AU504480B2 - Creación de Inventos y Patentes con Inteligencia Artificial

AU504480B2 – Anthracycline glycosides
– Google Patents

AU504480B2 – Anthracycline glycosides
– Google Patents
Anthracycline glycosides

Info

Publication number
AU504480B2

AU504480B2
AU18025/76A
AU1802576A
AU504480B2
AU 504480 B2
AU504480 B2
AU 504480B2
AU 18025/76 A
AU18025/76 A
AU 18025/76A
AU 1802576 A
AU1802576 A
AU 1802576A
AU 504480 B2
AU504480 B2
AU 504480B2
Authority
AU
Australia
Prior art keywords
anthracycline glycosides
anthracycline
glycosides
Prior art date
1975-09-26
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
AU18025/76A
Other versions

AU1802576A
(en

Inventor
Arcamone F. & Marco Ad Perico S.
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pfizer Italia SRL

Original Assignee
Farmaceutici Italia SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1975-09-26
Filing date
1976-09-22
Publication date
1979-10-18

1976-09-22
Application filed by Farmaceutici Italia SpA
filed
Critical
Farmaceutici Italia SpA

1978-04-06
Publication of AU1802576A
publication
Critical
patent/AU1802576A/en

1979-10-18
Application granted
granted
Critical

1979-10-18
Publication of AU504480B2
publication
Critical
patent/AU504480B2/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS

C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids

C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids

C07H13/04—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals attached to acyclic carbon atoms

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P35/00—Antineoplastic agents

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P35/00—Antineoplastic agents

A61P35/02—Antineoplastic agents specific for leukemia

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings

C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members

C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D309/14—Nitrogen atoms not forming part of a nitro radical

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS

C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals

C07H15/20—Carbocyclic rings

C07H15/24—Condensed ring systems having three or more rings

C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins

Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS

Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE

Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS

Y02P20/00—Technologies relating to chemical industry

Y02P20/50—Improvements relating to the production of bulk chemicals

Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

AU18025/76A
1975-09-26
1976-09-22
Anthracycline glycosides

Expired

AU504480B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

GB39471/75A

GB1511559A
(en)

1975-09-26
1975-09-26
Anthracycline glycosides

GBGB39471/75

1975-09-26

Publications (2)

Publication Number
Publication Date

AU1802576A

AU1802576A
(en)

1978-04-06

AU504480B2
true

AU504480B2
(en)

1979-10-18

Family
ID=10409731
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU18025/76A
Expired

AU504480B2
(en)

1975-09-26
1976-09-22
Anthracycline glycosides

Country Status (16)

Country
Link

US
(1)

US4067969A
(en)

JP
(1)

JPS5242869A
(en)

AT
(1)

AT347582B
(en)

AU
(1)

AU504480B2
(en)

BE
(1)

BE846548A
(en)

CA
(1)

CA1060002A
(en)

CH
(1)

CH606082A5
(en)

DE
(1)

DE2642837C3
(en)

DK
(1)

DK146626C
(en)

FR
(1)

FR2325659A1
(en)

GB
(1)

GB1511559A
(en)

HK
(1)

HK1182A
(en)

NL
(1)

NL174015C
(en)

SE
(2)

SE429655B
(en)

SU
(2)

SU670226A3
(en)

ZA
(1)

ZA765736B
(en)

Families Citing this family (31)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB1567456A
(en)

1976-11-16
1980-05-14
Farmaceutici Italia
Daunomycin derivatives

GB1550879A
(en)

1976-12-22
1979-08-22
Farmaceutici Italia
Antitumour glycosides

US4362720A
(en)

1977-04-14
1982-12-07
Chembiomed Ltd.
Synthesis of 2-amino-2-deoxyglycoses and 2-amino-2-deoxyglycosides from glycals

GB1573036A
(en)

1977-05-05
1980-08-13
Farmaceutici Italia
Anthracyclines

GB1573037A
(en)

1977-05-05
1980-08-13
Farmaceutici Italia
Anthracyclines

US4201773A
(en)

1978-07-26
1980-05-06
The United States Of America As Represented By The Department Of Health, Education And Welfare
7-O-(2,6-Dideoxy-α-L-lyxo-hexopyranosyl)-daunomycinone, desmethoxy daunomycinone, adriamycinone, and carminomycinone

US4259476A
(en)

1979-04-02
1981-03-31
Kende Andrew S
Novel heterocyclic anthracycline compounds

EP0024727B1
(en)

1979-09-01
1982-05-26
FARMITALIA CARLO ERBA S.p.A.
Anthracycline glycosides, processes for their preparation and pharmaceutical composition containing them

ZA814722B
(en)

1980-07-18
1982-07-28
Hoffmann La Roche
Novel anthracycline glycosides

CA1174669A
(en)

1980-07-18
1984-09-18
Michael J. Broadhurst
Anthracycline glycosides

US4345070A
(en)

1980-09-29
1982-08-17
Farmitalia Carlo Erba S.P.A.
Process for the preparation of 4′-deoxy-daunorubicin and 4′-deoxy-doxorubicin

JPS57106695A
(en)

1980-11-01
1982-07-02
Erba Carlo Spa
Anthracycline g lycoside compound

EP0051279B1
(en)

1980-11-01
1985-09-04
FARMITALIA CARLO ERBA S.p.A.
Anthracycline glycosides, intermediate compounds, process for preparing both and pharmaceutical compositions

JPS57142981A
(en)

1981-01-21
1982-09-03
Erba Carlo Spa
Anthracycline glycoside, manufacture and tumor generation inhibiting drug containing same

DE3200809C2
(en)

1981-01-21
1986-08-28
Farmitalia Carlo Erba S.p.A., Mailand/Milano

4′-Deoxy-3′-epi-daunorubicin and -doxorubicin, processes for their preparation and pharmaceuticals containing these compounds

US4325947A
(en)

1981-05-12
1982-04-20
Farmitalia Carlo Erba S.P.A.
4-Demethoxy-4′-deoxydoxorubicin

AU554416B2
(en)

1982-05-24
1986-08-21
Farmitalia Carlo Erba S.P.A.
Anthracycline glycosides

US4562177A
(en)

1982-08-17
1985-12-31
The Ohio State University Research Foundation
3′-Amino-2′ halo-anthracycline antibiotics

US4514561A
(en)

1983-04-15
1985-04-30
Research Corporation
Process for preparing α-L N-acetyl daunosaminide

DE3500023A1
(en)

1985-01-02
1986-07-10
Farmitalia Carlo Erba S.p.A., Mailand/Milano
4′-Deoxyanthracycline esters

GB2169285A
(en)

1985-01-05
1986-07-09
Erba Farmitalia
4′-Deoxydoxorubicin-14-esters

GB8519452D0
(en)

1985-08-02
1985-09-11
Erba Farmitalia
Injectable solutions

US5124317A
(en)

1985-08-02
1992-06-23
Farmitalia Carlo Erba S.P.A.
Injectable ready-to-use solutions containing an antitumor anthracycline glycoside

GB8708927D0
(en)

1987-04-14
1987-05-20
Erba Farmitalia
Chiral synthesis of anthracyclines

NZ224252A
(en)

1987-04-21
1991-09-25
Erba Carlo Spa
An anthracycline glycoside and its preparation

GB2212154B
(en)

1987-11-10
1991-03-27
Erba Carlo Spa
New 4-demethoxy anthracycline derivatives

WO1989006654A1
(en)

1988-01-19
1989-07-27
Board Of Regents, The University Of Texas System
Glycosides, liposomal compositions thereof, and methods for their use

GB8803076D0
(en)

1988-02-10
1988-03-09
Erba Carlo Spa
3′-deamino-4′-deoxy-4′-amino anthracyclines

AU4752190A
(en)

1988-12-28
1990-08-01
Board Of Regents, The University Of Texas System
3′-deamino analogs of esorubicin and methods for their use

US5948896A
(en)

1997-08-13
1999-09-07
Gem Pharmaceuticals
Processes for preparing 13-deoxy anthracycline derivatives

US5942605A
(en)

1998-03-03
1999-08-24
Gem Pharmaceuticals, Inc.
5-imino-13-deoxy anthracycline derivatives, their uses, and processes for preparing them

Family Cites Families (4)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US3803124A
(en)

1968-04-12
1974-04-09
Farmaceutici It Soc
Process for the preparation of adriamycin and adriamycinone and adriamycin derivatives

DE1792346C3
(en)

1968-08-22
1980-10-23
Rotta Research Laboratorium S.P.A., San Fruttuoso Di Monza, Mailand (Italien)

Pharmaceutical preparation for the treatment of degenerative joint diseases

FR2183710A1
(en)

1972-05-06
1973-12-21
Farmaceutici Italia
Daunomycin (hydrochloride) prepn – by reaction of daunomycinone with daunosamines, useful as antitumour agent and anti-leucemic

US4020270A
(en)

1974-05-02
1977-04-26
Societa’ Farmaceutici Italia S.P.A.
L-lyxohex-1-enopyranose derivative

1975

1975-09-26
GB
GB39471/75A
patent/GB1511559A/en
not_active
Expired

1976

1976-09-13
NL
NLAANVRAGE7610139,A
patent/NL174015C/en
not_active
IP Right Cessation

1976-09-13
US
US05/722,689
patent/US4067969A/en
not_active
Expired – Lifetime

1976-09-22
DK
DK426076A
patent/DK146626C/en
not_active
IP Right Cessation

1976-09-22
AU
AU18025/76A
patent/AU504480B2/en
not_active
Expired

1976-09-23
AT
AT707276A
patent/AT347582B/en
not_active
IP Right Cessation

1976-09-23
FR
FR7628582A
patent/FR2325659A1/en
active
Granted

1976-09-23
DE
DE2642837A
patent/DE2642837C3/en
not_active
Expired

1976-09-23
CA
CA261,920A
patent/CA1060002A/en
not_active
Expired

1976-09-23
SE
SE7610564A
patent/SE429655B/en
not_active
IP Right Cessation

1976-09-24
BE
BE170901A
patent/BE846548A/en
not_active
IP Right Cessation

1976-09-24
CH
CH1215876A
patent/CH606082A5/xx
not_active
IP Right Cessation

1976-09-24
JP
JP51115356A
patent/JPS5242869A/en
active
Granted

1976-09-24
SU
SU762403408A
patent/SU670226A3/en
active

1976-09-24
ZA
ZA765736A
patent/ZA765736B/en
unknown

1977

1977-09-22
SU
SU772523451A
patent/SU730310A3/en
active

1980

1980-02-29
SE
SE8001616A
patent/SE435514B/en
not_active
IP Right Cessation

1982

1982-01-14
HK
HK11/82A
patent/HK1182A/en
unknown

Also Published As

Publication number
Publication date

CA1060002A
(en)

1979-08-07

DE2642837C3
(en)

1982-08-12

FR2325659A1
(en)

1977-04-22

DE2642837B2
(en)

1982-01-07

HK1182A
(en)

1982-01-22

NL174015C
(en)

1984-04-16

DE2642837A1
(en)

1977-04-07

BE846548A
(en)

1977-03-24

SE8001616L
(en)

1980-02-29

US4067969A
(en)

1978-01-10

CH606082A5
(en)

1978-10-13

JPS5242869A
(en)

1977-04-04

ZA765736B
(en)

1977-11-30

SU670226A3
(en)

1979-06-25

SE7610564L
(en)

1977-03-27

GB1511559A
(en)

1978-05-24

SU730310A3
(en)

1980-04-25

SE429655B
(en)

1983-09-19

JPS6123189B2
(en)

1986-06-04

NL7610139A
(en)

1977-03-29

ATA707276A
(en)

1978-05-15

DK426076A
(en)

1977-03-27

SE435514B
(en)

1984-10-01

DK146626C
(en)

1984-04-30

FR2325659B1
(en)

1982-08-20

NL174015B
(en)

1983-11-16

AT347582B
(en)

1979-01-10

AU1802576A
(en)

1978-04-06

DK146626B
(en)

1983-11-21

Información de contacto