AU1297083A - Creation of Inventions and Patents with Artificial Intelligence

AU1297083A – Cycloalka(c)pyrrolcarboxylates
– Google Patents

AU1297083A – Cycloalka(c)pyrrolcarboxylates
– Google Patents
Cycloalka(c)pyrrolcarboxylates

Info

Publication number
AU1297083A

AU1297083A
AU12970/83A
AU1297083A
AU1297083A
AU 1297083 A
AU1297083 A
AU 1297083A
AU 12970/83 A
AU12970/83 A
AU 12970/83A
AU 1297083 A
AU1297083 A
AU 1297083A
AU 1297083 A
AU1297083 A
AU 1297083A
Authority
AU
Australia
Prior art keywords
pyrrolcarboxylates
cycloalka
Prior art date
1982-03-30
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU12970/83A
Other versions

AU560124B2
(en

Inventor
Reinhard Becker
Rolf Geiger
Rainer Henning
Volker Teetz
Hansjorg Urbach
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Hoechst AG

Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1982-03-30
Filing date
1983-03-29
Publication date
1983-10-06

1983-03-29
Application filed by Hoechst AG
filed
Critical
Hoechst AG

1983-10-06
Publication of AU1297083A
publication
Critical
patent/AU1297083A/en

1987-04-02
Application granted
granted
Critical

1987-04-02
Publication of AU560124B2
publication
Critical
patent/AU560124B2/en

2003-03-29
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom

C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring

C07D209/04—Indoles; Hydrogenated indoles

C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring

C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07K—PEPTIDES

C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof

C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link

C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2

C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P9/00—Drugs for disorders of the cardiovascular system

A61P9/12—Antihypertensives

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom

C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring

C07D209/44—Iso-indoles; Hydrogenated iso-indoles

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom

C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring

C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems

C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring

C07D217/24—Oxygen atoms

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES

A61K38/00—Medicinal preparations containing peptides

AU12970/83A
1982-03-30
1983-03-29
Cycloalka(c)pyrrolcarboxylates

Ceased

AU560124B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

DE19823211676

DE3211676A1
(en)

1982-03-30
1982-03-30

NEW DERIVATIVES OF CYCLOALKA (C) PYRROL CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF, THEIR SUBSTANCES AND THE USE THEREOF AND NEW CYCLOALKA (C) PYRROL CARBONIC ACIDS AS THE INTERMEDIATE LEVELS AND METHODS

DE32116764

1982-03-30

Publications (2)

Publication Number
Publication Date

AU1297083A
true

AU1297083A
(en)

1983-10-06

AU560124B2

AU560124B2
(en)

1987-04-02

Family
ID=6159702
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU12970/83A
Ceased

AU560124B2
(en)

1982-03-30
1983-03-29
Cycloalka(c)pyrrolcarboxylates

Country Status (17)

Country
Link

EP
(1)

EP0090362A3
(en)

JP
(1)

JPS58177967A
(en)

KR
(1)

KR840004069A
(en)

AU
(1)

AU560124B2
(en)

CA
(1)

CA1198118A
(en)

DE
(1)

DE3211676A1
(en)

DK
(1)

DK144783A
(en)

ES
(2)

ES521041A0
(en)

FI
(1)

FI831049L
(en)

GR
(1)

GR78157B
(en)

HU
(1)

HU193876B
(en)

IL
(1)

IL68267A
(en)

NO
(2)

NO831168L
(en)

NZ
(1)

NZ203719A
(en)

PH
(1)

PH19003A
(en)

PT
(1)

PT76472B
(en)

ZA
(1)

ZA832229B
(en)

Families Citing this family (44)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

DE3226768A1
(en)

1981-11-05
1983-05-26
Hoechst Ag, 6230 Frankfurt

DERIVATIVES OF CIS, ENDO-2-AZABICYCLO- (3.3.0) -OCTAN-3-CARBONIC ACID, METHOD FOR THE PRODUCTION THEREOF, THE MEANS CONTAINING THEM AND THE USE THEREOF

GR78413B
(en)

1981-12-29
1984-09-27
Hoechst Ag

DE3246503A1
(en)

1982-12-16
1984-06-20
Hoechst Ag, 6230 Frankfurt

DERIVATIVES OF CIS, ENDO-2-AZABICYCLO- (5.3.0) -DECAN-3-CARBONIC ACID, METHOD FOR THE PRODUCTION THEREOF, THESE AGENTS AND THE USE THEREOF

US5175306A
(en)

1983-01-31
1992-12-29
Hoechst Aktiengesellschaft
Process for the resolution of racemates of optically active bicyclic imino-α-carboxylic esters

DE3303344A1
(en)

1983-02-02
1984-08-02
Hoechst Ag, 6230 Frankfurt

METHOD FOR PRODUCING N-ALKYLATED AMINO ACIDS AND THEIR ESTERS

DK156484A
(en)

1983-03-16
1984-09-17
Usv Pharma Corp

AMINO ACID DERIVATIVES

FR2546886B2
(en)

1983-06-06
1986-05-16
Adir

DERIVATIVES OF ISOINDOLEDICARBOXYLIC ACIDS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

DE3333454A1
(en)

1983-09-16
1985-04-11
Hoechst Ag, 6230 Frankfurt

METHOD FOR PRODUCING N-ALKYLATED DIPEPTIDES AND THEIR ESTERS

DE3333455A1
(en)

1983-09-16
1985-04-11
Hoechst Ag, 6230 Frankfurt

METHOD FOR PRODUCING N-ALKYLATED DIPEPTIDES AND THEIR ESTERS

DE3410732A1
(en)

1984-03-23
1985-09-26
Hoechst Ag, 6230 Frankfurt

METHOD FOR TREATING GLAUCOMA

US5684016A
(en)

1984-04-12
1997-11-04
Hoechst Aktiengesellschaft
Method of treating cardiac insufficiency

DE3413710A1
(en)

1984-04-12
1985-10-24
Hoechst Ag, 6230 Frankfurt

METHOD FOR TREATING HEART INSUFFICIENCY

AU581919B2
(en)

1984-07-30
1989-03-09
Schering Corporation
Process for the preparation of cis, endooctahydrocyclopenta (b) pyrrole-2-carboxylate

DE3431541A1
(en)

1984-08-28
1986-03-06
Hoechst Ag, 6230 Frankfurt

CIS, ENDO-2-AZABICYCLOALKAN-3-CARBONIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AND INTERMEDIATE PRODUCTS IN THEIR PRODUCTION

US5231080A
(en)

1985-10-15
1993-07-27
Hoechst Aktiengesellschaft
Method for the treatment of atherosclerosis, thrombosis, and peripheral vessel disease

US5231084A
(en)

1986-03-27
1993-07-27
Hoechst Aktiengesellschaft
Compounds having a cognition adjuvant action, agents containing them, and the use thereof for the treatment and prophylaxis of cognitive dysfuncitons

DE3633496A1
(en)

1986-10-02
1988-04-14
Hoechst Ag

COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITORS WITH CALCIUMANTAGONISTS AND THEIR USE IN MEDICINAL PRODUCTS

DE3639879A1
(en)

1986-11-21
1988-06-01
Hoechst Ag

METHOD FOR PRODUCING MONO, BI AND TRICYCLIC AMINO ACIDS, INTERMEDIATE PRODUCTS OF THIS METHOD, AND A METHOD FOR PRODUCING THE SAME

DE3722007A1
(en)

1987-07-03
1989-01-12
Hoechst Ag

METHOD FOR PRODUCING BICYCLIC AMINOCARBONIC ACIDS, INTERMEDIATE PRODUCTS OF THIS METHOD AND THE USE THEREOF

JPH0278659A
(en)

1988-09-12
1990-03-19
Shionogi & Co Ltd
Compound of azabicycloalkanes

DE3839127A1
(en)

1988-11-19
1990-05-23
Hoechst Ag

PYRROLIDONE-2-CARBONIC ACID DERIVATIVES WITH PSYCHOTROPER EFFECT

DD284030A5
(en)

1988-11-24
1990-10-31
Hoechst Ag,De

PROCESS FOR THE PREPARATION OF PEPTIDES WITH BRADYKININ-ANTAGONISTIC EFFECT

LT3872B
(en)

1993-12-06
1996-04-25
Hoechst Ag
Novel peptides and pharmaceutical compositions containing them

EP0796855B1
(en)

1996-03-20
2002-02-06
Hoechst Aktiengesellschaft
Inhibitors of bone resorption and vitronectin receptor antagonists

FR2746394B1
(en)

1996-03-20
1998-05-29
Roussel Uclaf

NOVEL TRICYCLIC COMPOUNDS, THEIR PREPARATION PROCESS, AND INTERMEDIATES THEREOF, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

CN1133649C
(en)

1996-10-18
2004-01-07
沃泰克斯药物股份有限公司
Inhibitors of serine proteases, particularly hepatitis C virus NS3 protease

DE19653647A1
(en)

1996-12-20
1998-06-25
Hoechst Ag

Vitronectin receptor antagonists, their preparation and their use

DE19741235A1
(en)

1997-09-18
1999-03-25
Hoechst Marion Roussel De Gmbh

Novel imidazolidine derivatives, their preparation, their use and pharmaceutical compositions containing them

DE19741873A1
(en)

1997-09-23
1999-03-25
Hoechst Marion Roussel De Gmbh

New 5-ring heterocycles, their preparation, their use and pharmaceutical preparations containing them

DE19751251A1
(en)

1997-11-19
1999-05-20
Hoechst Marion Roussel De Gmbh

Substituted imidazolidine derivatives, their manufacture, their use and pharmaceutical preparations containing them

DE19821483A1
(en)

1998-05-14
1999-11-18
Hoechst Marion Roussel De Gmbh
New imidazolidine derivatives useful as leukocyte adhesion and migration inhibitors and/or VLA-4 receptor antagonists for treating E.G. inflammatory and allergic disorders

SV2003000617A
(en)

2000-08-31
2003-01-13
Lilly Co Eli

INHIBITORS OF PROTEASA PEPTIDOMIMETICA REF. X-14912M

AR045596A1
(en)

2003-09-05
2005-11-02
Vertex Pharma

INHIBITORS OF SERINE PROTEASES IN PARTICULAR HCV PROTEASA NS3-NS4A

WO2007022459A2
(en)

2005-08-19
2007-02-22
Vertex Pharmaceuticals Incorporated
Processes and intermediates

US8399615B2
(en)

2005-08-19
2013-03-19
Vertex Pharmaceuticals Incorporated
Processes and intermediates

AR055395A1
(en)

2005-08-26
2007-08-22
Vertex Pharma

INHIBITING COMPOUNDS OF THE ACTIVITY OF SERINA PROTEASA NS3-NS4A OF HEPATITIS C VIRUS

US7964624B1
(en)

2005-08-26
2011-06-21
Vertex Pharmaceuticals Incorporated
Inhibitors of serine proteases

AU2007217355B2
(en)

2006-02-27
2012-06-21
Vertex Pharmaceuticals Incorporated
Co-crystals comprising VX-950 and pharmaceutical compositions comprising the same

BRPI0709567A2
(en)

2006-03-16
2011-07-12
Vertex Pharma

deuterated hepatitis c protease inhibitors

KR20090115970A
(en)

2007-02-27
2009-11-10
버텍스 파마슈티칼스 인코포레이티드
Co-crystals and pharmaceutical compositions comprising the same

CA2679426A1
(en)

2007-02-27
2008-09-04
Luc Farmer
Inhibitors of serine proteases

JP5443360B2
(en)

2007-08-30
2014-03-19
バーテックスファーマシューティカルズインコーポレイテッド

Co-crystal and pharmaceutical composition containing the same

EP2307419B1
(en)

2008-06-24
2013-11-06
Codexis, Inc.
Biocatalytic processes for the preparation of substantially stereomerically pure fused bicyclic proline compounds

JP5829529B2
(en)

2011-08-29
2015-12-09
日本曹達株式会社

Optically active quaternary ammonium salt and method for producing optically active compound

Family Cites Families (7)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

IL58849A
(en)

1978-12-11
1983-03-31
Merck & Co Inc
Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them

FR2487829A2
(en)

1979-12-07
1982-02-05
Science Union & Cie

NOVEL SUBSTITUTED IMINO ACIDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS AN ENZYME INHIBITOR

EP0050800B2
(en)

1980-10-23
1995-06-07
Schering Corporation
Carboxyalkyl dipeptides, processes for their production and pharmaceutical compositions containing them

DE3276311D1
(en)

1981-02-17
1987-06-19
Warner Lambert Co
Octahydro-2-(omega-mercaptoalkanoyl)3-oxo-1h-isoindole-1-carboxylic acids and esters

ZA826022B
(en)

1981-08-21
1983-08-31
Univ Miami
Novel complex amido and imido derivatives of carboxyalkyl peptides and thioethers and ethers of peptides

EP0081094A1
(en)

1981-11-12
1983-06-15
Merck & Co. Inc.
Substituted omega-amino-carboxymethyldipeptide antihypertensive agents

DE3360065D1
(en)

1982-03-08
1985-03-28
Schering Corp
Carboxyalkyl dipeptides, processes for their production and pharmaceutical compositions containing them

1982

1982-03-30
DE
DE19823211676
patent/DE3211676A1/en
not_active
Withdrawn

1983

1983-03-24
EP
EP83102961A
patent/EP0090362A3/en
not_active
Withdrawn

1983-03-28
NZ
NZ203719A
patent/NZ203719A/en
unknown

1983-03-28
FI
FI831049A
patent/FI831049L/en
not_active
Application Discontinuation

1983-03-28
KR
KR1019830001244A
patent/KR840004069A/en
not_active
Application Discontinuation

1983-03-28
GR
GR70912A
patent/GR78157B/el
unknown

1983-03-28
ES
ES521041A
patent/ES521041A0/en
active
Granted

1983-03-29
PH
PH28723A
patent/PH19003A/en
unknown

1983-03-29
HU
HU831064A
patent/HU193876B/en
unknown

1983-03-29
NO
NO831168A
patent/NO831168L/en
unknown

1983-03-29
PT
PT76472A
patent/PT76472B/en
unknown

1983-03-29
JP
JP58051780A
patent/JPS58177967A/en
active
Pending

1983-03-29
AU
AU12970/83A
patent/AU560124B2/en
not_active
Ceased

1983-03-29
CA
CA000424770A
patent/CA1198118A/en
not_active
Expired

1983-03-29
ZA
ZA832229A
patent/ZA832229B/en
unknown

1983-03-29
DK
DK144783A
patent/DK144783A/en
not_active
Application Discontinuation

1983-03-30
IL
IL68267A
patent/IL68267A/en
unknown

1983-04-22
ES
ES521741A
patent/ES8402570A1/en
not_active
Expired

1983-11-25
NO
NO834352A
patent/NO834352L/en
unknown

Also Published As

Publication number
Publication date

PH19003A
(en)

1985-12-03

FI831049A0
(en)

1983-03-28

EP0090362A2
(en)

1983-10-05

DK144783A
(en)

1983-10-01

JPS58177967A
(en)

1983-10-18

NZ203719A
(en)

1986-02-21

PT76472A
(en)

1983-04-01

ES521741A0
(en)

1984-02-01

ES8401937A1
(en)

1984-01-01

GR78157B
(en)

1984-09-26

PT76472B
(en)

1986-01-24

KR840004069A
(en)

1984-10-06

ZA832229B
(en)

1983-12-28

ES8402570A1
(en)

1984-02-01

CA1198118A
(en)

1985-12-17

HU193876B
(en)

1987-12-28

ES521041A0
(en)

1984-01-01

AU560124B2
(en)

1987-04-02

DK144783D0
(en)

1983-03-29

IL68267A
(en)

1987-03-31

IL68267A0
(en)

1983-06-15

EP0090362A3
(en)

1985-09-18

FI831049L
(en)

1983-10-01

DE3211676A1
(en)

1983-10-06

NO834352L
(en)

1983-10-03

NO831168L
(en)

1983-10-03

Contact information