AU6536086A - Creation of Inventions and Patents with Artificial Intelligence

AU6536086A – Bicyclic sulphonamide derivatives
– Google Patents

AU6536086A – Bicyclic sulphonamide derivatives
– Google Patents
Bicyclic sulphonamide derivatives

Info

Publication number
AU6536086A

AU6536086A
AU65360/86A
AU6536086A
AU6536086A
AU 6536086 A
AU6536086 A
AU 6536086A
AU 65360/86 A
AU65360/86 A
AU 65360/86A
AU 6536086 A
AU6536086 A
AU 6536086A
AU 6536086 A
AU6536086 A
AU 6536086A
Authority
AU
Australia
Prior art keywords
bicyclic
sulphonamide derivatives
sulphonamide
derivatives
bicyclic sulphonamide
Prior art date
1985-11-18
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Granted

Application number
AU65360/86A
Other versions

AU595554B2
(en

Inventor
Nobuhiro Haga
Sanji Hagishita
Susumu Kamata
Kenji Kawada
Masayuki Narisada
Mitsuaki Ohtani
Kaoru Seno
Tatsuo Tsuri
Tadahiko Tsushima
Fumihiko Watanabe
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Shionogi and Co Ltd

Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1985-11-18
Filing date
1986-11-18
Publication date
1987-05-21

1986-11-18
Application filed by Shionogi and Co Ltd
filed
Critical
Shionogi and Co Ltd

1987-05-21
Publication of AU6536086A
publication
Critical
patent/AU6536086A/en

1990-04-05
Application granted
granted
Critical

1990-04-05
Publication of AU595554B2
publication
Critical
patent/AU595554B2/en

2006-11-18
Anticipated expiration
legal-status
Critical

Status
Ceased
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system

C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings

C07D493/08—Bridged systems

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P11/00—Drugs for disorders of the respiratory system

A61P11/08—Bronchodilators

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P7/00—Drugs for disorders of the blood or the extracellular fluid

A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

A—HUMAN NECESSITIES

A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE

A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS

A61P9/00—Drugs for disorders of the cardiovascular system

A61P9/08—Vasodilators for multiple indications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members

C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom

C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms

C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms

C07D213/32—Sulfur atoms

C07D213/34—Sulfur atoms to which a second hetero atom is attached

Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS

Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE

Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS

Y02P20/00—Technologies relating to chemical industry

Y02P20/50—Improvements relating to the production of bulk chemicals

Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

AU65360/86A
1985-11-18
1986-11-18
Bicyclic sulphonamide derivatives

Ceased

AU595554B2
(en)

Applications Claiming Priority (10)

Application Number
Priority Date
Filing Date
Title

JP60-259154

1985-11-18

JP25915485

1985-11-18

JP61-30130

1986-02-13

JP3013086

1986-02-13

JP11559986

1986-05-19

JP61-115599

1986-05-19

JP61-129011

1986-06-03

JP12901186

1986-06-03

JP61-169257

1986-07-17

JP16925786

1986-07-17

Publications (2)

Publication Number
Publication Date

AU6536086A
true

AU6536086A
(en)

1987-05-21

AU595554B2

AU595554B2
(en)

1990-04-05

Family
ID=27521199
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

AU65360/86A
Ceased

AU595554B2
(en)

1985-11-18
1986-11-18
Bicyclic sulphonamide derivatives

Country Status (20)

Country
Link

US
(6)

US4861913A
(en)

EP
(1)

EP0226346B1
(en)

JP
(1)

JPS63139161A
(en)

CN
(1)

CN1019194B
(en)

AR
(1)

AR245102A1
(en)

AT
(1)

ATE66207T1
(en)

AU
(1)

AU595554B2
(en)

CA
(1)

CA1278577C
(en)

DE
(1)

DE3680884D1
(en)

DK
(1)

DK169918B1
(en)

ES
(1)

ES2051693T3
(en)

FI
(1)

FI90064C
(en)

GB
(1)

GB2184118B
(en)

GR
(1)

GR3002489T3
(en)

HU
(1)

HU203078B
(en)

IE
(1)

IE58988B1
(en)

IL
(1)

IL80670A
(en)

NO
(1)

NO165442C
(en)

NZ
(1)

NZ218115A
(en)

PT
(1)

PT83744B
(en)

Families Citing this family (42)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

CA1278577C
(en)

1985-11-18
1991-01-02
Tatsuo Tsuri
Bicyclic sulfonamide derivatives

GB8708233D0
(en)

1987-04-07
1987-05-13
Smith Kline French Lab
Pharmaceutically active compounds

CA1294974C
(en)

1987-05-08
1992-01-28
Sanji Hagishita
Bicyclic sulfonamide derivatives and process therefor

GB8717374D0
(en)

1987-07-22
1987-08-26
Smith Kline French Lab
Pharmaceutically active compounds

EP0516181A1
(en)

1987-10-23
1992-12-02
Ono Pharmaceutical Co., Ltd.
Novel sulfonamide derivatives

JP2565746B2
(en)

1987-10-23
1996-12-18
小野薬品工業株式会社

New carbocyclic sulfonamide derivative

EP0312906A3
(en)

1987-10-23
1990-09-05
Ono Pharmaceutical Co., Ltd.
Novel sulfonamide derivatives

EP0516180A1
(en)

1988-04-19
1992-12-02
Ono Pharmaceutical Co., Ltd.
Novel sulfonamide derivatives

CA1332607C
(en)

1988-07-19
1994-10-18
Masayuki Narisada
Alkenyltetrazole derivatives

US5047574A
(en)

1988-12-14
1991-09-10
Shionogi & Co., Ltd.
Certain optically active mono esters of dicarboxylic acids

US5241104A
(en)

1988-12-14
1993-08-31
Shionogi & Co., Ltd.
Mono ester of dicarboxylic acid and process thereof

US5117039A
(en)

1988-12-14
1992-05-26
Shionogi & Co., Ltd.
Monoesters of arylacetic acid and the process thereof

KR0138528B1
(en)

1988-12-14
1998-05-01
Shionogi Seiyaku Kk
Preparation of 2,3-trans-1,4-bridged cyclohexane sulfonamide derivatives

US5008409A
(en)

1988-12-14
1991-04-16
Shionogi & Co., Ltd.
Process for preparing 1,4-bridged cyclohexane carboxylic acid derivatives

JP2756689B2
(en)

1989-02-20
1998-05-25
塩野義製薬株式会社

Substituted hexenoic acid derivatives

US5124462A
(en)

1989-10-18
1992-06-23
Shiongi & Co., Ltd.
Preparation of norbornyl sulfonamide derivatives

JP2891740B2
(en)

1990-03-30
1999-05-17
塩野義製薬株式会社

Method for producing optically active norbornane-based amine derivative

US5763647A
(en)

1990-03-30
1998-06-09
Shionogi & Co., Ltd.
Preparation of optically active 1,4-bridged-cyclohexane carboxylic acid derivatives

JP2984077B2
(en)

1990-04-19
1999-11-29
塩野義製薬株式会社

Sulfonylamino-substituted bicyclo ring system hydroxamic acid derivatives

FR2665440B1
(en)

1990-07-31
1994-02-04
Lipha

NOVEL SUBSTITUTED CYCLOALKYLSULFONAMIDES, METHODS OF PREPARATION AND MEDICAMENTS CONTAINING THEM.

US5550248A
(en)

1990-11-29
1996-08-27
E.R. Squibb & Sons, Inc.
Substituted stryl heterocyclic amido prostaglandin analogs

US5334369A
(en)

1991-06-11
1994-08-02
Medical University Of South Carolina
Platelet receptor antagonists useful in detecting intravascular platelet aggregation

US5827868A
(en)

1991-10-07
1998-10-27
E. R. Squibb & Sons, Inc.
Prostaglandin analogs

CA2113787A1
(en)

1993-01-29
1994-07-30
Nobuyuki Hamanaka
Carbocyclic sulfonamides

ES2270438T3
(en)

1995-06-21
2007-04-01
SHIONOGI & CO., LTD.

BICYCLE AMINO DERIVATIVES AND PGD2 AGONIST CONTAINING THE SAME.

IL118727A
(en)

1995-06-29
2003-01-12
Lilly Co Eli
(-)-2-spiro-5-hydantoinbicyclo [3.1.0] hexane-6-carboxylic acid, salts thereof and use thereof for the preparation of (+)-(2) aminobicyclo [3.1.0] hexane-2,6-dicarboxylic acid

AU703093B2
(en)

1995-11-16
1999-03-18
Eli Lilly And Company
Excitatory amino acid receptor antagonists

ZA969485B
(en)

1995-11-16
1998-05-12
Lilly Co Eli
Excitatory amino acid receptor antagonists.

EP0906754B1
(en)

1996-04-26
2002-12-11
Shionogi & Co., Ltd.
Rapid-release s1452 tablets

ATE295360T1
(en)

1996-12-12
2005-05-15
Shionogi & Co

CONDENSED HETEROCYCLIC BENZENECARBONIC ACID AMIDE DERIVATIVES AND PGD2 ANTAGONISTS CONTAINING SAME

TR199901280T2
(en)

1996-12-13
1999-10-21
Shionogi & Co., Ltd.

Benzothiophenecarboxamide derivatives and PGD2 antagonists containing them.

ZA984040B
(en)

1997-05-15
1998-11-20
Ono Pharmaceutical Co
Benzenesulfonamide compounds

US6225336B1
(en)

1997-09-19
2001-05-01
Shionogi & Co., Ltd.
Compounds having [2.2.1] bicyclo skeleton

EP1528060A1
(en)

1998-03-31
2005-05-04
Shionogi & Co., Ltd.
Process for preparing 5-hydroxy[b]thiophene-3-carboxylic acid derivatives

PA8469401A1
(en)

1998-04-10
2000-05-24
Pfizer Prod Inc

BICYCLE DERIVATIVES OF HYDROXAMIC ACID

WO2000030683A1
(en)

1998-11-19
2000-06-02
Shionogi & C0., Ltd.
Preventives and/or remedies for central nervous system diseases containing compounds having txa2 receptor antagonism and/or txa2 synthase inhibitory effect

JP2000351729A
(en)

1999-06-08
2000-12-19
Shionogi & Co Ltd
Percutaneous absorption preparation of thromboxane a2 receptor antagonist

ATE405257T1
(en)

1999-11-26
2008-09-15
Shionogi & Co

NPYY5 ANTAGONISTS

WO2001070677A1
(en)

2000-03-20
2001-09-27
Merck Sharp & Dohme Limited
Sulphonamido-substituted bridged bicycloalkyl derivatives

US6727277B1
(en)

2002-11-12
2004-04-27
Kansas State University Research Foundation
Compounds affecting cholesterol absorption

JP5861884B2
(en)

2012-03-29
2016-02-16
荒川化学工業株式会社

Method for producing exo-type norbornene compound

CN110563006A
(en)

2019-09-25
2019-12-13
新乡市锦源化工有限公司
Sodium bisulfite treatment method in production of para-ester

Family Cites Families (14)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

IL33813A
(en)

1969-02-14
1973-10-25
Sparamedica Ag
Bornanocarboxamides and their salts,and their preparation

US3988362A
(en)

1972-08-10
1976-10-26
Hoffmann-La Roche Inc.
Intermediates for preparation of 2,2,3-endotrimethyl-7-anti-amino-norbornanes

JPH025739B2
(en)

1979-01-05
1990-02-05
Nat Res Dev

EP0044711B1
(en)

1980-07-22
1984-03-14
Ono Pharmaceutical Co., Ltd.
9,11-methano-13-aza-11a-carbathrombanoic acid analogues and pharmaceutical use thereof

JPS5813551A
(en)

1981-07-16
1983-01-26
Ono Pharmaceut Co Ltd
13-azathromboxane analogus compound, its preparation, and remedy for disease caused by thromboxane comprising it as active ingredient

GB2113678B
(en)

1981-12-23
1985-06-19
Nat Res Dev
Prostaglandins

US4456615A
(en)

1982-10-25
1984-06-26
E. R. Squibb & Sons, Inc.
7-Oxabicycloheptane substituted amino prostaglandin analogs and their use in inhibiting platelet aggregation and bronchoconstriction

US4456616A
(en)

1982-12-27
1984-06-26
E. R. Squibb & Sons, Inc.
7-Oxabicycloheptane substituted amino prostaglandin analogs and their use in inhibiting platelet aggregation and bronchoconstriction

US4647585A
(en)

1984-11-08
1987-03-03
E. R. Squibb & Sons, Inc.
Bicycloheptane substituted ethers

US4663336A
(en)

1985-07-01
1987-05-05
E. R. Squibb & Sons, Inc.
7-oxabicycloheptane substituted diamide and its congener prostaglandin analogs useful in the treatment of thrombotic disease

US4654357A
(en)

1985-08-09
1987-03-31
E. R. Squibb & Sons, Inc.
7-oxabicycloheptane substituted sulfonamide prostaglandin analogs

CA1278577C
(en)

1985-11-18
1991-01-02
Tatsuo Tsuri
Bicyclic sulfonamide derivatives

US4734424A
(en)

1986-09-24
1988-03-29
E. R. Squibb & Sons, Inc.
Bicycloheptane substituted diamide and its congener prostaglandin analogs

CA1294974C
(en)

1987-05-08
1992-01-28
Sanji Hagishita
Bicyclic sulfonamide derivatives and process therefor

1986

1986-10-30
CA
CA000521812A
patent/CA1278577C/en
not_active
Expired – Fee Related

1986-10-30
NZ
NZ218115A
patent/NZ218115A/en
unknown

1986-11-05
US
US06/927,823
patent/US4861913A/en
not_active
Expired – Lifetime

1986-11-13
IE
IE300286A
patent/IE58988B1/en
not_active
IP Right Cessation

1986-11-14
PT
PT83744A
patent/PT83744B/en
not_active
IP Right Cessation

1986-11-14
NO
NO864542A
patent/NO165442C/en
not_active
IP Right Cessation

1986-11-16
AR
AR86305933A
patent/AR245102A1/en
active

1986-11-17
FI
FI864675A
patent/FI90064C/en
not_active
IP Right Cessation

1986-11-17
DK
DK549086A
patent/DK169918B1/en
not_active
IP Right Cessation

1986-11-17
JP
JP61273372A
patent/JPS63139161A/en
active
Granted

1986-11-17
IL
IL80670A
patent/IL80670A/en
unknown

1986-11-17
HU
HU864742A
patent/HU203078B/en
not_active
IP Right Cessation

1986-11-18
GB
GB8627561A
patent/GB2184118B/en
not_active
Expired – Fee Related

1986-11-18
CN
CN86108584A
patent/CN1019194B/en
not_active
Expired

1986-11-18
ES
ES86309016T
patent/ES2051693T3/en
not_active
Expired – Lifetime

1986-11-18
EP
EP86309016A
patent/EP0226346B1/en
not_active
Expired – Lifetime

1986-11-18
AT
AT86309016T
patent/ATE66207T1/en
not_active
IP Right Cessation

1986-11-18
AU
AU65360/86A
patent/AU595554B2/en
not_active
Ceased

1986-11-18
DE
DE8686309016T
patent/DE3680884D1/en
not_active
Expired – Fee Related

1989

1989-03-23
US
US07/327,778
patent/US4976891A/en
not_active
Expired – Lifetime

1989-03-23
US
US07/327,772
patent/US4960909A/en
not_active
Expired – Lifetime

1990

1990-04-27
US
US07/516,141
patent/US5043456A/en
not_active
Expired – Lifetime

1990-04-27
US
US07/516,140
patent/US5043451A/en
not_active
Expired – Lifetime

1990-06-20
US
US07/541,491
patent/US5041635A/en
not_active
Expired – Lifetime

1991

1991-08-16
GR
GR91401163T
patent/GR3002489T3/en
unknown

Also Published As

Publication number
Publication date

CN86108584A
(en)

1987-07-29

AU595554B2
(en)

1990-04-05

NO165442C
(en)

1991-02-13

GB8627561D0
(en)

1986-12-17

DK549086D0
(en)

1986-11-17

NZ218115A
(en)

1990-02-26

FI90064C
(en)

1993-12-27

US4976891A
(en)

1990-12-11

IE58988B1
(en)

1993-12-15

JPS63139161A
(en)

1988-06-10

GB2184118B
(en)

1990-01-17

US5043451A
(en)

1991-08-27

ES2051693T3
(en)

1994-07-01

FI864675A0
(en)

1986-11-17

PT83744A
(en)

1986-12-01

HUT44765A
(en)

1988-04-28

GR3002489T3
(en)

1992-12-30

CN1019194B
(en)

1992-11-25

NO864542L
(en)

1987-05-19

IE863002L
(en)

1987-05-18

GB2184118A
(en)

1987-06-17

US4861913A
(en)

1989-08-29

AR245102A1
(en)

1993-12-30

IL80670A0
(en)

1987-02-27

DK549086A
(en)

1987-05-19

FI864675A
(en)

1987-05-19

FI90064B
(en)

1993-09-15

JPH0579060B2
(en)

1993-11-01

EP0226346B1
(en)

1991-08-14

ATE66207T1
(en)

1991-08-15

PT83744B
(en)

1988-08-17

NO165442B
(en)

1990-11-05

US5041635A
(en)

1991-08-20

HU203078B
(en)

1991-05-28

NO864542D0
(en)

1986-11-14

DK169918B1
(en)

1995-04-03

DE3680884D1
(en)

1991-09-19

IL80670A
(en)

1991-06-10

US5043456A
(en)

1991-08-27

EP0226346A1
(en)

1987-06-24

CA1278577C
(en)

1991-01-02

US4960909A
(en)

1990-10-02

Contact information