AU2713184A – 5-acyl-2-(1h)-pyridinones
– Google Patents
AU2713184A – 5-acyl-2-(1h)-pyridinones
– Google Patents
5-acyl-2-(1h)-pyridinones
Info
Publication number
AU2713184A
AU2713184A
AU27131/84A
AU2713184A
AU2713184A
AU 2713184 A
AU2713184 A
AU 2713184A
AU 27131/84 A
AU27131/84 A
AU 27131/84A
AU 2713184 A
AU2713184 A
AU 2713184A
AU 2713184 A
AU2713184 A
AU 2713184A
Authority
AU
Australia
Prior art keywords
pyridinones
acyl
Prior art date
1983-04-29
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU27131/84A
Other versions
AU557543B2
(en
Inventor
Richard C. Dage
Winton D. Jones
Richard A. Schettler
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Merrell Dow Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1983-04-29
Filing date
1984-04-19
Publication date
1984-11-01
1984-04-19
Application filed by Merrell Dow Pharmaceuticals Inc
filed
Critical
Merrell Dow Pharmaceuticals Inc
1984-11-01
Publication of AU2713184A
publication
Critical
patent/AU2713184A/en
1986-12-24
Application granted
granted
Critical
1986-12-24
Publication of AU557543B2
publication
Critical
patent/AU557543B2/en
2004-04-19
Anticipated expiration
legal-status
Critical
Status
Ceased
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
C07D213/84—Nitriles
C07D213/85—Nitriles in position 3
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P9/00—Drugs for disorders of the cardiovascular system
A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P9/00—Drugs for disorders of the cardiovascular system
A61P9/06—Antiarrhythmics
AU27131/84A
1983-04-29
1984-04-19
5-acyl-2-(1h)-pyridinones
Ceased
AU557543B2
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
US490081
1983-04-29
US06/490,081
US4568751A
(en)
1983-04-29
1983-04-29
5-Acyl-2-(1H)-pyridinones
Publications (2)
Publication Number
Publication Date
AU2713184A
true
AU2713184A
(en)
1984-11-01
AU557543B2
AU557543B2
(en)
1986-12-24
Family
ID=23946554
Family Applications (2)
Application Number
Title
Priority Date
Filing Date
AU27131/84A
Ceased
AU557543B2
(en)
1983-04-29
1984-04-19
5-acyl-2-(1h)-pyridinones
AU27141/84A
Ceased
AU571219B2
(en)
1983-04-29
1984-04-19
5-acyl-2-(1h)-pyridinones
Family Applications After (1)
Application Number
Title
Priority Date
Filing Date
AU27141/84A
Ceased
AU571219B2
(en)
1983-04-29
1984-04-19
5-acyl-2-(1h)-pyridinones
Country Status (22)
Country
Link
US
(1)
US4568751A
(en)
EP
(2)
EP0124089B1
(en)
JP
(2)
JPS59206356A
(en)
KR
(2)
KR900005010B1
(en)
AR
(1)
AR240313A1
(en)
AT
(2)
ATE25678T1
(en)
AU
(2)
AU557543B2
(en)
CA
(2)
CA1242443A
(en)
DD
(1)
DD223444A5
(en)
DE
(2)
DE3462889D1
(en)
DK
(2)
DK159424C
(en)
ES
(2)
ES531910A0
(en)
GR
(2)
GR81967B
(en)
HU
(2)
HU191753B
(en)
IE
(2)
IE57273B1
(en)
IL
(2)
IL71648A
(en)
NO
(2)
NO164415C
(en)
NZ
(2)
NZ207961A
(en)
PH
(1)
PH20256A
(en)
PT
(2)
PT78491B
(en)
SU
(1)
SU1299505A3
(en)
ZA
(2)
ZA843033B
(en)
Cited By (1)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
AU571219B2
(en)
*
1983-04-29
1988-04-14
Merrell Dow Pharmaceuticals Inc.
5-acyl-2-(1h)-pyridinones
Families Citing this family (9)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
US5428045A
(en)
*
1983-04-29
1995-06-27
Merrell Dow Pharmaceuticals Inc.
5-acyl-2-(1H)-pyridinoes
US5118696A
(en)
*
1983-04-29
1992-06-02
Merrell Dow Pharmaceuticals Inc.
5-Acyl-2-(1H)-pyridinones useful for treating cardiac failure
US4992452A
(en)
*
1983-04-29
1991-02-12
Merrell Dow Pharmaceuticals Inc.
Certain 5-acyl-2-(1H)-pyridinones useful in treating cardiac failure
US4853395A
(en)
*
1983-04-29
1989-08-01
Merrell Dow Pharmaceuticals Inc.
Certain 3-carboxylate or 3-carbamyl-5-acyl-2-(1H)-pyridinones having cardiotonic properties
US4731371A
(en)
*
1984-03-29
1988-03-15
Merrell Dow Pharmaceuticals Inc.
Certain 5-acyl-1,2-dihydro-2-oxo-3-pyridinecarbonitriles which are useful as cardiotonic agents
US4732982A
(en)
*
1983-11-03
1988-03-22
Merrell Dow Pharmaceuticals Inc.
Novel alkoxyimino ether derivatives of 5-acyl-2(1H)-pyridinones
US5212314A
(en)
*
1983-11-03
1993-05-18
Merrell Dow Pharmaceuticals Inc.
Alkoxyimino ether derivatives of 5-acyl-2(1H)-pyridinones
US4657919A
(en)
*
1984-08-03
1987-04-14
E. I. Du Pont De Nemours & Co.
Pyridone esters as inotropic agents
US4650806A
(en)
*
1985-01-14
1987-03-17
Sterling Drug Inc.
Cardiotonic 5-(heterylcarbonyl)-pyridones
Family Cites Families (9)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
DE2531035A1
(en)
*
1975-07-11
1977-01-27
Basf Ag
PROCESS FOR THE PRODUCTION OF 5-CYANPYRIDONE- (6)
US4072746A
(en)
*
1975-10-14
1978-02-07
Sterling Drug Inc.
3-Amino-5-(pyridinyl)-2(1H)-pyridinones
GB1596887A
(en)
*
1977-07-15
1981-09-03
Rohm & Haas
2-pyridone derivatives and their use as plant growth regulators
DE3005069A1
(en)
*
1980-02-11
1981-08-20
Cassella Ag, 6000 Frankfurt
2-Oxo-6-hydroxy-1,2-di:hydro-pyridine-5- carboxylic acid derivs. – prepd. by reaction of alkoxy:methylene-malonate cpds. with substd. acetamide cpds.
DE3106460A1
(en)
*
1980-03-03
1982-01-28
Sandoz-Patent-GmbH, 7850 Lörrach
2 (1H) -PYRIDINONE DERIVATIVES, THEIR PRODUCTION AND THE PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME
US4524149A
(en)
*
1982-03-15
1985-06-18
Sterling Drug Inc.
5-Alkanoyl-6-alkyl-2(1H)-pyridinones, their preparation and their cardiotonic use
US4412077A
(en)
*
1982-03-15
1983-10-25
Sterling Drug Inc.
Process for preparing 5-(lower-alkanoyl)-6-(lower-alkyl)-2(1H)-pyridinone
US4568751A
(en)
*
1983-04-29
1986-02-04
Merrell Dow Pharmaceuticals Inc.
5-Acyl-2-(1H)-pyridinones
DE3406329A1
(en)
*
1984-02-22
1985-08-22
Merck Patent Gmbh, 6100 Darmstadt
PYRIDONE
1983
1983-04-29
US
US06/490,081
patent/US4568751A/en
not_active
Expired – Lifetime
1984
1984-04-19
AU
AU27131/84A
patent/AU557543B2/en
not_active
Ceased
1984-04-19
AU
AU27141/84A
patent/AU571219B2/en
not_active
Ceased
1984-04-24
ZA
ZA843033A
patent/ZA843033B/en
unknown
1984-04-24
AR
AR296404A
patent/AR240313A1/en
active
1984-04-24
ZA
ZA843034A
patent/ZA843034B/en
unknown
1984-04-25
ES
ES531910A
patent/ES531910A0/en
active
Granted
1984-04-25
ES
ES531911A
patent/ES531911A0/en
active
Granted
1984-04-26
AT
AT84104703T
patent/ATE25678T1/en
active
1984-04-26
NZ
NZ207961A
patent/NZ207961A/en
unknown
1984-04-26
IL
IL71648A
patent/IL71648A/en
unknown
1984-04-26
EP
EP84104703A
patent/EP0124089B1/en
not_active
Expired
1984-04-26
DE
DE8484104704T
patent/DE3462889D1/en
not_active
Expired
1984-04-26
CA
CA000452888A
patent/CA1242443A/en
not_active
Expired
1984-04-26
NZ
NZ207960A
patent/NZ207960A/en
unknown
1984-04-26
HU
HU841619A
patent/HU191753B/en
not_active
IP Right Cessation
1984-04-26
HU
HU841618A
patent/HU191928B/en
not_active
IP Right Cessation
1984-04-26
PT
PT78491A
patent/PT78491B/en
not_active
IP Right Cessation
1984-04-26
PT
PT78493A
patent/PT78493B/en
not_active
IP Right Cessation
1984-04-26
PH
PH30602A
patent/PH20256A/en
unknown
1984-04-26
AT
AT84104704T
patent/ATE26262T1/en
not_active
IP Right Cessation
1984-04-26
EP
EP84104704A
patent/EP0124090B1/en
not_active
Expired
1984-04-26
IL
IL71649A
patent/IL71649A/en
unknown
1984-04-26
CA
CA000452889A
patent/CA1256880A/en
not_active
Expired
1984-04-26
DE
DE8484104703T
patent/DE3462503D1/en
not_active
Expired
1984-04-27
NO
NO841691A
patent/NO164415C/en
unknown
1984-04-27
IE
IE1046/84A
patent/IE57273B1/en
not_active
IP Right Cessation
1984-04-27
NO
NO841690A
patent/NO164416C/en
unknown
1984-04-27
DD
DD84262415A
patent/DD223444A5/en
not_active
IP Right Cessation
1984-04-27
IE
IE1047/84A
patent/IE57285B1/en
not_active
IP Right Cessation
1984-04-27
DK
DK213284A
patent/DK159424C/en
not_active
IP Right Cessation
1984-04-27
GR
GR74536A
patent/GR81967B/el
unknown
1984-04-27
JP
JP59084235A
patent/JPS59206356A/en
active
Granted
1984-04-27
DK
DK213584A
patent/DK159425C/en
not_active
IP Right Cessation
1984-04-27
JP
JP59084234A
patent/JPS59206355A/en
active
Granted
1984-04-27
GR
GR74535A
patent/GR81990B/el
unknown
1984-04-28
KR
KR1019840002297A
patent/KR900005010B1/en
not_active
IP Right Cessation
1984-04-28
KR
KR1019840002298A
patent/KR900005011B1/en
not_active
IP Right Cessation
1984-04-28
SU
SU843732701A
patent/SU1299505A3/en
active
Cited By (1)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
AU571219B2
(en)
*
1983-04-29
1988-04-14
Merrell Dow Pharmaceuticals Inc.
5-acyl-2-(1h)-pyridinones
Also Published As
Publication number
Publication date
NO164416C
(en)
1990-10-03
JPH0579668B2
(en)
1993-11-04
IE57285B1
(en)
1992-07-15
DK213584A
(en)
1984-10-30
PT78493A
(en)
1984-05-01
PT78493B
(en)
1986-05-20
DK159425B
(en)
1990-10-15
DK213584D0
(en)
1984-04-27
KR840008323A
(en)
1984-12-14
NO164416B
(en)
1990-06-25
EP0124090A1
(en)
1984-11-07
JPS59206356A
(en)
1984-11-22
AU571219B2
(en)
1988-04-14
AU2714184A
(en)
1984-11-01
PT78491A
(en)
1984-05-01
US4568751A
(en)
1986-02-04
DK159424B
(en)
1990-10-15
KR900005010B1
(en)
1990-07-16
DE3462889D1
(en)
1987-05-07
DD223444A5
(en)
1985-06-12
ATE26262T1
(en)
1987-04-15
IL71649A
(en)
1987-10-30
JPH058192B2
(en)
1993-02-01
AR240313A1
(en)
1990-03-30
HUT34007A
(en)
1985-01-28
PT78491B
(en)
1986-05-22
EP0124089B1
(en)
1987-03-04
EP0124089A1
(en)
1984-11-07
ZA843034B
(en)
1984-11-28
GR81967B
(en)
1984-12-12
IL71648A0
(en)
1984-07-31
NO164415C
(en)
1990-10-03
NZ207960A
(en)
1987-05-29
DK213284A
(en)
1984-10-30
NZ207961A
(en)
1986-09-10
ATE25678T1
(en)
1987-03-15
ES8505956A1
(en)
1985-06-01
SU1299505A3
(en)
1987-03-23
JPS59206355A
(en)
1984-11-22
DK213284D0
(en)
1984-04-27
KR900005011B1
(en)
1990-07-16
IE841047L
(en)
1984-10-29
AU557543B2
(en)
1986-12-24
CA1242443A
(en)
1988-09-27
ES8505955A1
(en)
1985-06-01
CA1256880A
(en)
1989-07-04
EP0124090B1
(en)
1987-04-01
PH20256A
(en)
1986-11-14
IL71648A
(en)
1987-11-30
NO164415B
(en)
1990-06-25
NO841690L
(en)
1984-10-30
ES531911A0
(en)
1985-06-01
IE57273B1
(en)
1992-07-01
HUT34006A
(en)
1985-01-28
IL71649A0
(en)
1984-07-31
DK159424C
(en)
1991-03-18
DK159425C
(en)
1991-03-18
DE3462503D1
(en)
1987-04-09
NO841691L
(en)
1984-10-30
KR840008322A
(en)
1984-12-14
ES531910A0
(en)
1985-06-01
ZA843033B
(en)
1984-11-28
GR81990B
(en)
1984-12-12
HU191928B
(en)
1987-04-28
IE841046L
(en)
1984-10-29
HU191753B
(en)
1987-04-28
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