AU3717489A – New compounds
– Google Patents
AU3717489A – New compounds
– Google Patents
New compounds
Info
Publication number
AU3717489A
AU3717489A
AU37174/89A
AU3717489A
AU3717489A
AU 3717489 A
AU3717489 A
AU 3717489A
AU 37174/89 A
AU37174/89 A
AU 37174/89A
AU 3717489 A
AU3717489 A
AU 3717489A
AU 3717489 A
AU3717489 A
AU 3717489A
Authority
AU
Australia
Prior art keywords
new compounds
compounds
new
Prior art date
1988-07-07
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU37174/89A
Other versions
AU622188B2
(en
Inventor
Hans-Georg Capraro
Giorgio Caravatti
Jorg Frei
Jaroslav Stanek
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1988-07-07
Filing date
1989-06-28
Publication date
1990-01-11
1989-06-28
Application filed by Ciba Geigy AG
filed
Critical
Ciba Geigy AG
1990-01-11
Publication of AU3717489A
publication
Critical
patent/AU3717489A/en
1992-04-02
Application granted
granted
Critical
1992-04-02
Publication of AU622188B2
publication
Critical
patent/AU622188B2/en
2009-06-28
Anticipated expiration
legal-status
Critical
Status
Ceased
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P35/00—Antineoplastic agents
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
C07D213/81—Amides; Imides
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
C07D213/83—Thioacids; Thioesters; Thioamides; Thioimides
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
C07D213/84—Nitriles
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
AU37174/89A
1988-07-07
1989-06-28
New compounds
Ceased
AU622188B2
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
CH258888
1988-07-07
CH2588/88
1988-07-07
Publications (2)
Publication Number
Publication Date
AU3717489A
true
AU3717489A
(en)
1990-01-11
AU622188B2
AU622188B2
(en)
1992-04-02
Family
ID=4237163
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU37174/89A
Ceased
AU622188B2
(en)
1988-07-07
1989-06-28
New compounds
Country Status (15)
Country
Link
US
(2)
US4968804A
(en)
EP
(1)
EP0350448A1
(en)
JP
(1)
JPH0276843A
(en)
KR
(1)
KR900001677A
(en)
AU
(1)
AU622188B2
(en)
DD
(1)
DD284004A5
(en)
DK
(1)
DK336089A
(en)
FI
(1)
FI893266A
(en)
HU
(1)
HU208811B
(en)
IL
(1)
IL90793A0
(en)
MX
(1)
MX16687A
(en)
NO
(1)
NO892810L
(en)
NZ
(1)
NZ229841A
(en)
PT
(1)
PT91068B
(en)
ZA
(1)
ZA895141B
(en)
Families Citing this family (27)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
EP0495749A1
(en)
*
1991-01-14
1992-07-22
Ciba-Geigy Ag
Bipyridines
US5608059A
(en)
*
1993-04-21
1997-03-04
Eastman Kodak Company
Ion-sensitive compounds
EP1231910B1
(en)
*
1999-11-16
2009-05-20
Oncozyme Pharma Inc.
Pentamidine for treating cancer
DE10035908A1
(en)
*
2000-07-21
2002-03-07
Asta Medica Ag
New heteroaryl derivatives and their use as medicines
GB0124939D0
(en)
*
2001-10-17
2001-12-05
Glaxo Group Ltd
Chemical compounds
GB0124941D0
(en)
*
2001-10-17
2001-12-05
Glaxo Group Ltd
Chemical compounds
GB0124938D0
(en)
*
2001-10-17
2001-12-05
Glaxo Group Ltd
Chemical compounds
GB0124934D0
(en)
*
2001-10-17
2001-12-05
Glaxo Group Ltd
Chemical compounds
GB0124931D0
(en)
*
2001-10-17
2001-12-05
Glaxo Group Ltd
Chemical compounds
GB0124936D0
(en)
*
2001-10-17
2001-12-05
Glaxo Group Ltd
Chemical compounds
GB0124933D0
(en)
*
2001-10-17
2001-12-05
Glaxo Group Ltd
Chemical compounds
MXPA04007838A
(en)
2002-02-12
2004-10-15
Smithkline Beecham Corp
Nicotinamide derivates useful as p38 inhibitors.
GB0217757D0
(en)
2002-07-31
2002-09-11
Glaxo Group Ltd
Novel compounds
GB0308185D0
(en)
*
2003-04-09
2003-05-14
Smithkline Beecham Corp
Novel compounds
GB0402143D0
(en)
*
2004-01-30
2004-03-03
Smithkline Beecham Corp
Novel compounds
US20080051416A1
(en)
*
2004-10-05
2008-02-28
Smithkline Beecham Corporation
Novel Compounds
GB0512429D0
(en)
*
2005-06-17
2005-07-27
Smithkline Beecham Corp
Novel compound
US20100216796A1
(en)
*
2007-10-04
2010-08-26
Solomon Kattar
N-hydroxy-naphthalene dicarboxamide and n-hydroxy-biphenyl-dicarboxamide compounds as histone deacetylase inhibitors
MX2011001349A
(en)
2008-08-04
2011-08-17
Chidi Inc
Certain kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof.
NZ601547A
(en)
*
2010-01-25
2014-04-30
Chdi Foundation Inc
Certain kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof
CA2844128C
(en)
2011-08-30
2020-09-01
Chdi Foundation, Inc.
Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof
CA2844521A1
(en)
2011-08-30
2013-03-07
Chdi Foundation, Inc.
Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof
KR20170026633A
(en)
2014-07-17
2017-03-08
씨에이치디아이 파운데이션, 인코포레이티드
Methods and compositions for treating hiv-related disorders
CN106407739B
(en)
*
2016-04-22
2019-02-22
三峡大学
Small molecule covalency inhibitor computational screening method and its screening S adenosylmethionine decarboxylase covalency inhibitor application
CN106389403B
(en)
*
2016-04-22
2019-02-19
三峡大学
Application and screening technique of the small molecule covalency inhibitor on the drug that preparation inhibits S adenosylmethionine decarboxylase
CN106389399B
(en)
*
2016-04-22
2019-02-19
三峡大学
The application and its screening technique of a kind of small molecule covalency inhibitor on the drug that preparation inhibits S adenosylmethionine decarboxylase
CN106389415B
(en)
*
2016-04-22
2019-02-19
三峡大学
Application and its screening technique of the small molecule covalency inhibitor on the drug that preparation inhibits S adenosylmethionine decarboxylase
Family Cites Families (9)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
US4086244A
(en)
*
1976-12-10
1978-04-25
E. R. Squibb & Sons, Inc.
Amidines
US4495934A
(en)
*
1978-07-25
1985-01-29
Shaw Jr Seth T
IUD Arrangement
US4233968A
(en)
*
1978-07-26
1980-11-18
Shaw Jr Seth T
IUD Arrangement
US4284074A
(en)
*
1978-07-26
1981-08-18
Shaw Jr Seth T
IUD Arrangement
AU538963B2
(en)
*
1979-07-09
1984-09-06
Seth Thomas Shaw Jr.
Drug for use with an iud
US4359046A
(en)
*
1979-07-09
1982-11-16
Shaw Jr Seth T
IUD Arrangement
US4381001A
(en)
*
1979-07-09
1983-04-26
Shaw Jr Seth T
IUD Arrangement
DOP1981004033A
(en)
*
1980-12-23
1990-12-29
Ciba Geigy Ag
PROCEDURE TO PROTECT CROP PLANTS FROM PHYTOTOXIC ACTION OF HERBICIDES.
US4598073A
(en)
*
1982-12-06
1986-07-01
Research Corporation
Certain polycyclo-palladium-bipyridine complexes having anti-tumor activity
1989
1989-06-05
MX
MX1668789A
patent/MX16687A/en
unknown
1989-06-28
EP
EP89810491A
patent/EP0350448A1/en
not_active
Ceased
1989-06-28
AU
AU37174/89A
patent/AU622188B2/en
not_active
Ceased
1989-06-29
IL
IL90793A
patent/IL90793A0/en
not_active
IP Right Cessation
1989-07-05
PT
PT91068A
patent/PT91068B/en
active
IP Right Grant
1989-07-05
DD
DD89330468A
patent/DD284004A5/en
not_active
IP Right Cessation
1989-07-05
FI
FI893266A
patent/FI893266A/en
not_active
IP Right Cessation
1989-07-05
US
US07/375,760
patent/US4968804A/en
not_active
Expired – Fee Related
1989-07-05
NZ
NZ229841A
patent/NZ229841A/en
unknown
1989-07-06
KR
KR1019890009573A
patent/KR900001677A/en
not_active
Application Discontinuation
1989-07-06
ZA
ZA895141A
patent/ZA895141B/en
unknown
1989-07-06
DK
DK336089A
patent/DK336089A/en
not_active
Application Discontinuation
1989-07-06
JP
JP1173144A
patent/JPH0276843A/en
active
Pending
1989-07-06
HU
HU893434A
patent/HU208811B/en
not_active
IP Right Cessation
1989-07-06
NO
NO89892810A
patent/NO892810L/en
unknown
1990
1990-08-16
US
US07/568,371
patent/US5064832A/en
not_active
Expired – Fee Related
Also Published As
Publication number
Publication date
NZ229841A
(en)
1990-11-27
AU622188B2
(en)
1992-04-02
ZA895141B
(en)
1990-02-28
JPH0276843A
(en)
1990-03-16
DD284004A5
(en)
1990-10-31
HUT50778A
(en)
1990-03-28
NO892810D0
(en)
1989-07-06
EP0350448A1
(en)
1990-01-10
US5064832A
(en)
1991-11-12
FI893266A0
(en)
1989-07-05
HU208811B
(en)
1994-01-28
KR900001677A
(en)
1990-02-27
US4968804A
(en)
1990-11-06
IL90793A0
(en)
1990-01-18
FI893266A
(en)
1990-01-08
DK336089A
(en)
1990-01-08
PT91068B
(en)
1994-12-30
NO892810L
(en)
1990-01-08
PT91068A
(en)
1990-02-08
MX16687A
(en)
1994-01-31
DK336089D0
(en)
1989-07-06
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