AU3436578A

AU3436578A – Heterocyclic substituted imidazo (1, 2-a)pyridines
– Google Patents

AU3436578A – Heterocyclic substituted imidazo (1, 2-a)pyridines
– Google Patents
Heterocyclic substituted imidazo (1, 2-a)pyridines

Info

Publication number
AU3436578A

AU3436578A
AU34365/78A
AU3436578A
AU3436578A
AU 3436578 A
AU3436578 A
AU 3436578A
AU 34365/78 A
AU34365/78 A
AU 34365/78A
AU 3436578 A
AU3436578 A
AU 3436578A
AU 3436578 A
AU3436578 A
AU 3436578A
Authority
AU
Australia
Prior art keywords
pyridines
heterocyclic substituted
substituted imidazo
imidazo
heterocyclic
Prior art date
1977-03-28
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU34365/78A
Other versions

AU516695B2
(en

Inventor
R. J. and Telman R. L Buchta
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Merck and Co Inc

Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1977-03-28
Filing date
1978-03-21
Publication date
1979-09-27

1978-03-21
Application filed by Merck and Co Inc
filed
Critical
Merck and Co Inc

1979-09-27
Publication of AU3436578A
publication
Critical
patent/AU3436578A/en

1981-06-18
Application granted
granted
Critical

1981-06-18
Publication of AU516695B2
publication
Critical
patent/AU516695B2/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

125000000623
heterocyclic group
Chemical group

0.000
title
1

150000005234
imidazo[1,2-a]pyridines
Chemical class

0.000
title
1

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members

C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D213/62—Oxygen or sulfur atoms

C07D213/63—One oxygen atom

C07D213/64—One oxygen atom attached in position 2 or 6

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members

C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D213/72—Nitrogen atoms

C07D213/73—Unsubstituted amino or imino radicals

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members

C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals

C07D213/79—Acids; Esters

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 – C07D463/00

C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 – C07D463/00 in which the condensed system contains two hetero rings

C07D471/04—Ortho-condensed systems

AU34365/78A
1977-03-28
1978-03-21
Heterocyclic substituted imidazo (1, 2-a)pyridines

Expired

AU516695B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

USUS781902

1977-03-28

US05/781,902

US4105767A
(en)

1977-03-28
1977-03-28
Imidazo [1,2-a] pyridines substituted with a thienyl, thiazolyl, or thiadiazolyl group

Publications (2)

Publication Number
Publication Date

AU3436578A
true

AU3436578A
(en)

1979-09-27

AU516695B2

AU516695B2
(en)

1981-06-18

Family
ID=25124326
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU34365/78A
Expired

AU516695B2
(en)

1977-03-28
1978-03-21
Heterocyclic substituted imidazo (1, 2-a)pyridines

Country Status (9)

Country
Link

US
(2)

US4105767A
(en)

AU
(1)

AU516695B2
(en)

DE
(1)

DE2812914A1
(en)

FR
(1)

FR2385715A1
(en)

GB
(1)

GB1575781A
(en)

IT
(1)

IT7848582D0
(en)

NL
(1)

NL7802661A
(en)

NZ
(1)

NZ186711A
(en)

ZA
(1)

ZA781711B
(en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4250174A
(en)

*

1979-05-02
1981-02-10
Merck & Co., Inc.
3-Substituted imidazo [1,2-A] pyridines

US4221796A
(en)

*

1979-09-19
1980-09-09
E. R. Squibb & Sons, Inc.
Substituted imidazolo-pyridines and method

ZA81219B
(en)

*

1980-01-23
1982-01-27
Schering Corp
Imidazo (1,2-a) pyridines ,process for their preparation and pharmaceutical compositions containing them

JPS61218589A
(en)

*

1985-03-26
1986-09-29
Eisai Co Ltd
Imidazo(1,2-a)pyridinylpyridine derivative

GB8719368D0
(en)

*

1987-08-15
1987-09-23
Wellcome Found
Heterocyclic compounds

US5382110A
(en)

*

1992-12-30
1995-01-17
Esco Corporation
Quick coupling device

JPH0717971A
(en)

*

1993-07-02
1995-01-20
Takeda Chem Ind Ltd
Imidazole derivative, production and use thereof

AU2682695A
(en)

*

1994-06-20
1996-01-15
Takeda Chemical Industries Ltd.
Condensed imidazole compounds, their production and use

IL117620A0
(en)

*

1995-03-27
1996-07-23
Fujisawa Pharmaceutical Co
Heterocyclic compounds processes for the preparation thereof and pharmaceutical compositions containing the same

DE10117184A1
(en)

*

2001-04-05
2002-10-17
Gruenenthal Gmbh

Substituted imidazole [1,2-a] pyridin-3-yl amide and amine compounds

JP2007529496A
(en)

*

2004-03-19
2007-10-25
ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー

Imidazopyridine and imidazopyrimidine derivatives as antibacterial agents

EP1799680A2
(en)

*

2004-10-07
2007-06-27
Warner-Lambert Company LLC
Triazolopyridine derivatives as antibacterial agents

EP2277881A4
(en)

2008-04-18
2011-09-07
Shionogi & Co
Heterocyclic compound having inhibitory activity on p13k

Family Cites Families (3)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US3701780A
(en)

*

1970-09-18
1972-10-31
Merck & Co Inc
Imidazo(1,2-a)pyridines

JPS5154583A
(en)

*

1974-11-01
1976-05-13
Kyorin Seiyaku Kk
Shinkipirazoro * 1 55a * pirijinjudotaino seizoho

US4096264A
(en)

*

1975-12-09
1978-06-20
Merck & Co., Inc.
Certain substituted imidazo [1,2-a] pyridines

1977

1977-03-28
US
US05/781,902
patent/US4105767A/en
not_active
Expired – Lifetime

1978

1978-03-10
NL
NL7802661A
patent/NL7802661A/en
not_active
Application Discontinuation

1978-03-16
NZ
NZ186711A
patent/NZ186711A/en
unknown

1978-03-21
AU
AU34365/78A
patent/AU516695B2/en
not_active
Expired

1978-03-22
GB
GB11436/78A
patent/GB1575781A/en
not_active
Expired

1978-03-22
FR
FR7808308A
patent/FR2385715A1/en
active
Granted

1978-03-23
ZA
ZA00781711A
patent/ZA781711B/en
unknown

1978-03-23
IT
IT7848582A
patent/IT7848582D0/en
unknown

1978-03-23
DE
DE19782812914
patent/DE2812914A1/en
not_active
Withdrawn

1978-05-30
US
US05/910,418
patent/US4146642A/en
not_active
Expired – Lifetime

Also Published As

Publication number
Publication date

US4105767A
(en)

1978-08-08

NZ186711A
(en)

1981-02-11

FR2385715A1
(en)

1978-10-27

ZA781711B
(en)

1979-11-28

DE2812914A1
(en)

1978-10-12

GB1575781A
(en)

1980-09-24

IT7848582D0
(en)

1978-03-23

NL7802661A
(en)

1978-10-02

AU516695B2
(en)

1981-06-18

FR2385715B1
(en)

1981-09-04

US4146642A
(en)

1979-03-27

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