AU5444486A

AU5444486A – Pyridine derivatives
– Google Patents

AU5444486A – Pyridine derivatives
– Google Patents
Pyridine derivatives

Info

Publication number
AU5444486A

AU5444486A
AU54444/86A
AU5444486A
AU5444486A
AU 5444486 A
AU5444486 A
AU 5444486A
AU 54444/86 A
AU54444/86 A
AU 54444/86A
AU 5444486 A
AU5444486 A
AU 5444486A
AU 5444486 A
AU5444486 A
AU 5444486A
Authority
AU
Australia
Prior art keywords
pyridine derivatives
pyridine
derivatives
Prior art date
1985-03-08
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU54444/86A
Other versions

AU585586B2
(en

Inventor
Ian Ahnfelt-Ronne
Ole Bent Tvaermose Nielsen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Leo Pharma AS

Original Assignee
Leo Pharmaceutical Products Ltd AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1985-03-08
Filing date
1986-03-07
Publication date
1986-09-18

1985-03-08
Priority claimed from GB858506094A
external-priority
patent/GB8506094D0/en

1985-10-11
Priority claimed from GB858525153A
external-priority
patent/GB8525153D0/en

1986-03-07
Application filed by Leo Pharmaceutical Products Ltd AS
filed
Critical
Leo Pharmaceutical Products Ltd AS

1986-09-18
Publication of AU5444486A
publication
Critical
patent/AU5444486A/en

1989-06-22
Application granted
granted
Critical

1989-06-22
Publication of AU585586B2
publication
Critical
patent/AU585586B2/en

2006-03-07
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members

C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms

C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms

C07D213/30—Oxygen atoms

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members

C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms

C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms

C07D213/32—Sulfur atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members

C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms

C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms

C07D213/32—Sulfur atoms

C07D213/34—Sulfur atoms to which a second hetero atom is attached

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems

C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom

C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems

C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom

C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms

C07D215/14—Radicals substituted by oxygen atoms

AU54444/86A
1985-03-08
1986-03-07
Pyridine derivatives

Ceased

AU585586B2
(en)

Applications Claiming Priority (4)

Application Number
Priority Date
Filing Date
Title

GB8506094

1985-03-08

GB858506094A

GB8506094D0
(en)

1985-03-08
1985-03-08
Chemical products

GB858525153A

GB8525153D0
(en)

1985-10-11
1985-10-11
Chemical compounds

GB8525153

1985-10-11

Publications (2)

Publication Number
Publication Date

AU5444486A
true

AU5444486A
(en)

1986-09-18

AU585586B2

AU585586B2
(en)

1989-06-22

Family
ID=26288945
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU54444/86A
Ceased

AU585586B2
(en)

1985-03-08
1986-03-07
Pyridine derivatives

Country Status (18)

Country
Link

US
(2)

US4826987A
(en)

JP
(1)

JPH0764813B2
(en)

AU
(1)

AU585586B2
(en)

BE
(1)

BE904368A
(en)

CA
(1)

CA1276640C
(en)

DE
(1)

DE3607382A1
(en)

DK
(1)

DK166582B1
(en)

ES
(1)

ES8802610A1
(en)

FR
(1)

FR2578540B1
(en)

GB
(1)

GB2173788B
(en)

GR
(1)

GR860628B
(en)

IE
(1)

IE58870B1
(en)

IT
(1)

IT1221079B
(en)

LU
(1)

LU86349A1
(en)

NL
(1)

NL8600596A
(en)

NZ
(1)

NZ215347A
(en)

PT
(1)

PT82147B
(en)

SE
(1)

SE463819B
(en)

Families Citing this family (24)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

ATE68789T1
(en)

*

1985-10-16
1991-11-15
Merck Frosst Canada Inc

2-SUBSTITUTED QUINOLINES.

DK196688A
(en)

*

1987-04-28
1988-10-29
Fujisawa Pharmaceutical Co

BICYCLIC RELATIONS AND PROCEDURES FOR PRODUCING THEREOF

US4826990A
(en)

*

1987-09-30
1989-05-02
American Home Products Corporation
2-aryl substituted heterocyclic compounds as antiallergic and antiinflammatory agents

GB8728051D0
(en)

*

1987-12-01
1988-01-06
Leo Pharm Prod Ltd
Chemical compounds

US4889935A
(en)

*

1987-12-18
1989-12-26
American Home Products Corporation
Aminoguanidine derivatives

WO1990012006A1
(en)

*

1989-04-07
1990-10-18
Pfizer Inc.
Substituted 1-[3-(heteroarylmethoxy)phenyl]alkanols and related compounds in the treatment of asthma, arthritis and related diseases

DE3927369A1
(en)

*

1989-08-19
1991-02-21
Bayer Ag

SUBSTITUTED N- (CHINOLIN-2-YL-METHOXY) BENZYL-SULFONYL-UREAS

DE3935139A1
(en)

*

1989-10-21
1991-04-25
Bayer Ag

SUBSTITUTED (CHINOLIN-2-YL-METHOXY) PHENYL-THINARNES

US5021576A
(en)

*

1989-10-27
1991-06-04
American Home Products Corporation
2-Anilino phenylacetic acid derivatives

US5324747A
(en)

*

1992-07-15
1994-06-28
Hoffmann-La Roche Inc.
N-substituted anilines, inhibitors of phospholipases A2

US5840318A
(en)

*

1993-05-11
1998-11-24
Immunom Technologies, Inc.
Methods and compositions for modulating immune systems of animals

US7189834B2
(en)

*

1993-05-11
2007-03-13
Marshall William E
Oligoribonucleotides alert the immune system of animals to the imminence of microbial infection

US5508408A
(en)

*

1993-09-10
1996-04-16
Ciba-Geigy Corporation
Quinoline compound

US5795900A
(en)

*

1995-10-03
1998-08-18
Abbott Laboratories
Symmetrical bis-heteroaryl-methoxy-phenylalkyl carboxylates as inhibitors of leukotriene biosynthesis

US5668150A
(en)

*

1996-07-26
1997-09-16
Abbott Laboratories
Non-symmetrical bis-heteroarylmethoxyphenylalkyl carboxylates as inhibitors of leukotriene biosynthesis

CA2317008C
(en)

*

1997-12-31
2009-01-20
The University Of Kansas
Water soluble prodrugs of tertiary amine containing drugs and methods of making thereof

HN2001000008A
(en)

*

2000-01-21
2003-12-11
Inc Agouron Pharmaceuticals

AMIDA COMPOSITE AND PHARMACEUTICAL COMPOSITIONS TO INHIBIT PROTEINKINASES, AND THE INSTRUCTIONS FOR USE

GB2431927B
(en)

*

2005-11-04
2010-03-17
Amira Pharmaceuticals Inc
5-Lipoxygenase-activating protein (FLAP) inhibitors

US8399666B2
(en)

*

2005-11-04
2013-03-19
Panmira Pharmaceuticals, Llc
5-lipoxygenase-activating protein (FLAP) inhibitors

US7977359B2
(en)

*

2005-11-04
2011-07-12
Amira Pharmaceuticals, Inc.
5-lipdxygenase-activating protein (FLAP) inhibitors

TW200920369A
(en)

*

2007-10-26
2009-05-16
Amira Pharmaceuticals Inc
5-lipoxygenase activating protein (flap) inhibitor

EP2285803A4
(en)

*

2008-05-23
2011-10-05
Amira Pharmaceuticals Inc
5-lipoxygenase-activating protein inhibitor

US8546431B2
(en)

2008-10-01
2013-10-01
Panmira Pharmaceuticals, Llc
5-lipoxygenase-activating protein (FLAP) inhibitors

TW201215607A
(en)

2010-07-02
2012-04-16
Lundbeck & Co As H
Aryl-and heteroarylamid derivatives as PDE10A enzyme inhibitor

Family Cites Families (12)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US31624A
(en)

*

1861-03-05

Tatting-frame

US2761865A
(en)

*

1954-07-07
1956-09-04
Hoffmann La Roche
Pyridylalkyl sulfones

US4003906A
(en)

*

1974-01-22
1977-01-18
The Dow Chemical Company
Substituted pyridinyl methylthio or (methylsulfonyl)benzeneamines

GB2069492B
(en)

*

1980-02-20
1984-02-29
Wyeth John & Brother Ltd
Sulphur compounds

GB2069493B
(en)

*

1980-02-20
1984-02-29
Wyeth John & Brother Ltd
Pyridine derivatives

US4567184A
(en)

*

1982-12-01
1986-01-28
Usv Pharmaceutical Corporation
Certain aryl or hetero-aryl derivatives of 1-hydroxy-pentane or 1-hydroxy-hexane which are useful for treating inflammation and allergies

IE56702B1
(en)

*

1982-12-01
1991-11-06
Usv Pharma Corp
Antiinflammatory antiallergic compounds

JPS5988835U
(en)

*

1982-12-06
1984-06-15
ホシデン株式会社

switch

US4486593A
(en)

*

1983-01-19
1984-12-04
The Upjohn Company
2-,3-, or 4-Pyridinylmethylamino arylic acids as thromboxane A2 synthetase and 5-lipoxygenase inhibitors

US4563463A
(en)

*

1983-03-18
1986-01-07
Usv Pharmaceutical Corp.
2-Oxo-1,3-oxazolo[4,5-h] quinolines useful as anti-allergy agents

US4554355A
(en)

*

1984-07-19
1985-11-19
American Home Products Corporation
Heterocyclic compounds as antiallergic agents

US5109009A
(en)

*

1985-03-08
1992-04-28
Leo Pharmaceutical Products Ltd.
Quinoline and pyridine compounds and inhibition of 5-lipoxygenases therewith

1986

1986-02-10
IE
IE37086A
patent/IE58870B1/en
not_active
IP Right Cessation

1986-02-20
GB
GB08604183A
patent/GB2173788B/en
not_active
Expired

1986-02-28
US
US06/834,542
patent/US4826987A/en
not_active
Expired – Fee Related

1986-02-28
SE
SE8600913A
patent/SE463819B/en
not_active
IP Right Cessation

1986-03-03
NZ
NZ215347A
patent/NZ215347A/en
unknown

1986-03-04
DK
DK096986A
patent/DK166582B1/en
not_active
IP Right Cessation

1986-03-06
GR
GR860628A
patent/GR860628B/en
unknown

1986-03-06
IT
IT67183/86A
patent/IT1221079B/en
active

1986-03-06
DE
DE19863607382
patent/DE3607382A1/en
not_active
Ceased

1986-03-06
CA
CA000503464A
patent/CA1276640C/en
not_active
Expired – Fee Related

1986-03-06
PT
PT82147A
patent/PT82147B/en
not_active
IP Right Cessation

1986-03-07
ES
ES552805A
patent/ES8802610A1/en
not_active
Expired

1986-03-07
FR
FR868603268A
patent/FR2578540B1/en
not_active
Expired – Fee Related

1986-03-07
AU
AU54444/86A
patent/AU585586B2/en
not_active
Ceased

1986-03-07
BE
BE0/216378A
patent/BE904368A/en
not_active
IP Right Cessation

1986-03-07
LU
LU86349A
patent/LU86349A1/en
unknown

1986-03-07
NL
NL8600596A
patent/NL8600596A/en
not_active
Application Discontinuation

1986-03-08
JP
JP61051286A
patent/JPH0764813B2/en
not_active
Expired – Lifetime

1990

1990-12-31
US
US07/633,390
patent/US5157039A/en
not_active
Expired – Fee Related

Also Published As

Publication number
Publication date

ES552805A0
(en)

1988-09-16

LU86349A1
(en)

1987-04-02

GB2173788A
(en)

1986-10-22

PT82147A
(en)

1986-04-01

AU585586B2
(en)

1989-06-22

JPH0764813B2
(en)

1995-07-12

FR2578540A1
(en)

1986-09-12

FR2578540B1
(en)

1990-11-16

SE8600913L
(en)

1986-09-09

SE8600913D0
(en)

1986-02-28

DK166582B1
(en)

1993-06-14

GB8604183D0
(en)

1986-03-26

PT82147B
(en)

1988-07-29

SE463819B
(en)

1991-01-28

DE3607382A1
(en)

1986-09-11

IE860370L
(en)

1986-09-08

BE904368A
(en)

1986-09-08

IT8667183D0
(en)

1986-03-06

ES8802610A1
(en)

1988-09-16

JPS61207374A
(en)

1986-09-13

DK96986A
(en)

1986-09-09

GB2173788B
(en)

1988-08-10

CA1276640C
(en)

1990-11-20

US4826987A
(en)

1989-05-02

DK96986D0
(en)

1986-03-04

GR860628B
(en)

1986-06-26

NL8600596A
(en)

1986-10-01

US5157039A
(en)

1992-10-20

NZ215347A
(en)

1990-02-26

IT1221079B
(en)

1990-06-21

IE58870B1
(en)

1993-11-17

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