AU6581086A - Creación de Inventos y Patentes con Inteligencia Artificial

AU6581086A – New thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same
– Google Patents

AU6581086A – New thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same
– Google Patents
New thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same

Info

Publication number
AU6581086A

AU6581086A
AU65810/86A
AU6581086A
AU6581086A
AU 6581086 A
AU6581086 A
AU 6581086A
AU 65810/86 A
AU65810/86 A
AU 65810/86A
AU 6581086 A
AU6581086 A
AU 6581086A
AU 6581086 A
AU6581086 A
AU 6581086A
Authority
AU
Australia
Prior art keywords
processes
preparation
pharmaceutical composition
same
thiazole compounds
Prior art date
1985-12-05
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU65810/86A
Other versions

AU601911B2
(en

Inventor
Takashi Manabe
Hiroshi Matsuda
Masaaki Matsuo
Ikuo Ueda
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Fujisawa Pharmaceutical Co Ltd

Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1985-12-05
Filing date
1986-11-28
Publication date
1987-06-11

1986-11-28
Application filed by Fujisawa Pharmaceutical Co Ltd
filed
Critical
Fujisawa Pharmaceutical Co Ltd

1987-06-11
Publication of AU6581086A
publication
Critical
patent/AU6581086A/en

1990-09-20
Application granted
granted
Critical

1990-09-20
Publication of AU601911B2
publication
Critical
patent/AU601911B2/en

2006-11-28
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom

C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom

C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings

C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P11/00—Drugs for disorders of the respiratory system

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P27/00—Drugs for disorders of the senses

A61P27/16—Otologicals

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P37/00—Drugs for immunological or allergic disorders

A61P37/08—Antiallergic agents

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00

C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

AU65810/86A
1985-12-05
1986-11-28
New thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same

Ceased

AU601911B2
(en)

Applications Claiming Priority (4)

Application Number
Priority Date
Filing Date
Title

JP27446585

1985-12-05

JP60-274465

1985-12-05

JP61-236879

1986-10-03

JP23687986

1986-10-03

Publications (2)

Publication Number
Publication Date

AU6581086A
true

AU6581086A
(en)

1987-06-11

AU601911B2

AU601911B2
(en)

1990-09-20

Family
ID=26532916
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU65810/86A
Ceased

AU601911B2
(en)

1985-12-05
1986-11-28
New thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same

Country Status (20)

Country
Link

US
(1)

US4742057A
(en)

EP
(1)

EP0224919B1
(en)

JP
(1)

JPS63225374A
(en)

KR
(1)

KR890003356B1
(en)

CN
(1)

CN1017707B
(en)

AR
(1)

AR242574A1
(en)

AT
(1)

ATE66224T1
(en)

AU
(1)

AU601911B2
(en)

CA
(1)

CA1311754C
(en)

DE
(1)

DE3680877D1
(en)

DK
(1)

DK575386A
(en)

ES
(1)

ES2040206T3
(en)

FI
(1)

FI87212C
(en)

GR
(1)

GR3002606T3
(en)

HU
(1)

HU207315B
(en)

IE
(1)

IE59624B1
(en)

IL
(1)

IL80729A0
(en)

NO
(1)

NO165397C
(en)

PH
(1)

PH23004A
(en)

SU
(2)

SU1597102A3
(en)

Cited By (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

AU583607B2
(en)

1985-04-10
1989-05-04
H. Lundbeck A/S
Indole derivatives

Families Citing this family (23)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB8726763D0
(en)

1987-11-16
1987-12-23
Fujisawa Pharmaceutical Co
Thiazole compounds

DK733788A
(en)

1988-01-14
1989-07-15
Fujisawa Pharmaceutical Co

INDOLYL PIPERIDE INGREDIENTS AND PROCEDURES FOR PREPARING THEREOF

GB8908085D0
(en)

1989-04-11
1989-05-24
Lundbeck & Co As H
New therapeutic use

US5238945A
(en)

1989-04-11
1993-08-24
H. Lundbeck A/S
Method of treating psychoses

US5643784A
(en)

1990-12-04
1997-07-01
H, Lundbeck A/S
Indan derivatives

NZ243065A
(en)

1991-06-13
1995-07-26
Lundbeck & Co As H
Piperidine derivatives and pharmaceutical compositions

JP2600644B2
(en)

1991-08-16
1997-04-16
藤沢薬品工業株式会社

Thiazolyl benzofuran derivative

DK78692D0
(en)

1992-06-12
1992-06-12
Lundbeck & Co As H

DIMER PIPERIDINE AND PIPERAZINE DERIVATIVES

US5457099A
(en)

1992-07-02
1995-10-10
Sawai Pharmaceutical Co., Ltd.
Carbostyril derivatives and antiallergic agent

JP3719612B2
(en)

1993-06-14
2005-11-24
塩野義製薬株式会社

Urea derivatives containing heterocycles

US5521196A
(en)

1994-10-05
1996-05-28
Eli Lilly And Company
5-HT1F agonists for the treatment of migraine

US5521197A
(en)

1994-12-01
1996-05-28
Eli Lilly And Company
3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT1F agonists

CA2215322A1
(en)

1995-03-20
1996-09-26
Stephen Warren Kaldor
5-substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)-and 3-(piperidin-4-yl)-1h-indoles: new 5-ht1f agonists

CZ168896A3
(en)

1995-06-27
1997-01-15
Egyt Gyogyszervegyeszeti Gyar
Oxaindene derivatives and process for preparing thereof

ES2165274B1
(en)

1999-06-04
2003-04-01
Almirall Prodesfarma Sa

NEW DERIVATIVES OF INDOLILPIPERIDINE AS ANTIHISTAMINIC AND ANTIALERGIC AGENTS.

ES2172436B1
(en)

2000-10-31
2004-01-16
Almirall Prodesfarma Sa

INDOLILPIPERIDINE DERIVATIVES AS ANTIHISTAMINIC AND ANTIALERGIC AGENTS.

ES2201907B1
(en)

2002-05-29
2005-06-01
Almirall Prodesfarma, S.A.

NEW DERIVATIVES OF INDOLILPIPERIDINE AS POWERFUL ANTIHISTAMINIC AND ANTIALERGIC AGENTS.

GB0328909D0
(en)

2003-12-12
2004-01-14
Syngenta Participations Ag
Chemical compounds

AU2006306497A1
(en)

2005-10-24
2007-05-03
Janssen Pharmaceutica, N.V.
3-piperidin-4-yl-indole ORL-1 receptor modulators

LT3027603T
(en)

2013-08-02
2018-08-10
Pfizer Inc.
Heterobicycloaryl rorc2 inhibitors and methods of use thereof

US20150315179A1
(en)

2014-05-02
2015-11-05
Torrey Pines Institute For Molecular Studies
Compounds and methods of treating neurological disorders

JP2018510131A
(en)

2015-01-30
2018-04-12
ファイザー・インク

RORC2 sulfonamide substituted indole modulator and method of use thereof

EP3250570A1
(en)

2015-01-30
2017-12-06
Pfizer Inc
Methoxy-substituted pyrrolopyridine modulators of rorc2 and methods of use thereof

Family Cites Families (14)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US3361759A
(en)

1963-10-07
1968-01-02
Upjohn Co
3-(2-pyrrolidinyl)-indoles and method of preparation

FR2193584B1
(en)

1972-07-28
1975-08-08
Roussel Uclaf

US3873559A
(en)

1973-03-30
1975-03-25
Squibb & Sons Inc
Heterocyclic carboxamido thiazolinyl indoles

DE2322470A1
(en)

1973-05-04
1974-11-21
Boehringer Sohn Ingelheim

NEW INDOLYL-PIPERIDINO- (OR 1,2,5,6TETRAHYDRO-PYRIDYL-) BUTYROPHENONE AND METHOD FOR THEIR PRODUCTION

IL48508A
(en)

1974-12-09
1979-10-31
Roussel Uclaf
Pharmaceutical compositions comprising piperidylindole derivatives

FR2349331A1
(en)

1976-04-30
1977-11-25
Roussel Uclaf

NEW DERIVATIVES OF 2,3 DIHYDRO A / 4- (3-INDOLYL) 1-PIPERIDINYL / METHYL 1,4-BENZODIOXIN-2-METHANOL, A PROCESS FOR THEIR PREPARATION AND APPLICATION AS MEDICINAL PRODUCTS

FR2362628A1
(en)

1976-08-26
1978-03-24
Roussel Uclaf

NEW DERIVATIVES OF PIPERIDYL-INDOLE AND THEIR SALTS, METHOD OF PREPARATION AND APPLICATION AS MEDICINAL PRODUCTS

FR2426465B1
(en)

1978-01-16
1983-04-29
Roussel Uclaf

FR2421899A1
(en)

1978-01-16
1979-11-02
Roussel Uclaf

NEW TETRAHYDROPYRIDINYL-INDOLE DERIVATIVES AND THEIR SALTS, THE PREPARATION PROCESS AND THE MEDICINAL APPLICATION OF THESE NEW PRODUCTS

FR2460947A1
(en)

1979-07-13
1981-01-30
Roussel Uclaf

NOVEL N-SUBSTITUTED TETRAHYDROPYRIDINYL-INDOLE DERIVATIVES, THEIR SALTS, PREPARATION METHOD, MEDICAMENT APPLICATION AND COMPOSITIONS COMPRISING SAME

US4359468A
(en)

1981-02-25
1982-11-16
Boehringer Ingelheim Ltd.
Antiallergic N-[4-(indolyl)-piperidino-alkyl]-benzimidazolones

FR2533924A1
(en)

1982-10-05
1984-04-06
Roussel Uclaf

NOVEL 4- (1H-INDOL-3-YL) A-METHYL PIPERIDINE-1-ETHANOL DERIVATIVES, THEIR SALTS, THE PREPARATION PROCESS, THE MEDICINAL APPLICATION AND THE COMPOSITIONS COMPRISING THE SAME

US4548939A
(en)

1984-10-01
1985-10-22
Janssen Pharmaceutica N. V.
1H-Indol-3-yl containing 1,3-dimethyl-1H-purine-2,6-diones

IE58370B1
(en)

1985-04-10
1993-09-08
Lundbeck & Co As H
Indole derivatives

1986

1986-11-20
US
US06/932,592
patent/US4742057A/en
not_active
Expired – Fee Related

1986-11-23
IL
IL80729A
patent/IL80729A0/en
not_active
IP Right Cessation

1986-11-25
CA
CA000523787A
patent/CA1311754C/en
not_active
Expired – Fee Related

1986-11-25
IE
IE310386A
patent/IE59624B1/en
not_active
IP Right Cessation

1986-11-28
DK
DK575386A
patent/DK575386A/en
not_active
Application Discontinuation

1986-11-28
AU
AU65810/86A
patent/AU601911B2/en
not_active
Ceased

1986-11-28
PH
PH34537A
patent/PH23004A/en
unknown

1986-12-01
FI
FI864879A
patent/FI87212C/en
not_active
IP Right Cessation

1986-12-03
EP
EP86116829A
patent/EP0224919B1/en
not_active
Expired – Lifetime

1986-12-03
DE
DE8686116829T
patent/DE3680877D1/en
not_active
Expired – Fee Related

1986-12-03
AT
AT86116829T
patent/ATE66224T1/en
not_active
IP Right Cessation

1986-12-03
ES
ES198686116829T
patent/ES2040206T3/en
not_active
Expired – Lifetime

1986-12-04
JP
JP61289450A
patent/JPS63225374A/en
active
Pending

1986-12-04
NO
NO864879A
patent/NO165397C/en
unknown

1986-12-04
HU
HU865027A
patent/HU207315B/en
not_active
IP Right Cessation

1986-12-04
SU
SU864028638A
patent/SU1597102A3/en
active

1986-12-05
CN
CN86108205A
patent/CN1017707B/en
not_active
Expired

1986-12-05
KR
KR1019860010414A
patent/KR890003356B1/en
not_active
IP Right Cessation

1986-12-05
AR
AR86306103A
patent/AR242574A1/en
active

1988

1988-07-12
SU
SU884356048A
patent/SU1753948A3/en
active

1991

1991-08-26
GR
GR91400945T
patent/GR3002606T3/en
unknown

Cited By (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

AU583607B2
(en)

1985-04-10
1989-05-04
H. Lundbeck A/S
Indole derivatives

Also Published As

Publication number
Publication date

FI864879A
(en)

1987-06-06

AU601911B2
(en)

1990-09-20

NO165397C
(en)

1991-02-06

DK575386D0
(en)

1986-11-28

IE59624B1
(en)

1994-03-09

ES2040206T3
(en)

1993-10-16

CN1017707B
(en)

1992-08-05

CA1311754C
(en)

1992-12-22

KR890003356B1
(en)

1989-09-19

AR242574A1
(en)

1993-04-30

IE863103L
(en)

1987-06-05

PH23004A
(en)

1989-02-24

US4742057A
(en)

1988-05-03

FI87212C
(en)

1992-12-10

EP0224919A2
(en)

1987-06-10

ATE66224T1
(en)

1991-08-15

EP0224919A3
(en)

1988-03-30

KR870006039A
(en)

1987-07-08

IL80729A0
(en)

1987-02-27

FI87212B
(en)

1992-08-31

NO165397B
(en)

1990-10-29

HUT46320A
(en)

1988-10-28

NO864879D0
(en)

1986-12-04

JPS63225374A
(en)

1988-09-20

FI864879A0
(en)

1986-12-01

SU1753948A3
(en)

1992-08-07

SU1597102A3
(en)

1990-09-30

NO864879L
(en)

1987-06-09

DK575386A
(en)

1987-06-06

GR3002606T3
(en)

1993-01-25

DE3680877D1
(en)

1991-09-19

CN86108205A
(en)

1987-06-17

EP0224919B1
(en)

1991-08-14

HU207315B
(en)

1993-03-29

Información de contacto