AU3924978A – Novel 5-hydroxymethyl oxazolidinones, the method of preparing them and their application in therapeutics
– Google Patents
AU3924978A – Novel 5-hydroxymethyl oxazolidinones, the method of preparing them and their application in therapeutics
– Google Patents
Novel 5-hydroxymethyl oxazolidinones, the method of preparing them and their application in therapeutics
Info
Publication number
AU3924978A
AU3924978A
AU39249/78A
AU3924978A
AU3924978A
AU 3924978 A
AU3924978 A
AU 3924978A
AU 39249/78 A
AU39249/78 A
AU 39249/78A
AU 3924978 A
AU3924978 A
AU 3924978A
AU 3924978 A
AU3924978 A
AU 3924978A
Authority
AU
Australia
Prior art keywords
therapeutics
preparing
novel
application
oxazolidinones
Prior art date
1977-08-26
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU39249/78A
Other versions
AU526714B2
(en
Inventor
Et Al Philippe Hostert
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1977-08-26
Filing date
1978-08-24
Publication date
1980-02-28
1977-08-26
Priority claimed from FR7726105A
external-priority
patent/FR2381037A2/en
1978-05-23
Priority claimed from FR7815342A
external-priority
patent/FR2426684A2/en
1978-08-24
Application filed by Delalande SA
filed
Critical
Delalande SA
1980-02-28
Publication of AU3924978A
publication
Critical
patent/AU3924978A/en
1983-01-27
Application granted
granted
Critical
1983-01-27
Publication of AU526714B2
publication
Critical
patent/AU526714B2/en
Status
Expired
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D263/18—Oxygen atoms
C07D263/20—Oxygen atoms attached in position 2
C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P25/00—Drugs for disorders of the nervous system
A61P25/24—Antidepressants
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P25/00—Drugs for disorders of the nervous system
A61P25/26—Psychostimulants, e.g. nicotine, cocaine
AU39249/78A
1977-08-26
1978-08-24
Novel 5-hydroxymethyl oxazolidinones, the method of preparing them and their application in therapeutics
Expired
AU526714B2
(en)
Applications Claiming Priority (4)
Application Number
Priority Date
Filing Date
Title
FR7726105A
FR2381037A2
(en)
1977-02-22
1977-08-26
NEW HYDROXYMETHYL-5 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION
FRFR7726105
1977-08-26
FR7815342A
FR2426684A2
(en)
1978-05-23
1978-05-23
3-Phenyl-5-hydroxymethyl-oxazolidin-2-one derivs. – useful as antidepressants
FRFR7815342
1978-05-23
Publications (2)
Publication Number
Publication Date
AU3924978A
true
AU3924978A
(en)
1980-02-28
AU526714B2
AU526714B2
(en)
1983-01-27
Family
ID=26220188
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU39249/78A
Expired
AU526714B2
(en)
1977-08-26
1978-08-24
Novel 5-hydroxymethyl oxazolidinones, the method of preparing them and their application in therapeutics
Country Status (13)
Country
Link
US
(2)
US4250318A
(en)
JP
(1)
JPS5441871A
(en)
AU
(1)
AU526714B2
(en)
CA
(1)
CA1113093A
(en)
CH
(1)
CH634836A5
(en)
DE
(1)
DE2836305A1
(en)
ES
(1)
ES472825A1
(en)
GB
(1)
GB2003151B
(en)
GR
(1)
GR64146B
(en)
IT
(1)
IT1118099B
(en)
LU
(1)
LU80081A1
(en)
NL
(1)
NL7808817A
(en)
SE
(1)
SE444813B
(en)
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* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
JPS53108278A
(en)
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1977-11-14
1978-09-20
Nec Corp
Manufacture of semiconductor device
US4348393A
(en)
1978-06-09
1982-09-07
Delalande S.A.
N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
FR2460940A2
(en)
*
1979-07-10
1981-01-30
Delalande Sa
Antidepressant oxazolidinone(s) – with 5-hydroxymethyl -3-phenyl substituents
CA1171865A
(en)
*
1980-06-04
1984-07-31
Alain Lacour
N-aryl azolone derivatives, the process for preparing the same and their application in therapeutics
US4340606A
(en)
1980-10-23
1982-07-20
E. I. Du Pont De Nemours And Company
3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents
JPS57128058A
(en)
*
1980-12-15
1982-08-09
Seiko Epson Corp
Manufacture of semiconductor device
FR2500450A1
(en)
*
1981-02-25
1982-08-27
Delalande Sa
NOVEL AMINOMETHYL-5-OXAZOLIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC USE THEREOF
ES517852A0
(en)
*
1981-12-04
1984-01-16
Du Pont
A PROCEDURE FOR THE PREPARATION OF BENZENE-SULPHONAMID DERIVATIVES.
US4405794A
(en)
*
1981-12-18
1983-09-20
The Dow Chemical Company
Preparation of 2-oxazolidinone and ethyleneurea
FR2528046B1
(en)
*
1982-06-08
1985-06-21
Delalande Sa
OPTICALLY ACTIVE OXAZOLIDINONE-2 N-ARYLATED DERIVATIVES, SPECIFIC AND REVERSIBLE INHIBITORS OF TYPE B MONOAMINE OXYDASE AND PROCESS FOR THEIR PREPARATION
US4461773A
(en)
*
1982-09-15
1984-07-24
E. I. Dupont De Nemours And Company
P-Oxooxazolidinylbenzene compounds as antibacterial agents
US4500717A
(en)
*
1983-03-28
1985-02-19
The Dow Chemical Company
Process for preparation of 2-oxazolidinones
US4705799A
(en)
*
1983-06-07
1987-11-10
E. I. Du Pont De Nemours And Company
Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents
US4732956A
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*
1984-06-18
1988-03-22
Loctite (Ireland) Ltd.
Styryloxy resins and compositions thereof
CA1260948A
(en)
1984-12-05
1989-09-26
E. I. Du Pont De Nemours And Company
Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents
US4985429A
(en)
*
1987-10-09
1991-01-15
E. I. Du Pont De Nemours And Company
Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5036093A
(en)
*
1987-10-09
1991-07-30
Du Pont Merck Pharmaceutical
Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US5036092A
(en)
*
1987-10-09
1991-07-30
Du Pont Merck Pharmaceutical
Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US4801600A
(en)
*
1987-10-09
1989-01-31
E. I. Du Pont De Nemours And Company
Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5032605A
(en)
*
1987-10-09
1991-07-16
Du Pont Merck Pharmaceutical Company
Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US4965268A
(en)
*
1987-10-09
1990-10-23
E. I. Du Pont De Nemours And Company
Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5039690A
(en)
*
1987-10-09
1991-08-13
Du Pont Merck Pharmaceutical Company
Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US4921869A
(en)
*
1987-10-09
1990-05-01
E. I. Du Pont De Nemours And Company
Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4942183A
(en)
*
1987-10-16
1990-07-17
E. I. Du Pont De Nemours And Company
Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
US4977173A
(en)
*
1987-10-21
1990-12-11
E. I. Du Pont De Nemours And Company
Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents
US5254577A
(en)
*
1988-07-29
1993-10-19
The Du Pont Merck Pharmaceutical Company
Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
US5182403A
(en)
*
1988-09-15
1993-01-26
The Upjohn Company
Substituted 3(5’indazolyl) oxazolidin-2-ones
US5225565A
(en)
*
1988-09-15
1993-07-06
The Upjohn Company
Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones
US5196543A
(en)
*
1989-10-17
1993-03-23
Delalande S.A.
3-aryloxazolidinone derivatives, process for their preparation and their use in therapy
US5235063A
(en)
*
1989-10-17
1993-08-10
Delalande S.A.
Process of preparing by condensation certain
FR2653017B1
(en)
*
1989-10-17
1995-05-05
Delalande Sa
DERIVATIVES OF ARYL-3 OXAZOLIDINONE-2, THEIR PREPARATION PROCESS AND THEIR APPLICATION IN THERAPEUTICS.
US5231188A
(en)
*
1989-11-17
1993-07-27
The Upjohn Company
Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents
JP2841976B2
(en)
*
1990-11-28
1998-12-24
日本電気株式会社
Semiconductor device and manufacturing method thereof
JP3176626B2
(en)
*
1991-11-01
2001-06-18
ファルマシア・アンド・アップジョン・カンパニー
Substituted aryl- and heteroarylphenyloxazolidinones useful as antimicrobial agents
PL175782B1
(en)
*
1992-12-08
1999-02-26
Upjohn Co
Thropone substituted phenyloxazodinonic bactericides
TW286317B
(en)
*
1993-12-13
1996-09-21
Hoffmann La Roche
MX9703040A
(en)
*
1995-09-12
1997-07-31
Upjohn Co
Phenyloxazolidinone antimicrobials.
FR2741071B1
(en)
*
1995-11-09
1997-12-12
Synthelabo
DERIVATIVES OF 3- (BENZOFURAN-5-YL) OXAZOLIDIN-2-ONE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
US5795985A
(en)
*
1996-03-05
1998-08-18
Ciba Specialty Chemicals Corporation
Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof
EP0892792B1
(en)
*
1996-04-11
2001-11-21
PHARMACIA & UPJOHN COMPANY
Process to prepare oxazolidinones
US6037354A
(en)
1997-06-18
2000-03-14
Merck & Co., Inc.
Alpha 1a adrenergic receptor antagonists
BR9813187A
(en)
1997-11-07
2000-08-22
Upjohn Co
Process for producing oxazolidinones
DE19962924A1
(en)
1999-12-24
2001-07-05
Bayer Ag
Substituted oxazolidinones and their use
DE60118241T2
(en)
*
2000-10-17
2006-12-28
Pharmacia & Upjohn Co. Llc, Kalamazoo
METHOD FOR PRODUCING OXAZOLIDINONE COMPOUNDS
DE10129725A1
(en)
*
2001-06-20
2003-01-02
Bayer Ag
Combination therapy of substituted oxazolidinones
TW200302095A
(en)
*
2002-01-25
2003-08-01
Upjohn Co
Oxazolidinone cotherapy
DE10300111A1
(en)
*
2003-01-07
2004-07-15
Bayer Healthcare Ag
Process for the preparation of 5-chloro-N – ({(5S) -2-oxo-3- [4- (3-oxo-4-morpholinyl) phenyl] -1,3-oxazolidin-5-yl} methyl ) -2-thiophenecarboxamide
DE10355461A1
(en)
2003-11-27
2005-06-23
Bayer Healthcare Ag
Solid, high bioavailabilty oral formulations of N-substituted 5-chloro-2-thiophene-carboxamide derivative in hydrophilized form, useful for combating thrombo-embolic diseases
KR100854211B1
(en)
*
2003-12-18
2008-08-26
동아제약주식회사
Novel oxazolidinone derivatives, a process for the preparation thereof and pharmaceutical composition comprising the same for antibiotics
DE102004062475A1
(en)
*
2004-12-24
2006-07-06
Bayer Healthcare Ag
Solid, orally administrable, modified release pharmaceutical dosage forms
EP1685841A1
(en)
*
2005-01-31
2006-08-02
Bayer Health Care Aktiengesellschaft
Prevention and treatment of thromboembolic disorders
DE102005045518A1
(en)
*
2005-09-23
2007-03-29
Bayer Healthcare Ag
New 5-thienylaminocarbonylmethyl-oxazolidin-2-one derivatives, useful for treating and preventing thromboembolic disease, are selective inhibitors of coagulation factor Xa
DE502006009169D1
(en)
2005-10-04
2011-05-05
Bayer Schering Pharma Ag
NEUE POLYMORPHE FORM VON 5-CHLOR-N-(ä ( 5S )-2-0X0-3-Ä4-( 3-OXO-4-MORPHOLINYL)-PHENYLÜ-1,3-OXAZOLIDIN-5-YLü -METHYL)-2-THIOPHENCARBOXAMID
DE102005047558A1
(en)
*
2005-10-04
2008-02-07
Bayer Healthcare Ag
Combination therapy of substituted oxazolidinones for the prophylaxis and treatment of cerebral circulatory disorders
DE102005047561A1
(en)
2005-10-04
2007-04-05
Bayer Healthcare Ag
Drug delivery system, useful to treat and/or prevent e.g. thromboembolic disease, comprises 5-chloro-N-(((5S)-2-oxo-3-(4-(3-oxo-4-morpholinyl)-phenyl)-1,3-oxazolidine-5-yl)-methyl)-2-thiophene carboxamide with fast release active substance
DE102005048824A1
(en)
*
2005-10-10
2007-04-12
Bayer Healthcare Ag
Treatment and prophylaxis of microangiopathies
DE102006051625A1
(en)
*
2006-11-02
2008-05-08
Bayer Materialscience Ag
Combination therapy of substituted oxazolidinones
MX2011003820A
(en)
2008-10-10
2011-06-16
Trius Therapeutics
Methods for preparing oxazolidinones and compositions containing them.
UA114068C2
(en)
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2009-02-03
2017-04-25
Crystalline particles
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2009-05-28
2013-11-12
Trius Therapeutics, Inc.
Oxazolidinone containing dimer compounds, compositions and methods to make and use
CN103601724B
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2013-11-14
2016-05-25
暨南大学
A kind of novel oxazolidinone compounds and its preparation method and application
CN103965085B
(en)
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2014-04-17
2016-02-24
上海恒晟药业有限公司
A kind of preparation method replacing 1,2-amino alcohol medicine
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Publication number
Priority date
Publication date
Assignee
Title
GB1180089A
(en)
*
1967-10-20
1970-02-04
Delalande Sa
Acetylenic Derivatives of 2-Oxazolidinones and processes of preparation
GB1224995A
(en)
*
1968-09-20
1971-03-10
Delalande Sa
New 5-propargyloxymethyl-2-substituted oxazolidinones and their process of preparation
GB1222708A
(en)
*
1968-10-22
1971-02-17
Delalande Sa
Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation
GB1252101A
(en)
*
1969-03-18
1971-11-03
DE2538424C2
(en)
*
1975-08-29
1983-01-05
Nordmark-Werke Gmbh, 2000 Hamburg
4-substituted 5-phenyl-oxazolidone- (2) – compounds and a pharmaceutical preparation containing them
FR2356422A1
(en)
*
1976-03-01
1978-01-27
Delalande Sa
NEW HYDROXYMETHYL-5 OXAZOLIDINONE-2, THEIR PREPARATION PROCESS AND THEIR APPLICATION IN THERAPEUTICS
JPS6040428A
(en)
*
1983-08-12
1985-03-02
Wakachiku Kensetsu Kk
Installation work of caisson
1978
1978-08-04
LU
LU80081A
patent/LU80081A1/en
unknown
1978-08-08
GR
GR56962A
patent/GR64146B/en
unknown
1978-08-09
US
US05/932,212
patent/US4250318A/en
not_active
Expired – Lifetime
1978-08-14
CH
CH861378A
patent/CH634836A5/en
not_active
IP Right Cessation
1978-08-16
GB
GB7833478A
patent/GB2003151B/en
not_active
Expired
1978-08-18
DE
DE19782836305
patent/DE2836305A1/en
not_active
Ceased
1978-08-18
JP
JP10082478A
patent/JPS5441871A/en
active
Granted
1978-08-21
SE
SE7808804A
patent/SE444813B/en
not_active
IP Right Cessation
1978-08-24
AU
AU39249/78A
patent/AU526714B2/en
not_active
Expired
1978-08-24
ES
ES472825A
patent/ES472825A1/en
not_active
Expired
1978-08-24
CA
CA310,018A
patent/CA1113093A/en
not_active
Expired
1978-08-25
IT
IT68979/78A
patent/IT1118099B/en
active
1978-08-25
NL
NL7808817A
patent/NL7808817A/en
not_active
Application Discontinuation
1980
1980-08-01
US
US06/174,415
patent/US4338451A/en
not_active
Expired – Lifetime
Also Published As
Publication number
Publication date
US4250318A
(en)
1981-02-10
GR64146B
(en)
1980-01-31
US4338451A
(en)
1982-07-06
JPS6354710B2
(en)
1988-10-28
CH634836A5
(en)
1983-02-28
GB2003151A
(en)
1979-03-07
IT1118099B
(en)
1986-02-24
SE444813B
(en)
1986-05-12
ES472825A1
(en)
1979-02-16
SE7808804L
(en)
1979-02-27
DE2836305A1
(en)
1979-03-01
AU526714B2
(en)
1983-01-27
IT7868979D0
(en)
1978-08-25
JPS5441871A
(en)
1979-04-03
GB2003151B
(en)
1982-10-06
NL7808817A
(en)
1979-02-28
CA1113093A
(en)
1981-11-24
LU80081A1
(en)
1979-05-15
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