)
GR79058B
(en)
IE
(1)
IE56148B1
(en)
Families Citing this family (14)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
US5099019A
(en)
*
1985-09-12
1992-03-24
Upjohn Company
Amines useful in producing pharmaceutically active CNS compounds
USRE35053E
(en)
*
1985-09-12
1995-10-10
The Upjohn Company
Amines useful in producing pharmaceutically active CNS compounds
LU86695A1
(en)
*
1986-12-01
1988-07-14
Oreal
NOVEL PIPERAZINYL-1 PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPEUTICS AND COSMETICS
HUT64323A
(en)
*
1992-06-09
1993-12-28
Richter Gedeon Vegyeszet
Process for production new piperazinyl-bis(alkyl-amino)-pyrimidine derivatives
DE4320570C2
(en)
*
1993-02-26
2002-07-11
Max Delbrueck Centrum
Process for the production of C-nucleosides and C-nucleoside analogs, new C-nucleosides and C-nucleoside analogues and their use
ATE166347T1
(en)
*
1993-02-26
1998-06-15
Max Delbrueck Centrum
METHOD FOR PRODUCING C-NUCLEOSIDES AND C-NUCLEOSIDE ANALOGAS, NEW C-NUCLEOSIDES AND C-NUCLEOSIDE ANALOGAS, AND USE THEREOF
GB9801392D0
(en)
1998-01-22
1998-03-18
Smithkline Beecham Plc
Novel compounds
EP1057818A4
(en)
1998-01-30
2003-01-29
Meiji Seika Kaisha
PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS
US20040006042A1
(en)
*
1998-08-13
2004-01-08
Berry David Allen
Diaminopyrimidines and combination therapies effective for treatment of P-glycoprotein positive cancers
WO2000009131A1
(en)
*
1998-08-13
2000-02-24
Warner-Lambert Company
Diaminopyrimidines and combination therapies effective for treatment of p-glycoprotein positive cancers
JP2005515961A
(en)
2001-05-22
2005-06-02
ニューロジェン コーポレイション
Melanin-concentrating hormone receptor ligand: substituted 1-benzyl-4-arylpiperazine analogues
GB0412072D0
(en)
*
2004-05-28
2004-06-30
Syngenta Participations Ag
Chemical compounds
CA3013760A1
(en)
*
2016-02-05
2017-08-10
Vyera Pharmaceuticals, LLC
Compositions and methods for treating infections
US20200270233A1
(en)
*
2017-08-07
2020-08-27
Vyera Pharmaceuticais LLC
Dhfr inhibitors, compositions, and methods related thereto
Family Cites Families (7)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
US416404A
(en)
1889-12-03
Automatic lath-feeder for paper-carriers
BE485737A
(en)
*
1947-11-12
US2748125A
(en)
*
1954-04-26
1956-05-29
American Cyanamid Co
1-substituted-4-sulfamylpiperazine and method of preparing the same
AT340933B
(en)
*
1973-08-20
1978-01-10
Thomae Gmbh Dr K
PROCESS FOR THE PRODUCTION OF NEW PYRIMIDE DERIVATIVES AND THEIR ACID ADDITIONAL SALTS
US4166852A
(en)
*
1974-08-09
1979-09-04
Produits Chimiques Ugine Kuhlmann
Piperazino-pyrimidines and their use as spasmolytic agents
US4287338A
(en)
*
1980-03-10
1981-09-01
The Upjohn Company
Sulfooxy-pyrimidinium, -pyridinium, and -triazinium hydroxide inner salts
US4351832A
(en)
*
1980-04-18
1982-09-28
American Home Products Corporation
2-(Piperazinyl)-4-pyrimidinamines
1983
1983-08-09
US
US06/520,653
patent/US4532240A/en
not_active
Expired – Lifetime
1983-08-16
IE
IE1920/83A
patent/IE56148B1/en
not_active
IP Right Cessation
1983-09-05
AU
AU18699/83A
patent/AU560971B2/en
not_active
Ceased
1983-09-07
GR
GR72395A
patent/GR79058B/el
unknown
1983-09-08
CA
CA000436240A
patent/CA1251447A/en
not_active
Expired
1983-09-08
DK
DK407383A
patent/DK158310C/en
not_active
IP Right Cessation
1983-09-08
EP
EP83305229A
patent/EP0103464B1/en
not_active
Expired
1983-09-08
ES
ES525490A
patent/ES8502989A1/en
not_active
Expired
1983-09-08
DE
DE8383305229T
patent/DE3378469D1/en
not_active
Expired
1984
1984-03-27
ES
ES531004A
patent/ES531004A0/en
active
Granted
1987
1987-02-13
AU
AU68787/87A
patent/AU568997B2/en
not_active
Ceased
Also Published As
Publication number
Publication date
DK407383D0
(en)
1983-09-08
ES525490A0
(en)
1985-02-01
IE56148B1
(en)
1991-05-08
DK407383A
(en)
1984-03-10
DK158310B
(en)
1990-04-30
ES8502989A1
(en)
1985-02-01
AU568997B2
(en)
1988-01-14
EP0103464A2
(en)
1984-03-21
CA1251447A
(en)
1989-03-21
EP0103464A3
(en)
1985-07-03
AU6878787A
(en)
1987-05-14
DE3378469D1
(en)
1988-12-22
US4532240A
(en)
1985-07-30
ES8504775A1
(en)
1985-05-01
AU560971B2
(en)
1987-04-30
GR79058B
(en)
1984-10-02
DK158310C
(en)
1990-10-15
EP0103464B1
(en)
1988-11-17
IE831920L
(en)
1984-03-09
ES531004A0
(en)
1985-05-01
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