AU5183279A – Compounds
– Google Patents
AU5183279A – Compounds
– Google Patents
Compounds
Info
Publication number
AU5183279A
AU5183279A
AU51832/79A
AU5183279A
AU5183279A
AU 5183279 A
AU5183279 A
AU 5183279A
AU 51832/79 A
AU51832/79 A
AU 51832/79A
AU 5183279 A
AU5183279 A
AU 5183279A
AU 5183279 A
AU5183279 A
AU 5183279A
Authority
AU
Australia
Prior art keywords
carboxy
hydrogen
physiologically acceptable
salt
base
Prior art date
1978-10-18
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU51832/79A
Other versions
AU529643B2
(en
Inventor
Helmut Biere
Dr. Irmgard Bottcher
Joachim-Friedrich Kapp
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Pharma AG
Original Assignee
Schering AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1978-10-18
Filing date
1979-10-16
Publication date
1980-04-24
1979-10-16
Application filed by Schering AG
filed
Critical
Schering AG
1980-04-24
Publication of AU5183279A
publication
Critical
patent/AU5183279A/en
1983-06-16
Application granted
granted
Critical
1983-06-16
Publication of AU529643B2
publication
Critical
patent/AU529643B2/en
1999-10-16
Anticipated expiration
legal-status
Critical
Status
Expired – Fee Related
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 – C07D463/00
C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 – C07D463/00 in which the condensed system contains two hetero rings
C07D471/04—Ortho-condensed systems
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P25/00—Drugs for disorders of the nervous system
A61P25/04—Centrally acting analgesics, e.g. opioids
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P37/00—Drugs for immunological or allergic disorders
A61P37/08—Antiallergic agents
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
C07D209/04—Indoles; Hydrogenated indoles
C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
C07D209/32—Oxygen atoms
C07D209/38—Oxygen atoms in positions 2 and 3, e.g. isatin
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D213/61—Halogen atoms or nitro radicals
Abstract
Pyrido[2,1-b]quinazolinones of the formula
AU51832/79A
1978-10-18
1979-10-16
Compounds
Expired – Fee Related
AU529643B2
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
DE28457661
1978-10-18
DE19782845766
DE2845766A1
(en)
1978-10-18
1978-10-18
PYRIDO ANGLE CLAMP ON 2,1-B ANGLE CLAMP ON -CHINAZOLINONE DERIVATIVES, THEIR PRODUCTION AND USE
Publications (2)
Publication Number
Publication Date
AU5183279A
true
AU5183279A
(en)
1980-04-24
AU529643B2
AU529643B2
(en)
1983-06-16
Family
ID=6052696
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU51832/79A
Expired – Fee Related
AU529643B2
(en)
1978-10-18
1979-10-16
Compounds
Country Status (25)
Country
Link
US
(1)
US4457927A
(en)
EP
(1)
EP0011142B1
(en)
JP
(1)
JPS5557588A
(en)
AT
(1)
ATE2146T1
(en)
AU
(1)
AU529643B2
(en)
CA
(1)
CA1130805A
(en)
CS
(1)
CS216512B2
(en)
DD
(1)
DD147242A5
(en)
DE
(2)
DE2845766A1
(en)
DK
(1)
DK154297C
(en)
EG
(1)
EG14028A
(en)
ES
(1)
ES8103745A1
(en)
FI
(1)
FI793229A
(en)
FR
(1)
FR2439199A1
(en)
GB
(1)
GB2034705B
(en)
GR
(1)
GR73819B
(en)
IE
(1)
IE48852B1
(en)
IL
(1)
IL58474A0
(en)
NO
(1)
NO793344L
(en)
NZ
(1)
NZ191828A
(en)
PL
(3)
PL123075B1
(en)
PT
(1)
PT70329A
(en)
RO
(1)
RO78339A
(en)
SU
(1)
SU1001857A3
(en)
ZA
(1)
ZA795559B
(en)
Families Citing this family (18)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
DE3300477A1
(en)
*
1983-01-08
1984-07-12
Boehringer Ingelheim KG, 6507 Ingelheim
NEW HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE
US4587339A
(en)
*
1983-10-14
1986-05-06
Sun Chemical Corporation
Nickel complex pigments of bis-azomethines
JPH06509576A
(en)
*
1991-07-29
1994-10-27
ワーナー−ランバート・コンパニー
Quinazoline derivatives as acetylcholinesterase inhibitors
CA2238283C
(en)
1997-05-30
2002-08-20
Cell Pathways, Inc.
Method for identifying compounds for inhibition of neoplastic lesions, pharmaceutical compositions from such compounds and uses of such compounds and compositions for treating neoplastic lesions
US5858694A
(en)
*
1997-05-30
1999-01-12
Cell Pathways, Inc.
Method for identifying compounds for inhibition of cancerous lesions
US6410584B1
(en)
*
1998-01-14
2002-06-25
Cell Pathways, Inc.
Method for inhibiting neoplastic cells with indole derivatives
US6200771B1
(en)
1998-10-15
2001-03-13
Cell Pathways, Inc.
Method of using a novel phosphodiesterase in pharmaceutical screeing to identify compounds for treatment of neoplasia
US6130053A
(en)
*
1999-08-03
2000-10-10
Cell Pathways, Inc.
Method for selecting compounds for inhibition of neoplastic lesions
US6133271A
(en)
*
1998-11-19
2000-10-17
Cell Pathways, Inc.
Method for inhibiting neoplastic cells and related conditions by exposure thienopyrimidine derivatives
US6187779B1
(en)
1998-11-20
2001-02-13
Cell Pathways, Inc.
Method for inhibiting neoplastic cells and related conditions by exposure to 2,8-disubstituted quinazoline derivatives
US6369092B1
(en)
1998-11-23
2002-04-09
Cell Pathways, Inc.
Method for treating neoplasia by exposure to substituted benzimidazole derivatives
US6077842A
(en)
*
1998-11-24
2000-06-20
Cell Pathways, Inc.
Method of inhibiting neoplastic cells with pyrazolopyridylpyridazinone derivatives
US6486155B1
(en)
1998-11-24
2002-11-26
Cell Pathways Inc
Method of inhibiting neoplastic cells with isoquinoline derivatives
US6034099A
(en)
*
1998-11-24
2000-03-07
Cell Pathways, Inc.
Method for inhibiting neoplastic lesions by administering 4-(arylmethylene)- 2, 3- dihydro-pyrazol-3-ones
US6025394A
(en)
1999-01-29
2000-02-15
Cell Pathways, Inc.
Method for treating patients with acne by administering substituted sulfonyl indenyl acetic acids, amides and alcohols
US6020379A
(en)
*
1999-02-19
2000-02-01
Cell Pathways, Inc.
Position 7 substituted indenyl-3-acetic acid derivatives and amides thereof for the treatment of neoplasia
US6555547B1
(en)
2000-02-28
2003-04-29
Cell Pathways, Inc.
Method for treating a patient with neoplasia by treatment with a vinca alkaloid derivative
US6569638B1
(en)
2000-03-03
2003-05-27
Cell Pathways, Inc
Method for screening compounds for the treatment of neoplasia
Family Cites Families (5)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
GB1064259A
(en)
*
1963-12-19
1967-04-05
Union Pharma Scient Appl
New derivatives of 2-anilino-nicotinic acid and process for their preparation
US4033961A
(en)
*
1975-10-07
1977-07-05
Warner-Lambert Company
Pyrido[2-1-b]quinazolin-ones and their methods of preparation
DE2557425A1
(en)
*
1975-12-19
1977-06-30
Boehringer Sohn Ingelheim
CHINAZOLONE DERIVATIVES
US4066767A
(en)
*
1976-11-01
1978-01-03
Warner-Lambert Company
8-(1H-Tetrazol-5-yl)-11H-pyrido[2,1-b]quinazolin-11-ones and method of treating bronchial asthma using them
ES468126A1
(en)
*
1977-03-24
1979-09-01
Hoffmann La Roche
Pyridol(2,1-b)quinazoline derivatives
1978
1978-10-18
DE
DE19782845766
patent/DE2845766A1/en
not_active
Withdrawn
1979
1979-10-11
NZ
NZ191828A
patent/NZ191828A/en
unknown
1979-10-15
DD
DD79216232A
patent/DD147242A5/en
unknown
1979-10-15
EP
EP79103974A
patent/EP0011142B1/en
not_active
Expired
1979-10-15
AT
AT79103974T
patent/ATE2146T1/en
not_active
IP Right Cessation
1979-10-15
DE
DE7979103974T
patent/DE2964431D1/en
not_active
Expired
1979-10-16
AU
AU51832/79A
patent/AU529643B2/en
not_active
Expired – Fee Related
1979-10-16
RO
RO7998984A
patent/RO78339A/en
unknown
1979-10-16
PL
PL1979227126A
patent/PL123075B1/en
unknown
1979-10-16
PL
PL1979218993A
patent/PL119174B1/en
unknown
1979-10-16
PL
PL1979227124A
patent/PL123430B1/en
unknown
1979-10-16
GR
GR60275A
patent/GR73819B/el
unknown
1979-10-17
NO
NO793344A
patent/NO793344L/en
unknown
1979-10-17
DK
DK438379A
patent/DK154297C/en
active
1979-10-17
IE
IE1969/79A
patent/IE48852B1/en
unknown
1979-10-17
CA
CA337,796A
patent/CA1130805A/en
not_active
Expired
1979-10-17
IL
IL58474A
patent/IL58474A0/en
unknown
1979-10-17
PT
PT70329A
patent/PT70329A/en
unknown
1979-10-17
SU
SU792832051A
patent/SU1001857A3/en
active
1979-10-18
FI
FI793229A
patent/FI793229A/en
not_active
Application Discontinuation
1979-10-18
ES
ES485162A
patent/ES8103745A1/en
not_active
Expired
1979-10-18
GB
GB7936147A
patent/GB2034705B/en
not_active
Expired
1979-10-18
CS
CS797083A
patent/CS216512B2/en
unknown
1979-10-18
EG
EG624/79A
patent/EG14028A/en
active
1979-10-18
ZA
ZA00795559A
patent/ZA795559B/en
unknown
1979-10-18
FR
FR7925883A
patent/FR2439199A1/en
not_active
Withdrawn
1979-10-18
JP
JP13363479A
patent/JPS5557588A/en
active
Granted
1982
1982-12-22
US
US06/452,009
patent/US4457927A/en
not_active
Expired – Fee Related
Also Published As
Publication number
Publication date
EP0011142B1
(en)
1982-12-29
DD147242A5
(en)
1981-03-25
IL58474A0
(en)
1980-01-31
FR2439199A1
(en)
1980-05-16
SU1001857A3
(en)
1983-02-28
DE2964431D1
(en)
1983-02-03
CS216512B2
(en)
1982-11-26
DK438379A
(en)
1980-04-19
ZA795559B
(en)
1980-09-24
ES485162A0
(en)
1981-03-16
NZ191828A
(en)
1983-03-15
DE2845766A1
(en)
1980-04-30
US4457927A
(en)
1984-07-03
ES8103745A1
(en)
1981-03-16
JPS5557588A
(en)
1980-04-28
DK154297B
(en)
1988-10-31
PT70329A
(en)
1979-11-01
EP0011142A1
(en)
1980-05-28
IE791969L
(en)
1980-04-18
RO78339A
(en)
1982-04-12
PL218993A1
(en)
1980-06-16
PL123430B1
(en)
1982-10-30
PL119174B1
(en)
1981-12-31
NO793344L
(en)
1980-04-21
CA1130805A
(en)
1982-08-31
IE48852B1
(en)
1985-05-29
ATE2146T1
(en)
1983-01-15
GB2034705A
(en)
1980-06-11
GR73819B
(en)
1984-05-03
AU529643B2
(en)
1983-06-16
GB2034705B
(en)
1982-12-08
EG14028A
(en)
1982-09-30
JPS634537B2
(en)
1988-01-29
PL123075B1
(en)
1982-09-30
FI793229A
(en)
1980-04-19
DK154297C
(en)
1989-03-28
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None