AU3878585A - Creation of Inventions and Patents with Artificial Intelligence

AU3878585A – Isoxazole derivatives
– Google Patents

AU3878585A – Isoxazole derivatives
– Google Patents
Isoxazole derivatives

Info

Publication number
AU3878585A

AU3878585A
AU38785/85A
AU3878585A
AU3878585A
AU 3878585 A
AU3878585 A
AU 3878585A
AU 38785/85 A
AU38785/85 A
AU 38785/85A
AU 3878585 A
AU3878585 A
AU 3878585A
AU 3878585 A
AU3878585 A
AU 3878585A
Authority
AU
Australia
Prior art keywords
compounds
carbon atoms
isoxazole derivatives
denotes
halogenoalkyl
Prior art date
1984-02-17
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU38785/85A
Other versions

AU572612B2
(en

Inventor
Friedrich-Johannes Kammerer
Rudolf Schleyerbach
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Hoechst AG

Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1984-02-17
Filing date
1985-02-15
Publication date
1985-09-05

1985-02-15
Application filed by Hoechst AG
filed
Critical
Hoechst AG

1985-09-05
Publication of AU3878585A
publication
Critical
patent/AU3878585A/en

1988-05-12
Application granted
granted
Critical

1988-05-12
Publication of AU572612B2
publication
Critical
patent/AU572612B2/en

2005-02-15
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms

C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings

C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms

C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings

C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P25/00—Drugs for disorders of the nervous system

A61P25/04—Centrally acting analgesics, e.g. opioids

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings

C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings

C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members

C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen

Abstract

4-Isoxazolecarboxylic acid amides of the general formula I (I) in which R denotes hydrogen, alkyl with up to 4 carbon atoms or halogenoalkyl with up to 2 carbon atoms and W denotes a direct bond, CH2, CH-CH3, CH-C2H5, CHOH, O or S, processes for their preparation, medicaments which contain these compounds and the use of the compounds for the treatment of pain and/or fever.

AU38785/85A
1984-02-17
1985-02-15
Isoxazole derivatives

Ceased

AU572612B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

DE3405727

1984-02-17

DE19843405727

DE3405727A1
(en)

1984-02-17
1984-02-17

ISOXAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS

Publications (2)

Publication Number
Publication Date

AU3878585A
true

AU3878585A
(en)

1985-09-05

AU572612B2

AU572612B2
(en)

1988-05-12

Family
ID=6228020
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU38785/85A
Ceased

AU572612B2
(en)

1984-02-17
1985-02-15
Isoxazole derivatives

Country Status (19)

Country
Link

US
(1)

US4636513A
(en)

EP
(1)

EP0152868B1
(en)

JP
(1)

JPS60193973A
(en)

KR
(1)

KR850006411A
(en)

AT
(1)

ATE44142T1
(en)

AU
(1)

AU572612B2
(en)

CA
(1)

CA1247616A
(en)

DE
(2)

DE3405727A1
(en)

DK
(1)

DK165981C
(en)

ES
(1)

ES8602776A1
(en)

FI
(1)

FI81094C
(en)

GR
(1)

GR850416B
(en)

HU
(1)

HU194192B
(en)

IL
(1)

IL74351A
(en)

MA
(1)

MA20352A1
(en)

NO
(1)

NO158677C
(en)

NZ
(1)

NZ211139A
(en)

PH
(1)

PH21434A
(en)

PT
(1)

PT79969B
(en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US5268382A
(en)

1985-09-27
1993-12-07
Hoechst Aktiengesellschaft
Medicaments to combat autoimmune diseases, in particular systemic lupus erythematosus

DE3534440A1
(en)

1985-09-27
1987-04-02
Hoechst Ag

DRUGS AGAINST CHRONIC GRAFT VERSUS HOST DISEASES AND AUTO AUTO DISEASES, IN PARTICULAR SYSTEMIC LUPUS ERYTHEMATODES

IT1228288B
(en)

1989-01-09
1991-06-07
Zambon Spa

COMPOUNDS WITH ANTI-SEROTONIN ACTIVITY

ZA913762B
(en)

1990-05-18
1992-01-29
Hoechst Ag
Isoxazole-4-carboxamides and hydroxyalkylidenecyanoacetamides,pharmaceuticals containing these compounds and their use

EP0527736B1
(en)

1990-05-18
1997-04-16
Hoechst Aktiengesellschaft
Isoxazole-4-carboxamides and hydroxyalkylidene-cyanoacetamides, drugs containing these compounds and use of such drugs

US6133301A
(en)

1991-08-22
2000-10-17
Aventis Pharma Deutschland Gmbh
Pharmaceuticals for the treatment of rejection reactions in organ transplantations

DE4127737A1
(en)

1991-08-22
1993-02-25
Hoechst Ag

MEDICINAL PRODUCTS FOR TREATMENT OF REPELLATION REACTIONS IN ORGAN PLANTING

GB9219779D0
(en)

1992-09-18
1992-10-28
Rhone Poulenc Agriculture
Compositions of new matter

US5624946A
(en)

1994-07-05
1997-04-29
Williams; James
Use of leflunomide to control and reverse chronic allograft rejection

ES2247749T3
(en)

1999-07-02
2006-03-01
Cognis Ip Management Gmbh

MICROCAPSULES III.

Family Cites Families (5)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

DE634286C
(en)

1935-02-23
1936-08-26
Hoffmann La Roche & Co Akt Ges

Process for the preparation of dialkyl-substituted amides of isoxazole carboxylic acids

DE653835C
(en)

1936-03-20
1937-12-03
Hoffmanni La Roche & Co Akt Ge

Process for the preparation of amide-like derivatives of isoxazole carboxylic acids

US2126329A
(en)

1936-03-20
1938-08-09
Hoffmann La Roche
Amide derivatives of isoxazole carboxylic acids

US2212767A
(en)

1938-01-17
1940-08-27
Hoffmann La Roche
Amide derivatives of 3,5-dimethylisoxazole carboxylic acids

DE2524959C2
(en)

1975-06-05
1983-02-10
Hoechst Ag, 6000 Frankfurt

5-methyl-isoxazole-4-carboxylic acid anilides, process for their preparation, agents containing these compounds

1984

1984-02-17
DE
DE19843405727
patent/DE3405727A1/en
not_active
Withdrawn

1985

1985-02-07
EP
EP85101264A
patent/EP0152868B1/en
not_active
Expired

1985-02-07
DE
DE8585101264T
patent/DE3571130D1/en
not_active
Expired

1985-02-07
AT
AT85101264T
patent/ATE44142T1/en
not_active
IP Right Cessation

1985-02-12
HU
HU85524A
patent/HU194192B/en
not_active
IP Right Cessation

1985-02-14
FI
FI850613A
patent/FI81094C/en
not_active
IP Right Cessation

1985-02-14
NO
NO850580A
patent/NO158677C/en
unknown

1985-02-15
GR
GR850416A
patent/GR850416B/el
unknown

1985-02-15
IL
IL74351A
patent/IL74351A/en
not_active
IP Right Cessation

1985-02-15
US
US06/702,312
patent/US4636513A/en
not_active
Expired – Fee Related

1985-02-15
MA
MA20576A
patent/MA20352A1/en
unknown

1985-02-15
CA
CA000474482A
patent/CA1247616A/en
not_active
Expired

1985-02-15
ES
ES540438A
patent/ES8602776A1/en
not_active
Expired

1985-02-15
JP
JP60026671A
patent/JPS60193973A/en
active
Granted

1985-02-15
PT
PT79969A
patent/PT79969B/en
not_active
IP Right Cessation

1985-02-15
DK
DK074085A
patent/DK165981C/en
active

1985-02-15
PH
PH31872A
patent/PH21434A/en
unknown

1985-02-15
NZ
NZ211139A
patent/NZ211139A/en
unknown

1985-02-15
AU
AU38785/85A
patent/AU572612B2/en
not_active
Ceased

1985-02-16
KR
KR1019850000966A
patent/KR850006411A/en
not_active
Application Discontinuation

Also Published As

Publication number
Publication date

NO850580L
(en)

1985-08-19

CA1247616A
(en)

1988-12-28

IL74351A
(en)

1988-11-15

KR850006411A
(en)

1985-10-05

JPH03866B2
(en)

1991-01-09

EP0152868A3
(en)

1986-10-08

ES540438A0
(en)

1985-12-01

NO158677B
(en)

1988-07-11

JPS60193973A
(en)

1985-10-02

DK74085A
(en)

1985-08-18

GR850416B
(en)

1985-06-18

HU194192B
(en)

1988-01-28

IL74351A0
(en)

1985-05-31

NO158677C
(en)

1988-10-19

FI81094B
(en)

1990-05-31

NZ211139A
(en)

1988-04-29

AU572612B2
(en)

1988-05-12

DE3571130D1
(en)

1989-07-27

HUT37767A
(en)

1986-02-28

DE3405727A1
(en)

1985-08-22

PH21434A
(en)

1987-10-15

EP0152868A2
(en)

1985-08-28

EP0152868B1
(en)

1989-06-21

DK165981C
(en)

1993-07-26

FI81094C
(en)

1990-09-10

DK74085D0
(en)

1985-02-15

PT79969B
(en)

1987-02-02

PT79969A
(en)

1985-03-01

FI850613A0
(en)

1985-02-14

ATE44142T1
(en)

1989-07-15

US4636513A
(en)

1987-01-13

DK165981B
(en)

1993-02-22

FI850613L
(en)

1985-08-18

ES8602776A1
(en)

1985-12-01

MA20352A1
(en)

1985-10-01

Contact information