AU504599B2 - Creation of Inventions and Patents with Artificial Intelligence

AU504599B2 – Benzisothiazolone derivatives
– Google Patents

AU504599B2 – Benzisothiazolone derivatives
– Google Patents
Benzisothiazolone derivatives

Info

Publication number
AU504599B2

AU504599B2
AU19163/76A
AU1916376A
AU504599B2
AU 504599 B2
AU504599 B2
AU 504599B2
AU 19163/76 A
AU19163/76 A
AU 19163/76A
AU 1916376 A
AU1916376 A
AU 1916376A
AU 504599 B2
AU504599 B2
AU 504599B2
Authority
AU
Australia
Prior art keywords
benzisothiazolone derivatives
benzisothiazolone
derivatives
Prior art date
1975-11-18
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Ceased

Application number
AU19163/76A
Other versions

AU1916376A
(en

Inventor
Keith Howard Baggaley
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Beecham Group PLC

Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1975-11-18
Filing date
1976-10-29
Publication date
1979-10-18

1976-10-29
Application filed by Beecham Group PLC
filed
Critical
Beecham Group PLC

1978-05-04
Publication of AU1916376A
publication
Critical
patent/AU1916376A/en

1979-10-18
Application granted
granted
Critical

1979-10-18
Publication of AU504599B2
publication
Critical
patent/AU504599B2/en

1992-10-29
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00

C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings

C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES

A61K31/00—Medicinal preparations containing organic active ingredients

A61K31/33—Heterocyclic compounds

A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins

A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES

A61K31/00—Medicinal preparations containing organic active ingredients

A61K31/33—Heterocyclic compounds

A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins

A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom

A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES

A61K31/00—Medicinal preparations containing organic active ingredients

A61K31/33—Heterocyclic compounds

A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins

A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom

A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof

A61K31/445—Non condensed piperidines, e.g. piperocaine

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES

A61K31/00—Medicinal preparations containing organic active ingredients

A61K31/33—Heterocyclic compounds

A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins

A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom

A61K31/47—Quinolines; Isoquinolines

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings

C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems

AU19163/76A
1975-11-18
1976-10-29
Benzisothiazolone derivatives

Ceased

AU504599B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

GB4737375

1975-11-18

GB47373/75

1975-11-18

Related Child Applications (1)

Application Number
Title
Priority Date
Filing Date

AU47163/79A
Division

AU520890B2
(en)

1975-11-18
1979-05-17
Benzisothiazolones

Publications (2)

Publication Number
Publication Date

AU1916376A

AU1916376A
(en)

1978-05-04

AU504599B2
true

AU504599B2
(en)

1979-10-18

Family
ID=10444739
Family Applications (2)

Application Number
Title
Priority Date
Filing Date

AU19163/76A
Ceased

AU504599B2
(en)

1975-11-18
1976-10-29
Benzisothiazolone derivatives

AU47163/79A
Expired – Fee Related

AU520890B2
(en)

1975-11-18
1979-05-17
Benzisothiazolones

Family Applications After (1)

Application Number
Title
Priority Date
Filing Date

AU47163/79A
Expired – Fee Related

AU520890B2
(en)

1975-11-18
1979-05-17
Benzisothiazolones

Country Status (28)

Country
Link

US
(5)

US4113728A
(en)

JP
(1)

JPS5262273A
(en)

AR
(3)

AR217411A1
(en)

AT
(1)

AT355017B
(en)

AU
(2)

AU504599B2
(en)

BE
(1)

BE848371A
(en)

BG
(4)

BG24811A3
(en)

CA
(1)

CA1064511A
(en)

CH
(1)

CH627465A5
(en)

CS
(4)

CS192570B2
(en)

DD
(1)

DD127645A5
(en)

DE
(1)

DE2652201A1
(en)

DK
(1)

DK517776A
(en)

ES
(3)

ES453420A1
(en)

FI
(1)

FI763285A
(en)

FR
(1)

FR2332019A1
(en)

HU
(1)

HU173958B
(en)

IL
(1)

IL50690A
(en)

NL
(1)

NL7612796A
(en)

NO
(1)

NO763922L
(en)

NZ
(1)

NZ182325A
(en)

PH
(1)

PH13918A
(en)

PL
(1)

PL193742A1
(en)

PT
(1)

PT65851B
(en)

RO
(4)

RO69608A
(en)

SE
(1)

SE7612919L
(en)

SU
(4)

SU682129A3
(en)

ZA
(1)

ZA766489B
(en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

NZ182325A
(en)

1975-11-18
1979-03-16
Beecham Group Ltd
2-substituted-1,2-benzisothiazol-3-ones

DE2602643C2
(en)

1976-01-24
1984-12-20
Bayer Ag, 5090 Leverkusen

1,2-Benzisothiazolinone-3, process for their preparation, as well as pharmaceuticals

US4190663A
(en)

1976-01-24
1980-02-26
Bayer Aktiengesellschaft
Anti-thrombotic 1,2-benzisothiazolin-3-ones

DE2860750D1
(en)

1977-06-20
1981-09-17
Beecham Group Plc
Antithrombotic 2-(gamma-(1-piperidinyl)propyl)1,2-benzisothiazol 3-one, its pharmaceutically acceptable acid addition salts, their preparation and their compositions

DE2860430D1
(en)

1977-10-08
1981-02-26
Beecham Group Ltd
Antithrombotic compositions containing benzisothiazolones

DE2966957D1
(en)

1979-10-08
1984-06-07
Merck & Co Inc
2-aryl-1,2-benzisothiazolinone-1,1-dioxides and pharmaceutical compositions containing them

DE3226284A1
(en)

1982-07-14
1984-01-19
A. Nattermann & Cie GmbH, 5000 Köln

NEW BENZISOSELENAZOLONES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM

DE3238006A1
(en)

1982-10-13
1984-04-19
Bayer Ag, 5090 Leverkusen

AZOLYL METHYLAMINE, THEIR PRODUCTION AND USE IN MICROBICIDES

DE3500577A1
(en)

1985-01-10
1986-07-10
Basf Ag, 6700 Ludwigshafen

METHOD FOR PRODUCING 1,2-BENZISOTHIAZOLONES

US4732984A
(en)

1985-10-17
1988-03-22
American Home Products Corporation
Piperazinoisothiazolones with psychotropic activity

DE3617976A1
(en)

1986-05-28
1988-01-14
Alter Sa

1,4-DIHYDROPYRIDINE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE IN ANTITHROMBOTIC MEDICATIONS

US4831031A
(en)

1988-01-22
1989-05-16
Pfizer Inc.
Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity

CA1340759C
(en)

1988-07-01
1999-09-21
James P. Albarella
Isobenzothiazolone chromogenic thiol indicators and their derivatives

US5128457A
(en)

1988-07-01
1992-07-07
Miles Inc.
Chromogenic thiol indicators based on an isobenzothiazolone ring system

US5236917A
(en)

1989-05-04
1993-08-17
Sterling Winthrop Inc.
Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof

EP2344479B1
(en)

2008-09-23
2015-04-08
Georgetown University
1,2-benzisothiazolinone and isoindolinone derivatives

AU2012296543B2
(en)

2011-08-16
2016-08-11
Georgetown University
Methods of treating bacterial infections with 1,2-benzisothiazolinone and isoindolinone derivatives

US20180318818A1
(en)

2015-10-19
2018-11-08
Emory University
Redox Dehydration Coupling Catalysts and Methods Related Thereto

Family Cites Families (8)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

BE565380A
(en)

1957-03-08

US3012039A
(en)

1958-03-14
1961-12-05
Ici Ltd
2-p-chlorobenzyl-1, 2-benzisothiazolone

DE1147947B
(en)

1961-07-25
1963-05-02
Knoll Ag

Process for the preparation of new 1,2-benzisothiazolones

SE392103B
(en)

1970-04-27
1977-03-14
Sherwin Williams Co

METHOD OF PRODUCING 1,2-BENSISOTIAZOLINE-3-ONERS

US3661974A
(en)

1970-04-27
1972-05-09
Sherwin Williams Co
2-carbalkoxy-phenyl sulfenamides

NZ182325A
(en)

1975-11-18
1979-03-16
Beecham Group Ltd
2-substituted-1,2-benzisothiazol-3-ones

GB1582214A
(en)

1977-05-31
1981-01-07
Beecham Group Ltd
Antithrombotic compositions

DE2734882A1
(en)

1977-08-03
1979-02-22
Basf Ag

3-SQUARE BRACKETS ON 4- (1,3-DIAZACYCLOALKEN-2-YL) -PHENYL SQUARE BRACKETS FOR -1,2-BENZISOTHIAZOLS, THE METHOD FOR THEIR MANUFACTURING AND THE MEDICINAL PRODUCTS CONTAINED

1976

1976-10-13
NZ
NZ182325A
patent/NZ182325A/en
unknown

1976-10-15
IL
IL50690A
patent/IL50690A/en
unknown

1976-10-20
PH
PH19020A
patent/PH13918A/en
unknown

1976-10-29
ZA
ZA766489A
patent/ZA766489B/en
unknown

1976-10-29
AU
AU19163/76A
patent/AU504599B2/en
not_active
Ceased

1976-11-02
US
US05/738,000
patent/US4113728A/en
not_active
Expired – Lifetime

1976-11-10
AR
AR265414A
patent/AR217411A1/en
active

1976-11-15
FR
FR7634296A
patent/FR2332019A1/en
active
Granted

1976-11-15
AT
AT849176A
patent/AT355017B/en
not_active
IP Right Cessation

1976-11-16
BE
BE172385A
patent/BE848371A/en
not_active
IP Right Cessation

1976-11-16
DE
DE19762652201
patent/DE2652201A1/en
not_active
Withdrawn

1976-11-16
HU
HU76BE1280A
patent/HU173958B/en
unknown

1976-11-16
FI
FI763285A
patent/FI763285A/fi
not_active
Application Discontinuation

1976-11-17
ES
ES453420A
patent/ES453420A1/en
not_active
Expired

1976-11-17
CS
CS767392A
patent/CS192570B2/en
unknown

1976-11-17
CA
CA265,874A
patent/CA1064511A/en
not_active
Expired

1976-11-17
DD
DD195824A
patent/DD127645A5/xx
unknown

1976-11-17
RO
RO7688476A
patent/RO69608A/en
unknown

1976-11-17
CS
CS775980A
patent/CS192593B2/en
unknown

1976-11-17
BG
BG7600035568A
patent/BG24811A3/en
unknown

1976-11-17
CH
CH1448376A
patent/CH627465A5/en
not_active
IP Right Cessation

1976-11-17
BG
BG7600034711A
patent/BG24808A3/en
unknown

1976-11-17
PL
PL19374276A
patent/PL193742A1/en
unknown

1976-11-17
BG
BG7600035567A
patent/BG24810A3/en
unknown

1976-11-17
BG
BG7600035566A
patent/BG24809A3/en
unknown

1976-11-17
RO
RO7696010A
patent/RO75540A/en
unknown

1976-11-17
NL
NL7612796A
patent/NL7612796A/en
not_active
Application Discontinuation

1976-11-17
PT
PT65851A
patent/PT65851B/en
unknown

1976-11-17
CS
CS775981A
patent/CS192594B2/en
unknown

1976-11-17
DK
DK517776A
patent/DK517776A/en
not_active
Application Discontinuation

1976-11-17
NO
NO763922A
patent/NO763922L/no
unknown

1976-11-17
CS
CS775979A
patent/CS192592B2/en
unknown

1976-11-17
SU
SU762422503A
patent/SU682129A3/en
active

1976-11-17
RO
RO7696012A
patent/RO75777A/en
unknown

1976-11-17
RO
RO7696011A
patent/RO75730A/en
unknown

1976-11-18
SE
SE7612919A
patent/SE7612919L/en
not_active
Application Discontinuation

1976-11-18
JP
JP51139026A
patent/JPS5262273A/en
active
Pending

1977

1977-04-04
SU
SU772466684A
patent/SU679141A3/en
active

1977-04-04
SU
SU772466683A
patent/SU701536A3/en
active

1977-04-04
SU
SU772466669A
patent/SU671728A3/en
active

1977-10-17
AR
AR269610A
patent/AR217449A1/en
active

1977-10-17
AR
AR269611A
patent/AR215271A1/en
active

1977-11-11
US
US05/850,786
patent/US4212979A/en
not_active
Expired – Lifetime

1977-12-16
ES
ES465174A
patent/ES465174A1/en
not_active
Expired

1977-12-16
ES
ES465173A
patent/ES465173A1/en
not_active
Expired

1978

1978-08-25
US
US05/936,861
patent/US4212872A/en
not_active
Expired – Lifetime

1979

1979-05-17
AU
AU47163/79A
patent/AU520890B2/en
not_active
Expired – Fee Related

1979-08-20
US
US06/067,949
patent/US4243669A/en
not_active
Expired – Lifetime

1980

1980-10-31
US
US06/202,711
patent/US4350702A/en
not_active
Expired – Lifetime

Also Published As

Publication number
Publication date

AT355017B
(en)

1980-02-11

AR215271A1
(en)

1979-09-28

SE7612919L
(en)

1977-05-19

FI763285A
(en)

1977-05-19

SU701536A3
(en)

1979-11-30

CS192570B2
(en)

1979-08-31

PH13918A
(en)

1980-11-04

AR217449A1
(en)

1980-03-31

AU4716379A
(en)

1979-09-27

NZ182325A
(en)

1979-03-16

US4243669A
(en)

1981-01-06

RO75777A
(en)

1981-02-28

DK517776A
(en)

1977-05-19

AU1916376A
(en)

1978-05-04

BE848371A
(en)

1977-05-16

DE2652201A1
(en)

1977-06-02

NL7612796A
(en)

1977-05-23

SU679141A3
(en)

1979-08-05

BG24809A3
(en)

1978-05-12

RO75540A
(en)

1980-11-30

ES465173A1
(en)

1978-10-01

CA1064511A
(en)

1979-10-16

BG24808A3
(en)

1978-05-12

FR2332019B1
(en)

1983-05-20

US4212979A
(en)

1980-07-15

HU173958B
(en)

1979-09-28

PL193742A1
(en)

1979-05-21

IL50690A
(en)

1980-01-31

DD127645A5
(en)

1977-10-05

PT65851B
(en)

1978-05-15

RO69608A
(en)

1982-07-06

US4212872A
(en)

1980-07-15

CS192592B2
(en)

1979-08-31

SU682129A3
(en)

1979-08-25

ZA766489B
(en)

1977-10-26

US4350702A
(en)

1982-09-21

NO763922L
(en)

1977-05-20

ES465174A1
(en)

1978-10-01

ES453420A1
(en)

1978-02-16

RO75730A
(en)

1981-02-28

ATA849176A
(en)

1979-07-15

CS192593B2
(en)

1979-08-31

BG24811A3
(en)

1978-05-12

IL50690A0
(en)

1976-12-31

AU520890B2
(en)

1982-03-04

CH627465A5
(en)

1982-01-15

CS192594B2
(en)

1979-08-31

AR217411A1
(en)

1980-03-31

US4113728A
(en)

1978-09-12

JPS5262273A
(en)

1977-05-23

BG24810A3
(en)

1978-05-12

FR2332019A1
(en)

1977-06-17

SU671728A3
(en)

1979-06-30

PT65851A
(en)

1976-12-01

Contact information