AU4330685A - Creation of Inventions and Patents with Artificial Intelligence

AU4330685A – Cephems, carbacephems and oxacephmes derivatives
– Google Patents

AU4330685A – Cephems, carbacephems and oxacephmes derivatives
– Google Patents
Cephems, carbacephems and oxacephmes derivatives

Info

Publication number
AU4330685A

AU4330685A
AU43306/85A
AU4330685A
AU4330685A
AU 4330685 A
AU4330685 A
AU 4330685A
AU 43306/85 A
AU43306/85 A
AU 43306/85A
AU 4330685 A
AU4330685 A
AU 4330685A
AU 4330685 A
AU4330685 A
AU 4330685A
Authority
AU
Australia
Prior art keywords
oxacephmes
cephems
carbacephems
derivatives
oxacephmes derivatives
Prior art date
1984-06-07
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU43306/85A
Other versions

AU576588B2
(en

Inventor
Masahiko Fujino
Masahiro Kondo
Akio Miyake
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Takeda Pharmaceutical Co Ltd

Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1984-06-07
Filing date
1985-06-03
Publication date
1985-12-12

1984-06-07
Priority claimed from PCT/JP1984/000295
external-priority
patent/WO1986000070A1/en

1985-04-01
Priority claimed from PCT/JP1985/000155
external-priority
patent/WO1986005787A1/en

1985-06-03
Application filed by Takeda Chemical Industries Ltd
filed
Critical
Takeda Chemical Industries Ltd

1985-12-12
Publication of AU4330685A
publication
Critical
patent/AU4330685A/en

1988-09-01
Application granted
granted
Critical

1988-09-01
Publication of AU576588B2
publication
Critical
patent/AU576588B2/en

2005-06-03
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

C07D501/14—Compounds having a nitrogen atom directly attached in position 7

C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3

C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids

C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3

C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof

C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D463/00—Heterocyclic compounds containing 1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

C07D463/10—Heterocyclic compounds containing 1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2

C07D463/14—Heterocyclic compounds containing 1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hetero atoms directly attached in position 7

C07D463/16—Nitrogen atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D463/16—Nitrogen atoms

C07D463/18—Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof

C07D463/20—Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof with the acylating radicals further substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

C07D463/22—Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof with the acylating radicals further substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen further substituted by nitrogen atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS

Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE

Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS

Y02P20/00—Technologies relating to chemical industry

Y02P20/50—Improvements relating to the production of bulk chemicals

Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

AU43306/85A
1984-06-07
1985-06-03
Cephems, carbacephems and oxacephmes derivatives

Ceased

AU576588B2
(en)

Applications Claiming Priority (4)

Application Number
Priority Date
Filing Date
Title

WOJP8400295

1984-06-07

PCT/JP1984/000295

WO1986000070A1
(en)

1984-06-07
1984-06-07
Cephem compounds

PCT/JP1985/000155

WO1986005787A1
(en)

1985-04-01
1985-04-01
Antibacterial compounds

WOJP8500155

1985-04-01

Publications (2)

Publication Number
Publication Date

AU4330685A
true

AU4330685A
(en)

1985-12-12

AU576588B2

AU576588B2
(en)

1988-09-01

Family
ID=26425045
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU43306/85A
Ceased

AU576588B2
(en)

1984-06-07
1985-06-03
Cephems, carbacephems and oxacephmes derivatives

Country Status (15)

Country
Link

US
(1)

US4665065A
(en)

EP
(1)

EP0164113B1
(en)

KR
(1)

KR920004823B1
(en)

AU
(1)

AU576588B2
(en)

CA
(1)

CA1264052A
(en)

DE
(1)

DE3577707D1
(en)

DK
(1)

DK256085A
(en)

ES
(2)

ES8609343A1
(en)

FI
(1)

FI852289L
(en)

GR
(1)

GR851384B
(en)

HU
(1)

HU194894B
(en)

NO
(1)

NO852294L
(en)

NZ
(1)

NZ212320A
(en)

PH
(1)

PH22107A
(en)

PT
(1)

PT80595B
(en)

Cited By (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

AU617154B2
(en)

1988-03-09
1991-11-21
Fujisawa Pharmaceutical Co., Ltd.
New cephem compounds and processes for preparation thereof

Families Citing this family (13)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4788185A
(en)

1984-04-23
1988-11-29
Takeda Chemical Industries, Ltd.
Cephalosporin compounds

ATE89826T1
(en)

1985-03-01
1993-06-15
Takeda Chemical Industries Ltd

ANTIBACTERIAL COMPOUNDS, THEIR PREPARATION AND USE.

DE3688477T2
(en)

1985-03-01
1993-09-16
Takeda Chemical Industries Ltd

ANTIBACTERIAL CONNECTIONS, THEIR PRODUCTION AND USE.

DE3687200T2
(en)

1985-09-03
1993-05-27
Otsuka Kagaku Kk

CEPHALOSPORINE DERIVATIVES.

US4826834A
(en)

1985-09-27
1989-05-02
Takeda Chemical Industries, Ltd.
Cephem compounds

US4760140A
(en)

1986-10-20
1988-07-26
American Cyanamid Company
3-substituted-7-[5-substituted-2-thiazolyl)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-3-ene-2-carboxylic acid, diphenylmethyl esters

CA1293719C
(en)

1986-09-22
1991-12-31
Takao Takaya
Cephem compounds and processes for preparation thereof

US5019571A
(en)

1988-01-25
1991-05-28
Eli Lilly And Company
1-carbacephalosporin antibiotics

DE3803169A1
(en)

1988-02-03
1989-08-17
Bayer Ag

SS LACTAM ANTIBIOTICS, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS AND IN MEDICINAL PRODUCTS

US5173485A
(en)

1988-03-09
1992-12-22
Fujisawa Pharmaceutical Company, Ltd.
Cephem compounds

US5215982A
(en)

1989-11-10
1993-06-01
Fujisawa Pharmaceutical Co., Ltd.
Cephem compounds

KR930009796B1
(en)

1991-05-25
1993-10-11
주식회사 대웅제약
Cephalosporin derivatives

WO1998000159A1
(en)

1996-06-28
1998-01-08
Oxigene, Inc.
Useful formulations of acid addition salt drugs

Family Cites Families (14)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4024133A
(en)

1971-05-14
1977-05-17
Glaxo Laboratories Limited
7β-[2-Etherified oximino-2-(thienyl-,furyl- or pyridylacetamido)]cephalosporins

US4033950A
(en)

1971-05-14
1977-07-05
Glaxo Laboratories Limited
3-Hydroxymethyl-7β-(2-alkoxy-or benzyloxyimino-2-arylacetamido)ceph-3-em-4-carboxylic acids and salts thereof

DK154939C
(en)

1974-12-19
1989-06-12
Takeda Chemical Industries Ltd

METHOD OF ANALOGUE FOR THE PREPARATION OF THIAZOLYLACETAMIDO-CEPHEM COMPOUNDS OR PHARMACEUTICAL ACCEPTABLE SALTS OR ESTERS THEREOF

GR63088B
(en)

1976-04-14
1979-08-09
Takeda Chemical Industries Ltd
Preparation process of novel cephalosporins

DE2714880A1
(en)

1977-04-02
1978-10-26
Hoechst Ag

CEPHEMDER DERIVATIVES AND PROCESS FOR THEIR PRODUCTION

AR229883A1
(en)

1978-05-26
1983-12-30
Glaxo Group Ltd

PROCEDURE FOR THE PREPARATION OF ANTIBIOTIC (6R, 7R) -7 – ((Z) -2- (2-AMINOTIAZOL-4-IL) -2- (2-CARBOXIPROP-2-OXIIMINO) -ACETAMIDO) -3- (1 -PIRIDINOMETIL) -CEF-3-EM-4-CARBOXYLATE

GB2037281B
(en)

1978-11-15
1983-01-19
Glaxo Group Ltd
7( -(2-amino-4-thiozolyl)-2-hydroximino-acetanuds)-cephalosporins

ES511101A0
(en)

1981-04-03
1983-05-01
Fujisawa Pharmaceutical Co

“PROCEDURE TO PREPARE A NEW CEFEM COMPOUND”.

US4501739A
(en)

1982-01-19
1985-02-26
Eli Lilly And Company
Thieno and furopyridinium-substituted cephalosporins

US4500526A
(en)

1982-06-28
1985-02-19
Bristol-Myers Company
Cephalosporin derivatives

DE3336757A1
(en)

1983-10-08
1985-04-25
Hoechst Ag, 6230 Frankfurt

CEPHALOSPORINE DERIVATIVES AND METHOD FOR THEIR PRODUCTION

GB2148289B
(en)

1983-10-17
1987-09-23
Lilly Co Eli
3-bicyclicpyridinium-methyl cephalosporins

GB8401093D0
(en)

1984-01-16
1984-02-15
Fujisawa Pharmaceutical Co
Cephem compounds

NO165842C
(en)

1984-04-23
1991-04-17
Takeda Chemical Industries Ltd

ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE CEFEM COMPOUNDS.

1985

1985-05-29
PH
PH32333A
patent/PH22107A/en
unknown

1985-05-30
US
US06/739,440
patent/US4665065A/en
not_active
Expired – Lifetime

1985-06-03
AU
AU43306/85A
patent/AU576588B2/en
not_active
Ceased

1985-06-05
EP
EP85106979A
patent/EP0164113B1/en
not_active
Expired – Lifetime

1985-06-05
ES
ES543932A
patent/ES8609343A1/en
not_active
Expired

1985-06-05
PT
PT80595A
patent/PT80595B/en
unknown

1985-06-05
DE
DE8585106979T
patent/DE3577707D1/en
not_active
Expired – Fee Related

1985-06-06
HU
HU852256A
patent/HU194894B/en
not_active
IP Right Cessation

1985-06-06
NO
NO852294A
patent/NO852294L/en
unknown

1985-06-06
NZ
NZ212320A
patent/NZ212320A/en
unknown

1985-06-06
GR
GR851384A
patent/GR851384B/el
unknown

1985-06-06
DK
DK256085A
patent/DK256085A/en
not_active
Application Discontinuation

1985-06-06
CA
CA000483303A
patent/CA1264052A/en
not_active
Expired

1985-06-07
KR
KR1019850004012A
patent/KR920004823B1/en
not_active
IP Right Cessation

1985-06-07
FI
FI852289A
patent/FI852289L/en
not_active
Application Discontinuation

1986

1986-01-21
ES
ES551064A
patent/ES8800240A1/en
not_active
Expired

Cited By (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

AU617154B2
(en)

1988-03-09
1991-11-21
Fujisawa Pharmaceutical Co., Ltd.
New cephem compounds and processes for preparation thereof

Also Published As

Publication number
Publication date

ES551064A0
(en)

1987-11-01

FI852289L
(en)

1985-12-08

ES8800240A1
(en)

1987-11-01

HUT41034A
(en)

1987-03-30

HU194894B
(en)

1988-03-28

EP0164113B1
(en)

1990-05-16

PT80595B
(en)

1987-04-21

EP0164113A3
(en)

1987-01-28

DK256085A
(en)

1985-12-08

ES543932A0
(en)

1986-08-16

FI852289A0
(en)

1985-06-07

NZ212320A
(en)

1988-09-29

KR920004823B1
(en)

1992-06-18

PH22107A
(en)

1988-06-01

DK256085D0
(en)

1985-06-06

AU576588B2
(en)

1988-09-01

KR860000302A
(en)

1986-01-27

ES8609343A1
(en)

1986-08-16

GR851384B
(en)

1985-11-25

CA1264052A
(en)

1989-12-27

EP0164113A2
(en)

1985-12-11

PT80595A
(en)

1985-07-01

NO852294L
(en)

1985-12-09

DE3577707D1
(en)

1990-06-21

US4665065A
(en)

1987-05-12

Contact information