AU1982483A – Dichloro derivatives of 16alpha-methyl pregnanes
– Google Patents
AU1982483A – Dichloro derivatives of 16alpha-methyl pregnanes
– Google Patents
Dichloro derivatives of 16alpha-methyl pregnanes
Info
Publication number
AU1982483A
AU1982483A
AU19824/83A
AU1982483A
AU1982483A
AU 1982483 A
AU1982483 A
AU 1982483A
AU 19824/83 A
AU19824/83 A
AU 19824/83A
AU 1982483 A
AU1982483 A
AU 1982483A
AU 1982483 A
AU1982483 A
AU 1982483A
Authority
AU
Australia
Prior art keywords
16alpha
pregnanes
methyl
dichloro derivatives
dichloro
Prior art date
1982-10-05
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU19824/83A
Other versions
AU563739B2
(en
Inventor
Josette Benzoni
Roger Deraedt
Jean Georges Teutsch
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1982-10-05
Filing date
1983-09-30
Publication date
1984-04-12
1983-09-30
Application filed by Roussel Uclaf SA
filed
Critical
Roussel Uclaf SA
1984-04-12
Publication of AU1982483A
publication
Critical
patent/AU1982483A/en
1987-07-23
Application granted
granted
Critical
1987-07-23
Publication of AU563739B2
publication
Critical
patent/AU563739B2/en
2003-09-30
Anticipated expiration
legal-status
Critical
Status
Ceased
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 – C07J43/00
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C29/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
C07C29/36—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal
C07C29/38—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal by reaction with aldehydes or ketones
C07C29/40—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal by reaction with aldehydes or ketones with compounds containing carbon-to-metal bonds
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C31/00—Saturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
C07C31/13—Monohydroxylic alcohols containing saturated rings
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C68/00—Preparation of esters of carbonic or haloformic acids
C07C68/02—Preparation of esters of carbonic or haloformic acids from phosgene or haloformates
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
C07F7/02—Silicon compounds
C07F7/08—Compounds having one or more C—Si linkages
C07F7/0803—Compounds with Si-C or Si-Si linkages
C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07J—STEROIDS
C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
C07J5/0007—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa
C07J5/0023—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa substituted in position 16
C07J5/003—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group including 16-alkylidene substitutes
C07J5/0038—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group including 16-alkylidene substitutes by an alkyl group
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C2601/00—Systems containing only non-condensed rings
C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
AU19824/83A
1982-10-05
1983-09-30
Dichloro derivatives of 16alpha-methyl pregnanes
Ceased
AU563739B2
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
FR8216668
1982-10-05
FR8216668A
FR2533928A1
(en)
1982-10-05
1982-10-05
NOVEL DICHLORIC DERIVATIVES OF THE 16A-METHYL PREGNANE SERIES, PROCESS FOR PREPARING THEM AND THEIR APPLICATION AS MEDICAMENTS
Publications (2)
Publication Number
Publication Date
AU1982483A
true
AU1982483A
(en)
1984-04-12
AU563739B2
AU563739B2
(en)
1987-07-23
Family
ID=9277977
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU19824/83A
Ceased
AU563739B2
(en)
1982-10-05
1983-09-30
Dichloro derivatives of 16alpha-methyl pregnanes
Country Status (22)
Country
Link
US
(1)
US4515787A
(en)
JP
(1)
JPS59116300A
(en)
AT
(1)
AT385996B
(en)
AU
(1)
AU563739B2
(en)
BE
(1)
BE897906A
(en)
CA
(1)
CA1203234A
(en)
CH
(1)
CH659251A5
(en)
DE
(1)
DE3336292A1
(en)
DK
(1)
DK164062C
(en)
ES
(1)
ES8405812A1
(en)
FI
(1)
FI77668C
(en)
FR
(1)
FR2533928A1
(en)
GB
(1)
GB2127827B
(en)
HU
(1)
HU190506B
(en)
IE
(1)
IE56022B1
(en)
IT
(1)
IT1197713B
(en)
MA
(1)
MA19909A1
(en)
NL
(1)
NL8303409A
(en)
NO
(1)
NO157864C
(en)
OA
(1)
OA07558A
(en)
SE
(1)
SE447388B
(en)
ZA
(1)
ZA836538B
(en)
Families Citing this family (8)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
FR2561919B1
(en)
*
1984-04-03
1986-12-19
Roussel Uclaf
PHARMACEUTICAL COMPOSITION CONSTITUTED ON THE ONE HAND, AS ACTIVE INGREDIENT, BY 9A, 11B-DICHLORO 16A-METHYL 21-OXYCARBONYLDICYCLOHEXYL METHYLOXY PREGNA-1,4-DIENE 3,20-DIONE AND ON THE OTHER HAND, BY A PHARM EXCIPIENT INERTE CAPABLE OF ALLOWING THE ACTION OF THE PRODUCT IN THE RECTUM OR THE COLON
GB8512738D0
(en)
*
1984-09-04
1985-06-26
Gen Electric
Silylation method
AU4093799A
(en)
1998-05-22
1999-12-13
Board Of Trustees Of The Leland Stanford Junior University
Bifunctional molecules and therapies based thereon
US7247607B2
(en)
*
2001-11-08
2007-07-24
Green & Clean, Inc.
Active soluble cleaning composite of natural state using soybean fatty acids and the making method thereof
EP1889198B1
(en)
2005-04-28
2014-11-26
Proteus Digital Health, Inc.
Pharma-informatics system
EP1945240B1
(en)
2005-09-16
2016-12-28
Raptor Pharmaceutical Inc
Compositions comprising receptor-associated protein (rap) variants specific for cr-containing proteins and uses thereof
AU2010216512B2
(en)
2009-02-20
2016-06-30
2-Bbb Medicines B.V.
Glutathione-based drug delivery system
BRPI1011188B1
(en)
2009-05-06
2019-10-15
Laboratory Skin Care, Inc.
DERMAL RELEASE COMPOSITIONS UNDERSTANDING CALCIUM ACTIVE-PHOSPHATE PARTICLE COMPLEXES AND METHODS FOR USING THE SAME
Family Cites Families (3)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
FR2342738A1
(en)
*
1976-03-02
1977-09-30
Roussel Uclaf
NEW HALOGEN DERIVATIVES OF THE 16A-METHYL PREGNANE SERIES
FR2381065A2
(en)
*
1977-02-22
1978-09-15
Roussel Uclaf
9-Alpha-11-beta-di:chloro-16-alpha-methyl pregnadiene di:one cpds. – having topical antiinflammatory activity with little general activity
FR2462443A1
(en)
*
1979-07-26
1981-02-13
Roussel Uclaf
NEW HALOGENIC DERIVATIVE OF THE 16A-METHYL PREGNANE SERIES, PREPARATION METHOD AND APPLICATION AS MEDICINE
1982
1982-10-05
FR
FR8216668A
patent/FR2533928A1/en
active
Granted
1983
1983-07-20
SE
SE8304062A
patent/SE447388B/en
not_active
IP Right Cessation
1983-07-27
NO
NO832738A
patent/NO157864C/en
unknown
1983-09-03
ZA
ZA836538A
patent/ZA836538B/en
unknown
1983-09-15
US
US06/532,739
patent/US4515787A/en
not_active
Expired – Fee Related
1983-09-19
IT
IT48990/83A
patent/IT1197713B/en
active
1983-09-28
MA
MA20132A
patent/MA19909A1/en
unknown
1983-09-30
AU
AU19824/83A
patent/AU563739B2/en
not_active
Ceased
1983-10-04
GB
GB08326527A
patent/GB2127827B/en
not_active
Expired
1983-10-04
ES
ES526212A
patent/ES8405812A1/en
not_active
Expired
1983-10-04
FI
FI833602A
patent/FI77668C/en
not_active
IP Right Cessation
1983-10-04
BE
BE0/211641A
patent/BE897906A/en
not_active
IP Right Cessation
1983-10-04
HU
HU833444A
patent/HU190506B/en
not_active
IP Right Cessation
1983-10-04
CA
CA000438264A
patent/CA1203234A/en
not_active
Expired
1983-10-04
CH
CH5395/83A
patent/CH659251A5/en
not_active
IP Right Cessation
1983-10-04
IE
IE2337/83A
patent/IE56022B1/en
not_active
IP Right Cessation
1983-10-04
DK
DK456483A
patent/DK164062C/en
not_active
IP Right Cessation
1983-10-05
OA
OA58129A
patent/OA07558A/en
unknown
1983-10-05
NL
NL8303409A
patent/NL8303409A/en
not_active
Application Discontinuation
1983-10-05
AT
AT0352783A
patent/AT385996B/en
not_active
IP Right Cessation
1983-10-05
JP
JP58185211A
patent/JPS59116300A/en
active
Granted
1983-10-05
DE
DE19833336292
patent/DE3336292A1/en
active
Granted
Also Published As
Publication number
Publication date
JPH0412279B2
(en)
1992-03-04
DE3336292A1
(en)
1984-04-05
DK164062B
(en)
1992-05-04
DK456483D0
(en)
1983-10-04
FI833602A0
(en)
1983-10-04
AU563739B2
(en)
1987-07-23
NO832738L
(en)
1984-04-06
FR2533928A1
(en)
1984-04-06
SE8304062L
(en)
1984-04-06
MA19909A1
(en)
1984-04-01
FI833602A
(en)
1984-04-06
NO157864C
(en)
1988-06-01
JPS59116300A
(en)
1984-07-05
ES526212A0
(en)
1984-06-16
DE3336292C2
(en)
1992-09-10
GB2127827A
(en)
1984-04-18
BE897906A
(en)
1984-04-04
ES8405812A1
(en)
1984-06-16
ATA352783A
(en)
1987-11-15
OA07558A
(en)
1985-03-31
ZA836538B
(en)
1984-10-31
FI77668C
(en)
1989-04-10
SE447388B
(en)
1986-11-10
GB2127827B
(en)
1986-01-29
IE832337L
(en)
1984-04-05
DK164062C
(en)
1992-09-28
DK456483A
(en)
1984-04-06
AT385996B
(en)
1988-06-10
SE8304062D0
(en)
1983-07-20
US4515787A
(en)
1985-05-07
CA1203234A
(en)
1986-04-15
FI77668B
(en)
1988-12-30
CH659251A5
(en)
1987-01-15
HU190506B
(en)
1986-09-29
NL8303409A
(en)
1984-05-01
IT1197713B
(en)
1988-12-06
IE56022B1
(en)
1991-03-27
NO157864B
(en)
1988-02-22
FR2533928B1
(en)
1985-05-03
GB8326527D0
(en)
1983-11-02
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