AU539177B2 - Creation of Inventions and Patents with Artificial Intelligence

AU539177B2 – Amino alkoxy pyrazoles
– Google Patents

AU539177B2 – Amino alkoxy pyrazoles
– Google Patents
Amino alkoxy pyrazoles

Info

Publication number
AU539177B2

AU539177B2
AU68926/81A
AU6892681A
AU539177B2
AU 539177 B2
AU539177 B2
AU 539177B2
AU 68926/81 A
AU68926/81 A
AU 68926/81A
AU 6892681 A
AU6892681 A
AU 6892681A
AU 539177 B2
AU539177 B2
AU 539177B2
Authority
AU
Australia
Prior art keywords
general formula
hydrogen atom
phenyl
alkyl group
alkyl
Prior art date
1980-04-01
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
AU68926/81A
Other versions

AU6892681A
(en

Inventor
Francois-Xavier Jarreau
Jean-Jacques Koenig
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Nativelle Sa Ets

Original Assignee
Nativelle SA Ets
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1980-04-01
Filing date
1981-03-31
Publication date
1984-09-13

1981-03-31
Application filed by Nativelle SA Ets
filed
Critical
Nativelle SA Ets

1981-10-08
Publication of AU6892681A
publication
Critical
patent/AU6892681A/en

1984-09-13
Application granted
granted
Critical

1984-09-13
Publication of AU539177B2
publication
Critical
patent/AU539177B2/en

2001-03-31
Anticipated expiration
legal-status
Critical

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

-1
Amino alkoxy pyrazoles
Chemical class

0.000
title
abstract
3

125000000217
alkyl group
Chemical group

0.000
abstract
3

125000004435
hydrogen atom
Chemical group

[H]*

0.000
abstract
2

125000001997
phenyl group
Chemical group

[H]C1=C([H])C([H])=C(*)C([H])=C1[H]

0.000
abstract
2

125000003341
7 membered heterocyclic group
Chemical group

0.000
abstract
1

208000024172
Cardiovascular disease
Diseases

0.000
abstract
1

208000020401
Depressive disease
Diseases

0.000
abstract
1

208000019695
Migraine disease
Diseases

0.000
abstract
1

125000003545
alkoxy group
Chemical group

0.000
abstract
1

125000001797
benzyl group
Chemical group

[H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])*

0.000
abstract
1

125000004093
cyano group
Chemical group

*C#N

0.000
abstract
1

208000037265
diseases, disorders, signs and symptoms
Diseases

0.000
abstract
1

208000035475
disorder
Diseases

0.000
abstract
1

229940079593
drug
Drugs

0.000
abstract
1

239000003814
drug
Substances

0.000
abstract
1

125000005843
halogen group
Chemical group

0.000
abstract
1

229910052500
inorganic mineral
Inorganic materials

0.000
abstract
1

238000002483
medication
Methods

0.000
abstract
1

239000011707
mineral
Substances

0.000
abstract
1

150000007522
mineralic acids
Chemical class

0.000
abstract
1

125000001624
naphthyl group
Chemical group

0.000
abstract
1

229910052757
nitrogen
Inorganic materials

0.000
abstract
1

125000004433
nitrogen atom
Chemical group

0.000
abstract
1

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings

C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings

C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members

C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D231/18—One oxygen or sulfur atom

C07D231/20—One oxygen atom attached in position 3 or 5

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P25/00—Drugs for disorders of the nervous system

A61P25/24—Antidepressants

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P25/00—Drugs for disorders of the nervous system

A61P25/26—Psychostimulants, e.g. nicotine, cocaine

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P9/00—Drugs for disorders of the cardiovascular system

Abstract

An aminoalkoxypyrazole of the general formula (I) (I) wherein Ar is a phenyl, benzyl or naphthyl group, or a phenyl group substituted by one or more halogen atoms, or by one or more alkyl, cyano, nitro, hydroxy or alkoxy groups; R1 is a hydrogen atom or an alkyl group; R2 and R3, which may be the same or different, are a hydrogen atom or an alkyl group, or form, with the nitrogen atom to which they are attached, a 5- to 7-membered heterocyclic ring; n is an integer of from 1 to 4; as well as the mineral or organic acid salts thereof. A further embodiment of the invention is the application of the derivatives of the general formula (I) as medications, in particular, for the treatment of depression, polyfunctional disorders, migraines and cardiovascular diseases.

AU68926/81A
1980-04-01
1981-03-31
Amino alkoxy pyrazoles

Expired

AU539177B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

FR8007301

1980-04-01

FR8007301A

FR2479219A1
(en)

1980-04-01
1980-04-01

AMINO-ALCOXY PYRAZOLES, PROCESS FOR THEIR PREPARATION, AND MEDICAMENTS CONTAINING SAME

Publications (2)

Publication Number
Publication Date

AU6892681A

AU6892681A
(en)

1981-10-08

AU539177B2
true

AU539177B2
(en)

1984-09-13

Family
ID=9240402
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU68926/81A
Expired

AU539177B2
(en)

1980-04-01
1981-03-31
Amino alkoxy pyrazoles

Country Status (12)

Country
Link

US
(1)

US4330544A
(en)

EP
(1)

EP0037344B1
(en)

JP
(1)

JPS56152465A
(en)

AT
(1)

ATE8389T1
(en)

AU
(1)

AU539177B2
(en)

CA
(1)

CA1152992A
(en)

DE
(1)

DE3164667D1
(en)

DK
(1)

DK153547C
(en)

ES
(1)

ES500810A0
(en)

FR
(1)

FR2479219A1
(en)

GR
(1)

GR75618B
(en)

IE
(1)

IE51963B1
(en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

FR2513996A1
(en)

1981-10-02
1983-04-08
Nativelle Sa Ets

PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC APPLICATION

US4550119A
(en)

1983-05-23
1985-10-29
Warner-Lambert Company
2,4-Dihydro-5-[(substituted)phenyl]-4,4-disubstituted-3H-pyrazol-3-ones

DE3532880A1
(en)

1985-09-14
1987-03-26
Basf Ag

1,4-DISUBSTITUTED PYRAZOLE DERIVATIVES

US4806554A
(en)

1988-01-11
1989-02-21
Hoechst-Roussel Pharmaceuticals, Inc.
Pyrazol and indazolpyridinamines

US4962120A
(en)

1989-03-22
1990-10-09
Sterling Drug Inc.
1H-imidazole-1-acetamides

DE4341749A1
(en)

1993-12-08
1995-06-14
Kali Chemie Pharma Gmbh

3- (Phenylalkylaminoalkyloxy) -5-phenylpyrazole compounds and methods and intermediates for their preparation and medicaments containing these compounds

US5547967A
(en)

1993-12-08
1996-08-20
Kali-Chemie Pharma Gmbh
(Phenylalkylaminoalkyloxy)-heteroaryl-compounds, processes and intermediates for their production and pharmaceutical compositions containing them

Family Cites Families (1)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB1385811A
(en)

1972-01-14
1975-03-05
Nativelle Sa Ets
1-amino pyrazole derivatives and pharmaceutical compositions containing them

1980

1980-04-01
FR
FR8007301A
patent/FR2479219A1/en
active
Granted

1981

1981-03-27
JP
JP4421781A
patent/JPS56152465A/en
active
Granted

1981-03-27
ES
ES500810A
patent/ES500810A0/en
active
Granted

1981-03-30
IE
IE728/81A
patent/IE51963B1/en
not_active
IP Right Cessation

1981-03-31
AU
AU68926/81A
patent/AU539177B2/en
not_active
Expired

1981-03-31
DK
DK144981A
patent/DK153547C/en
not_active
IP Right Cessation

1981-03-31
CA
CA000374331A
patent/CA1152992A/en
not_active
Expired

1981-04-01
AT
AT81400520T
patent/ATE8389T1/en
active

1981-04-01
EP
EP81400520A
patent/EP0037344B1/en
not_active
Expired

1981-04-01
US
US06/250,952
patent/US4330544A/en
not_active
Expired – Lifetime

1981-04-01
GR
GR64550A
patent/GR75618B/el
unknown

1981-04-01
DE
DE8181400520T
patent/DE3164667D1/en
not_active
Expired

Also Published As

Publication number
Publication date

JPS56152465A
(en)

1981-11-26

ES8201977A1
(en)

1982-01-01

ATE8389T1
(en)

1984-07-15

EP0037344A1
(en)

1981-10-07

GR75618B
(en)

1984-08-01

ES500810A0
(en)

1982-01-01

CA1152992A
(en)

1983-08-30

DK153547B
(en)

1988-07-25

AU6892681A
(en)

1981-10-08

US4330544A
(en)

1982-05-18

DE3164667D1
(en)

1984-08-16

FR2479219A1
(en)

1981-10-02

FR2479219B1
(en)

1982-04-09

DK153547C
(en)

1988-12-05

JPH0446953B2
(en)

1992-07-31

IE810728L
(en)

1981-10-01

DK144981A
(en)

1981-10-02

IE51963B1
(en)

1987-05-13

EP0037344B1
(en)

1984-07-11

Contact information