GB1112347A

GB1112347A – Salts of organic bases with n-carbamyl-l-glutamic acid
– Google Patents

GB1112347A – Salts of organic bases with n-carbamyl-l-glutamic acid
– Google Patents
Salts of organic bases with n-carbamyl-l-glutamic acid

Info

Publication number
GB1112347A

GB1112347A
GB3590065A
GB3590065A
GB1112347A
GB 1112347 A
GB1112347 A
GB 1112347A
GB 3590065 A
GB3590065 A
GB 3590065A
GB 3590065 A
GB3590065 A
GB 3590065A
GB 1112347 A
GB1112347 A
GB 1112347A
Authority
GB
United Kingdom
Prior art keywords
carbamyl
lysine
glutamic acid
acid
salt
Prior art date
1965-08-20
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
GB3590065A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Individual

Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1965-08-20
Filing date
1965-08-20
Publication date
1968-05-01

1965-08-20
Application filed by Individual
filed
Critical
Individual

1965-08-20
Priority to GB3590065A
priority
Critical
patent/GB1112347A/en

1968-05-01
Publication of GB1112347A
publication
Critical
patent/GB1112347A/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS

C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups

C07C275/04—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms

C07C275/06—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton

C07C275/16—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton being further substituted by carboxyl groups

Abstract

The invention comprises the salts of N-carbamyl-l-glumatic acid with organic bases other than lysine, the neutral salt of N-carbamyl-l-glutamic acid with lysine and the acid salt of N-carbamyl-l-glutamic acid with lysine in the pure state having a melting point of 191-3 DEG C. and an optical rotation of +11.7 DEG , which are prepared by salifying the acid with the appropriate organic base in an aqueous or alcoholic medium at room temperature or at about 80-90 DEG C. Suitable organic bases mentioned are morpholine, methylglucamine, amphetamine, pyridoxine, choline, arginine, ornithine, piperazine, dimethylaminoethanol and di-isopropylamine.ALSO:The invention comprises pharmaceutical compositions comprising as active ingredient a salt of N-carbamyl-l-glutamic acid with an organic base other than lysine, or the neutral salt of N-carbamyl-l-glutamic acid with lysine, and also pharmaceutical compositions in the form of a sterile injectable solution, suppository, tablet or capsule comprising as active ingredient the acid salt of N-carbamyl-l-glutamic acid with lysine. The compounds possess, in general, a hepatotropic effect and one or more of the following properties:- a favourable effect on growth, a restorative and regenerative action, a reducing effect on hyperammoniaemia, a neuro-regulating and neuro-stimulating action and an anti-fatigue action.

GB3590065A
1965-08-20
1965-08-20
Salts of organic bases with n-carbamyl-l-glutamic acid

Expired

GB1112347A
(en)

Priority Applications (1)

Application Number
Priority Date
Filing Date
Title

GB3590065A

GB1112347A
(en)

1965-08-20
1965-08-20
Salts of organic bases with n-carbamyl-l-glutamic acid

Applications Claiming Priority (1)

Application Number
Priority Date
Filing Date
Title

GB3590065A

GB1112347A
(en)

1965-08-20
1965-08-20
Salts of organic bases with n-carbamyl-l-glutamic acid

Publications (1)

Publication Number
Publication Date

GB1112347A
true

GB1112347A
(en)

1968-05-01

Family
ID=10382790
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

GB3590065A
Expired

GB1112347A
(en)

1965-08-20
1965-08-20
Salts of organic bases with n-carbamyl-l-glutamic acid

Country Status (1)

Country
Link

GB
(1)

GB1112347A
(en)

Cited By (15)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US7105486B2
(en)

2002-02-22
2006-09-12
New River Pharmaceuticals Inc.
Abuse-resistant amphetamine compounds

US7223735B2
(en)

2003-05-29
2007-05-29
New River Pharmaceuticals Inc.
Abuse resistant lysine amphetamine compounds

WO2008004610A1
(en)

*

2006-07-05
2008-01-10
The University Of Tokyo
Method of treating genetic disease caused by nonsense mutation

US7375083B2
(en)

2003-09-30
2008-05-20
Shire Llc
Pharmaceutical compositions for prevention of overdose or abuse

US7427600B2
(en)

2000-08-22
2008-09-23
Shire Llc
Active agent delivery systems and methods for protecting and administering active agents

US7622441B2
(en)

2002-02-22
2009-11-24
Shire Llc
Sustained release pharmaceutical compounds to prevent abuse of controlled substances

US7655630B2
(en)

2002-02-22
2010-02-02
Shire Llc
Abuse-resistant amphetamine prodrugs

US7659253B2
(en)

2002-02-22
2010-02-09
Shire Llc
Abuse-resistant amphetamine prodrugs

WO2011160259A1
(en)

*

2010-06-24
2011-12-29
上海永颐生物科技有限公司
Use of n-carbamoyl glutamic acid, salts or esters thereof in manufacture of health care products for protecting liver or promoting muscle growth

US8106016B2
(en)

2003-09-30
2012-01-31
Shire Llc
Compounds and compositions for prevention of overdose of oxycodone

US8343927B2
(en)

2001-08-22
2013-01-01
Shire Llc
Pharmaceutical compositions for prevention of overdose or abuse

US8394813B2
(en)

2000-11-14
2013-03-12
Shire Llc
Active agent delivery systems and methods for protecting and administering active agents

CN108017561A
(en)

*

2016-11-04
2018-05-11
武汉武药科技有限公司
A kind of method of refined card glutamic acid

EP3323410A1
(en)

*

2016-11-22
2018-05-23
RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.p.a.
Pharmaceutical parenteral formulation containing carglumic acid

CN112028794A
(en)

*

2019-06-03
2020-12-04
武汉武药科技有限公司
High-purity kaglutamic acid and preparation method thereof

1965

1965-08-20
GB
GB3590065A
patent/GB1112347A/en
not_active
Expired

Cited By (35)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US7427600B2
(en)

2000-08-22
2008-09-23
Shire Llc
Active agent delivery systems and methods for protecting and administering active agents

US8394813B2
(en)

2000-11-14
2013-03-12
Shire Llc
Active agent delivery systems and methods for protecting and administering active agents

US8343927B2
(en)

2001-08-22
2013-01-01
Shire Llc
Pharmaceutical compositions for prevention of overdose or abuse

US7659253B2
(en)

2002-02-22
2010-02-09
Shire Llc
Abuse-resistant amphetamine prodrugs

US7671030B2
(en)

2002-02-22
2010-03-02
Shire Llc
Abuse-resistant amphetamine prodrugs

US7622441B2
(en)

2002-02-22
2009-11-24
Shire Llc
Sustained release pharmaceutical compounds to prevent abuse of controlled substances

US7655630B2
(en)

2002-02-22
2010-02-02
Shire Llc
Abuse-resistant amphetamine prodrugs

US7659254B2
(en)

2002-02-22
2010-02-09
Shire Llc
Abuse-resistant amphetamine prodrugs

US7105486B2
(en)

2002-02-22
2006-09-12
New River Pharmaceuticals Inc.
Abuse-resistant amphetamine compounds

US7713936B2
(en)

2002-02-22
2010-05-11
Shire Llc
Abuse-resistant amphetamine prodrugs

US7662788B2
(en)

2002-02-22
2010-02-16
Shire Llc
Abuse-resistant amphetamine prodrugs

US7671031B2
(en)

2002-02-22
2010-03-02
Shire Llc
Abuse-resistant amphetamine prodrugs

US7718619B2
(en)

2002-02-22
2010-05-18
Shire Llc
Abuse-resistant amphetamine prodrugs

US7674774B2
(en)

2002-02-22
2010-03-09
Shire Llc
Abuse-resistant amphetamine prodrugs

US7678771B2
(en)

2002-02-22
2010-03-16
Shire Llc
Abuse-resistant amphetamine prodrugs

US7678770B2
(en)

2002-02-22
2010-03-16
Shire Llc
Abuse-resistant amphetamine prodrugs

US7687466B2
(en)

2002-02-22
2010-03-30
Shire Llc
Abuse-resistant amphetamine prodrugs

US7687467B2
(en)

2002-02-22
2010-03-30
Shire Llc
Abuse-resistant amphetamine prodrugs

US7700561B2
(en)

2002-02-22
2010-04-20
Shire Llc
Abuse-resistant amphetamine prodrugs

US7723305B2
(en)

2002-02-22
2010-05-25
Shire Llc
Abuse-resistant amphetamine prodrugs

US7223735B2
(en)

2003-05-29
2007-05-29
New River Pharmaceuticals Inc.
Abuse resistant lysine amphetamine compounds

US7662787B2
(en)

2003-05-29
2010-02-16
Shire Llc
Abuse resistant lysine amphetamine compounds

US8106016B2
(en)

2003-09-30
2012-01-31
Shire Llc
Compounds and compositions for prevention of overdose of oxycodone

US7375083B2
(en)

2003-09-30
2008-05-20
Shire Llc
Pharmaceutical compositions for prevention of overdose or abuse

WO2008004610A1
(en)

*

2006-07-05
2008-01-10
The University Of Tokyo
Method of treating genetic disease caused by nonsense mutation

WO2011160259A1
(en)

*

2010-06-24
2011-12-29
上海永颐生物科技有限公司
Use of n-carbamoyl glutamic acid, salts or esters thereof in manufacture of health care products for protecting liver or promoting muscle growth

CN108017561B
(en)

*

2016-11-04
2021-03-30
武汉武药科技有限公司
Method for refining carglutamic acid

CN108017561A
(en)

*

2016-11-04
2018-05-11
武汉武药科技有限公司
A kind of method of refined card glutamic acid

EP3323410A1
(en)

*

2016-11-22
2018-05-23
RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.p.a.
Pharmaceutical parenteral formulation containing carglumic acid

KR20190086662A
(en)

*

2016-11-22
2019-07-23
레코다티인더스트리아치미카이파마슈티카에스.피.에이.

Pharmaceutical parenteral formulations containing carglum acid

WO2018095848A1
(en)

*

2016-11-22
2018-05-31
Recordati Industria Chimica E Farmaceutica S.P.A.
Pharmaceutical parenteral formulation containing carglumic acid

US11103474B2
(en)

2016-11-22
2021-08-31
Recordati Industria Chimica E Farmaceutica S.P.A.
Pharmaceutical parenteral formulation containing carglumic acid

EA039003B1
(en)

*

2016-11-22
2021-11-19
Рекордати Индустрия Кимика Э Фармасеутика С.П.А.
Pharmaceutical parenteral formulation containing carglumic acid

AU2017364135B2
(en)

*

2016-11-22
2023-06-15
Recordati Industria Chimica E Farmaceutica S.P.A.
Pharmaceutical parenteral formulation containing carglumic acid

CN112028794A
(en)

*

2019-06-03
2020-12-04
武汉武药科技有限公司
High-purity kaglutamic acid and preparation method thereof

Similar Documents

Publication
Publication Date
Title

GB1112347A
(en)

1968-05-01

Salts of organic bases with n-carbamyl-l-glutamic acid

SE8300623D0
(en)

1983-02-07

PHARMACEUTICAL COMPOSITION CONTAINING STABLE MICROCRISTALLIN CIS-PLATINA (II) -DIAMMINE DICHLORIDE (CISPLATIN)

ES427079A1
(en)

1976-07-16

Phenothiazine derivatives, compositions thereof and methods of preparation thereof

GB1091089A
(en)

1967-11-15

Organic base salts of n-carbamyl-aspartic acids

DE3773017D1
(en)

1991-10-24

PREPARATION FOR INJECTION CONTAINING NICORANDIL.

IE44339L
(en)

1977-08-07

Piperazine derivatives.

IE44030L
(en)

1977-05-25

Ó-amino-ketones.

GB1225462A
(en)

1971-03-17

GB1362845A
(en)

1974-08-07

Benzyl alcohol derivatives

ES8200363A1
(en)

1981-11-01

Piperidine derivatives of 4,5-dialkyl-3-hydroxy-pyrrole-2-carboxylic acid esters, their preparation and pharmaceutical compositions containing them.

GB1262292A
(en)

1972-02-02

Novel thiazoline derivatives, the preparation thereof and compositions containing the same

GB1231250A
(en)

1971-05-12

GB1512101A
(en)

1978-05-24

Piperazinopyrimidines process for their preparation and use

ATE4808T1
(en)

1983-10-15

PIPERIDINE DERIVATIVES OF 3-HYDROXY-THIOPHEN-2CARBONS[UREESTERS, THEIR PRODUCTION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM.

IL42201A
(en)

1976-02-29

2-((1-benzylcyclopentyl)-imino)pyrrolidine

ES440208A1
(en)

1977-03-01

Piperazine compounds

AR010942A1
(en)

2000-07-12

DERIVED FROM PIPERIDINYLMETILOXAZOLIDINONE, THE PROCEDURES TO PREPARE IT, ITS USE IN THE PREPARATION OF MEDICINES, THE PHARMACEUTICAL PREPARATIONS THAT CONTAIN IT AND A PROCEDURE TO PREPARE THESE PHARMACEUTICAL PREPARATIONS.

GB850298A
(en)

1960-10-05

ª‡,ª‡[(p-chlorophenyl)-(4-pyridyl)] carbinols and method of preparing same

GB1246727A
(en)

1971-09-15

Therapeutic hypotensive compositions comprising 5-alkylpicolinic acids

GB1116775A
(en)

1968-06-12

ªß-hydroxy-acrylic acid derivatives and process for their manufacture

GB486449A
(en)

1938-06-02

Preparation of new therapeutically active diamines

ES455692A1
(en)

1978-01-01

Alkylenedioxy piperazine derivatives

ES369646A1
(en)

1971-06-01

A procedure for the preparation of the derivatives of 5-thzolol carboxylic acid. (Machine-translation by Google Translate, not legally binding)

GB1420976A
(en)

1976-01-14

Pharmaceutical compositions for use in the treatment of certain respiratory diseases or conditions in prematurely born children

FR2451380A1
(en)

1980-10-10

NOVEL DITHIEPINNO (1,4) (2,3-C) PYRROLE DERIVATIVES, THEIR PREPARATION AND THE MEDICINAL PRODUCTS CONTAINING THEM

Download PDF in English

None