AU504599B2 – Benzisothiazolone derivatives
– Google Patents
AU504599B2 – Benzisothiazolone derivatives
– Google Patents
Benzisothiazolone derivatives
Info
Publication number
AU504599B2
AU504599B2
AU19163/76A
AU1916376A
AU504599B2
AU 504599 B2
AU504599 B2
AU 504599B2
AU 19163/76 A
AU19163/76 A
AU 19163/76A
AU 1916376 A
AU1916376 A
AU 1916376A
AU 504599 B2
AU504599 B2
AU 504599B2
Authority
AU
Australia
Prior art keywords
benzisothiazolone derivatives
benzisothiazolone
derivatives
Prior art date
1975-11-18
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU19163/76A
Other versions
AU1916376A
(en
Inventor
Keith Howard Baggaley
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1975-11-18
Filing date
1976-10-29
Publication date
1979-10-18
1976-10-29
Application filed by Beecham Group PLC
filed
Critical
Beecham Group PLC
1978-05-04
Publication of AU1916376A
publication
Critical
patent/AU1916376A/en
1979-10-18
Application granted
granted
Critical
1979-10-18
Publication of AU504599B2
publication
Critical
patent/AU504599B2/en
1992-10-29
Anticipated expiration
legal-status
Critical
Status
Ceased
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
A61K31/00—Medicinal preparations containing organic active ingredients
A61K31/33—Heterocyclic compounds
A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
A61K31/00—Medicinal preparations containing organic active ingredients
A61K31/33—Heterocyclic compounds
A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
A61K31/00—Medicinal preparations containing organic active ingredients
A61K31/33—Heterocyclic compounds
A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
A61K31/445—Non condensed piperidines, e.g. piperocaine
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
A61K31/00—Medicinal preparations containing organic active ingredients
A61K31/33—Heterocyclic compounds
A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
A61K31/47—Quinolines; Isoquinolines
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
AU19163/76A
1975-11-18
1976-10-29
Benzisothiazolone derivatives
Ceased
AU504599B2
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
GB4737375
1975-11-18
GB47373/75
1975-11-18
Related Child Applications (1)
Application Number
Title
Priority Date
Filing Date
AU47163/79A
Division
AU520890B2
(en)
1975-11-18
1979-05-17
Benzisothiazolones
Publications (2)
Publication Number
Publication Date
AU1916376A
AU1916376A
(en)
1978-05-04
AU504599B2
true
AU504599B2
(en)
1979-10-18
Family
ID=10444739
Family Applications (2)
Application Number
Title
Priority Date
Filing Date
AU19163/76A
Ceased
AU504599B2
(en)
1975-11-18
1976-10-29
Benzisothiazolone derivatives
AU47163/79A
Expired – Fee Related
AU520890B2
(en)
1975-11-18
1979-05-17
Benzisothiazolones
Family Applications After (1)
Application Number
Title
Priority Date
Filing Date
AU47163/79A
Expired – Fee Related
AU520890B2
(en)
1975-11-18
1979-05-17
Benzisothiazolones
Country Status (28)
Country
Link
US
(5)
US4113728A
(en)
JP
(1)
JPS5262273A
(en)
AR
(3)
AR217411A1
(en)
AT
(1)
AT355017B
(en)
AU
(2)
AU504599B2
(en)
BE
(1)
BE848371A
(en)
BG
(4)
BG24811A3
(en)
CA
(1)
CA1064511A
(en)
CH
(1)
CH627465A5
(en)
CS
(4)
CS192570B2
(en)
DD
(1)
DD127645A5
(en)
DE
(1)
DE2652201A1
(en)
DK
(1)
DK517776A
(en)
ES
(3)
ES453420A1
(en)
FI
(1)
FI763285A
(en)
FR
(1)
FR2332019A1
(en)
HU
(1)
HU173958B
(en)
IL
(1)
IL50690A
(en)
NL
(1)
NL7612796A
(en)
NO
(1)
NO763922L
(en)
NZ
(1)
NZ182325A
(en)
PH
(1)
PH13918A
(en)
PL
(1)
PL193742A1
(en)
PT
(1)
PT65851B
(en)
RO
(4)
RO69608A
(en)
SE
(1)
SE7612919L
(en)
SU
(4)
SU682129A3
(en)
ZA
(1)
ZA766489B
(en)
Families Citing this family (18)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
NZ182325A
(en)
*
1975-11-18
1979-03-16
Beecham Group Ltd
2-substituted-1,2-benzisothiazol-3-ones
DE2602643C2
(en)
*
1976-01-24
1984-12-20
Bayer Ag, 5090 Leverkusen
1,2-Benzisothiazolinone-3, process for their preparation, as well as pharmaceuticals
US4190663A
(en)
*
1976-01-24
1980-02-26
Bayer Aktiengesellschaft
Anti-thrombotic 1,2-benzisothiazolin-3-ones
DE2860750D1
(en)
*
1977-06-20
1981-09-17
Beecham Group Plc
Antithrombotic 2-(gamma-(1-piperidinyl)propyl)1,2-benzisothiazol 3-one, its pharmaceutically acceptable acid addition salts, their preparation and their compositions
DE2860430D1
(en)
*
1977-10-08
1981-02-26
Beecham Group Ltd
Antithrombotic compositions containing benzisothiazolones
DE2966957D1
(en)
*
1979-10-08
1984-06-07
Merck & Co Inc
2-aryl-1,2-benzisothiazolinone-1,1-dioxides and pharmaceutical compositions containing them
DE3226284A1
(en)
*
1982-07-14
1984-01-19
A. Nattermann & Cie GmbH, 5000 Köln
NEW BENZISOSELENAZOLONES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM
DE3238006A1
(en)
*
1982-10-13
1984-04-19
Bayer Ag, 5090 Leverkusen
AZOLYL METHYLAMINE, THEIR PRODUCTION AND USE IN MICROBICIDES
DE3500577A1
(en)
*
1985-01-10
1986-07-10
Basf Ag, 6700 Ludwigshafen
METHOD FOR PRODUCING 1,2-BENZISOTHIAZOLONES
US4732984A
(en)
*
1985-10-17
1988-03-22
American Home Products Corporation
Piperazinoisothiazolones with psychotropic activity
DE3617976A1
(en)
*
1986-05-28
1988-01-14
Alter Sa
1,4-DIHYDROPYRIDINE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE IN ANTITHROMBOTIC MEDICATIONS
US4831031A
(en)
*
1988-01-22
1989-05-16
Pfizer Inc.
Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity
CA1340759C
(en)
*
1988-07-01
1999-09-21
James P. Albarella
Isobenzothiazolone chromogenic thiol indicators and their derivatives
US5128457A
(en)
*
1988-07-01
1992-07-07
Miles Inc.
Chromogenic thiol indicators based on an isobenzothiazolone ring system
US5236917A
(en)
*
1989-05-04
1993-08-17
Sterling Winthrop Inc.
Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
EP2344479B1
(en)
*
2008-09-23
2015-04-08
Georgetown University
1,2-benzisothiazolinone and isoindolinone derivatives
AU2012296543B2
(en)
2011-08-16
2016-08-11
Georgetown University
Methods of treating bacterial infections with 1,2-benzisothiazolinone and isoindolinone derivatives
US20180318818A1
(en)
2015-10-19
2018-11-08
Emory University
Redox Dehydration Coupling Catalysts and Methods Related Thereto
Family Cites Families (8)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
BE565380A
(en)
*
1957-03-08
US3012039A
(en)
*
1958-03-14
1961-12-05
Ici Ltd
2-p-chlorobenzyl-1, 2-benzisothiazolone
DE1147947B
(en)
*
1961-07-25
1963-05-02
Knoll Ag
Process for the preparation of new 1,2-benzisothiazolones
SE392103B
(en)
*
1970-04-27
1977-03-14
Sherwin Williams Co
METHOD OF PRODUCING 1,2-BENSISOTIAZOLINE-3-ONERS
US3661974A
(en)
*
1970-04-27
1972-05-09
Sherwin Williams Co
2-carbalkoxy-phenyl sulfenamides
NZ182325A
(en)
*
1975-11-18
1979-03-16
Beecham Group Ltd
2-substituted-1,2-benzisothiazol-3-ones
GB1582214A
(en)
*
1977-05-31
1981-01-07
Beecham Group Ltd
Antithrombotic compositions
DE2734882A1
(en)
*
1977-08-03
1979-02-22
Basf Ag
3-SQUARE BRACKETS ON 4- (1,3-DIAZACYCLOALKEN-2-YL) -PHENYL SQUARE BRACKETS FOR -1,2-BENZISOTHIAZOLS, THE METHOD FOR THEIR MANUFACTURING AND THE MEDICINAL PRODUCTS CONTAINED
1976
1976-10-13
NZ
NZ182325A
patent/NZ182325A/en
unknown
1976-10-15
IL
IL50690A
patent/IL50690A/en
unknown
1976-10-20
PH
PH19020A
patent/PH13918A/en
unknown
1976-10-29
ZA
ZA766489A
patent/ZA766489B/en
unknown
1976-10-29
AU
AU19163/76A
patent/AU504599B2/en
not_active
Ceased
1976-11-02
US
US05/738,000
patent/US4113728A/en
not_active
Expired – Lifetime
1976-11-10
AR
AR265414A
patent/AR217411A1/en
active
1976-11-15
FR
FR7634296A
patent/FR2332019A1/en
active
Granted
1976-11-15
AT
AT849176A
patent/AT355017B/en
not_active
IP Right Cessation
1976-11-16
BE
BE172385A
patent/BE848371A/en
not_active
IP Right Cessation
1976-11-16
DE
DE19762652201
patent/DE2652201A1/en
not_active
Withdrawn
1976-11-16
HU
HU76BE1280A
patent/HU173958B/en
unknown
1976-11-16
FI
FI763285A
patent/FI763285A/fi
not_active
Application Discontinuation
1976-11-17
ES
ES453420A
patent/ES453420A1/en
not_active
Expired
1976-11-17
CS
CS767392A
patent/CS192570B2/en
unknown
1976-11-17
CA
CA265,874A
patent/CA1064511A/en
not_active
Expired
1976-11-17
DD
DD195824A
patent/DD127645A5/xx
unknown
1976-11-17
RO
RO7688476A
patent/RO69608A/en
unknown
1976-11-17
CS
CS775980A
patent/CS192593B2/en
unknown
1976-11-17
BG
BG7600035568A
patent/BG24811A3/en
unknown
1976-11-17
CH
CH1448376A
patent/CH627465A5/en
not_active
IP Right Cessation
1976-11-17
BG
BG7600034711A
patent/BG24808A3/en
unknown
1976-11-17
PL
PL19374276A
patent/PL193742A1/en
unknown
1976-11-17
BG
BG7600035567A
patent/BG24810A3/en
unknown
1976-11-17
BG
BG7600035566A
patent/BG24809A3/en
unknown
1976-11-17
RO
RO7696010A
patent/RO75540A/en
unknown
1976-11-17
NL
NL7612796A
patent/NL7612796A/en
not_active
Application Discontinuation
1976-11-17
PT
PT65851A
patent/PT65851B/en
unknown
1976-11-17
CS
CS775981A
patent/CS192594B2/en
unknown
1976-11-17
DK
DK517776A
patent/DK517776A/en
not_active
Application Discontinuation
1976-11-17
NO
NO763922A
patent/NO763922L/no
unknown
1976-11-17
CS
CS775979A
patent/CS192592B2/en
unknown
1976-11-17
SU
SU762422503A
patent/SU682129A3/en
active
1976-11-17
RO
RO7696012A
patent/RO75777A/en
unknown
1976-11-17
RO
RO7696011A
patent/RO75730A/en
unknown
1976-11-18
SE
SE7612919A
patent/SE7612919L/en
not_active
Application Discontinuation
1976-11-18
JP
JP51139026A
patent/JPS5262273A/en
active
Pending
1977
1977-04-04
SU
SU772466684A
patent/SU679141A3/en
active
1977-04-04
SU
SU772466683A
patent/SU701536A3/en
active
1977-04-04
SU
SU772466669A
patent/SU671728A3/en
active
1977-10-17
AR
AR269610A
patent/AR217449A1/en
active
1977-10-17
AR
AR269611A
patent/AR215271A1/en
active
1977-11-11
US
US05/850,786
patent/US4212979A/en
not_active
Expired – Lifetime
1977-12-16
ES
ES465174A
patent/ES465174A1/en
not_active
Expired
1977-12-16
ES
ES465173A
patent/ES465173A1/en
not_active
Expired
1978
1978-08-25
US
US05/936,861
patent/US4212872A/en
not_active
Expired – Lifetime
1979
1979-05-17
AU
AU47163/79A
patent/AU520890B2/en
not_active
Expired – Fee Related
1979-08-20
US
US06/067,949
patent/US4243669A/en
not_active
Expired – Lifetime
1980
1980-10-31
US
US06/202,711
patent/US4350702A/en
not_active
Expired – Lifetime
Also Published As
Publication number
Publication date
AT355017B
(en)
1980-02-11
AR215271A1
(en)
1979-09-28
SE7612919L
(en)
1977-05-19
FI763285A
(en)
1977-05-19
SU701536A3
(en)
1979-11-30
CS192570B2
(en)
1979-08-31
PH13918A
(en)
1980-11-04
AR217449A1
(en)
1980-03-31
AU4716379A
(en)
1979-09-27
NZ182325A
(en)
1979-03-16
US4243669A
(en)
1981-01-06
RO75777A
(en)
1981-02-28
DK517776A
(en)
1977-05-19
AU1916376A
(en)
1978-05-04
BE848371A
(en)
1977-05-16
DE2652201A1
(en)
1977-06-02
NL7612796A
(en)
1977-05-23
SU679141A3
(en)
1979-08-05
BG24809A3
(en)
1978-05-12
RO75540A
(en)
1980-11-30
ES465173A1
(en)
1978-10-01
CA1064511A
(en)
1979-10-16
BG24808A3
(en)
1978-05-12
FR2332019B1
(en)
1983-05-20
US4212979A
(en)
1980-07-15
HU173958B
(en)
1979-09-28
PL193742A1
(en)
1979-05-21
IL50690A
(en)
1980-01-31
DD127645A5
(en)
1977-10-05
PT65851B
(en)
1978-05-15
RO69608A
(en)
1982-07-06
US4212872A
(en)
1980-07-15
CS192592B2
(en)
1979-08-31
SU682129A3
(en)
1979-08-25
ZA766489B
(en)
1977-10-26
US4350702A
(en)
1982-09-21
NO763922L
(en)
1977-05-20
ES465174A1
(en)
1978-10-01
ES453420A1
(en)
1978-02-16
RO75730A
(en)
1981-02-28
ATA849176A
(en)
1979-07-15
CS192593B2
(en)
1979-08-31
BG24811A3
(en)
1978-05-12
IL50690A0
(en)
1976-12-31
AU520890B2
(en)
1982-03-04
CH627465A5
(en)
1982-01-15
CS192594B2
(en)
1979-08-31
AR217411A1
(en)
1980-03-31
US4113728A
(en)
1978-09-12
JPS5262273A
(en)
1977-05-23
BG24810A3
(en)
1978-05-12
FR2332019A1
(en)
1977-06-17
SU671728A3
(en)
1979-06-30
PT65851A
(en)
1976-12-01
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