AU4334885A - Creation of Inventions and Patents with Artificial Intelligence

AU4334885A – Triazole derivatives
– Google Patents

AU4334885A – Triazole derivatives
– Google Patents
Triazole derivatives

Info

Publication number
AU4334885A

AU4334885A
AU43348/85A
AU4334885A
AU4334885A
AU 4334885 A
AU4334885 A
AU 4334885A
AU 43348/85 A
AU43348/85 A
AU 43348/85A
AU 4334885 A
AU4334885 A
AU 4334885A
AU 4334885 A
AU4334885 A
AU 4334885A
Authority
AU
Australia
Prior art keywords
compounds
triazole derivatives
ethers
esters
susbtituents
Prior art date
1984-06-07
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU43348/85A
Other versions

AU554476B2
(en

Inventor
Robert John Bass
Kelvin Cooper
Kenneth Richardson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pfizer Corp

Original Assignee
Pfizer Corp
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1984-06-07
Filing date
1985-06-06
Publication date
1985-12-12

1985-06-06
Application filed by Pfizer Corp, Pfizer Inc
filed
Critical
Pfizer Corp

1985-12-12
Publication of AU4334885A
publication
Critical
patent/AU4334885A/en

1986-08-21
Application granted
granted
Critical

1986-08-21
Publication of AU554476B2
publication
Critical
patent/AU554476B2/en

2005-06-06
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00

C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings

C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings

C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members

C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

A—HUMAN NECESSITIES

A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING

A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS

A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds

A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms

A01N43/647—Triazoles; Hydrogenated triazoles

A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics

A61P31/04—Antibacterial agents

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings

C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members

C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms

C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings

C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Abstract

Compounds of the formula:

where R is a phenyl group optionally substituted by 1 to 3 susbtituents each independently selected from F, Cl, Br, I, CF3, C1-C4 alkyl and C1-C4 alkoxy, or R is a 5-chloropyrid-2-yl group; and X is OH, F, Cl or Br;
and the O-esters and O-ethers of the compounds in which X is OH; and the pharmaceutically and agriculturally acceptable salts of said compounds and O-esters and O-ethers.
The compounds are useful as human and agricultural fungicides.

AU43348/85A
1984-06-07
1985-06-06
Triazole derivatives

Ceased

AU554476B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

GB8414519

1984-06-07

GB848414519A

GB8414519D0
(en)

1984-06-07
1984-06-07
Triazole antifungal agents

Publications (2)

Publication Number
Publication Date

AU4334885A
true

AU4334885A
(en)

1985-12-12

AU554476B2

AU554476B2
(en)

1986-08-21

Family
ID=10562061
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU43348/85A
Ceased

AU554476B2
(en)

1984-06-07
1985-06-06
Triazole derivatives

Country Status (25)

Country
Link

US
(1)

US4618616A
(en)

EP
(1)

EP0164246B1
(en)

JP
(1)

JPS611672A
(en)

KR
(1)

KR870001829B1
(en)

CN
(1)

CN85104471B
(en)

AT
(1)

ATE36328T1
(en)

AU
(1)

AU554476B2
(en)

CA
(1)

CA1287059C
(en)

DD
(1)

DD235641A5
(en)

DE
(1)

DE3564266D1
(en)

DK
(1)

DK170301B1
(en)

ES
(1)

ES8604170A1
(en)

FI
(1)

FI86176C
(en)

GB
(1)

GB8414519D0
(en)

GR
(1)

GR851382B
(en)

HU
(1)

HU195647B
(en)

IE
(1)

IE57804B1
(en)

IL
(1)

IL75410A
(en)

NO
(1)

NO852287L
(en)

NZ
(1)

NZ212317A
(en)

PH
(1)

PH22870A
(en)

PL
(1)

PL144920B1
(en)

PT
(1)

PT80598B
(en)

YU
(1)

YU94985A
(en)

ZA
(1)

ZA854250B
(en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

DE3440117A1
(en)

1984-11-02
1986-05-15
Bayer Ag, 5090 Leverkusen

SUBSTITUTED AZOLYLCYCLOPROPYL AZOLYL METHYL CARBINOL DERIVATIVES

DE3440114A1
(en)

1984-11-02
1986-05-07
Bayer Ag, 5090 Leverkusen

ANTIMYCOTIC AGENTS

EP0180850A3
(en)

1984-11-02
1987-05-27
Bayer Ag
Antimycotic azolyl-methyl-cyclopropyl-carbinol derivatives

GB8429932D0
(en)

1984-11-27
1985-01-03
Pfizer Ltd
Triazole antifungal agents

DE3608792A1
(en)

1986-03-15
1987-09-24
Hoechst Ag

1,1-DISUBSTITUTED CYCLOPROPANE DERIVATIVES, METHOD FOR THEIR PRODUCTION AND THEIR USE

DE3608727A1
(en)

1986-03-15
1987-09-17
Hoechst Ag

1,1-DISUBSTITUTED CYCLOPROPANDERIVATES, METHODS FOR THE PRODUCTION THEREOF AND THEIR USE AS AN ANTIMYCOTICS OR AS AN INTERMEDIATE PRODUCT

DE3837463A1
(en)

1988-11-04
1990-05-10
Bayer Ag

SUBSTITUTED BISAZOLE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS

DE3921162A1
(en)

1989-06-28
1991-01-10
Bayer Ag

USE OF SUBSTITUTED BIS-AZOLYL DERIVATIVES FOR CONTROLLING MUSHROOMS IN PLANT PROTECTION

US5247094A
(en)

1990-01-24
1993-09-21
Bayer Aktiengesellschaft
1-(3- or 5-halo-1,2,4-triazol-1-yl)ethyl phenyl ketone intermediates

US5039676A
(en)

1990-05-11
1991-08-13
Schering Corporation
Tri- and tetra-substituted-oxetanes and tetrahydrofurans and intermediates thereof

US5488035A
(en)

1991-12-06
1996-01-30
Pioneer Hi-Bred International, Inc.
Peptide with inhibitory activity towards plant pathogenic fungi

JPH06340636A
(en)

1993-05-31
1994-12-13
Ss Pharmaceut Co Ltd
Triazole derivative or its salt and antimycotic agent containing the compound

WO2014118170A1
(en)

2013-02-04
2014-08-07
Syngenta Participations Ag
Novel microbiocides

Family Cites Families (7)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

EP0051565A1
(en)

1980-11-03
1982-05-12
Ciba-Geigy Ag
1-N,N-dimethylcarbamoyl-3(5)-cyclopropyl-1,2,4-triazoles, their preparation and use as pesticides

DE3337937A1
(en)

1982-10-28
1984-05-03
Sandoz-Patent-GmbH, 7850 Lörrach

NEW AZOLE DERIVATIVES

GB8302500D0
(en)

1983-01-29
1983-03-02
Pfizer Ltd
Antifungal agents

DE3305834A1
(en)

1983-02-19
1984-08-23
Bayer Ag, 5090 Leverkusen

MICROBICIDAL AGENT FOR PROTECTING TECHNICAL MINERALS

DE3440114A1
(en)

1984-11-02
1986-05-07
Bayer Ag, 5090 Leverkusen

ANTIMYCOTIC AGENTS

EP0180850A3
(en)

1984-11-02
1987-05-27
Bayer Ag
Antimycotic azolyl-methyl-cyclopropyl-carbinol derivatives

GB8429932D0
(en)

1984-11-27
1985-01-03
Pfizer Ltd
Triazole antifungal agents

1984

1984-06-07
GB
GB848414519A
patent/GB8414519D0/en
active
Pending

1985

1985-05-24
US
US06/738,143
patent/US4618616A/en
not_active
Expired – Fee Related

1985-05-28
PL
PL1985253666A
patent/PL144920B1/en
unknown

1985-05-29
EP
EP85303764A
patent/EP0164246B1/en
not_active
Expired

1985-05-29
DE
DE8585303764T
patent/DE3564266D1/en
not_active
Expired

1985-05-29
AT
AT85303764T
patent/ATE36328T1/en
not_active
IP Right Cessation

1985-05-31
JP
JP60118701A
patent/JPS611672A/en
active
Granted

1985-06-03
FI
FI852223A
patent/FI86176C/en
not_active
IP Right Cessation

1985-06-05
NZ
NZ212317A
patent/NZ212317A/en
unknown

1985-06-05
PT
PT80598A
patent/PT80598B/en
not_active
IP Right Cessation

1985-06-05
PH
PH32370A
patent/PH22870A/en
unknown

1985-06-05
IL
IL75410A
patent/IL75410A/en
unknown

1985-06-05
ZA
ZA854250A
patent/ZA854250B/en
unknown

1985-06-05
CA
CA000483188A
patent/CA1287059C/en
not_active
Expired – Fee Related

1985-06-05
KR
KR1019850003935A
patent/KR870001829B1/en
not_active
IP Right Cessation

1985-06-05
DD
DD85277055A
patent/DD235641A5/en
unknown

1985-06-06
IE
IE1416/85A
patent/IE57804B1/en
unknown

1985-06-06
GR
GR851382A
patent/GR851382B/el
unknown

1985-06-06
NO
NO852287A
patent/NO852287L/en
unknown

1985-06-06
DK
DK253685A
patent/DK170301B1/en
not_active
IP Right Cessation

1985-06-06
HU
HU852247A
patent/HU195647B/en
unknown

1985-06-06
YU
YU00949/85A
patent/YU94985A/en
unknown

1985-06-06
AU
AU43348/85A
patent/AU554476B2/en
not_active
Ceased

1985-06-07
ES
ES543998A
patent/ES8604170A1/en
not_active
Expired

1985-06-11
CN
CN198585104471A
patent/CN85104471B/en
not_active
Expired

Also Published As

Publication number
Publication date

PL144920B1
(en)

1988-07-30

ATE36328T1
(en)

1988-08-15

DK170301B1
(en)

1995-07-31

GR851382B
(en)

1985-11-25

ES543998A0
(en)

1986-01-16

DD235641A5
(en)

1986-05-14

PT80598B
(en)

1987-04-23

EP0164246A2
(en)

1985-12-11

GB8414519D0
(en)

1984-07-11

IE57804B1
(en)

1993-04-07

FI86176B
(en)

1992-04-15

DK253685A
(en)

1985-12-08

FI852223L
(en)

1985-12-08

FI86176C
(en)

1992-07-27

NO852287L
(en)

1985-12-09

PH22870A
(en)

1989-01-19

ZA854250B
(en)

1987-01-28

JPS611672A
(en)

1986-01-07

PT80598A
(en)

1985-07-01

AU554476B2
(en)

1986-08-21

KR860000288A
(en)

1986-01-27

YU94985A
(en)

1987-10-31

ES8604170A1
(en)

1986-01-16

CN85104471B
(en)

1987-10-21

JPH0521108B2
(en)

1993-03-23

PL253666A1
(en)

1986-06-17

HU195647B
(en)

1988-06-28

EP0164246B1
(en)

1988-08-10

CA1287059C
(en)

1991-07-30

DK253685D0
(en)

1985-06-06

NZ212317A
(en)

1988-04-29

HUT38326A
(en)

1986-05-28

EP0164246A3
(en)

1987-01-28

IL75410A
(en)

1989-02-28

FI852223A0
(en)

1985-06-03

CN85104471A
(en)

1986-12-10

DE3564266D1
(en)

1988-09-15

US4618616A
(en)

1986-10-21

KR870001829B1
(en)

1987-10-15

IE851416L
(en)

1985-12-07

Contact information