AU7869081A – Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates
– Google Patents
AU7869081A – Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates
– Google Patents
Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates
Info
Publication number
AU7869081A
AU7869081A
AU78690/81A
AU7869081A
AU7869081A
AU 7869081 A
AU7869081 A
AU 7869081A
AU 78690/81 A
AU78690/81 A
AU 78690/81A
AU 7869081 A
AU7869081 A
AU 7869081A
AU 7869081 A
AU7869081 A
AU 7869081A
Authority
AU
Australia
Prior art keywords
carbon atoms
alkyl
optionally substituted
case
aryl
Prior art date
1980-12-20
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU78690/81A
Other versions
AU547689B2
(en
Inventor
Wilhelm Brandes
Karl Heinz Buchel
Hans-Ludwig Elbe
Paul-Ernst Frohberger
Udo Kraatz
Wolfgang Kramer
Erik Regel
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1980-12-20
Filing date
1981-12-21
Publication date
1982-07-01
1981-12-21
Application filed by Bayer AG
filed
Critical
Bayer AG
1982-07-01
Publication of AU7869081A
publication
Critical
patent/AU7869081A/en
1985-10-31
Application granted
granted
Critical
1985-10-31
Publication of AU547689B2
publication
Critical
patent/AU547689B2/en
2001-12-21
Anticipated expiration
legal-status
Critical
Status
Ceased
legal-status
Critical
Current
Links
Espacenet
Global Dossier
Discuss
Classifications
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
A—HUMAN NECESSITIES
A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
A—HUMAN NECESSITIES
A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
A01N43/647—Triazoles; Hydrogenated triazoles
A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
A—HUMAN NECESSITIES
A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
A01N47/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
C07C49/04—Saturated compounds containing keto groups bound to acyclic carbon atoms
C07C49/16—Saturated compounds containing keto groups bound to acyclic carbon atoms containing halogen
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
C—CHEMISTRY; METALLURGY
C07—ORGANIC CHEMISTRY
C07D—HETEROCYCLIC COMPOUNDS
C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Abstract
1. Substituted 1-azolyl-butan-2-ones of the formula see diagramm : EP0054865,P68,F1 in which Az represents 1,2,4-triazol-1-yl and 4-yl or imidazol-1-yl ; R**1 represents hydrogen, alkyl with 1 to 12 and alkenyl and alkinyl with in each case 2 to 12 carbon atoms, and represents optionally C1 -C4 -alkyl-substituted cycloalkyl with 3 to 7 carbon atoms or cycloalkylalkyl with 3 to 7 carbon atoms in the cycloalkyl part and 1 to 4 carbon atoms in the alkyl part, and represents optionally substituted phenoxyalkyl with 1 to 4 carbon atoms in the alkyl part or optionally substituted phenylalkyl with 1 to 4 carbon atoms in the alkyl part, the phenyl substituents to be mentioned in each case being : halogen ; alkyl, alkoxy and alkylthio with in each case 1 to 6 carbon atoms ; cyclohexyl ; dialkylamino with in each case 1 to 4 carbon atoms in each alkyl part ; halogenoalkyl, halogenoalkoxy and halogenoalkylthio with in each case 1 to 4 carbon atoms and 1 to 5 identical or different halogen atoms ; nitro ; cyano ; alkoxycarbonyl with 1 to 4 carbon atoms in the alkyl part ; and optionally halogensubstituted phenyl and phenoxy ; and the grouping -CO-NR**6 R**7 ; n represents the numbers 0 or 1, R**2 represents cyano or the groupings -X-R**3 and -CO-NR**4 R**5 , and, in the case where n does not represent 0 at the same time as R**1 represents hydrogen and Az represents 1,2,4-triazolyl, also additionally represents optionally substituted aryl with 6 to 10 carbon atoms, possible substituents being the aryl substituents already mentioned under R**1 , and represents alkoxycarbonyl with 1 to 4 carbon atoms in the alkyl part ; X represents oxygen, sulphur, or the SO or SO2 group, R**3 represents alkyl with 1 to 6 carbon atoms, halogenoalkyl with 1 to 4 carbon atoms and 1 to 5 identical or different halogen atoms, and represents optionally substituted aryl with 6 to 10 carbon atoms and aralkyl with 6 to 10 carbon atoms in the aryl part and 1 to 2 carbon atoms in the alkyl part, possible substituents being the aryl substituents already mentioned under R**1 ; R**4 represents hydrogen, alkyl with 1 to 4 carbon atoms or optionally substituted aryl with 1 to 10 carbon atoms, possible substituents being the aryl substituents already mentioned under R**1 ; R**5 represents hydrogen or alkyl with 1 to 4 carbon atoms ; and R**6 and R**7 represent hydrogen, alkyl with 1 to 4 carbon atoms, phenyl which is optionally substituted by halogen and alkyl with 1 to 4 carbon atoms, or both together with the adjacent nitrogen atom represent a saturated 5- or 6-membered ring system which can contain nitrogen or oxygen as additional hetero atoms ; and plant-tolerated acid addition salts and metal salt complexes thereof.
AU78690/81A
1980-12-20
1981-12-21
Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates
Ceased
AU547689B2
(en)
Applications Claiming Priority (2)
Application Number
Priority Date
Filing Date
Title
DE19803048266
DE3048266A1
(en)
1980-12-20
1980-12-20
SUBSTITUTED 1-AZOLYL-BUTANE-2ONE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS FUNGICIDES AND AS INTERMEDIATE PRODUCTS
DE30482667
1980-12-20
Publications (2)
Publication Number
Publication Date
AU7869081A
true
AU7869081A
(en)
1982-07-01
AU547689B2
AU547689B2
(en)
1985-10-31
Family
ID=6119802
Family Applications (1)
Application Number
Title
Priority Date
Filing Date
AU78690/81A
Ceased
AU547689B2
(en)
1980-12-20
1981-12-21
Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates
Country Status (15)
Country
Link
EP
(1)
EP0054865B1
(en)
JP
(1)
JPS57128676A
(en)
AT
(1)
ATE18213T1
(en)
AU
(1)
AU547689B2
(en)
BR
(1)
BR8108274A
(en)
CA
(1)
CA1178587A
(en)
DE
(2)
DE3048266A1
(en)
DK
(1)
DK563081A
(en)
EG
(1)
EG15306A
(en)
ES
(1)
ES508134A0
(en)
GR
(1)
GR77634B
(en)
HU
(1)
HU189549B
(en)
IL
(1)
IL64572A
(en)
PT
(1)
PT74109B
(en)
ZA
(1)
ZA818757B
(en)
Families Citing this family (16)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
DE3209431A1
(en)
*
1982-03-16
1983-09-22
Bayer Ag, 5090 Leverkusen
PHENOXYPROPYLTRIAZOLYL KETONES AND CARBINOLS, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS FUNGICIDES
DE3229274A1
(en)
*
1982-08-05
1984-02-09
Bayer Ag, 5090 Leverkusen
SUBSTITUTED AZOLYLVINYL KETONES AND CARBINOLS
DE3229273A1
(en)
*
1982-08-05
1984-02-09
Bayer Ag, 5090 Leverkusen
SUBSTITUTED AZOLYLALLYL KETONES AND CARBINOLS
DE3313941A1
(en)
*
1983-04-15
1984-10-18
Schering AG, 1000 Berlin und 4709 Bergkamen
4-AZOLYL-PENTANNITRILE, METHOD FOR THE PRODUCTION OF THESE COMPOUNDS AND THE BIOCIDES CONTAINING THEM
DE3322526A1
(en)
*
1983-06-23
1985-01-10
Basf Ag, 6700 Ludwigshafen
FUNGICIDAL AZOL COMPOUNDS, THEIR PRODUCTION AND USE
DE3329128A1
(en)
*
1983-08-11
1985-02-28
Bayer Ag, 5090 Leverkusen
3-CYCLOALKYL-1- (1,3-DIOXAN-5-YL) -2- (1,2,4-TRIAZOL-1-YL) -PROPAN-1-ONE AND -PROPAN-1-OLE
DE3336861A1
(en)
*
1983-10-11
1985-04-25
Bayer Ag, 5090 Leverkusen
AZOLYL-TETRAHYDROFURAN-2-YLIDEN-METHANE DERIVATIVES
DE3434158A1
(en)
*
1984-09-18
1986-03-20
Bayer Ag, 5090 Leverkusen
SUBSTITUTED 1,1-BIS-AZOLYL-BUTAN-2-ONE AND -OLE
DE3702962A1
(en)
*
1987-01-31
1988-08-11
Bayer Ag
PYRIMIDINE DERIVATIVE-BASED PEST CONTROL
DE3725397A1
(en)
*
1987-07-31
1989-02-09
Bayer Ag
1,4-DISUBSTITUTED 1-AZOLYL-3,3-DIMETHYLBUTANE DERIVATIVES
DE3813253A1
(en)
*
1988-04-20
1989-11-02
Bayer Ag
SUBSTITUTED TRIAZOLYL METHYLCARBINOLS
USRE37303E1
(en)
*
1992-01-10
2001-07-31
Institut National Del La Sante Et De La Recherche Medicale
Imidazole compounds and their therapeutic applications
FR2686084B1
(en)
*
1992-01-10
1995-12-22
Bioprojet Soc Civ
NEW IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATIONS.
DE4222542A1
(en)
*
1992-07-09
1994-01-13
Bayer Ag
Triazolyl butane derivatives
DE4222541A1
(en)
*
1992-07-09
1994-01-13
Bayer Ag
Triazolyl butane derivatives
DE4318916A1
(en)
*
1993-06-07
1994-12-08
Bayer Ag
Cyclobutylazole
Family Cites Families (2)
* Cited by examiner, † Cited by third party
Publication number
Priority date
Publication date
Assignee
Title
DE2842137A1
(en)
*
1978-09-28
1980-04-17
Bayer Ag
HALOGENED 1-AZOLYL-1-FLUORPHENOXYBUTANE DERIVATIVES, METHODS FOR THE PRODUCTION THEREOF AND THEIR USE AS FUNGICIDES
DE2951164A1
(en)
*
1979-12-19
1981-07-16
Bayer Ag, 5090 Leverkusen
SUBSTITUTED TRIAZOLYL METHYL-TERT.-BUTYL-KETONE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A PLANT PROTECTANT AND AS AN INTERMEDIATE PRODUCT
1980
1980-12-20
DE
DE19803048266
patent/DE3048266A1/en
not_active
Withdrawn
1981
1981-12-10
PT
PT74109A
patent/PT74109B/en
unknown
1981-12-11
EP
EP81110365A
patent/EP0054865B1/en
not_active
Expired
1981-12-11
DE
DE8181110365T
patent/DE3173926D1/en
not_active
Expired
1981-12-11
AT
AT81110365T
patent/ATE18213T1/en
not_active
IP Right Cessation
1981-12-17
IL
IL64572A
patent/IL64572A/en
unknown
1981-12-18
JP
JP56203841A
patent/JPS57128676A/en
active
Pending
1981-12-18
ZA
ZA818757A
patent/ZA818757B/en
unknown
1981-12-18
HU
HU813865A
patent/HU189549B/en
not_active
IP Right Cessation
1981-12-18
BR
BR8108274A
patent/BR8108274A/en
unknown
1981-12-18
ES
ES508134A
patent/ES508134A0/en
active
Granted
1981-12-18
CA
CA000392632A
patent/CA1178587A/en
not_active
Expired
1981-12-18
DK
DK563081A
patent/DK563081A/en
not_active
Application Discontinuation
1981-12-18
GR
GR66841A
patent/GR77634B/el
unknown
1981-12-20
EG
EG759/81A
patent/EG15306A/en
active
1981-12-21
AU
AU78690/81A
patent/AU547689B2/en
not_active
Ceased
Also Published As
Publication number
Publication date
PT74109A
(en)
1982-01-01
GR77634B
(en)
1984-09-25
EP0054865A1
(en)
1982-06-30
EP0054865B1
(en)
1986-02-26
PT74109B
(en)
1983-05-16
IL64572A
(en)
1985-05-31
AU547689B2
(en)
1985-10-31
EG15306A
(en)
1986-09-30
CA1178587A
(en)
1984-11-27
HU189549B
(en)
1986-07-28
ES8300712A1
(en)
1982-11-01
ATE18213T1
(en)
1986-03-15
ES508134A0
(en)
1982-11-01
BR8108274A
(en)
1982-10-05
ZA818757B
(en)
1982-11-24
DK563081A
(en)
1982-06-21
JPS57128676A
(en)
1982-08-10
IL64572A0
(en)
1982-03-31
DE3048266A1
(en)
1982-07-29
DE3173926D1
(en)
1986-04-03
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