AU571090B2

AU571090B2 – 3, 17beta-estriol diesters
– Google Patents

AU571090B2 – 3, 17beta-estriol diesters
– Google Patents
3, 17beta-estriol diesters

Info

Publication number
AU571090B2

AU571090B2
AU43301/85A
AU4330185A
AU571090B2
AU 571090 B2
AU571090 B2
AU 571090B2
AU 43301/85 A
AU43301/85 A
AU 43301/85A
AU 4330185 A
AU4330185 A
AU 4330185A
AU 571090 B2
AU571090 B2
AU 571090B2
Authority
AU
Australia
Prior art keywords
estriol
17beta
diesters
esters
surpass
Prior art date
1984-05-16
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Ceased

Application number
AU43301/85A
Other versions

AU4330185A
(en

Inventor
Sybille Dr. Beier
Dieter Bittler
Walter Elger
Henry Laurent
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bayer Pharma AG

Original Assignee
Schering AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1984-05-16
Filing date
1985-06-04
Publication date
1988-03-31

1985-06-04
Application filed by Schering AG
filed
Critical
Schering AG

1986-01-09
Publication of AU4330185A
publication
Critical
patent/AU4330185A/en

1988-03-31
Application granted
granted
Critical

1988-03-31
Publication of AU571090B2
publication
Critical
patent/AU571090B2/en

2005-06-04
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07J—STEROIDS

C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane

C07J1/0051—Estrane derivatives

C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa

C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified

C07J1/0074—Esters

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07J—STEROIDS

C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 – C07J43/00

Abstract

Estriol esters of Formula I (I) wherein R, in each case, means the residue of a monocarboxylic acid of 2-10 carbon atoms. The novel estriol esters surpass estriol in strength and duration of estrogen effect.

AU43301/85A
1984-05-16
1985-06-04
3, 17beta-estriol diesters

Ceased

AU571090B2
(en)

Applications Claiming Priority (2)

Application Number
Priority Date
Filing Date
Title

DE3418562

1984-05-16

DE3418562

1984-05-16

Publications (2)

Publication Number
Publication Date

AU4330185A

AU4330185A
(en)

1986-01-09

AU571090B2
true

AU571090B2
(en)

1988-03-31

Family
ID=6236262
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU43301/85A
Ceased

AU571090B2
(en)

1984-05-16
1985-06-04
3, 17beta-estriol diesters

Country Status (19)

Country
Link

US
(1)

US4681875A
(en)

EP
(1)

EP0163596B1
(en)

JP
(1)

JPS6194A
(en)

CN
(1)

CN1003856B
(en)

AT
(1)

ATE55610T1
(en)

AU
(1)

AU571090B2
(en)

CA
(1)

CA1285274C
(en)

DD
(1)

DD232920A5
(en)

DE
(1)

DE3579193D1
(en)

DK
(1)

DK159323C
(en)

ES
(1)

ES8603193A1
(en)

FI
(1)

FI83087C
(en)

GR
(1)

GR851164B
(en)

HU
(1)

HU191789B
(en)

IE
(1)

IE58116B1
(en)

IL
(1)

IL75206A
(en)

NO
(2)

NO160520C
(en)

PT
(1)

PT80472B
(en)

ZA
(1)

ZA853715B
(en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

DE3510555A1
(en)

*

1985-03-21
1986-09-25
Schering AG, 1000 Berlin und 4709 Bergkamen

ESTRIOLESTER

DE3511587A1
(en)

*

1985-03-27
1986-10-02
Schering AG, Berlin und Bergkamen, 1000 Berlin

GLYCOESTER OF ESTRADIOL AND ESTRIOLS

US4757062A
(en)

*

1985-11-01
1988-07-12
E. I. Du Pont De Nemours And Company
Substituted benzoate ester prodrugs of estrogens

JPH03500049A
(en)

*

1987-08-25
1991-01-10
ジー、ケルビン・ダブリュー

Compositions and methods for alleviating stress, anxiety and seizure activity

US5208227A
(en)

*

1987-08-25
1993-05-04
University Of Southern California
Method, compositions, and compounds for modulating brain excitability

ES2081823T3
(en)

1988-10-27
1996-03-16
Schering Ag

AGENT FOR TRANSDERMIC APPLICATION, CONTAINING GESTODEN.

JPH07101977A
(en)

*

1993-10-05
1995-04-18
Kureha Chem Ind Co Ltd
New estradiol derivative with reduced hormone action and growth factor inhibitor thereof

US5861431A
(en)

*

1995-06-07
1999-01-19
Iotek, Inc.
Incontinence treatment

EP1358881A1
(en)

*

2002-04-30
2003-11-05
Schering Aktiengesellschaft
Use of biogenic estriol diester prodrugs for the treatment of autoimmune diseases

KR101582726B1
(en)

*

2013-12-27
2016-01-06
재단법인대구경북과학기술원
Apparatus and method for recognizing distance of stereo type

Citations (3)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB879014A
(en)

*

1959-05-29
1961-10-04

Organon Labor Ltd

Water-soluble derivatives of estriol

GB1006802A
(en)

*

1962-04-12
1965-10-06

Mochida Seiyaku Kabushikikaish

Estra-1,3,5(10)-triene-3,16,17-triol tripropionate

AU418344B2
(en)

*

1966-10-12
1971-10-27

Gonatriene derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

BE788500A
(en)

*

1971-09-10
1973-03-07
Roussel Uclaf

NEW AROMATIC STEROIDS AND PREPARATION PROCESS

JPS5124511A
(en)

*

1974-08-23
1976-02-27
Nisshin Steel Co Ltd

NETSUKANATSUENKOTAINO KEISHAREIKYAKUHO

IT1037092B
(en)

*

1974-12-13
1979-11-10
Farmila Farma Milano

TETRAIDOPIRANIL ETHERS OF EXTRUGENS

1985

1985-05-08
FI
FI851826A
patent/FI83087C/en
not_active
IP Right Cessation

1985-05-10
AT
AT85730070T
patent/ATE55610T1/en
not_active
IP Right Cessation

1985-05-10
EP
EP85730070A
patent/EP0163596B1/en
not_active
Expired – Lifetime

1985-05-10
DE
DE8585730070T
patent/DE3579193D1/en
not_active
Expired – Lifetime

1985-05-11
CN
CN85103839.5A
patent/CN1003856B/en
not_active
Expired

1985-05-13
DD
DD85276276A
patent/DD232920A5/en
not_active
IP Right Cessation

1985-05-14
HU
HU851816A
patent/HU191789B/en
not_active
IP Right Cessation

1985-05-14
DK
DK213385A
patent/DK159323C/en
not_active
IP Right Cessation

1985-05-14
GR
GR851164A
patent/GR851164B/el
unknown

1985-05-14
ES
ES543152A
patent/ES8603193A1/en
not_active
Expired

1985-05-15
JP
JP60101663A
patent/JPS6194A/en
active
Granted

1985-05-15
PT
PT80472A
patent/PT80472B/en
active
IP Right Revival

1985-05-15
IE
IE120685A
patent/IE58116B1/en
unknown

1985-05-15
NO
NO851966A
patent/NO160520C/en
unknown

1985-05-15
CA
CA000481616A
patent/CA1285274C/en
not_active
Expired – Lifetime

1985-05-15
ZA
ZA853715A
patent/ZA853715B/en
unknown

1985-05-16
US
US06/734,737
patent/US4681875A/en
not_active
Expired – Fee Related

1985-05-16
IL
IL75206A
patent/IL75206A/en
not_active
IP Right Cessation

1985-06-04
AU
AU43301/85A
patent/AU571090B2/en
not_active
Ceased

1986

1986-01-22
NO
NO86860233A
patent/NO161375C/en
unknown

Patent Citations (3)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

GB879014A
(en)

*

1959-05-29
1961-10-04
Organon Labor Ltd
Water-soluble derivatives of estriol

GB1006802A
(en)

*

1962-04-12
1965-10-06
Mochida Seiyaku Kabushikikaish
Estra-1,3,5(10)-triene-3,16,17-triol tripropionate

AU418344B2
(en)

*

1966-10-12
1971-10-27

Gonatriene derivatives

Also Published As

Publication number
Publication date

FI851826A0
(en)

1985-05-08

IL75206A
(en)

1989-03-31

CA1285274C
(en)

1991-06-25

NO860233L
(en)

1985-11-18

JPS6194A
(en)

1986-01-06

DK213385D0
(en)

1985-05-14

DK213385A
(en)

1985-11-17

PT80472A
(en)

1985-06-01

ZA853715B
(en)

1986-01-29

NO160520B
(en)

1989-01-16

FI83087B
(en)

1991-02-15

CN1003856B
(en)

1989-04-12

GR851164B
(en)

1985-11-25

IE58116B1
(en)

1993-07-14

ES543152A0
(en)

1986-01-01

ATE55610T1
(en)

1990-09-15

HUT37943A
(en)

1986-03-28

DK159323C
(en)

1991-03-25

CN85103839A
(en)

1986-12-24

FI83087C
(en)

1991-05-27

EP0163596A1
(en)

1985-12-04

NO161375C
(en)

1989-08-09

DK159323B
(en)

1990-10-01

DD232920A5
(en)

1986-02-12

AU4330185A
(en)

1986-01-09

NO851966L
(en)

1985-11-18

US4681875A
(en)

1987-07-21

IL75206A0
(en)

1985-09-29

NO160520C
(en)

1989-04-26

ES8603193A1
(en)

1986-01-01

HU191789B
(en)

1987-04-28

EP0163596B1
(en)

1990-08-16

JPH0564637B2
(en)

1993-09-16

DE3579193D1
(en)

1990-09-20

PT80472B
(en)

1987-08-19

FI851826L
(en)

1985-11-17

NO161375B
(en)

1989-05-02

IE851206L
(en)

1985-11-16

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(en)

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(en)

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Legal Events

Date
Code
Title
Description

2000-01-20
MK14
Patent ceased section 143(a) (annual fees not paid) or expired

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