GB1242863A

GB1242863A – 2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF
– Google Patents

GB1242863A – 2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF
– Google Patents
2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF

Info

Publication number
GB1242863A

GB1242863A
GB2222368A
GB2222368A
GB1242863A
GB 1242863 A
GB1242863 A
GB 1242863A
GB 2222368 A
GB2222368 A
GB 2222368A
GB 2222368 A
GB2222368 A
GB 2222368A
GB 1242863 A
GB1242863 A
GB 1242863A
Authority
GB
United Kingdom
Prior art keywords
signify
alkoxy
alkyl
quinazolines
thiazolo
Prior art date
1968-05-10
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

Expired

Application number
GB2222368A
Inventor
Kurt Rubinstein
Erik Falch
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pharmacia AS

Original Assignee
Pharmacia AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
1968-05-10
Filing date
1968-05-10
Publication date
1971-08-18

1968-05-10
Application filed by Pharmacia AS
filed
Critical
Pharmacia AS

1968-05-10
Priority to GB2222368A
priority
Critical
patent/GB1242863A/en

1971-08-18
Publication of GB1242863A
publication
Critical
patent/GB1242863A/en

Status
Expired
legal-status
Critical
Current

Links

Espacenet

Global Dossier

Discuss

Classifications

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 – C07D507/00

C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 – C07D507/00 in which the condensed system contains two hetero rings

C07D513/04—Ortho-condensed systems

C—CHEMISTRY; METALLURGY

C07—ORGANIC CHEMISTRY

C07D—HETEROCYCLIC COMPOUNDS

C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings

C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings

C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member

C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

C07D277/16—Sulfur atoms

Abstract

1,242,863. Anti-inflammatory &c. medicines. PHARMACIA AS. 9 May, 1969 [10 May, 1968], No. 22223/68. Heading A5B. [Also in Division C2] Pharmaceutical preparations showing, in particular, anti-inflammatory, analgesic, hypothermic and sedative properties, contain as active ingredient compounds I (including salts and hydrates thereof) wherein X is O, S, NH or alkylidene (especially CH 2 ), R 1 and R 2 signify H, alkyl or alkoxy or R 1 and R 3 together signify alkylidene, R 3 and R 4 signify H, OH, alkyl, alkoxy, CO 2 H, alkoxycarbonyl or CONH 2 and R 5 , R 6 , R 7 and R 8 signify H, halogen, CF 3 , OH, alkyl, alkoxy, alkylthio, CO 2 H, alkoxycarbonyl, CONH 2 , NO 2 CN, NH 2 or dialkylamino. Administration may be orally, parenterally or topically and the other actives can be incorporated in the preparations.

GB2222368A
1968-05-10
1968-05-10
2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF

Expired

GB1242863A
(en)

Priority Applications (1)

Application Number
Priority Date
Filing Date
Title

GB2222368A

GB1242863A
(en)

1968-05-10
1968-05-10
2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF

Applications Claiming Priority (1)

Application Number
Priority Date
Filing Date
Title

GB2222368A

GB1242863A
(en)

1968-05-10
1968-05-10
2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF

Publications (1)

Publication Number
Publication Date

GB1242863A
true

GB1242863A
(en)

1971-08-18

Family
ID=10175918
Family Applications (1)

Application Number
Title
Priority Date
Filing Date

GB2222368A
Expired

GB1242863A
(en)

1968-05-10
1968-05-10
2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF

Country Status (1)

Country
Link

GB
(1)

GB1242863A
(en)

Cited By (8)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4128648A
(en)

*

1978-03-24
1978-12-05
E. R. Squibb & Sons, Inc.
Substituted pyrano[4,3-d]-thiazolo[3,2-a]pyrimidines

US4128647A
(en)

*

1978-03-24
1978-12-05
E. R. Squibb & Sons, Inc.
Substituted thiazolo [3,2-a]-thiopyrano[4,3-d]pyrimidines

US4332802A
(en)

*

1975-12-19
1982-06-01
Boehringer Ingelheim Kg
11-Oxo-11H-pyrido[2,1-b]quinazoline-2-carboxylic acid and salts thereof, antiallergic compositions containing it and methods of suppressing allergic reactions with it

US4486221A
(en)

*

1981-10-28
1984-12-04
Basf Aktiengesellschaft
Thiazolo[2,3-b]quinazolones and their use for influencing plant growth

US5028705A
(en)

*

1987-09-11
1991-07-02
Basf Aktiengesellschaft
Preparation of pyrazolo[5,1-b]quinazolones

EP0564397A1
(en)

*

1992-03-03
1993-10-06
Sandoz Ltd.
Antiatherosclerotic substituted phenylquinazoline derivatives

DE10046728C1
(en)

*

2000-09-21
2001-09-27
Ibfb Gmbh Privates Inst Fuer B
New mercaptomethyl-substituted tricyclic quinazolinone derivatives, are matrix metalloprotease inhibitors useful for treating cancer, rheumatism, inflammatory reactions or allergies

CN108472267A
(en)

*

2015-12-01
2018-08-31
宝洁公司
Compounds and methods for for inhibiting trimethylamine to generate

1968

1968-05-10
GB
GB2222368A
patent/GB1242863A/en
not_active
Expired

Cited By (8)

* Cited by examiner, † Cited by third party

Publication number
Priority date
Publication date
Assignee
Title

US4332802A
(en)

*

1975-12-19
1982-06-01
Boehringer Ingelheim Kg
11-Oxo-11H-pyrido[2,1-b]quinazoline-2-carboxylic acid and salts thereof, antiallergic compositions containing it and methods of suppressing allergic reactions with it

US4128648A
(en)

*

1978-03-24
1978-12-05
E. R. Squibb & Sons, Inc.
Substituted pyrano[4,3-d]-thiazolo[3,2-a]pyrimidines

US4128647A
(en)

*

1978-03-24
1978-12-05
E. R. Squibb & Sons, Inc.
Substituted thiazolo [3,2-a]-thiopyrano[4,3-d]pyrimidines

US4486221A
(en)

*

1981-10-28
1984-12-04
Basf Aktiengesellschaft
Thiazolo[2,3-b]quinazolones and their use for influencing plant growth

US5028705A
(en)

*

1987-09-11
1991-07-02
Basf Aktiengesellschaft
Preparation of pyrazolo[5,1-b]quinazolones

EP0564397A1
(en)

*

1992-03-03
1993-10-06
Sandoz Ltd.
Antiatherosclerotic substituted phenylquinazoline derivatives

DE10046728C1
(en)

*

2000-09-21
2001-09-27
Ibfb Gmbh Privates Inst Fuer B
New mercaptomethyl-substituted tricyclic quinazolinone derivatives, are matrix metalloprotease inhibitors useful for treating cancer, rheumatism, inflammatory reactions or allergies

CN108472267A
(en)

*

2015-12-01
2018-08-31
宝洁公司
Compounds and methods for for inhibiting trimethylamine to generate

Similar Documents

Publication
Publication Date
Title

JO1502B1
(en)

1989-01-25

Novel pharmacological compounds

IT1207994B
(en)

1989-06-01

WATER SOLUBLE SALTS OF ANTI-INFLAMMATORY AND ANALGESIC ADAPTITY COMPOUNDS, THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS.

MY101177A
(en)

1991-07-31

Improvements in pharmaceutically acceptable salts

IE33269L
(en)

1970-02-20

Pyridobenzodiazepines.

GB1321509A
(en)

1973-06-27

Azepine derivatives

IT1208452B
(en)

1989-06-12

PHARMACEUTICAL PREPARATIONS WITH ANALGESIC EFFECT, AS WELL AS THEIR PRODUCTION AND USE

GB1242863A
(en)

1971-08-18

2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF

GB1290818A
(en)

1972-09-27

GB1174051A
(en)

1969-12-10

Aminophenol Derivatives and Analgesic and Antipyretic Compositions

ATE87313T1
(en)

1993-04-15

CEPHEM COMPOUNDS, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM.

GB1298603A
(en)

1972-12-06

Quinazolinone derivatives

GB1248430A
(en)

1971-10-06

4-phenyl-quinazolinone derivatives

IE34744L
(en)

1971-05-17

Biphenyl crotonic acids.

MY101821A
(en)

1992-01-31

Quinazolinediones and pyridopyrimidinediones

GB1256723A
(en)

1971-12-15

GB1332697A
(en)

1973-10-03

Benzodiazepine derivatives

GB1190680A
(en)

1970-05-06

Halocinnamoyl Piperidines and Morpholines and Pharmaceutical Compositions Containing Them

GB1359044A
(en)

1974-07-03

Quinoline derivatives

GB1352392A
(en)

1974-05-08

Phenylisopropylamine derivatives

GB1159271A
(en)

1969-07-23

1,5-Disubstituted Barbituric Acid Derivatives and process for the manufacture thereof

GB1092737A
(en)

1967-11-29

2-methoxy-4-[n-glutarylsulfanilamido]quinazoline and process for preparing the same

GB1159272A
(en)

1969-07-23

1,5-Disubstituted Barbituric Acid Derivatives and process for the manufacture thereof

GB1297043A
(en)

1972-11-22

GB1164579A
(en)

1969-09-17

Amino-Dibenz[b,f][[1,4]Oxazepine-11(10H)-Ones

GB1173985A
(en)

1969-12-10

Indole Derivatives

Download PDF in English

None