AU2747384A – Substituted piperazin-1-yl-acetic acid amides
– Google Patents
AU2747384A – Substituted piperazin-1-yl-acetic acid amides
– Google Patents
Substituted piperazin-1-yl-acetic acid amides
Info
Publication number
AU2747384A
AU2747384A
AU27473/84A
AU2747384A
AU2747384A
AU 2747384 A
AU2747384 A
AU 2747384A
AU 27473/84 A
AU27473/84 A
AU 27473/84A
AU 2747384 A
AU2747384 A
AU 2747384A
AU 2747384 A
AU2747384 A
AU 2747384A
Authority
AU
Australia
Prior art keywords
acetic acid
acid amides
substituted piperazin
piperazin
substituted
Prior art date
1983-04-28
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU27473/84A
Inventor
Rudi Beyerle
Piero Martorana
Rolf-Eberhard Nitz
Ursula Schindler
Karl Schonafinger
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis Deutschland GmbH
Original Assignee
Cassella AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1983-04-28
Filing date
1984-04-27
Publication date
1984-11-01
1984-04-27
Application filed by Cassella AG
filed
Critical
Cassella AG
1984-11-01
Publication of AU2747384A
publication
Critical
patent/AU2747384A/en
Status
Abandoned
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
C07D213/81—Amides; Imides
C07D213/82—Amides; Imides in position 3
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P25/00—Drugs for disorders of the nervous system
A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer’s disease or other forms of dementia
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
C07D295/182—Radicals derived from carboxylic acids
C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
C07D295/205—Radicals derived from carbonic acid
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
AU27473/84A
1983-04-28
1984-04-27
Substituted piperazin-1-yl-acetic acid amides
Abandoned
AU2747384A
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
DE19833315424
DE3315424A1
(en)
1983-04-28
1983-04-28
SUBSTITUTED PIPERAZIN-1-YL-ACETIC ACID AMIDES, METHOD FOR THEIR PRODUCTION AND THEIR USE
DE3315424
1983-04-28
Publications (1)
Publication Number
Publication Date
AU2747384A
true
AU2747384A
(en)
1984-11-01
Family
ID=6197594
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU27473/84A
Abandoned
AU2747384A
(en)
1983-04-28
1984-04-27
Substituted piperazin-1-yl-acetic acid amides
Country Status (19)
Country
Link
US
(1)
US4610984A
(en)
EP
(1)
EP0123977A1
(en)
JP
(1)
JPS59205363A
(en)
KR
(1)
KR840008347A
(en)
AU
(1)
AU2747384A
(en)
CA
(1)
CA1202304A
(en)
CS
(2)
CS244849B2
(en)
DD
(1)
DD223711A5
(en)
DE
(1)
DE3315424A1
(en)
DK
(1)
DK147784A
(en)
ES
(1)
ES532011A0
(en)
FI
(1)
FI841461A
(en)
GR
(1)
GR81494B
(en)
HU
(1)
HUT34178A
(en)
IL
(1)
IL71657A0
(en)
NO
(1)
NO841464L
(en)
PL
(2)
PL253669A1
(en)
PT
(1)
PT78488B
(en)
ZA
(1)
ZA843138B
(en)
Families Citing this family (5)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
GB8512163D0
(en)
*
1985-05-14
1985-06-19
Fujisawa Pharmaceutical Co
Oxothiazolidine compound
US5110929A
(en)
*
1986-08-07
1992-05-05
Medice Cham.-Pharm. Fabrik Putter Gmbh & Co. Kg
Process for the preparation of N-alkylated quaternary nitrogen containing aromatic heterocycles
IT1249728B
(en)
*
1991-11-06
1995-03-09
Sigma Tau Ind Farmaceuti
PROLINAMIDE DERIVATIVES AS ACTIVATORS OF MEMORY AND OF LEARNING PROCESSES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
DE19904710A1
(en)
*
1999-02-05
2000-08-10
Aventis Pharma Gmbh
Substituted 4-amino-2-aryl-tetrahydroquinazolines, their preparation, their use and pharmaceutical compositions containing them
US7851474B2
(en)
*
2005-08-02
2010-12-14
Neurogen Corporation
Dipiperazinyl ketones and related analogues
Family Cites Families (4)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
FR2081564A1
(en)
*
1970-03-05
1971-12-10
Delalande Sa
N-amino carbonyl-piperazines analgesics – antiinflammatories ,hypotensives and spasmolytics
BE774447A
(en)
*
1970-11-11
1972-02-14
Biasedra Lab
NEW DERIVATIVES OF SALICYLAMIDE AND THEIR APPLICATION IN THERAPEUTICS
US4247549A
(en)
*
1978-12-27
1981-01-27
Ici Americas Inc.
Piperazine-1-carboxylic acid esters possessing antidepressant or analgesic activity
AU535498B2
(en)
*
1981-05-08
1984-03-22
Otsuka Pharmaceutical Co., Ltd.
Aniline derivatives, process for their preparation, and cardiotonics
1983
1983-04-28
DE
DE19833315424
patent/DE3315424A1/en
not_active
Withdrawn
1984
1984-02-29
DK
DK147784A
patent/DK147784A/en
not_active
IP Right Cessation
1984-04-11
EP
EP84104042A
patent/EP0123977A1/en
not_active
Ceased
1984-04-12
NO
NO841464A
patent/NO841464L/en
unknown
1984-04-12
FI
FI841461A
patent/FI841461A/en
not_active
Application Discontinuation
1984-04-18
US
US06/601,637
patent/US4610984A/en
not_active
Expired – Fee Related
1984-04-23
JP
JP59080360A
patent/JPS59205363A/en
active
Pending
1984-04-25
CS
CS851217A
patent/CS244849B2/en
unknown
1984-04-25
CS
CS843071A
patent/CS244811B2/en
unknown
1984-04-25
DD
DD84262312A
patent/DD223711A5/en
unknown
1984-04-26
PT
PT78488A
patent/PT78488B/en
unknown
1984-04-26
PL
PL25366984A
patent/PL253669A1/en
unknown
1984-04-26
GR
GR74523A
patent/GR81494B/el
unknown
1984-04-26
IL
IL71657A
patent/IL71657A0/en
unknown
1984-04-26
PL
PL24741484A
patent/PL247414A1/en
unknown
1984-04-26
HU
HU841608A
patent/HUT34178A/en
unknown
1984-04-27
ES
ES532011A
patent/ES532011A0/en
active
Granted
1984-04-27
CA
CA000452963A
patent/CA1202304A/en
not_active
Expired
1984-04-27
ZA
ZA843138A
patent/ZA843138B/en
unknown
1984-04-27
AU
AU27473/84A
patent/AU2747384A/en
not_active
Abandoned
1984-04-28
KR
KR1019840002290A
patent/KR840008347A/en
not_active
Application Discontinuation
Also Published As
Publication number
Publication date
CA1202304A
(en)
1986-03-25
US4610984A
(en)
1986-09-09
DD223711A5
(en)
1985-06-19
CS307184A2
(en)
1985-09-17
ES8502103A1
(en)
1984-12-16
DK147784D0
(en)
1984-02-29
FI841461A
(en)
1984-10-29
FI841461A0
(en)
1984-04-12
NO841464L
(en)
1984-10-29
HUT34178A
(en)
1985-02-28
JPS59205363A
(en)
1984-11-20
PT78488B
(en)
1986-05-22
CS121785A2
(en)
1985-09-17
DK147784A
(en)
1984-10-29
PL247414A1
(en)
1985-10-08
IL71657A0
(en)
1984-07-31
GR81494B
(en)
1984-12-11
CS244811B2
(en)
1986-08-14
CS244849B2
(en)
1986-08-14
DE3315424A1
(en)
1984-12-20
ZA843138B
(en)
1984-11-28
KR840008347A
(en)
1984-12-14
PL253669A1
(en)
1986-02-11
EP0123977A1
(en)
1984-11-07
PT78488A
(en)
1984-05-01
ES532011A0
(en)
1984-12-16
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