AU7263081A – 3-aminopropoxyphenyl derivatives and their use as pharmaceutical compounds
– Google Patents
AU7263081A – 3-aminopropoxyphenyl derivatives and their use as pharmaceutical compounds
– Google Patents
3-aminopropoxyphenyl derivatives and their use as pharmaceutical compounds
Info
Publication number
AU7263081A
AU7263081A
AU72630/81A
AU7263081A
AU7263081A
AU 7263081 A
AU7263081 A
AU 7263081A
AU 72630/81 A
AU72630/81 A
AU 72630/81A
AU 7263081 A
AU7263081 A
AU 7263081A
AU 7263081 A
AU7263081 A
AU 7263081A
Authority
AU
Australia
Prior art keywords
pharmaceutical compounds
aminopropoxyphenyl
derivatives
aminopropoxyphenyl derivatives
pharmaceutical
Prior art date
1980-07-09
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU72630/81A
Other versions
AU547666B2
(en
Inventor
Richard Berthold
William John Louis
Andre Stoll
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1980-07-09
Filing date
1981-07-07
Publication date
1982-01-14
1981-07-07
Application filed by Individual
filed
Critical
Individual
1982-01-14
Publication of AU7263081A
publication
Critical
patent/AU7263081A/en
1985-10-31
Application granted
granted
Critical
1985-10-31
Publication of AU547666B2
publication
Critical
patent/AU547666B2/en
2001-07-07
Anticipated expiration
legal-status
Critical
Status
Expired
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
A61K31/00—Medicinal preparations containing organic active ingredients
A61K31/16—Amides, e.g. hydroxamic acids
A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
A61K31/00—Medicinal preparations containing organic active ingredients
A61K31/13—Amines
A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
A61K31/00—Medicinal preparations containing organic active ingredients
A61K31/275—Nitriles; Isonitriles
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
A61K31/00—Medicinal preparations containing organic active ingredients
A61K31/33—Heterocyclic compounds
A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P25/00—Drugs for disorders of the nervous system
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P25/00—Drugs for disorders of the nervous system
A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P25/00—Drugs for disorders of the nervous system
A61P25/04—Centrally acting analgesics, e.g. opioids
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P27/00—Drugs for disorders of the senses
A61P27/02—Ophthalmic agents
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P9/00—Drugs for disorders of the cardiovascular system
A61P9/08—Vasodilators for multiple indications
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P9/00—Drugs for disorders of the cardiovascular system
A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P9/00—Drugs for disorders of the cardiovascular system
A61P9/12—Antihypertensives
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
C07C217/28—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having one amino group and at least two singly-bound oxygen atoms, with at least one being part of an etherified hydroxy group, bound to the carbon skeleton, e.g. ethers of polyhydroxy amines
C07C217/30—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having one amino group and at least two singly-bound oxygen atoms, with at least one being part of an etherified hydroxy group, bound to the carbon skeleton, e.g. ethers of polyhydroxy amines having the oxygen atom of at least one of the etherified hydroxy groups further bound to a carbon atom of a six-membered aromatic ring
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C255/00—Carboxylic acid nitriles
C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C255/00—Carboxylic acid nitriles
C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
C07C255/53—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and hydroxy groups bound to the carbon skeleton
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C43/00—Ethers; Compounds having groups, groups or groups
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
C07D303/02—Compounds containing oxirane rings
C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
C07D303/18—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
C07D303/20—Ethers with hydroxy compounds containing no oxirane rings
C07D303/24—Ethers with hydroxy compounds containing no oxirane rings with polyhydroxy compounds
AU72630/81A
1980-07-09
1981-07-07
3-aminopropoxyphenyl derivatives and their use as pharmaceutical compounds
Expired
AU547666B2
(en)
Applications Claiming Priority (12)
Application Number
Priority Date
Filing Date
Title
GB8022412
1980-07-09
GB8022412
1980-07-09
CH5999/80
1980-08-07
CH599980
1980-08-07
CH824780
1980-11-06
CH824580
1980-11-06
CH8245/80
1980-11-06
CH8247/80
1980-11-06
GB8041155
1980-12-23
GB8041155
1980-12-23
GB8104585
1981-02-13
GB8104585
1981-02-13
Publications (2)
Publication Number
Publication Date
AU7263081A
true
AU7263081A
(en)
1982-01-14
AU547666B2
AU547666B2
(en)
1985-10-31
Family
ID=27543773
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU72630/81A
Expired
AU547666B2
(en)
1980-07-09
1981-07-07
3-aminopropoxyphenyl derivatives and their use as pharmaceutical compounds
Country Status (11)
Country
Link
US
(2)
US4816604A
(en)
AU
(1)
AU547666B2
(en)
DE
(1)
DE3125870C2
(en)
FR
(1)
FR2489316B1
(en)
GB
(1)
GB2132611B
(en)
IL
(1)
IL63245A
(en)
IT
(1)
IT1171374B
(en)
NZ
(1)
NZ197632A
(en)
PH
(1)
PH22546A
(en)
SE
(2)
SE8104236L
(en)
WO
(1)
WO1982000141A1
(en)
Families Citing this family (8)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
CA1262729A
(en)
*
1983-10-19
1989-11-07
Leo Alig
Phenoxypropanolamines
DE3907512C2
(en)
*
1989-03-08
1997-08-14
Laevosan Gmbh & Co Kg
Aryloxy-alkylamines, their preparation and medicaments containing them
US5304367A
(en)
*
1990-11-16
1994-04-19
New York University
In vivo brain imaging agent and method for diagnosis of psychiatric disorders
US5217994A
(en)
*
1991-08-09
1993-06-08
Merck & Co., Inc.
Method of inhibiting osteoclast-mediated bone resorption by administration of aminoalkyl-substituted phenyl derivatives
BR9306399A
(en)
*
1992-05-22
1998-09-15
Senju Pharma Co
Pharmaceutical composition for use in the treatment of glaucoma
EP0937030B1
(en)
*
1995-10-10
2004-03-31
William John Louis
3-amino-propoxyphenyl derivatives (i)
WO2012004549A1
(en)
2010-07-05
2012-01-12
The University Of Nottingham
Phenoxypropanol derivatives and their use in treating cardiac and cardiovascular diseases
GB201101959D0
(en)
*
2011-02-04
2011-03-23
Univ Nottingham
Novel ether linked compoundsand improved treatments for cardiac and cardiovascular disease
Family Cites Families (16)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
DE1957706C3
(en)
*
1968-11-18
1978-06-29
Pfizer Corp., Colon (Panama)
Nuclear-substituted 3-phenoxy-1-phenoxyalkylamino-propan-2-ols and drugs based on them
DE2023829C3
(en)
*
1970-05-15
1979-06-21
Pfizer Corp., Colon (Panama)
Nuclear-substituted 3-phenoxy-lphenoxyalkyl-aminopropane-2-oIe, process for their production and pharmaceuticals
AR204726A1
(en)
*
1973-01-17
1976-02-27
Ciba Geigy Ag
PROCEDURE FOR THE PREPARATION OF 1- (4- (ALKYLTHIO-ALCOXY) -PHENOXYL) -2-HYDROXY-3-ALKYLAMINOPROPANE
ZA741812B
(en)
*
1973-04-18
1975-04-30
Haessle A
New amines and process for their preparation
ZA754241B
(en)
*
1974-11-01
1976-06-30
Haessle Ab
New amines
DE2549745A1
(en)
*
1974-11-20
1976-05-26
Lipha
PROPIONIC ACIDS SUBSTITUTED BY A CHROMONYL RESIDUE AND THEIR DERIVATIVES AND USES
FR2330383A1
(en)
*
1975-11-06
1977-06-03
Synthelabo
NEW PHENOL SUBSTITUTE ETHERS, THEIR SALTS, THEIR PREPARATION AND THE MEDICINAL PRODUCTS CONTAINING THEM
DE2606140A1
(en)
*
1976-02-17
1977-08-25
Boehringer Sohn Ingelheim
NEW DERIVATIVES OF 2-PHENYL-2-HYDROXYAETHYLAMINE
DE2614875C2
(en)
*
1976-04-06
1978-06-15
Bayer Ag, 5090 Leverkusen
Process for the production of alkyl or arylthiomethylphenols
DE2645710C2
(en)
*
1976-10-09
1985-06-27
Merck Patent Gmbh, 6100 Darmstadt
Phenoxy-aminopropanols, process for their manufacture and pharmaceutical preparation
FR2368951A2
(en)
*
1976-10-27
1978-05-26
Synthelabo
Amino-hydroxypropoxy:phenyl ether cpds. – used as beta-blockers for cardiovascular disorders
JPS6022701B2
(en)
*
1977-06-02
1985-06-03
ウェルファイド株式会社
Phenoxyaminopropanol derivatives and their production method
SE7807408L
(en)
*
1978-06-30
1979-12-31
Haessle Ab
HEART ACTIVE ASSOCIATIONS
US4294966A
(en)
*
1978-07-28
1981-10-13
Ciba-Geigy Corporation
Process for inverting the configuration in optically active compounds
DE2838273A1
(en)
*
1978-09-01
1980-03-13
Bayer Ag
PROCESS FOR THE PRODUCTION OF ALKYL- OR. ARYLTHIOMETHYLPHENOLS
ZW9881A1
(en)
*
1980-06-02
1981-12-23
Hoffmann La Roche
Substituted phenoxyaminopropanol derivatives
1981
1981-07-01
DE
DE3125870A
patent/DE3125870C2/en
not_active
Expired – Fee Related
1981-07-06
FR
FR8113382A
patent/FR2489316B1/fr
not_active
Expired
1981-07-07
NZ
NZ197632A
patent/NZ197632A/en
unknown
1981-07-07
SE
SE8104236D
patent/SE8104236L/en
not_active
Application Discontinuation
1981-07-07
AU
AU72630/81A
patent/AU547666B2/en
not_active
Expired
1981-07-07
IL
IL63245A
patent/IL63245A/en
not_active
IP Right Cessation
1981-07-07
WO
PCT/CH1981/000074
patent/WO1982000141A1/en
unknown
1981-07-07
SE
SE8104236A
patent/SE457255B/en
not_active
IP Right Cessation
1981-07-07
PH
PH25876A
patent/PH22546A/en
unknown
1981-07-08
IT
IT48859/81A
patent/IT1171374B/en
active
1983
1983-09-19
GB
GB08324990A
patent/GB2132611B/en
not_active
Expired
1987
1987-03-09
US
US07/022,502
patent/US4816604A/en
not_active
Expired – Lifetime
1989
1989-03-10
US
US07/321,815
patent/US4970238A/en
not_active
Expired – Lifetime
Also Published As
Publication number
Publication date
FR2489316A1
(en)
1982-03-05
PH22546A
(en)
1988-10-17
DE3125870A1
(en)
1982-03-25
SE8104236L
(en)
1982-01-10
FR2489316B1
(en)
1985-01-18
AU547666B2
(en)
1985-10-31
US4970238A
(en)
1990-11-13
GB8324990D0
(en)
1983-10-19
SE457255B
(en)
1988-12-12
DE3125870C2
(en)
1994-09-15
GB2132611B
(en)
1985-01-16
US4816604A
(en)
1989-03-28
GB2132611A
(en)
1984-07-11
IT1171374B
(en)
1987-06-10
IL63245A
(en)
1985-06-30
IL63245A0
(en)
1981-10-30
IT8148859D0
(en)
1981-07-08
WO1982000141A1
(en)
1982-01-21
NZ197632A
(en)
1984-07-31
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Legal Events
Date
Code
Title
Description
2002-02-07
MK14
Patent ceased section 143(a) (annual fees not paid) or expired
