AU457015B2

AU457015B2 – Piperidine derivatives, their preparation and compositions containing them
– Google Patents

AU457015B2 – Piperidine derivatives, their preparation and compositions containing them
– Google Patents
Piperidine derivatives, their preparation and compositions containing them

Info

Publication number
AU457015B2

AU457015B2
AU35910/71A
AU3591071A
AU457015B2
AU 457015 B2
AU457015 B2
AU 457015B2
AU 35910/71 A
AU35910/71 A
AU 35910/71A
AU 3591071 A
AU3591071 A
AU 3591071A
AU 457015 B2
AU457015 B2
AU 457015B2
Authority
AU
Australia
Prior art keywords
preparation
compositions containing
piperidine derivatives
piperidine
derivatives
Prior art date
1970-12-10
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
AU35910/71A
Other versions

AU3591071A
(en

Inventor
Karl Schulte Joachim Borck Eike Pietsch Helmut Muller-Calnan Volker Hoppe
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Merck Patent GmbH

Original Assignee
Merck Patent GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1970-12-10
Filing date
1971-11-19
Publication date
1974-12-19

1971-11-19
Application filed by Merck Patent GmbH
filed
Critical
Merck Patent GmbH

1972-05-24
Publication of AU3591071A
publication
Critical
patent/AU3591071A/en

1974-12-19
Application granted
granted
Critical

1974-12-19
Publication of AU457015B2
publication
Critical
patent/AU457015B2/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

239000000203
mixture
Substances

0.000
title
1

150000003053
piperidines
Chemical class

0.000
title
1

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings

C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings

C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members

C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings

C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members

C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms

C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms

C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings

C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members

C07D211/82—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms

C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3

C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems

C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring

C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring

C07D317/58—Radicals substituted by nitrogen atoms

AU35910/71A
1970-12-10
1971-11-19
Piperidine derivatives, their preparation and compositions containing them

Expired

AU457015B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

DEDE820608

1970-12-10

DE2060816A

DE2060816C3
(en)

1970-12-10
1970-12-10

4-Phenylpiperidine derivatives Process for their production and pharmaceutical preparations containing these compounds

Publications (2)

Publication Number
Publication Date

AU3591071A

AU3591071A
(en)

1972-05-24

AU457015B2
true

AU457015B2
(en)

1974-12-19

Family
ID=5790598
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU35910/71A
Expired

AU457015B2
(en)

1970-12-10
1971-11-19
Piperidine derivatives, their preparation and compositions containing them

Country Status (24)

Country
Link

US
(1)

US3821234A
(en)

JP
(1)

JPS5518711B1
(en)

AT
(5)

AT317892B
(en)

AU
(1)

AU457015B2
(en)

BE
(1)

BE776406A
(en)

BR
(1)

BR7108208D0
(en)

CA
(1)

CA967575A
(en)

CH
(5)

CH570997A5
(en)

CS
(5)

CS166038B2
(en)

DD
(1)

DD94994A5
(en)

DE
(1)

DE2060816C3
(en)

DK
(1)

DK133780C
(en)

ES
(1)

ES397786A1
(en)

FR
(1)

FR2117971B1
(en)

GB
(1)

GB1322270A
(en)

HU
(1)

HU164941B
(en)

IL
(1)

IL38177A
(en)

IT
(1)

IT7948130D0
(en)

NL
(1)

NL7116991A
(en)

PL
(5)

PL84493B1
(en)

RO
(3)

RO59974A
(en)

SE
(1)

SE390306B
(en)

YU
(1)

YU34797B
(en)

ZA
(1)

ZA717685B
(en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB1345872A
(en)

*

1970-09-03
1974-02-06
Wyeth John & Brother Ltd
Amino-and acylamino-pyridine and hydropyridine derivatives

US3919242A
(en)

*

1970-09-03
1975-11-11
Wyeth John & Brother Ltd
1-(Benzodioxanylalkylene)piperidines

EP0007399B1
(en)

*

1978-06-24
1982-01-20
MERCK PATENT GmbH
Indolylalkyl amines, pharmaceutical preparations containing them and process for their manufacture

DE3441927A1
(en)

*

1984-11-16
1986-05-28
Basf Ag, 6700 Ludwigshafen

4- (P-TERT.BUTYL-PHENYL) -3-METHYL-PIPERIDINE SUBSTITUTED ON NITROGEN, THEIR QUARTAINE SALTS AND THEIR USE AS FUNGICIDES

US5212183A
(en)

*

1981-11-14
1993-05-18
Basf Aktiengesellschaft
4-(p-tert.-butylphenyl)-3-methylpiperidines substituted at the nitrogen, their quaternary salts and their use as fungicides

DE3236243A1
(en)

*

1982-09-30
1984-04-05
Merck Patent Gmbh, 6100 Darmstadt

SULFURIZED INDOLDER DERIVATIVES

JPS5995281A
(en)

*

1982-11-19
1984-06-01
Kotobuki Seiyaku Kk
Thiazole derivative and its preparation

DE3723797A1
(en)

*

1987-07-18
1989-01-26
Merck Patent Gmbh

OXAZOLIDINONE

US4935424A
(en)

*

1988-05-27
1990-06-19
Warner-Lambert Company
4 or 5-(substituted piperazinylalkyl)-2-aminothiazoles as antipsychotic agents

HU207310B
(en)

*

1988-12-02
1993-03-29
Pfizer
Process for producing aryl-piperidine derivatives

DE4017211A1
(en)

1990-05-29
1991-12-05
Merck Patent Gmbh

OXAZOLIDINONE

EP0568876B1
(en)

1992-05-04
1996-08-28
Bayer Ag
Reactive dyes, their preparation and their use

DE4425146A1
(en)

*

1994-07-15
1996-01-18
Basf Ag

Use of heterocyclic compounds

DE19602505A1
(en)

*

1996-01-25
1997-07-31
Merck Patent Gmbh

1- (pyrazol-4-indol-3-yl) piperidines

FR2803593B1
(en)

*

2000-01-06
2002-02-15
Sanofi Synthelabo

NOVEL TETRAHYDROPYRIDINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

CN102190536A
(en)

*

2010-03-08
2011-09-21
华东理工大学
Method for organically catalyzing asymmetric conjugated addition of ketene and organic phosphorus compound

BR102012024778A2
(en)

*

2012-09-28
2014-08-19
Cristalia Prod Quimicos Farm

Heteroaromatic compounds; PROCESS FOR PREPARING COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, USES AND TREATMENT METHOD FOR ACUTE AND CHRONIC PAIN

WO2021076835A1
(en)

*

2019-10-18
2021-04-22
Fmc Corporation
Methods for the preparation of 5-bromo-2-(3chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylic acid

1970

1970-12-10
DE
DE2060816A
patent/DE2060816C3/en
not_active
Expired

1971

1971-10-22
CH
CH86975A
patent/CH570997A5/xx
not_active
IP Right Cessation

1971-10-22
CH
CH86775A
patent/CH581650A5/xx
not_active
IP Right Cessation

1971-10-22
CH
CH86675A
patent/CH571514A5/xx
not_active
IP Right Cessation

1971-10-22
CH
CH1544271A
patent/CH571513A5/xx
not_active
IP Right Cessation

1971-10-22
CH
CH86875A
patent/CH571515A5/xx
not_active
IP Right Cessation

1971-11-16
ZA
ZA717685A
patent/ZA717685B/en
unknown

1971-11-19
GB
GB5385271A
patent/GB1322270A/en
not_active
Expired

1971-11-19
AU
AU35910/71A
patent/AU457015B2/en
not_active
Expired

1971-11-19
IL
IL38177A
patent/IL38177A/en
unknown

1971-11-26
YU
YU2992/71A
patent/YU34797B/en
unknown

1971-12-03
RO
RO72981A
patent/RO59974A/ro
unknown

1971-12-03
RO
RO72974A
patent/RO59096A/ro
unknown

1971-12-03
RO
RO68947A
patent/RO60110A/ro
unknown

1971-12-07
US
US00205707A
patent/US3821234A/en
not_active
Expired – Lifetime

1971-12-08
PL
PL1971175532A
patent/PL84493B1/pl
unknown

1971-12-08
JP
JP9872771A
patent/JPS5518711B1/ja
active
Pending

1971-12-08
PL
PL1971175535A
patent/PL84242B1/pl
unknown

1971-12-08
PL
PL1971175534A
patent/PL84241B1/xx
unknown

1971-12-08
PL
PL1971175553A
patent/PL84240B1/pl
unknown

1971-12-08
PL
PL1971152015A
patent/PL83235B1/pl
unknown

1971-12-08
DD
DD159585A
patent/DD94994A5/xx
unknown

1971-12-08
SE
SE7115736A
patent/SE390306B/en
unknown

1971-12-08
BE
BE776406A
patent/BE776406A/en
unknown

1971-12-09
ES
ES397786A
patent/ES397786A1/en
not_active
Expired

1971-12-09
AT
AT905973A
patent/AT317892B/en
not_active
IP Right Cessation

1971-12-09
DK
DK603271A
patent/DK133780C/en
active

1971-12-09
FR
FR7144205A
patent/FR2117971B1/fr
not_active
Expired

1971-12-09
AT
AT905773A
patent/AT320651B/en
not_active
IP Right Cessation

1971-12-09
AT
AT905873A
patent/AT320652B/en
not_active
IP Right Cessation

1971-12-09
AT
AT1058671A
patent/AT318604B/en
not_active
IP Right Cessation

1971-12-09
CA
CA129,750A
patent/CA967575A/en
not_active
Expired

1971-12-09
AT
AT905673A
patent/AT320650B/en
not_active
IP Right Cessation

1971-12-10
CS
CS2062*[A
patent/CS166038B2/cs
unknown

1971-12-10
CS
CS2064*[A
patent/CS166040B2/cs
unknown

1971-12-10
CS
CS2061*[A
patent/CS166037B2/cs
unknown

1971-12-10
CS
CS2063*[A
patent/CS166039B2/cs
unknown

1971-12-10
CS
CS8625A
patent/CS166036B2/cs
unknown

1971-12-10
HU
HUME1449A
patent/HU164941B/hu
unknown

1971-12-10
BR
BR8208/71A
patent/BR7108208D0/en
unknown

1971-12-10
NL
NL7116991A
patent/NL7116991A/xx
not_active
Application Discontinuation

1979

1979-02-26
IT
IT7948130A
patent/IT7948130D0/en
unknown

Also Published As

Publication number
Publication date

BR7108208D0
(en)

1973-07-03

YU34797B
(en)

1980-03-15

DE2060816A1
(en)

1972-06-29

ES397786A1
(en)

1975-05-16

IL38177A0
(en)

1972-01-27

ZA717685B
(en)

1972-08-30

US3821234A
(en)

1974-06-28

CA967575A
(en)

1975-05-13

RO60110A
(en)

1976-06-15

DE2060816B2
(en)

1980-01-10

AT320651B
(en)

1975-02-25

DK133780C
(en)

1976-12-13

GB1322270A
(en)

1973-07-04

IT7948130D0
(en)

1979-02-26

CH570997A5
(en)

1975-12-31

CS166040B2
(en)

1976-01-29

RO59974A
(en)

1976-05-15

DK133780B
(en)

1976-07-19

FR2117971B1
(en)

1974-10-18

DD94994A5
(en)

1973-01-12

AT320652B
(en)

1975-02-25

JPS5518711B1
(en)

1980-05-21

IL38177A
(en)

1975-05-22

SE390306B
(en)

1976-12-13

YU299271A
(en)

1979-09-10

AT317892B
(en)

1974-09-25

CH571514A5
(en)

1976-01-15

BE776406A
(en)

1972-06-08

PL83235B1
(en)

1975-12-31

CS166037B2
(en)

1976-01-29

CS166039B2
(en)

1976-01-29

CH581650A5
(en)

1976-11-15

CS166038B2
(en)

1976-01-29

AU3591071A
(en)

1972-05-24

CH571513A5
(en)

1976-01-15

PL84242B1
(en)

1976-03-31

CH571515A5
(en)

1976-01-15

DE2060816C3
(en)

1980-09-04

PL84240B1
(en)

1976-03-31

CS166036B2
(en)

1976-01-29

AT320650B
(en)

1975-02-25

AT318604B
(en)

1974-11-11

FR2117971A1
(en)

1972-07-28

HU164941B
(en)

1974-05-28

PL84493B1
(en)

1976-04-30

RO59096A
(en)

1976-01-15

PL84241B1
(en)

1976-03-31

NL7116991A
(en)

1972-06-13

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