AU7897787A

AU7897787A – Aminopyrazinone and aminotriazinones
– Google Patents

AU7897787A – Aminopyrazinone and aminotriazinones
– Google Patents
Aminopyrazinone and aminotriazinones

Info

Publication number
AU7897787A

AU7897787A
AU78977/87A
AU7897787A
AU7897787A
AU 7897787 A
AU7897787 A
AU 7897787A
AU 78977/87 A
AU78977/87 A
AU 78977/87A
AU 7897787 A
AU7897787 A
AU 7897787A
AU 7897787 A
AU7897787 A
AU 7897787A
Authority
AU
Australia
Prior art keywords
alkyl
hydrogen
alkoxy
halogenoalkyl
alkenyl
Prior art date
1986-09-26
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU78977/87A
Other versions

AU593945B2
(en

Inventor
Beat Bohner
Willy Meyer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Novartis AG

Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1986-09-26
Filing date
1987-09-25
Publication date
1988-03-31

1987-09-25
Application filed by Ciba Geigy AG
filed
Critical
Ciba Geigy AG

1988-03-31
Publication of AU7897787A
publication
Critical
patent/AU7897787A/en

1990-02-22
Application granted
granted
Critical

1990-02-22
Publication of AU593945B2
publication
Critical
patent/AU593945B2/en

2007-09-25
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D521/00—Heterocyclic compounds containing unspecified hetero rings

A—HUMAN NECESSITIES

A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING

A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS

A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid

A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms

A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< A01N47/36—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< directly attached to at least one heterocyclic ring; Thio analogues thereof C—CHEMISTRY; METALLURGY C07—ORGANIC CHEMISTRY C07D—HETEROCYCLIC COMPOUNDS C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms C07D241/20—Nitrogen atoms C—CHEMISTRY; METALLURGY C07—ORGANIC CHEMISTRY C07D—HETEROCYCLIC COMPOUNDS C07D253/00—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings C07D253/06—1,2,4-Triazines C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members C07D253/07—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms C—CHEMISTRY; METALLURGY C07—ORGANIC CHEMISTRY C07D—HETEROCYCLIC COMPOUNDS C07D253/00—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings C07D253/06—1,2,4-Triazines C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members C07D253/07—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms C07D253/075—Two hetero atoms, in positions 3 and 5 Abstract Aminopyrazinones and aminotriazinones of the formula (I) and the salts of these compounds with amines, alkali metal or alkaline earth metal bases or quaternary ammonium bases have good pre- and post-emergent selective herbicidal and growth-regulating properties. In this formula, E is nitrogen or =CR4-, R1 is C1-C4-alkyl, R2 is hydrogen, C1-C3-alkyl, C1-C3-halogenoalkyl, C1-C3-alkoxy, C1-C3-halogenoalkoxy, C1 -C3-alkylthio, C1-C3-alkylsulfinyl, C1-C2-alkoxyethoxy, C1-C3-alkylsulfonyl, halogen or -NR5R6, R3 is hydrogen or C1-C3-alkyl and Q is a group in which R4is hydrogen, C1-C3-alkyl, C1-C3-halogenoalkyl, C1-C3-alkoxy, cyclopropyl, C1-C3-halogenoalkoxy, C1-C3-alkylthio, C2-C4-alkoxyalkyl, C3-C5-dialkoxymethyl, halogen or -NR5R6, R5 and R6 independently of one another are hydrogen or C1-C3-alkyl, X is oxygen or sulfur and A is a group in which Y is oxygen, sulfur, -CH=CH-, – NR9-or -CR10=N-, R7 is hydrogen, halogen, C1-C3-alkyl C1-C3-alkoxy, nirtro or trifluoromethyl, R8 is hydrogen, halogen, C1-C3alkyl, C1-C3-alkoxy, nitro -C 3BOND CH, or one of the groups +TR SO2NR13R14, (Z)mR15 or OSO2R18, R9 and R10 independently of one another are hydrogen, C1-C3-alkyl or C2-C4-alkenyl, R11 is hydrogen, C1-C3-alkyl, C1-C3-halogenoalkyl, C3-C6-cycloalkyl or C2-C4-alkoxyalkyl, R12 is C1-C6-alkoxy, C3-C6-alkenyloxy, C3-C6-alkenyloxy, C3-C6-alkinyloxy, C2-C6-halogenoalkoxy, C1-C4-cyanoalkoxy, C1-C6-alkylthio, C3-C6-alkenylthio, C3-C6-alkinylthio, C5-C6-cycloalkoxy, C2-C6-alkoxyalkoxy or -NR16R17, R13 is hydrogen, C1-C3-alkyl or C3-C4-alkenyl, R14 is hydrogens C1-C3-alkyl, C1-C3-cyanoalkyl or C1-C3-alkoxy, R15 is C3-C6-alkinyl,C2-C6-alkenyl, C1-C6-alkyl, C1-C 4-halogenoalkyl, C2-C4-halogenoalkenyl or C1-C4-alkyl, substituted by cyano, methoxy, ethoxy, nitro, C1-C4-alkoxycarbonyl, methylthio, ethylthio, methylsulfonyl or ethylsulfonyl; or C3-C4-alkenyl substituted by nitro, cyano, methoxy or ethoxy, R16 is hydrogen, C1-C3-alkyl or C3-C4-alkenyl, R17 is hydrogen, C1-C3-alkyl, C1-C3-cyanoalkyl or C1-C3-alkoxy, R18 is C1-C3-alkyl and C1-C3-halogenoalkyl, W is oxygen or sulfur, Z is oxygen, sulfur, -SO- or -SO2- and m is the number zero or one.

AU78977/87A
1986-09-26
1987-09-25
Aminopyrazinone and aminotriazinones

Ceased

AU593945B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

CH3871/86

1986-09-26

CH387186

1986-09-26

Publications (2)

Publication Number
Publication Date

AU7897787A
true

AU7897787A
(en)

1988-03-31

AU593945B2

AU593945B2
(en)

1990-02-22

Family
ID=4265276
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU78977/87A
Ceased

AU593945B2
(en)

1986-09-26
1987-09-25
Aminopyrazinone and aminotriazinones

Country Status (11)

Country
Link

US
(4)

US4795486A
(en)

EP
(1)

EP0262096B1
(en)

JP
(1)

JPS6391378A
(en)

AT
(1)

ATE71096T1
(en)

AU
(1)

AU593945B2
(en)

CA
(1)

CA1292738C
(en)

DE
(1)

DE3775686D1
(en)

ES
(1)

ES2037738T3
(en)

GR
(1)

GR3003528T3
(en)

IL
(1)

IL83996A
(en)

ZA
(1)

ZA877223B
(en)

Families Citing this family (26)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4795486A
(en)

*

1986-09-26
1989-01-03
Boehner Beat
Aminopyrazinones and aminotriazinones

MY136106A
(en)

*

1990-09-06
2008-08-29
Novartis Ag
Synergistic composition comprising a sulfonylurea anda thiadiazolo (3,4-a)pyridazine and method of selective weed control.

DE69709727T2
(en)

*

1996-04-23
2002-08-08
Merck & Co Inc

PARAZINON THROMBIN INHIBITORS

US5872138A
(en)

*

1996-09-13
1999-02-16
Merck & Co., Inc.
Thrombin inhibitors

US5869487A
(en)

*

1996-10-24
1999-02-09
Merck & Co., Inc.
Pyrido 3,4-B!pyrazines for use as thrombin inhibitors

US5866573A
(en)

*

1997-04-21
1999-02-02
Merck & Co., Inc.
Pyrazinone thrombin inhibitors

US6011038A
(en)

*

1997-09-05
2000-01-04
Merck & Co., Inc.
Pyrazinone thrombin inhibitors

US6087373A
(en)

*

1997-09-23
2000-07-11
Merck & Co., Inc.
Thrombin inhibitors

US6133297A
(en)

*

1997-09-30
2000-10-17
Merck & Co., Inc.
Thrombin inhibitors

US6147078A
(en)

*

1998-05-19
2000-11-14
Merck & Co., Inc.
Pyrazinone thrombin inhibitors

WO2000018762A1
(en)

*

1998-09-28
2000-04-06
Merck & Co., Inc.
Thrombin inhibitors

JP2002528543A
(en)

1998-10-30
2002-09-03
メルク エンド カムパニー インコーポレーテッド

Thrombin inhibitor

CA2348530A1
(en)

1998-10-30
2000-05-11
Merck & Co., Inc.
Thrombin inhibitors

US6239132B1
(en)

1999-04-23
2001-05-29
Merck & Co., Inc.
Thrombin inhibitors

US6664255B1
(en)

*

1999-05-19
2003-12-16
Pharmacia Corporation
Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade

US6908919B2
(en)

*

1999-05-19
2005-06-21
Pharmacia Corporation
Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade

UA58636C2
(en)

1999-06-04
2003-08-15
Мерк Енд Ко., Інк.
Pyrazinone thrombin inhibitors, pharmaceutical composition, method for treatment conditions caused by thrombus formation

WO2000074682A1
(en)

1999-06-04
2000-12-14
Merck & Co., Inc.
Thrombin inhibitors

WO2001038323A1
(en)

1999-11-23
2001-05-31
Merck & Co., Inc.
Pyrazinone thrombin inhibitors

WO2001070229A1
(en)

2000-03-23
2001-09-27
Merck & Co., Inc.
Thrombin inhibitors

US7119094B1
(en)

2000-11-20
2006-10-10
Warner-Lambert Company
Substituted polycyclic aryl and heteroarpyl pyrazinones useful for selective inhibition of the coagulation cascade

SI3578547T1
(en)

2015-02-16
2021-09-30
The University Of Queensland
Sulfonylureas and related compounds and use of same

CA3067410A1
(en)

2017-07-07
2019-01-10
Inflazome Limited
Novel sulfonamide carboxamide compounds

WO2019008029A1
(en)

*

2017-07-07
2019-01-10
Inflazome Limited
Sulfonylureas and sulfonylthioureas as nlrp3 inhibitors

US11613542B2
(en)

2017-08-15
2023-03-28
Inflazome Limited
Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors

TW201910317A
(en)

2017-08-15
2019-03-16
愛爾蘭商英弗雷佐姆有限公司

Novel compound

Family Cites Families (9)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

CA1330438C
(en)

*

1980-07-17
1994-06-28
Willy Meyer
N-phenylsulfonyl-n’-pyrimidinyl-and-triazinylureas

US4443245A
(en)

*

1981-07-13
1984-04-17
Ciba-Geigy Corporation
N-Phenylsulfonyl-N’-triazinylureas

US4612037A
(en)

*

1982-05-28
1986-09-16
Ciba-Geigy Corporation
Novel sulfonylureas and sulfonylthioureas, and method of use thereof as herbicides and/or growth regulators

DE3479213D1
(en)

*

1983-05-16
1989-09-07
Ciba Geigy Ag
Herbicidally active and plant growth regulating pyrimidine derivatives, their preparation and use

AU576868B2
(en)

*

1984-06-11
1988-09-08
E.I. Du Pont De Nemours And Company
Thiophene and pyridine sulfonamides

US4659369A
(en)

*

1984-08-27
1987-04-21
E. I. Du Pont De Nemours And Company
Herbicidal acetals and ketals

US4690705A
(en)

*

1984-11-30
1987-09-01
E. I. Du Pont De Nemours And Company
Herbicidal sulfonamides

US4795486A
(en)

*

1986-09-26
1989-01-03
Boehner Beat
Aminopyrazinones and aminotriazinones

US4802908A
(en)

*

1987-01-22
1989-02-07
E. I. Du Pont De Nemours And Company
Herbicidal 2-(1H)-pyrazinones

1987

1987-09-21
US
US07/099,036
patent/US4795486A/en
not_active
Expired – Fee Related

1987-09-21
EP
EP87810545A
patent/EP0262096B1/en
not_active
Expired – Lifetime

1987-09-21
DE
DE8787810545T
patent/DE3775686D1/en
not_active
Expired – Lifetime

1987-09-21
ES
ES198787810545T
patent/ES2037738T3/en
not_active
Expired – Lifetime

1987-09-21
AT
AT87810545T
patent/ATE71096T1/en
active

1987-09-23
IL
IL83996A
patent/IL83996A/en
not_active
IP Right Cessation

1987-09-24
CA
CA000547731A
patent/CA1292738C/en
not_active
Expired – Lifetime

1987-09-25
ZA
ZA877223A
patent/ZA877223B/en
unknown

1987-09-25
AU
AU78977/87A
patent/AU593945B2/en
not_active
Ceased

1987-09-26
JP
JP62242411A
patent/JPS6391378A/en
active
Pending

1988

1988-10-21
US
US07/260,643
patent/US4871853A/en
not_active
Expired – Fee Related

1989

1989-07-25
US
US07/384,956
patent/US4920223A/en
not_active
Expired – Fee Related

1989-08-15
US
US07/394,389
patent/US4940482A/en
not_active
Expired – Fee Related

1992

1992-01-08
GR
GR910402042T
patent/GR3003528T3/el
unknown

Also Published As

Publication number
Publication date

GR3003528T3
(en)

1993-03-16

CA1292738C
(en)

1991-12-03

IL83996A0
(en)

1988-02-29

IL83996A
(en)

1992-03-29

ES2037738T3
(en)

1993-07-01

ZA877223B
(en)

1988-03-28

DE3775686D1
(en)

1992-02-13

US4871853A
(en)

1989-10-03

US4940482A
(en)

1990-07-10

US4920223A
(en)

1990-04-24

JPS6391378A
(en)

1988-04-22

US4795486A
(en)

1989-01-03

EP0262096A1
(en)

1988-03-30

ATE71096T1
(en)

1992-01-15

AU593945B2
(en)

1990-02-22

EP0262096B1
(en)

1992-01-02

Similar Documents

Publication
Publication Date
Title

AU7897787A
(en)

1988-03-31

Aminopyrazinone and aminotriazinones

IL69225A
(en)

1988-06-30

N-1,2-benzoxathiin-8-ylsulfonyl-n'-pyrimidinyl and-n'-triazinylureas,their preparation and their use as herbicides

AU591000B2
(en)

1989-11-23

Phenylsulfonyl derivatives as intermediates in herbicide manufacture

MY131297A
(en)

2007-08-30

Herbicides

WO2001077107A8
(en)

2003-02-13

Oxazole derivatives and their uses as tyrosine kinase inhibitors

IL66319A0
(en)

1982-11-30

N-phenylsulfonyl-n'-pyrimidinyl and-triazinylureas,their production and their use as herbicides and plant growth regulants

AU2002212598A1
(en)

2002-04-02

Pyridinone and pyridinethione derivatives having hiv inhibiting properties

CA2247167A1
(en)

1997-08-28

2-hetaroylcyclohexane-1,3-diones

ZA843522B
(en)

1984-12-24

Fused n-phenylsulfonyl-n'-pyrimidinylureas and n-phenylsulfonyl-n'-triazinylureas

ES2019163A6
(en)

1991-06-01

Imidazole derivatives and their use as hypercholesterolemia and hyperlipoproteinemia agents

AU5595490A
(en)

1990-11-29

Antispasmodic agents

MY129992A
(en)

2007-05-31

Benzanilide herbicides and process for the preparation thereof

AU8866482A
(en)

1983-03-31

Oxazolo- thiazolo- imidazolo (5,4-b) pyridines

IL104613A
(en)

1997-06-10

4-benzoylisoxazole herbicides, process for preparation thereof and compositions containing them

ATE108447T1
(en)

1994-07-15

SULFONYL UREAS AS HERBICIDES.

JPH0587510B2
(en)

1993-12-16

TH10189EX
(en)

1991-12-01

Acid derivatives (chemical formulas) with fluorine substituting groups

TH10189A
(en)

1991-12-01

Acid derivatives (chemical formulas) with fluorine substituting groups

Download PDF in English

None